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GPCR/G Protein Adrenergic Receptor

Adrenergic Receptor

The adrenergic receptors or adrenoceptors are a class of G protein-coupled receptors that are targets of many catecholamines like norepinephrine (noradrenaline) and epinephrine (adrenaline) produced by the body, but also many medications like beta blockers, β2 agonists and α2 agonists, which are used to treat high blood pressure and asthma.
Cat No. product name
T0007 Atenolol Atenolol is a selective β1 receptor antagonist.
T0031 Ziprasidone hydrochloride monohydrate Ziprasidone(CP88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
T0031L Ziprasidone hydrochloride Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
T0031L2 Ziprasidone Ziprasidone is an a typical antipsychotic used in the treatment of schizophrenia and bipolar disorder. Use of ziprasidone has not been consistently associate...
T0042 Xylometazoline hydrochloride Xylometazoline Hydrochloride is an α-adrenoceptor agonist usually used as nasal decongestant.
T0076 Paliperidone Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the p...
T0088 Urapidil hydrochloride Urapidil hydrochloride is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
T0091 Alfuzosin hydrochloride Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
T0101 Doxazosin mesylate Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
T0103 Dipivefrin hydrochloride Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
T0115 Idazoxan hydrochloride Idazoxan hydrochloride is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
T0137 Mirtazapine Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevat...
T0143 (±)-Bisoprolol hemifumarate Bisoprolol,a selective beta-1 adrenergic receptor antagonist,selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,th...
T0154 Nebivolol hydrochloride Nebivolol hydrochloride is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-argi...
T0162 Quetiapin Quetiapine is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapi...
T0165 Urapidil Urapidil, a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
T0172 Maprotiline hydrochloride Maprotiline hydrochloride is a bridged-ring tetracyclic antidepressant that is both mechanistically and functionally similar to the tricyclic antidepressants, i...
T0173 Nylidrin hydrochloride Nylidrin hydrochloride was an effective inhibitor of the IgG1-mediated release of histamine from passively sensitized guinea pig lung slices, and of the IgE-med...
T0197 Terazosin hydrochloride Terazosin, a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a drug of choice for pati...
T0210 Tamsulosin hydrochloride Tamsulosin Hydrochloride is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
T0226 Betaxolol hydrochloride Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induce...
T0248 Clorprenaline hydrochloride Clorprenaline Hydrochloride is a beta-2 adrenergic agonist with bronchodilator activity.
T0277 Orciprenaline sulfate Orciprenaline sulfate is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
T0279 Metaraminol bitartrate Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in th...
T0290 Tizanidine hydrochloride Tizanidine hydrochloride, an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
T0317 Buflomedil hydrochloride Buflomedil hydrochloride, a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
T0324 Isoxsuprine hydrochloride Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
T0342 Carvedilol phosphate Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intr...
T0348 Labetalol hydrochloride Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
T0351 Risperidal Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
T0365 Thioridazine hydrochloride Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
T0394 Moxisylyte hydrochloride Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
T0397 Tetryzoline Tetrahydrozoline, an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of the eye result...
T0445 Promethazine Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
T0445L Promethazine hydrochloride Promethazine HCl(NSC-231688), the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, mode...
T0446 Naphazoline hydrochloride Naphazoline hydrochloride is an adrenergic vasoconstrictor agent used as a decongestant.
T0447 Carvedilol Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intr...
T0453 Phenylephrine hydrochloride Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
T0455 Clozapine Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and display...
T0475 Timolol Maleate Timolol is a nonselective beta-adrenergic receptor blocker that is widely used for the therapy of hypertension, angina pectoris and prevention of vascular heada...
T0483 Sotalol hydrochloride Sotalol Hydrochloride is the hydrochloride salt form of sotalol, an ethanolamine derivative with Class III antiarrhythmic and antihypertensive properties.
T0487 Metoprolol tartrate Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
T0696 Naftopidil Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
T0766 Promazine hydrochloride Promazine hydrochloride is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treat...
T0783 Mianserin hydrochloride Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin ...
T0812 Propranolol hydrochloride Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGI...
T0871 Noradrenaline bitartrate Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic ph...
T0948 Adrenalone hydrochloride Adrenalone hydrochloride, a selective α1-adrenoceptor agonist, is used as a topical hemostatic and vasoconstrictor and used to extend the effect of local anest...
T0970 Anisodamine Anisodamine is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T0991 Desipramine hydrochloride Desipramine Hydrochloride a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), ...
T0993 Methoxamine hydrochloride An alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
T1012 Acebutolol hydrochloride Acebutolol acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutol...
T1045 Trimipramine maleate Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin a...
T1050 Prazosin hydrochloride Prazosin Hydrochloride reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not complet...
T1056 Isoprenaline hydrochlorideHOT Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
T1064 Noradrenaline bitartrate monohydrate Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.
T1071L DL-Adrenaline Hydrochloride DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular pressure-reducing acti...
T1073 Dronedarone hydrochloride Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
T1132 Nicergoline Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
T1139 Salbutamol Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3',...
T1158 Phenoxybenzamine hydrochloride Phenoxybenzamine Hydrochloride is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive an...
T1203 Nadolol Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. Nadolol competitively blocks beta-1 adrenergic recept...
T1215 Nicardipine hydrochloride Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nica...
T1239 Indacaterol maleate Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
T1247 Clonidine hydrochloride Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide...
T1275 Phentolamine mesilate Phentolamine mesylate is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma,...
T1282 Carteolol hydrochloride Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for b...
T1287 Synephrine Synephrine is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
T1327 Nortriptyline hydrochloride Nortriptyline hydrochloride is a metabolite of AMITRIPTYLINE that is also used as an antidepressive agent. Nortriptyline is used in major depression, dysthymia,...
T1433 Ritodrine hydrochloride Ritodrine binds to and activates beta-2 adrenergic receptors of myometrial cells in the uterus, which decreases the intensity and frequency of uterine contracti...
T1446 Bambuterol hydrochloride Bambuterol, a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
T1459 Cisatracurium besylate Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
T1496 Amiodarone hydrochloride Amiodarone hydrochloride is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting PO...
T1500 Xylazine hydrochloride Xylazine hydrochloride is an adrenergic alpha-2 agonist used as a sedative, analgesic and centrally acting muscle relaxant in veterinary medicine
T1503 Esmolol hydrochloride Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to insta...
T1504 Silodosin Silodosin is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
T1539 Iloperidone Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
T1540 Doxepin hydrochloride Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mec...
T1567 Olanzapine Olanzapine is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
T1577 Midodrine hydrochloride Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergi...
T1584 Terbutaline Sulfate Terbutaline sulfate is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
T1619 Trazodone hydrochloride Trazodone hydrochloride is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients with major depres...
T1632 Amitraz AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic m...
T1671 Mirabegron Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
T1680 Tolazoline hydrochloride Tolazoline is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
T1696 2-(1-Piperazinyl)pyrimidine 2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
T1738 Taxifolin Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
T1769 Pardoprunox Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying th...
T2142 Yohimbine hydrochloride Yohimbine hydrochloride is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of ERECTILE D...
T2150 Guanfacine hydrochloride Guanfacine hydrochloride is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
T2306 Brexpiprazole Brexpiprazole is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
T2320 Indacaterol Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
T2524 Dexmedetomidine Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect o...
T2535 Ivabradine hydrochloride Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, h...
T2547 Droxidopa Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auto...
T2580 Formoterol Arformoterol is an adrenergic β-2 receptor agonist with a prolonged duration of action. It is used to manage asthma and in the treatment of chronic obstructive...
T3046 BMY 7378 dihydrochloride BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
T3165 Metoprolol Succinate Metoprolol succinate is a selective adrenergic beta-1 blocking agent that is commonly used to treat ANGINA PECTORIS; HYPERTENSION; and CARDIAC ARRHYTHMIAS.
T3277 Tulobuterol hydrochloride Tulobuterol hydrochloride is a long-acting beta2-adrenergic receptor agonist.
T3278 Piribedil Piribedil is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
T3284 Carazolol Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
T3457 Olodaterol Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors l...
T3996 Dapiprazole Hydrochloride Dapiprazole Hydrochloride is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors in the smooth muscle of blood vessels (arteries, ...
T6241 Quetiapine Fumarate Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
T6408 Betaxolol Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
T6422 Brimonidine Tartrate Brimonidine tartrate is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated wit...
T6464 Detomidine HCl Detomidine HCl produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
T6466 Dexmedetomidine HCl Dexmedetomidine hydrochloride is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is ...
T6505 Formoterol Hemifumarate Formoterol Hemifumarate, an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of chronic obstructive pulmonary disease(...
T6522 Guanabenz Acetate Guanabenz Acetate is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is...
T6565 Levobetaxolol HCl Levobetaxolol hydrochloride is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treating conditions such as glaucom...
T6579 Medetomidine HCl Medetomidine is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
T6600 Naftopidil DiHCl Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
T6652 Salbutamol Sulfate Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
T6662 Scopine Scopine, the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
T6688 Synephrine HCl SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
T6701 Terazosin hydrochloride dihydrate Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
T6703 Tetrahydrozoline HCl Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
T6765 Atipamezole hydrochloride Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochl...
T6766 Atipamezole Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
T6860 ICI-118551 Hydrochloride ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
T6872 L755507 L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).
T4429 Rauwolscine hydrochloride Rauwolscine, a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which poten...
T2226 Pergolide mesylate salt PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due t...
T5S2178 Fargesin 1. Fargesin as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Fargesin improves ...
T4548 Procaterol hydrochloride Short-acting β2-adrenergic receptor agonist used to treat asthma.
T7046 Xylazine Xylazine is α2-adrenergic receptor agonist.
T7079 Batefenterol Batefenterol (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-a...
T4526 Piperoxan hydrochloride Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
T4560 Alprenolol Alprenolol is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT1B.
T4S0998 Trifolirhizin Trifolirhizin exerts varying degrees of inhibition on tyrosinase-dependent melanin biosynthesis, and therefore, are candidates as skin-whitening agents.Trifolir...
T4983 Isoetharine mesylate salt Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
T5105 1-(2-Pyridyl)piperazine 1-(2-Pyridyl)piperazine is a selective α2-adrenoceptor antagonists. 1-(2-Pyridyl)piperazine shows sympatholytic activity. 1-(2-Pyridyl)piperazine is also a met...
T5028 Landiolol hydrochloride Landiolol is an ultra-short-acting β1 selective adrenoceptor antagonist.
T5035 Methoxyphenamine Hydrochloride Methoxyphenamine is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
T4963 Higenamine Higenamine is a novel α1 -adrenoceptor antagonist.
T7045 Clonidine Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wid...
T5159 BI 1744 hydrochloride Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and...
T5327 Amezinium (methylsulfate) Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake.
T6519 Gramine Gramine, a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for...
T5450 DL-071-IT DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
T5471 GUANABENZ GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
T7160 Lofexidine Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
T7164 Levalbuterol tartrate Levosalbutamol tartrate is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
T1090 Perphenazine Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
T2546 Pimozide Pimozide is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic re...
T7044 Norepinephrine Norepinephrine can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascul...
T1415 Gemfibrozil Gemfibrozil interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation and an in...
TCS2185 Yohimbine Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
T8304 Anisodamine Hydrobromide Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
T8149 Dobutamine (hydrochloride) Dobutamine (hydrochloride) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
T8143 Bevantolol hydrochloride Bevantolol hydrochloride is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.
T8358 Fenoterol Fenoterol is an  agonist of  β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
TN1797 Isorhoifolin Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile ...
TN1922 Meranzin hydrate Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-...
TN2267 Tetrahydroalstonine Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogeno...
T8348 Phentolamine Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
T13804 OPC-28326 OPC-28326 is a selective peripheral vasodilator and an α2-adrenergic receptor angatonist(α2A-, α2B- and α2C-adrenoceptors with Ki of 2040, 285, and 55 nM,...
T12343 Benzquinamide Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
T11010 Detomidine carboxylic acid Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also...
T11015 Midaglizole hydrochloride Midaglizole hydrochloride (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6...
T11036 Diacetolol D7 Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
T13016 SR59230A SR59230A is a selective, and blood-brain barrier penetrating antagonist of β3-adrenergic receptor(IC50s of 40, 408, and 648 nM for β3, β1, and β2 receptors,...
T5134 Vilanterol trifenatate Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and ...
T7065 Tizanidine Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
T14287 Ancarolol Ancarolol is a blocking agent of beta-adrenergic.
T12643 (R)-Terazosin (R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values ...
T10364 Arbutamine Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure...
T15042 D2343 D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
T12815 (S)-Terazosin (S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor...
T11286 Fiduxosin Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively. 
T13285 Vatinoxan hydrochloride Vatinoxan hydrochloride is an antagonist of peripheral α2 adrenergic receptor.
T10778 CGP 20712 A CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
T13403 ZK-90055 hydrochloride ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
T13470 (±)-Methotrimeprazine (D6) (±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
T15943 M443 M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
T8366 Mitochonic acid 5 Mitochonic acid 5 is a derivative of the plant hormone indole-3-acetic acid. Mitochonic acid 5 binds mitochondria and ameliorates renal tubular and cardiac myoc...
T11786 KUL 7211 racemate KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211. 
T16759 Ritanserin Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM).
T16769 Ro 363 RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial cont...
T11894 Lusaperidone Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively. 
T22406 Prazosin Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
T8580 Bupranolol Bupranolol is an antagonist of β2-adrenergic receptor,and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombo...
T8595 Practolol Practolol is a selective β-adrenoceptor blocker.
TN3364 Agrimonolide Agrimonolide is a potential α1 adrenergic receptor antagonist, it exerts anti-inflammatory activity, at least in part, via suppressing LPS-induced activation o...
TN3368 Akuammigine Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding ...
TN3507 beta-Yohimbine Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor bloc...
TN4323 Isorauhimbine 3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities,it also has cardiovascular effects.
TN4882 Quinine HCl Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
TN5061 Stephanine l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of...
T8663 nifenalol.HCl Nifenalol is a antagonist of β-adrenergic receptor.
T21147 Clenbuterol Clenbuterol is a substituted phenylaminoethanol that has β2 adrenomimetic properties at very low doses, and is used as a bronchodilator in asthma.
T21066 Norepinephrine bitartrate salt Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
T8696 Propranolol hydrochloride Propranolol hydrochloride is a blocker of β1 and β2 adrenergic receptor
T12444 Phentolamine Analogue 1 Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of alpha-adrenergic.
Atenolol
T0007CAS 29122-68-7
Atenolol is a selective β1 receptor antagonist.
Ziprasidone hydrochloride monohydrate
T0031CAS 138982-67-9
Ziprasidone(CP88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic activity.
Ziprasidone hydrochloride
T0031LCAS 122883-93-6
Ziprasidone (hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.
Ziprasidone
T0031L2CAS 146939-27-7
Ziprasidone is an a typical antipsychotic used in the treatment of schizophrenia and bipolar disorder. Use of ziprasidone has not been consistently associate...
Xylometazoline hydrochloride
T0042CAS 1218-35-5
Xylometazoline Hydrochloride is an α-adrenoceptor agonist usually used as nasal decongestant.
Paliperidone
T0076CAS 144598-75-4
Paliperidone(Invega) is used as an atypical antipsychotic. It applies to the acute and maintenance treatment of schizophrenia. Chemically, paliperidone is the p...
Urapidil hydrochloride
T0088CAS 64887-14-5
Urapidil hydrochloride is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Alfuzosin hydrochloride
T0091CAS 81403-68-1
Alfuzosin hydrochloride is an α1 adrenergic receptor antagonist. It applies to treat benign prostatic hyperplasia (BPH).
Doxazosin mesylate
T0101CAS 77883-43-3
Doxazosin mesylate(UK 33274) is a quinazoline-derivative. It is a selectively antagonizes postsynaptic α1-adrenergic receptors.
Dipivefrin hydrochloride
T0103CAS 64019-93-8
Dipivefrin that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.
Idazoxan hydrochloride
T0115CAS 79944-56-2
Idazoxan hydrochloride is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.
Mirtazapine
T0137CAS 85650-52-8
Mirtazapine is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asymptomatic elevat...
(±)-Bisoprolol hemifumarate
T0143CAS 104344-23-2
Bisoprolol,a selective beta-1 adrenergic receptor antagonist,selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,th...
Nebivolol hydrochloride
T0154CAS 152520-56-4
Nebivolol hydrochloride is a cardioselective ADRENERGIC BETA-1 RECEPTOR ANTAGONIST (beta-blocker) that functions as a VASODILATOR through the endothelial L-argi...
Quetiapin
T0162CAS 111974-69-7
Quetiapine is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapi...
Urapidil
T0165CAS 34661-75-1
Urapidil, a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.
Maprotiline hydrochloride
T0172CAS 10347-81-6
Maprotiline hydrochloride is a bridged-ring tetracyclic antidepressant that is both mechanistically and functionally similar to the tricyclic antidepressants, i...
Nylidrin hydrochloride
T0173CAS 849-55-8
Nylidrin hydrochloride was an effective inhibitor of the IgG1-mediated release of histamine from passively sensitized guinea pig lung slices, and of the IgE-med...
Terazosin hydrochloride
T0197CAS 63074-08-8
Terazosin, a selective alpha1-antagonist, can treat the benign prostatic hyperplasia (BPH). It also can lower blood pressure, so it is a drug of choice for pati...
Tamsulosin hydrochloride
T0210CAS 106463-17-6
Tamsulosin Hydrochloride is the hydrochloride salt of tamsulosin, a sulfonamide derivative with α1 adrenergic antagonist activity.
Betaxolol hydrochloride
T0226CAS 63659-19-8
Betaxolol is a cardioselective beta-blocker used in the treatment of hypertension. Betaxolol has not been linked to instances of clinically apparent drug induce...
Clorprenaline hydrochloride
T0248CAS 6933-90-0
Clorprenaline Hydrochloride is a beta-2 adrenergic agonist with bronchodilator activity.
Orciprenaline sulfate
T0277CAS 5874-97-5
Orciprenaline sulfate is a beta-2 adrenergic agonist used in the treatment of ASTHMA and BRONCHIAL SPASM.
Metaraminol bitartrate
T0279CAS 33402-03-8
Metaraminol bitartrate is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors. It has been used primarily as a vasoconstrictor in th...
Tizanidine hydrochloride
T0290CAS 64461-82-1
Tizanidine hydrochloride, an α2-adrenergic receptor agonist, inhibits neurotransmitter release from CNS noradrenergic neurons.
Buflomedil hydrochloride
T0317CAS 35543-24-9
Buflomedil hydrochloride, a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.
Isoxsuprine hydrochloride
T0324CAS 579-56-6
Isoxsuprine hydrochloride is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
Carvedilol phosphate
T0342CAS 610309-89-2
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intr...
Labetalol hydrochloride
T0348CAS 32780-64-6
Labetalol hydrochloride, a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.
Risperidal
T0351CAS 106266-06-2
Risperidone is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.
Thioridazine hydrochloride
T0365CAS 130-61-0
Thioridazine, an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4 selectivity.
Moxisylyte hydrochloride
T0394CAS 964-52-3
Moxisylyte hydrochloride is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Tetryzoline
T0397CAS 84-22-0
Tetrahydrozoline, an alpha agonist, have an effect on the constriction of conjunctival blood vessels. This contributes to relieve the redness of the eye result...
Promethazine
T0445CAS 60-87-7
Tafluprost(AFP-168) is an analogue of anti-glaucoma prostaglandin (PG) .
Promethazine hydrochloride
T0445LCAS 58-33-3
Promethazine HCl(NSC-231688), the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, mode...
Naphazoline hydrochloride
T0446CAS 550-99-2
Naphazoline hydrochloride is an adrenergic vasoconstrictor agent used as a decongestant.
Carvedilol
T0447CAS 72956-09-3
Carvedilol Phosphate is the phosphate salt form of carvedilol, a racemic mixture and adrenergic blocking agent with antihypertensive activity and devoid of intr...
Phenylephrine hydrochloride
T0453CAS 61-76-7
Phenylephrine hydrochloride is a selective agonist of the α1-adrenergic receptor.
Clozapine
T0455CAS 5786-21-0
Clozapine is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, and display...
Timolol Maleate
T0475CAS 26921-17-5
Timolol is a nonselective beta-adrenergic receptor blocker that is widely used for the therapy of hypertension, angina pectoris and prevention of vascular heada...
Sotalol hydrochloride
T0483CAS 959-24-0
Sotalol Hydrochloride is the hydrochloride salt form of sotalol, an ethanolamine derivative with Class III antiarrhythmic and antihypertensive properties.
Metoprolol tartrate
T0487CAS 56392-17-7
Metoprolol Tartrate is a blocker of the cardioselective β-adrenergic receptor.
Naftopidil
T0696CAS 57149-07-2
Naftopidil (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
Promazine hydrochloride
T0766CAS 53-60-1
Promazine hydrochloride is a phenothiazine with actions similar to CHLORPROMAZINE but with less antipsychotic activity. It is primarily used in short-term treat...
Mianserin hydrochloride
T0783CAS 21535-47-7
Mianserin hydrochloride is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of serotonin ...
Propranolol hydrochloride
T0812CAS 318-98-9
Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGI...
Noradrenaline bitartrate
T0871CAS 69815-49-2
Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors. Norepinephrine Bitartrate is a bitartrate salt of norepinephrine, a synthetic ph...
Adrenalone hydrochloride
T0948CAS 62-13-5
Adrenalone hydrochloride, a selective α1-adrenoceptor agonist, is used as a topical hemostatic and vasoconstrictor and used to extend the effect of local anest...
Anisodamine
T0970CAS 17659-49-3
Anisodamine is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Desipramine hydrochloride
T0991CAS 58-28-6
Desipramine Hydrochloride a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine. In the central nervous system (CNS), ...
Methoxamine hydrochloride
T0993CAS 61-16-5
An alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.
Acebutolol hydrochloride
T1012CAS 34381-68-5
Acebutolol acts as a cardioselective beta-adrenergic antagonist with little effect on bronchial receptors and has intrinsic sympathomimetic properties. Acebutol...
Trimipramine maleate
T1045CAS 521-78-8
Trimipramine maleate appears to inhibit serotonin transport and norepinephrine uptake by nerve terminals. This increases available norepinephrine or serotonin a...
Prazosin hydrochloride
T1050CAS 19237-84-4
Prazosin Hydrochloride reduces peripheral resistance and relaxes vascular smooth muscles as a selective adrenergic alpha-1 antagonist by a mechanism not complet...
Isoprenaline hydrochloride HOT
T1056CAS 51-30-9
Isoproterenol is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.
Noradrenaline bitartrate monohydrate
T1064CAS 108341-18-0
Noradrenaline bitartrate monohydrate is a direct alpha-adrenergic receptors stimulator.
DL-Adrenaline Hydrochloride
T1071LCAS 329-63-5
DL-Adrenaline Hydrochloride is the hydrochloride salt of the naturally occurring sympathomimetic amine with vasoconstricting, intraocular pressure-reducing acti...
Dronedarone hydrochloride
T1073CAS 141625-93-6
Dronedarone hydrochloride is an amiodarone analog which has an effective and promising treatment for Atrial fibrillation.
Nicergoline
T1132CAS 27848-84-6
Nicergoline is an ergot derivative used to treat senile dementia and other disorders with vascular origins.
Salbutamol
T1139CAS 18559-94-9
Albuterol stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3',...
Phenoxybenzamine hydrochloride
T1158CAS 63-92-3
Phenoxybenzamine Hydrochloride is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive an...
Nadolol
T1203CAS 42200-33-9
Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities. Nadolol competitively blocks beta-1 adrenergic recept...
Nicardipine hydrochloride
T1215CAS 54527-84-3
Nicardipine Hydrochloride is the hydrochloride salt form of nicardipine, a synthetic derivative of nitrophenyl-pyridine and potent calcium channel blocker, Nica...
Indacaterol maleate
T1239CAS 753498-25-8
Indacaterol Maleate is an ultra-long-acting β-adrenoceptor agonist.
Clonidine hydrochloride
T1247CAS 4205-91-8
Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wide...
Phentolamine mesilate
T1275CAS 65-28-1
Phentolamine mesylate is a nonselective alpha-adrenergic antagonist. It is used in the treatment of hypertension and hypertensive emergencies, pheochromocytoma,...
Carteolol hydrochloride
T1282CAS 51781-21-6
Carteolol Hydrochloride is a synthetic quinolinone derivative, antihypertensive Carteolol Hydrochloride is a nonselective beta-adrenoceptor blocking agent for b...
Synephrine
T1287CAS 94-07-5
Synephrine is sympathetic alpha-adrenergic agonist used as a vasoconstrictor in circulatory failure, asthma, nasal congestion, and glaucoma.
Nortriptyline hydrochloride
T1327CAS 894-71-3
Nortriptyline hydrochloride is a metabolite of AMITRIPTYLINE that is also used as an antidepressive agent. Nortriptyline is used in major depression, dysthymia,...
Ritodrine hydrochloride
T1433CAS 23239-51-2
Ritodrine binds to and activates beta-2 adrenergic receptors of myometrial cells in the uterus, which decreases the intensity and frequency of uterine contracti...
Bambuterol hydrochloride
T1446CAS 81732-46-9
Bambuterol, a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.
Cisatracurium besylate
T1459CAS 96946-42-8
Cisatracurium Besylate is a nondepolarizing skeletal muscle relaxant for intravenous administration.
Amiodarone hydrochloride
T1496CAS 19774-82-4
Amiodarone hydrochloride is an antianginal and class III antiarrhythmic drug. It increases the duration of ventricular and atrial muscle action by inhibiting PO...
Xylazine hydrochloride
T1500CAS 23076-35-9
Xylazine hydrochloride is an adrenergic alpha-2 agonist used as a sedative, analgesic and centrally acting muscle relaxant in veterinary medicine
Esmolol hydrochloride
T1503CAS 81161-17-3
Esmolol is a cardioselective beta-blocker used in parenteral forms in the treatment of arrhythmias and severe hypertension. Esmolol has not been linked to insta...
Silodosin
T1504CAS 160970-54-7
Silodosin is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.
Iloperidone
T1539CAS 133454-47-4
Iloperidone is an atypical antipsychotic agent that is used for treatment of schizophrenia.
Doxepin hydrochloride
T1540CAS 1229-29-4
Doxepin Hydrochloride is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation. Its mec...
Olanzapine
T1567CAS 132539-06-1
Olanzapine is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
Midodrine hydrochloride
T1577CAS 3092-17-9
Midodrine is converted to its active metabolite, desglymidodrine by deglycination reaction. Desglymidodrine selectively binds to and activates alpha-1-adrenergi...
Terbutaline Sulfate
T1584CAS 23031-32-5
Terbutaline sulfate is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.
Trazodone hydrochloride
T1619CAS 25332-39-2
Trazodone hydrochloride is a serotonin uptake inhibitor that is used as an antidepressive agent. It has been shown to be effective in patients with major depres...
Amitraz
T1632CAS 33089-61-1
AMITRAZ is a white monoclinic crystals. Melting point 187-189°F (86-87°C). Insoluble in water. Used as an acaricide, insecticide and treatment of demodectic m...
Mirabegron
T1671CAS 223673-61-8
Mirabegron is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.
Tolazoline hydrochloride
T1680CAS 59-97-2
Tolazoline is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary hypertension of the newborn.
2-(1-Piperazinyl)pyrimidine
T1696CAS 20980-22-7
2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.
Taxifolin
T1738CAS 480-18-2
Taxifolin is a flavonoid in many plants such as Taxus chinensis, Siberian larch, Cedrus deodara and so on.
Pardoprunox
T1769CAS 269718-84-5
Pardoprunox is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties. Pardoprunox has been used in trials studying th...
Yohimbine hydrochloride
T2142CAS 65-19-0
Yohimbine hydrochloride is a plant alkaloid with alpha-2-adrenergic blocking activity. Yohimbine has been used as a mydriatic and in the treatment of ERECTILE D...
Guanfacine hydrochloride
T2150CAS 29110-48-3
Guanfacine hydrochloride is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.
Brexpiprazole
T2306CAS 913611-97-9
Brexpiprazole is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.
Indacaterol
T2320CAS 312753-06-3
Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.
Dexmedetomidine
T2524CAS 113775-47-6
Dexmedetomidine is a Central alpha-2 Adrenergic Agonist. The mechanism of action of dexmedetomidine is as an Adrenergic alpha2-Agonist. The physiologic effect o...
Ivabradine hydrochloride
T2535CAS 148849-67-6
Ivabradine hydrochloride is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, h...
Droxidopa
T2547CAS 23651-95-8
Droxidopa is an orally available prodrug of norepinephrine that is used in the treatment of symptomatic orthostatic hypotension due to neurogenic causes of auto...
Formoterol
T2580CAS 73573-87-2
Arformoterol is an adrenergic β-2 receptor agonist with a prolonged duration of action. It is used to manage asthma and in the treatment of chronic obstructive...
BMY 7378 dihydrochloride
T3046CAS 21102-95-4
BMY-7378, α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
Metoprolol Succinate
T3165CAS 98418-47-4
Metoprolol succinate is a selective adrenergic beta-1 blocking agent that is commonly used to treat ANGINA PECTORIS; HYPERTENSION; and CARDIAC ARRHYTHMIAS.
Tulobuterol hydrochloride
T3277CAS 56776-01-3
Tulobuterol hydrochloride is a long-acting beta2-adrenergic receptor agonist.
Piribedil
T3278CAS 3605-01-4
Piribedil is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
Carazolol
T3284CAS 57775-29-8
Carazolol is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.
Olodaterol
T3457CAS 868049-49-4
Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors l...
Dapiprazole Hydrochloride
T3996CAS 72822-13-0
Dapiprazole Hydrochloride is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors in the smooth muscle of blood vessels (arteries, ...
Quetiapine Fumarate
T6241CAS 111974-72-2
Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
Betaxolol
T6408CAS 63659-18-7
Betaxolol is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.
Brimonidine Tartrate
T6422CAS 70359-46-5
Brimonidine tartrate is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM) that is used to manage intraocular pressure associated wit...
Detomidine HCl
T6464CAS 90038-01-0
Detomidine HCl produce dose-dependent sedative and analgesic effects, mediatated by activation of α2 catecholamine receptors.
Dexmedetomidine HCl
T6466CAS 145108-58-3
Dexmedetomidine hydrochloride is an imidazole derivative that is an agonist of the adrenergic alpha-2 receptor. It is closely-related to MEDETOMIDINE, which is ...
Formoterol Hemifumarate
T6505CAS 43229-80-7
Formoterol Hemifumarate, an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of chronic obstructive pulmonary disease(...
Guanabenz Acetate
T6522CAS 23256-50-0
Guanabenz Acetate is a specific agonist of adrenergic receptor. The pEC50 for α2a-adrenergic receptor, α2b-adrenergic receptor and α2c-adrenergic receptor is...
Levobetaxolol HCl
T6565CAS 116209-55-3
Levobetaxolol hydrochloride is a beta-adrenergic receptor inhibitor (beta blocker), used to lower the pressure in the eye in treating conditions such as glaucom...
Medetomidine HCl
T6579CAS 86347-15-1
Medetomidine is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.
Naftopidil DiHCl
T6600CAS 57149-08-3
Naftopidil DiHCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
Salbutamol Sulfate
T6652CAS 51022-70-9
Salbutamol Sulfate is a short-acting β2-adrenergic receptor agonist with an IC50 of 8.93 μM.
Scopine
T6662CAS 498-45-3
Scopine, the metabolite of anisodine, is an α1-adrenergic receptor agonist used in the therapy of acute circulatory shock.
Synephrine HCl
T6688CAS 5985-28-4
SynephrineHCl (Oxedrine, p-Synephrine) is an agonist that acts on sympathomimetic α-adrenergic receptor (AR).
Terazosin hydrochloride dihydrate
T6701CAS 70024-40-7
Terazosin HCl is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).
Tetrahydrozoline HCl
T6703CAS 522-48-5
Tetrahydrozoline HCl is an imidazoline derivative with alpha receptor agonist activity.
Atipamezole hydrochloride
T6765CAS 104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochl...
Atipamezole
T6766CAS 104054-27-5
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
ICI-118551 Hydrochloride
T6860CAS 1217094-53-5
ICI-118551 is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3 receptors, respectively.
L755507
T6872CAS 159182-43-1
L755507 is an effective, selective agonist of β3-AR(IC50=35 nM).
Rauwolscine hydrochloride
T4429CAS 6211-32-1
Rauwolscine, a natural alkaloid, is a specific and reversible α2-adrenergic receptor antagonist (Ki: 12 nM) [1]. It is a stereoisomer of yohimbine, which poten...
Pergolide mesylate salt
T2226CAS 66104-23-2
PERGOLIDE MESYLATE is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some markets due t...
Fargesin
T5S2178CAS 31008-19-2
1. Fargesin as a potential β1AR antagonist through cAMP/PKA pathway could protect against myocardial ischemia/reperfusion injury in rats. 2. Fargesin improves ...
Procaterol hydrochloride
T4548CAS 81262-93-3
Short-acting β2-adrenergic receptor agonist used to treat asthma.
Xylazine
T7046CAS 7361-61-7
Xylazine is α2-adrenergic receptor agonist.
Batefenterol
T7079CAS 743461-65-6
Batefenterol (GSK961081, TD-5959) is a muscarinic receptor antagonist and β2-adrenoceptor agonist. It displays high affinity for hM2, hM3 muscarinic and hβ2-a...
Piperoxan hydrochloride
T4526CAS 135-87-5
Piperoxan hydrochloride is an α2 adrenoceptor antagonist. Piperoxan (benodaine) is a drug which was the very first antihistamine to be discovered.
Alprenolol
T4560CAS 13655-52-2
Alprenolol is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1A and 5-HT1B.
Trifolirhizin
T4S0998CAS 6807-83-6
Trifolirhizin exerts varying degrees of inhibition on tyrosinase-dependent melanin biosynthesis, and therefore, are candidates as skin-whitening agents.Trifolir...
Isoetharine mesylate salt
T4983CAS 7279-75-6
Isoetharine Mesylate Salt is a β-adrenergic receptor agonist. it also is pregnane X receptor (PXR) activator capable of upregulating CYP450 expression.
1-(2-Pyridyl)piperazine
T5105CAS 34803-66-2
1-(2-Pyridyl)piperazine is a selective α2-adrenoceptor antagonists. 1-(2-Pyridyl)piperazine shows sympatholytic activity. 1-(2-Pyridyl)piperazine is also a met...
Landiolol hydrochloride
T5028CAS 144481-98-1
Landiolol is an ultra-short-acting β1 selective adrenoceptor antagonist.
Methoxyphenamine Hydrochloride
T5035CAS 5588-10-3
Methoxyphenamine is a β-adrenergic receptor agonist of the amphetamine class used as a bronchodilator.
Higenamine
T4963CAS 5843-65-2
Higenamine is a novel α1 -adrenoceptor antagonist.
Clonidine
T7045CAS 4205-90-7
Clonidine is a centrally active alpha-adrenergic agonist used predominantly as an antihypertensive agent, usually in combination with other agents. Despite wid...
BI 1744 hydrochloride
T5159CAS 869477-96-3
Olodaterol is a novel, long-acting β2-adrenergic agonist (EC50s: 97.7 nM for the human β2-adrenoceptor) that exerts its pharmacological effect by binding and...
Amezinium (methylsulfate)
T5327CAS 30578-37-1
Amezinium metilsulfate has multiple mechanisms, including stimulation of alpha and beta-1 receptors and inhibition of noradrenaline and tyramine uptake.
Gramine
T6519CAS 87-52-5
Gramine, a natural indole alkaloid, present in several plant species, acts as an active adiponectin receptor (AdipoR) agonist, with IC50s of 3.2 and 4.2 μM for...
DL-071-IT
T5450CAS 55104-39-7
DL 071-IT is a potent non-selective beta-adrenoceptor antagonist. DL 071 IT showed intrinsic sympathomimetic activity and weak membrane stabilizing activity.
GUANABENZ
T5471CAS 5051-62-7
GUANABENZ is a Central alpha-2 Adrenergic Agonist. The mechanism of action of guanabenz is as an Adrenergic alpha2-Agonist.
Lofexidine
T7160CAS 31036-80-3
Lofexidine is a selective α2-receptor agonist, Lofexidine reduces narcotic withdrawal symptoms.
Levalbuterol tartrate
T7164CAS 661464-94-4
Levosalbutamol tartrate is the β2-adrenergic receptor agonist,and is used to treatment of asthma.
Perphenazine
T1090CAS 58-39-9
Perphenazine is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Pimozide
T2546CAS 2062-78-4
Pimozide is a diphenylbutylpiperidine derivative and a dopamine antagonist with the antipsychotic property. Pimozide selectively inhibits type 2 dopaminergic re...
Norepinephrine
T7044CAS 51-41-2
Norepinephrine can stimulate apoptosis in adult rat ventricular myocytes by activation of the β-adrenergic pathway. It can up-regulate the expression of vascul...
Gemfibrozil
T1415CAS 25812-30-0
Gemfibrozil interacts with peroxisome proliferator-activated receptors (PPARalpha) resulting in PPARalpha-mediated stimulation of fatty acid oxidation and an in...
Yohimbine
TCS2185CAS 146-48-5
Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)
Anisodamine Hydrobromide
T8304CAS 55449-49-5
Anisodamine Hydrobromide is an anticholinergic and α1-adrenergic receptor antagonist used in the treatment of acute circulatory shock.
Dobutamine (hydrochloride)
T8149CAS 49745-95-1
Dobutamine (hydrochloride) is a catecholamine that acts as a β-adrenergic receptor agonist with potent positive inotropic effects.
Bevantolol hydrochloride
T8143CAS 42864-78-8
Bevantolol hydrochloride is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.
Fenoterol
T8358CAS 13392-18-2
Fenoterol is an  agonist of  β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.
Isorhoifolin
TN1797CAS 552-57-8
Isorhoifolin and vicenin II are main compounds of ethyl acetate fraction (EAcF) obtained from Erythrina velutina leaves, EAcF increases the cardiac contractile ...
Meranzin hydrate
TN1922CAS 5875-49-0
Meranzin hydrate exhibits antidepressive and prokinetic-like effects through the regulation of the common mediator, the alpha 2-adrenoceptor , and α±-amino-3-...
Tetrahydroalstonine
TN2267CAS 6474-90-4
Tetrahydroalstonine and Raubasine preferentially block the pressor responses of post-synaptic alpha-adrenergic receptor activation due to exogenous and endogeno...
Phentolamine
T8348CAS 50-60-2
Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist
OPC-28326
T13804CAS 167626-17-7
OPC-28326 is a selective peripheral vasodilator and an α2-adrenergic receptor angatonist(α2A-, α2B- and α2C-adrenoceptors with Ki of 2040, 285, and 55 nM,...
Benzquinamide
T12343CAS 63-12-7
Benzquinamide is an antiemetic, can bind to the α2A, α2B, and α2C adrenergic receptors (α2-AR) (Ki of 1,365, 691, and 545 nM, respectively).
Detomidine carboxylic acid
T11010CAS 115664-39-6
Detomidine carboxylic acid is the main urine metabolite of detomidine. Detomidine is a synthetic α2-adrenergic agonist and an animal analgesic. Detomidine also...
Midaglizole hydrochloride
T11015CAS 79689-25-1
Midaglizole hydrochloride (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6...
Diacetolol D7
T11036CAS 1346604-19-0
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.
SR59230A
T13016CAS 174689-39-5
SR59230A is a selective, and blood-brain barrier penetrating antagonist of β3-adrenergic receptor(IC50s of 40, 408, and 648 nM for β3, β1, and β2 receptors,...
Vilanterol trifenatate
T5134CAS 503070-58-4
Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and ...
Tizanidine
T7065CAS 51322-75-9
Tizanidine is an α2-adrenergic receptor agonist and inhibits neurotransmitter release from CNS noradrenergic neurons.
Ancarolol
T14287CAS 75748-50-4
Ancarolol is a blocking agent of beta-adrenergic.
(R)-Terazosin
T12643CAS 109351-34-0
(R)-Terazosin is an active R-enantiomer of Terazosin. (R)-Terazosin is a potent antagonist of α1-adrenoceptor (α1a, α1b and α1d-adrenoceptor with Ki values ...
Arbutamine
T10364CAS 128470-16-6
Arbutamine is a short-acting synthetic potent nonselective β-adrenoceptor agonist that increases cardiac contractility, heart rate, and systolic blood pressure...
D2343
T15042CAS 72734-63-5
D2343 is an agonist of β2-adrenoceptor. It also is an inhibitor of α1- adrenoceptor.
(S)-Terazosin
T12815CAS 109351-33-9
(S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor...
Fiduxosin
T11286CAS 208993-54-8
Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively. 
Vatinoxan hydrochloride
T13285CAS 130466-38-5
Vatinoxan hydrochloride is an antagonist of peripheral α2 adrenergic receptor.
CGP 20712 A
T10778CAS 105737-62-0
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
ZK-90055 hydrochloride
T13403CAS 84638-81-3
ZK-90055 hydrochloride is an agonist of β2 adrenergic receptor.
(±)-Methotrimeprazine (D6)
T13470CAS 1189805-51-3
(±)-Methotrimeprazine (D6) is the deuterium labeled Methotrimeprazine, which is an antagonist of D3 dopamine and Histamine H1 receptor.
M443
T15943CAS 1820684-31-8
M443 is an irreversible and specific MRK inhibitor (IC50<125 nM).
Mitochonic acid 5
T8366CAS 1354707-41-7
Mitochonic acid 5 is a derivative of the plant hormone indole-3-acetic acid. Mitochonic acid 5 binds mitochondria and ameliorates renal tubular and cardiac myoc...
KUL 7211 racemate
T11786CAS 911196-40-2
KUL 7211 is a selective β-adrenoceptor agonist. KUL 7211 racemate is the racemate of KUL 7211. 
Ritanserin
T16759CAS 87051-43-2
Ritanserin is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM).
Ro 363
T16769CAS 74513-77-2
RO 363 is an effective inotropic stimulant and is a cardiovascular modulator that decreases diastolic blood pressure and pronounces increases in myocardial cont...
Lusaperidone
T11894CAS 214548-46-6
Lusaperidone is an α2 adrenergic receptor antagonist, with Kis of 0.13 and 0.15 nM for α2A and α2C, respectively. 
Prazosin
T22406CAS 19216-56-9
Prazosin, an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.
Bupranolol
T8580CAS 14556-46-8
Bupranolol is an antagonist of β2-adrenergic receptor,and has been used for angina pectoris, hypertension, glaucoma, cardiac arrhythmia and as an antithrombo...
Practolol
T8595CAS 6673-35-4
Practolol is a selective β-adrenoceptor blocker.
Agrimonolide
TN3364CAS 21499-24-1
Agrimonolide is a potential α1 adrenergic receptor antagonist, it exerts anti-inflammatory activity, at least in part, via suppressing LPS-induced activation o...
Akuammigine
TN3368CAS 642-17-1
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding ...
beta-Yohimbine
TN3507CAS 549-84-8
Beta-Yohimbine has approximately twice as toxic as yohimbine and corynanthine about one fifth as toxic. Beta-yohimbine has alpha-1 and alpha-2 adrenoceptor bloc...
Isorauhimbine
TN4323CAS 483-09-0
3-Epi-alpha-yohimbine(Isorauhimbine) has alpha adrenoceptor blocking activities,it also has cardiovascular effects.
Quinine HCl
TN4882CAS 130-89-2
Quinine HCl produces alpha-adrenergic blockade. Quinine modifies catecholamine- and calcium-induced myocardial contractile force responses.
Stephanine
TN5061CAS 517-63-5
l-Stephanine is a potent and highly selective alpha 1 adrenoceptor blocker, inhibits anococcygeus muscle contraction induced by phenylephrine with pA2 values of...
nifenalol.HCl
T8663CAS 5704-60-9
Nifenalol is a antagonist of β-adrenergic receptor.
Clenbuterol
T21147CAS 37148-27-9
Clenbuterol is a substituted phenylaminoethanol that has β2 adrenomimetic properties at very low doses, and is used as a bronchodilator in asthma.
Norepinephrine bitartrate salt
T21066CAS 3414-63-9
Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
Propranolol hydrochloride
T8696CAS 3506-09-0
Propranolol hydrochloride is a blocker of β1 and β2 adrenergic receptor
Phentolamine Analogue 1
T12444CAS 47142-51-8
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of alpha-adrenergic.