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Androgen Receptor

T0135 Estradiol valerate β-estradiol 17-valerate (EV) is a synthetic estrogen. In hormone replacement therapy drugs, it is widely used in combination with other steroid hormones.
T0272 Nilutamide Nilutamide, an antineoplastic hormonal agent, is mainly used in the treatment of prostate Y. Nilutamide is a pure, nonsteroidal anti-androgen with affinity for ...
T0380 Bicalutamide Bicalutamide, a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the receptor bin...
T0476 Abbolactone Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
T0489 Flutamide Flutamide is an antiandrogen with about the same potency as cyproterone in rodent and canine species.
T0856 Dehydroepiandrosterone acetate Dehydroepiandrosterone acetate is a primary C19 steroid generated by the adrenal cortex.
T0856L Dehydroepiandrosterone Dehydroepiandrosterone (DHEA) is an endogenous steroid hormone that is secreted primarily by the adrenal gland and is the most abundant sex steroid. Although th...
T1167 Cyproterone acetate Cyproterone binds the androgen receptor (AR), thereby preventing androgen-induced receptor activation in target tissues and inhibiting the growth of testosteron...
T1541 Drospirenone Drospirenone is a synthetic spironolactone analogue and progestin with progestational and anti-mineralocorticoid activity.
T1596 Chlormadinone acetate Chlormadinone acetate is an orally active synthetic progestational hormone used often in combinations as an oral contraceptive.
T2108 Andarine Andarine (S-4) is an active partial agonist and an investigational selective androgen receptor modulator (SARM).
T2195 Epiandrosterone Epiandrosterone is a dehydroepiandrosterone metabolite and a precursor of testosterone and estradiol with hypolipidemic and anabolic property.
T2207 Adrenosterone Adrenosterone is a steroid hormone isolated from the adrenal cortex.
T2236 RU58841 RU 58841 is a specific androgen receptor antagonist or anti-androgen; RU 58841 has a significant effect on hair regrowth.
T2339 Apalutamide Apalutamide is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
T2408 Ostarine Ostarine is a non-steroidal agent with anabolic activity. Selective androgen receptor modulator (SARM) GTx-024 is designed to work like testosterone, thus promo...
T2991 3,3'-Diindolylmethane DIM (3,3'-diindolylmethane), a small molecule compound, is a proposed Y preventive agent.
T3017 Trenbolone acetate Trenbolone acetate is a synthetic androgen steroid with anabolic properties.
T3137 Parenabol Boldenone undecylenate is a synthetic steroid.
T3357 17 alpha-propionate 17 alpha-propionate is a new topical and peripherally selective androgen antagonist.
T3618 GSK-2881078 GSK2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting t...
T6002 Enzalutamide Enzalutamide (MDV 3100) is a non-steroidal androgen receptor (AR) antagonist (IC50: 36 nM in LNCaP prostate cells).
T6400 AZD3514 AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.
T6509 Galeterone Galeterone is an orally bioavailable small-molecule androgen receptor modulator and CYP17 lyase inhibitor with potential antiandrogen activity. Galeterone exhib...
T6889 MI-136 MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.
T6915 Darolutamide ODM-201 is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).
T4358 Testolone RAD140 is an investigational selective androgen receptor modulator (SARM) for the treatment of conditions such as muscle wasting and breast cancer.
T7040 Angiotensin II human Angiotensin II is mediated by AT1 and AT2 receptors. AT1 and AT2 receptors have seven transmembrane glycoproteins with 30% sequence similarity.Angiotensin I con...
T4357 LGD-3303 LGD-3303 is an androgen receptor modulator, with good oral bioavailability.
T5591 Dihydrotestosterone(DHT) Dihydrotestosterone is a potent androgenic metabolite of testosterone. It is an agonist of the androgen receptor.
T7358 YK11 YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when us...
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