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Search Result

Search Results for " adrenergic-receptor "

Targets

Adrenergic Receptor

370

Compounds

31

Natural Products

6

Recombinant Proteins

2

Libraries

Cat No. Product Name Synonyms Targets
T13016 SR59230A Adrenergic Receptor
SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).
T37906 Dibenamine hydrochloride Adrenergic Receptor
Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.
T7065 Tizanidine Adrenergic Receptor
Tizanidine, an α2-adrenergic receptor agonist, suppresses the release of neurotransmitters from central nervous system (CNS) noradrenergic neurons.
T7160 Lofexidine Adrenergic Receptor
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
T40622 Mapenterol hydrochloride Adrenergic Receptor
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
T7045 Clonidine Nexiclon,Catapres,Kapvay Adrenergic Receptor
Clonidine (Kapvay) is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide-scale use for many years, clonidine has not been l...
T8348 Phentolamine Adrenergic Receptor
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
T7728 ACEPROMAZINE MALEATE Dopamine Receptor
ACEPROMAZINE MALEATE is a dopamine receptor antagonist
T19680 Zotepine Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM, 3.3 nM, 7.3 nM, and 8 nM, respectively. Zotepine is a second...
T8899 Metipranolol Adrenergic Receptor
Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta bloc...
T5471 GUANABENZ Adrenergic Receptor
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
T8580 Bupranolol Adrenergic Receptor
Bupranolol is an antagonist of β2-adrenergic receptor and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombotic.
T2524 Dexmedetomidine Adrenergic Receptor
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect of dexmedetomidine is by means of General Anesthesia.
T21640 Talinolol Adrenergic Receptor
(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.
T5511 L-765314 Adrenergic Receptor
L-765314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the role of α1B receptors in the regulation of blood pressure.
T10830 CL 316243 Adrenergic Receptor
CL316243 is a highly potent selective agonist of β3-adrenoceptor, with a EC50 of 3 nM. CL316243 is an effective stimulant of adipocyte lipolysis and increases brown adipose tissue thermogenesis and metabolic rate. CL3162...
T8708 Paroxetine Serotonin Transporter
Paroxetine is a inhibitor of serotonin uptake that is effective in the treatment of depression.
T0279 Metaraminol tartrate Metaradrine tartrate,Metaraminol bitartrate Adrenergic Receptor
Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in the treatment of HYPOTENSION.
T6641 Rilmenidine Phosphate Apoptosis , Adrenergic Receptor , Autophagy , Imidazoline Receptor
Rilmenidine Phosphate is a selective I(1) imidazoline receptor agonist, used to treat hypertension.
T22406 Prazosin Prazosine,Furazosin,Prazocin Adrenergic Receptor
Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T2320 Indacaterol Adrenergic Receptor
Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
T1584 Terbutaline Sulfate Terbutaline hemisulfate Antibacterial , Adrenergic Receptor , Antibiotic
Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
T0165 Urapidil Mediatensyl,Ebrantil,Eupressyl 5-HT Receptor , Adrenergic Receptor
Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T11318 Dopexamine hydrochloride FPL60278AR Adrenergic Receptor
Dopexamine hydrochloride (FPL60278AR) is a β2-adrenergic receptor agonist. Dopexamine can attenuate the inflammatory response and protect against organ injury in the absence of significant effects on hemodynamics or regi...
T12829 Salmeterol GR33343X Adrenergic Receptor
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
T6872 L755507 Adrenergic Receptor , CRISPR/Cas9
L755507 is an effective, selective agonist of β3-AR（IC50=35 nM）.
T12402 Penbutolol sulfate (-)-Terbuclomine Adrenergic Receptor
Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.
T16759 Ritanserin R 55667 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors.
T2344 LY 344864 LY344864 5-HT Receptor
LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.
T6647 Rotigotine- Neupro,N-0923,N-0437,SPM 962 Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome. Administered as a once-daily transdermal patch, Rotigotine has not been associated with ser...
T4983 Isoetharine mesylate salt Isoetarine mesilate Others , Adrenergic Receptor
Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T3284 Carazolol Conducton,Suacron Adrenergic Receptor
Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T21957 Guanabenz hydrochloride NE56490 Adrenergic Receptor
Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.
T1132 Nicergoline Nicergolinum,Nimergoline Adrenergic Receptor
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T13376 YS-49 RAAS , Akt , PI3K , Adrenergic Receptor
YS-49 is an activator of PI3K/Akt (a downstream target of RhoA).
T0088 Urapidil hydrochloride Urapidil HCl 5-HT Receptor , Adrenergic Receptor
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T1275 Phentolamine mesylate Phentolamine methanesulfonate,Phentolamine mesilate Adrenergic Receptor
Phentolamine mesylate (Phentolamine methanesulfonate) is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma, vasospasm of RAYNAUD DISEAS...
T17111 Todralazine hydrochloride Ecarazine hydrochloride Adrenergic Receptor
Todralazine hydrochloride (Ecarazine hydrochloride) is a β2AR blocker and has antioxidant and free radical scavenging activities. Todralazine hydrochloride can be used in anti-hypertensive research.
T1012 Acebutolol hydrochloride Acebutolol HCl Adrenergic Receptor
Acebutolol hydrochloride (Acebutolol HCl) acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutolol hydrochloride is the hydro...
T1247 Clonidine hydrochloride Clonidine HCl,Catapres Adrenergic Receptor
Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
T22316 Doxazosin UK 33274 Adrenergic Receptor
Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.
T0394 Moxisylyte hydrochloride Thymoxamine hydrochloride Adrenergic Receptor
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T1671 Mirabegron YM178 Adrenergic Receptor
Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T3278 Piribedil EU-4200,Trivastan,ET-495,Trivastal Dopamine Receptor , Histone Methyltransferase , Adrenergic Receptor
Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
T2546 Pimozide R6238 Potassium Channel , Dopamine Receptor , Adrenergic Receptor , STAT
Pimozide (R6238) is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic receptors in the central nervous system (CNS), thereby...
T0115 Idazoxan hydrochloride RX 781094 Adrenergic Receptor , Imidazoline Receptor
Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T0397 Tetrahydrozoline Tetryzolin,Tetryzoline Adrenergic Receptor
Tetrahydrozoline (Tetryzoline), an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of the eye resulted from minor ocular irritants.
T0993 Methoxamine hydrochloride Methoxamine HCl Adrenergic Receptor
Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
T7164 Levalbuterol tartrate Levosalbutamol tartrate Adrenergic Receptor
Levalbuterol tartrate (Levosalbutamol tartrate) is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T6766 Atipamezole Antisedan,MPV 1248 Adrenergic Receptor
Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.

Compounds

SR59230A
T13016
Synonym:
Target: Adrenergic Receptor
Dibenamine hydrochloride
T37906
Synonym:
Target: Adrenergic Receptor
Tizanidine
T7065
Synonym:
Target: Adrenergic Receptor
Lofexidine
T7160
Synonym:
Target: Adrenergic Receptor
Mapenterol hydrochloride
T40622
Synonym:
Target: Adrenergic Receptor
Clonidine
T7045
Synonym: Nexiclon,Catapres,Kapvay
Target: Adrenergic Receptor
Phentolamine
T8348
Synonym:
Target: Adrenergic Receptor
ACEPROMAZINE MALEATE
T7728
Synonym:
Target: Dopamine Receptor
Zotepine
T19680
Synonym:
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Metipranolol
T8899
Synonym:
Target: Adrenergic Receptor
GUANABENZ
T5471
Synonym:
Target: Adrenergic Receptor
Bupranolol
T8580
Synonym:
Target: Adrenergic Receptor
Dexmedetomidine
T2524
Synonym:
Target: Adrenergic Receptor
Talinolol
T21640
Synonym:
Target: Adrenergic Receptor
L-765314
T5511
Synonym:
Target: Adrenergic Receptor
CL 316243
T10830
Synonym:
Target: Adrenergic Receptor
Paroxetine
T8708
Synonym:
Target: Serotonin Transporter
Metaraminol tartrate
T0279
Synonym: Metaradrine tartrate,Metaraminol bitartrate
Target: Adrenergic Receptor
Rilmenidine Phosphate
T6641
Synonym:
Target: Apoptosis, Adrenergic Receptor, Autophagy, Imidazoline Receptor
Prazosin
T22406
Synonym: Prazosine,Furazosin,Prazocin
Target: Adrenergic Receptor
Indacaterol
T2320
Synonym:
Target: Adrenergic Receptor
Terbutaline Sulfate
T1584
Synonym: Terbutaline hemisulfate
Target: Antibacterial, Adrenergic Receptor, Antibiotic
Urapidil
T0165
Synonym: Mediatensyl,Ebrantil,Eupressyl
Target: 5-HT Receptor, Adrenergic Receptor
Dopexamine hydrochloride
T11318
Synonym: FPL60278AR
Target: Adrenergic Receptor
Salmeterol
T12829
Synonym: GR33343X
Target: Adrenergic Receptor
L755507
T6872
Synonym:
Target: Adrenergic Receptor, CRISPR/Cas9
Penbutolol sulfate
T12402
Synonym: (-)-Terbuclomine
Target: Adrenergic Receptor
Ritanserin
T16759
Synonym: R 55667
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
LY 344864
T2344
Synonym: LY344864
Target: 5-HT Receptor
Rotigotine-
T6647
Synonym: Neupro,N-0923,N-0437,SPM 962
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor
Isoetharine mesylate salt
T4983
Synonym: Isoetarine mesilate
Target: Others, Adrenergic Receptor
Carazolol
T3284
Synonym: Conducton,Suacron
Target: Adrenergic Receptor
Guanabenz hydrochloride
T21957
Synonym: NE56490
Target: Adrenergic Receptor
Nicergoline
T1132
Synonym: Nicergolinum,Nimergoline
Target: Adrenergic Receptor
YS-49
T13376
Synonym:
Target: RAAS, Akt, PI3K, Adrenergic Receptor
Urapidil hydrochloride
T0088
Synonym: Urapidil HCl
Target: 5-HT Receptor, Adrenergic Receptor
Phentolamine mesylate
T1275
Synonym: Phentolamine methanesulfonate,Phentolamine mesilate
Target: Adrenergic Receptor
Todralazine hydrochloride
T17111
Synonym: Ecarazine hydrochloride
Target: Adrenergic Receptor
Acebutolol hydrochloride
T1012
Synonym: Acebutolol HCl
Target: Adrenergic Receptor
Clonidine hydrochloride
T1247
Synonym: Clonidine HCl,Catapres
Target: Adrenergic Receptor
Doxazosin
T22316
Synonym: UK 33274
Target: Adrenergic Receptor
Moxisylyte hydrochloride
T0394
Synonym: Thymoxamine hydrochloride
Target: Adrenergic Receptor
Mirabegron
T1671
Synonym: YM178
Target: Adrenergic Receptor
Piribedil
T3278
Synonym: EU-4200,Trivastan,ET-495,Trivastal
Target: Dopamine Receptor, Histone Methyltransferase, Adrenergic Receptor
Pimozide
T2546
Synonym: R6238
Target: Potassium Channel, Dopamine Receptor, Adrenergic Receptor, STAT
Idazoxan hydrochloride
T0115
Synonym: RX 781094
Target: Adrenergic Receptor, Imidazoline Receptor
Tetrahydrozoline
T0397
Synonym: Tetryzolin,Tetryzoline
Target: Adrenergic Receptor
Methoxamine hydrochloride
T0993
Synonym: Methoxamine HCl
Target: Adrenergic Receptor
Levalbuterol tartrate
T7164
Synonym: Levosalbutamol tartrate
Target: Adrenergic Receptor
Atipamezole
T6766
Synonym: Antisedan,MPV 1248
Target: Adrenergic Receptor
1 2 3 4 5 6 7 8
Cat No. Product Name Synonyms Targets
TN1015 Meranzin Adrenergic Receptor , Immunology/Inflammation related
Meranzin, a bioactive compound derived from the Traditional Chinese Medicine (TCM) Chaihu-Shugan-San (CSS) and isolated from Murraya exotica L. leaves, targets the alpha 2-adrenoceptor and engages the AMPA-ERK1/2–BDNF si...
T1287 Synephrine Oxedrine Endogenous Metabolite , Adrenergic Receptor
Synephrine (Oxedrine) is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T6688 Synephrine hydrochloride Oxedrine hydrochloride,Synephrine HCl Endogenous Metabolite , Adrenergic Receptor
Synephrine hydrochloride (Oxedrine hydrochloride) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T6662 Scopine 6,7-Epoxytropine Adrenergic Receptor
Scopine (6,7-Epoxytropine), the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
TN1465 Cannabigerol NOS , 5-HT Receptor , ROS
Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also binds to the CB2 receptor; it can relieve interocular pressur...
T6519 Gramine NSC 16892,Donaxine Adiponectin receptor , Reverse Transcriptase , Adrenergic Receptor
Gramine (Donaxine), a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for AdipoR2 and AdipoR1, respectively. Gramine is als...
T0076 Paliperidone 9-hydroxyrisperidone Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor , Histamine Receptor
Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the primary active metabolite of the older...
T2142 Yohimbine hydrochloride Antagonil,Yohimbine HCl Adrenergic Receptor
Yohimbine hydrochloride (Antagonil) is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of ERECTILE DYSFUNCTION.
T8149 Dobutamine hydrochloride Dobutamine (hydrochloride) Adrenergic Receptor
Dobutamine hydrochloride (Dobutamine (hydrochloride)) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T17310 Phenylephrine L-Phenylephrine,(R)-(-)-Phenylephrine Adrenergic Receptor
Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).
T3158 Harmane Loturine,Harman,Aribine Adrenergic Receptor , Monoamine Oxidase , Imidazoline Receptor
Harmane (Loturine) is a bio-active β-Carboline and monoamine oxidase inhibitor found in coffee and tobacco smoke.
T13655 DL-Norepinephrine hydrochloride Lys,DL-lysine Adrenergic Receptor
DL-Norepinephrine hydrochloride (DL-lysine) is a high-affinity basic amino acid substrate of amino acid transporter b0 + with a Km value in the range of 100-400 μM.
T5S2059 Glaucine Calcium Channel , Dopamine Receptor , Influenza Virus , Adrenergic Receptor , PDE
Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 production. Glaucine can inhibit the migration and invasion of h...
T0453 Phenylephrine hydrochloride NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride Endogenous Metabolite , Adrenergic Receptor
Phenylephrine hydrochloride (NCI-c55641) is a selective agonist of the α1-adrenergic receptor.
T7044 Norepinephrine Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol MMP , Endogenous Metabolite , Adrenergic Receptor , Autophagy
Norepinephrine (Levophed) can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascular endothelial growth factor, matrix metalloprotei...
T2889 Isoferulic acid Isoferulate,Hesperetic acid,3-Hydroxy-4-methoxycinnamic acid,Hesperetate Influenza Virus , Adrenergic Receptor
Isoferulic acid (Hesperetate) exhibits hypoglycemic properties.
T0469 Octopamine hydrochloride (±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl Dopamine Receptor , Endogenous Metabolite , Adrenergic Receptor
Octopamine hydrochloride ((±)-p-Octopamine hydrochlorid) is a biogenic monoamine structurally associated with noradrenaline. It can serve as a neurohormone, a neurotransmitter, and a neuromodulator in invertebrates.
T0505 Methyldopa L-(-)-α-Methyldopa,MK-351 Dopamine Receptor , Adrenergic Receptor
Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or sympatholytic.
T7056 Dronedarone SR 33589 P450 , Potassium Channel , Calcium Channel , Sodium Channel , Adrenergic Receptor , AChR , Autophagy
Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.
TCS2185 Yohimbine Adrenergic Receptor
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T3232 Higenamine hydrochloride Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride Adrenergic Receptor
Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupled receptors, and are the most prominent...
T1064 Norepinephrine bitartrate monohydrate Levophed,Noradrenaline bitartrate monohydrate Endogenous Metabolite , Adrenergic Receptor , Autophagy
Norepinephrine bitartrate monohydrate (Levophed) is a direct alpha-adrenergic receptors stimulator.
T4429 Rauwolscine hydrochloride Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride Adrenergic Receptor
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) , a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which potently antagonizes b...
T1680 Tolazoline hydrochloride Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride) Adrenergic Receptor
Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
T8304 Anisodamine Hydrobromide 6-Hydroxyhyoscyamine Adrenergic Receptor , AChR
Anisodamine Hydrobromide (6-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T0970 Racanisodamine Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine Adrenergic Receptor , AChR
Racanisodamine (7β-Hydroxyhyoscyamine) is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
TN7129 Methyl maslinate Maslinic acid methyl ester,Crategolic acid methyl ester Adrenergic Receptor
Methyl maslinate (Maslinic acid methyl ester) is an antagonist of β- adrenergic receptor with cardiotonic and antidysrhythmic properties. Methyl maslinate can be used in studies about hypertension.
T5S1177 Aloin B Isobarbaloin Others
Aloin B (Isobarbaloin) is an isomer of aloin.1. The extract of A. vera and its active ingredient aloin cause melanin aggregation leading to skin lightening via alpha adrenergic receptor stimulation, the result opens new ...
T60245 Norepinephrine hydrochloride
Norepinephrine hydrochloride (Levarterenol hydrochloride) is a β1 -selective agonist of the adrenergic receptor with EC 50 of 5.37 μM [1].
TN1797 Isorhoifolin Adrenergic Receptor
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile force by increasing the l-type calcium current and activatin...
TN2001 Oblongine Others
Oblongine chloride may have potential haemodynamic effects, it can cause a dose-dependent reduction of systolic and diastolic blood pressure, and that these effects are not mediated by α²-adrenergic receptor stimulation.

Natural Products

Meranzin
TN1015
Synonym:
Target: Adrenergic Receptor, Immunology/Inflammation related
Synephrine
T1287
Synonym: Oxedrine
Target: Endogenous Metabolite, Adrenergic Receptor
Synephrine hydrochloride
T6688
Synonym: Oxedrine hydrochloride,Synephrine HCl
Target: Endogenous Metabolite, Adrenergic Receptor
Scopine
T6662
Synonym: 6,7-Epoxytropine
Target: Adrenergic Receptor
Cannabigerol
TN1465
Synonym:
Target: NOS, 5-HT Receptor, ROS
Gramine
T6519
Synonym: NSC 16892,Donaxine
Target: Adiponectin receptor, Reverse Transcriptase, Adrenergic Receptor
Paliperidone
T0076
Synonym: 9-hydroxyrisperidone
Target: Dopamine Receptor, 5-HT Receptor, Adrenergic Receptor, Histamine Receptor
Yohimbine hydrochloride
T2142
Synonym: Antagonil,Yohimbine HCl
Target: Adrenergic Receptor
Dobutamine hydrochloride
T8149
Synonym: Dobutamine (hydrochloride)
Target: Adrenergic Receptor
Phenylephrine
T17310
Synonym: L-Phenylephrine,(R)-(-)-Phenylephrine
Target: Adrenergic Receptor
Harmane
T3158
Synonym: Loturine,Harman,Aribine
Target: Adrenergic Receptor, Monoamine Oxidase, Imidazoline Receptor
DL-Norepinephrine hydrochloride
T13655
Synonym: Lys,DL-lysine
Target: Adrenergic Receptor
Glaucine
T5S2059
Synonym:
Target: Calcium Channel, Dopamine Receptor, Influenza Virus, Adrenergic Receptor, PDE
Phenylephrine hydrochloride
T0453
Synonym: NCI-c55641,Phenylephrine HCl,(R)-(-)-Phenylephrine hydrochloride
Target: Endogenous Metabolite, Adrenergic Receptor
Norepinephrine
T7044
Synonym: Levophed,Levonoradrenaline,Aktamin,Nor-Epirenan,Levonor,Arterenol
Target: MMP, Endogenous Metabolite, Adrenergic Receptor, Autophagy
Isoferulic acid
T2889
Synonym: Isoferulate,Hesperetic acid,3-Hydroxy-4-methoxycinnamic acid,Hesperetate
Target: Influenza Virus, Adrenergic Receptor
Octopamine hydrochloride
T0469
Synonym: (±)-p-Octopamine hydrochlorid,(+,-)-Octopamine HCl
Target: Dopamine Receptor, Endogenous Metabolite, Adrenergic Receptor
Methyldopa
T0505
Synonym: L-(-)-α-Methyldopa,MK-351
Target: Dopamine Receptor, Adrenergic Receptor
Dronedarone
T7056
Synonym: SR 33589
Target: P450, Potassium Channel, Calcium Channel, Sodium Channel, Adrenergic Receptor, AChR, Autophagy
Yohimbine
TCS2185
Synonym:
Target: Adrenergic Receptor
Higenamine hydrochloride
T3232
Synonym: Higenamine HCl,Demethylcoclaurine hydrochloride,norcoclaurine HCl,(+-)-Demethylcoclaurine hydrochloride,Higenamine Hydrochloride
Target: Adrenergic Receptor
Norepinephrine bitartrate monohydrate
T1064
Synonym: Levophed,Noradrenaline bitartrate monohydrate
Target: Endogenous Metabolite, Adrenergic Receptor, Autophagy
Rauwolscine hydrochloride
T4429
Synonym: Corynanthidine hydrochloride,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride
Target: Adrenergic Receptor
Tolazoline hydrochloride
T1680
Synonym: Imidaline hydrochloride,Imidaline (hydrochloride),Benzidazol hydrochloride,Tolazoline HCl,NSC35110 (hydrochloride)
Target: Adrenergic Receptor
Anisodamine Hydrobromide
T8304
Synonym: 6-Hydroxyhyoscyamine
Target: Adrenergic Receptor, AChR
Racanisodamine
T0970
Synonym: Anisodamine,7β-Hydroxyhyoscyamine,Raceanisodamine
Target: Adrenergic Receptor, AChR
Methyl maslinate
TN7129
Synonym: Maslinic acid methyl ester,Crategolic acid methyl ester
Target: Adrenergic Receptor
Aloin B
T5S1177
Synonym: Isobarbaloin
Target: Others
Norepinephrine hydrochloride
T60245
Synonym:
Target:
Isorhoifolin
TN1797
Synonym:
Target: Adrenergic Receptor
Oblongine
TN2001
Synonym:
Target: Others

Recombinant Proteins

Species：
Human (5)
Mouse (1)
Expression System：
E. coli (5)
Baculovirus-Insect Cells (1)
Tag：
N-terminal 6xHis-SUMO-tagged (2)
C-6His (1)
C-terminal 6xHis-tagged (1)
His,GST (1)
N-terminal 10xHis-tagged and C-terminal Myc-tagged (1)
Cat No. Product Name Species Expression System
TMPY-04562 GRK2 Protein, Human, Recombinant (His & GST) Human Baculovirus-Insect Cells
G-protein coupled receptor kinase 2 (GRK2), also referred as Adrenergic, beta, receptor kinase 1 (ADRBK1), is a ubiquitous member of the G protein-coupled receptor kinase (GRK) family that appears to play a central, inte...
TMPJ-00983 ARRB1 Protein, Human, Recombinant (His) Human E. coli
β-Arrestin-1 (ARRB1) is a cytoplasmic protein that belongs to the arrestin family. ARRB1 is expressed at high levels in peripheral blood leukocytes and the central nervous system. ARRB1 regulates agonist-mediated G-prote...
TMPH-01250 MAP2K3 Protein, Human, Recombinant (His & SUMO) Human E. coli
Dual specificity kinase. Is activated by cytokines and environmental stress in vivo. Catalyzes the concomitant phosphorylation of a threonine and a tyrosine residue in the MAP kinase p38. Part of a signaling cascade that...
TMPH-02540 GRK2 Protein, Mouse, Recombinant (His & SUMO) Mouse E. coli
Specifically phosphorylates the agonist-occupied form of the beta-adrenergic and closely related receptors, probably inducing a desensitization of them. Key regulator of LPAR1 signaling. Competes with RALA for binding to...
TMPH-01857 PIK3CG Protein, Human, Recombinant (His & Myc) Human E. coli
Phosphoinositide-3-kinase (PI3K) that phosphorylates PtdIns(4,5)P2 (Phosphatidylinositol 4,5-bisphosphate) to generate phosphatidylinositol 3,4,5-trisphosphate (PIP3). PIP3 plays a key role by recruiting PH domain-contai...
TMPH-01027 CAMK2D Protein, Human, Recombinant (His) Human E. coli
Calcium/calmodulin-dependent protein kinase involved in the regulation of Ca(2+) homeostatis and excitation-contraction coupling (ECC) in heart by targeting ion channels, transporters and accessory proteins involved in C...
Cat No. Product Name
L2700 Adrenergic Receptor-Targeted Compound Library

219 compounds
A unique collection of 219 bioactive compounds specifically targeting adrenergic receptors, effective tool for screening new drugs or new target identification;
L2610 Neurotransmitter Receptor Compound Library

1513 compounds
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；

Libraries

Adrenergic Receptor-Targeted Compound Library
L2700
Compounds: 219
Neurotransmitter Receptor Compound Library
L2610
Compounds: 1513
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