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Androgen Receptor

The androgen receptor (AR), also known as NR3C4 (nuclear receptor subfamily 3, group C, member 4), is a type of nuclear receptor that is activated by binding any of the androgenic hormones, including testosterone and dihydrotestosterone in the cytoplasm and then translocating into the nucleus.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T6002 Enzalutamide 915087-33-1 99.48%
Enzalutamide
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP). Enzalutamide activates autophagy, has antitumor activity, and is commonly u...
T10896L CSRM617 hydrochloride 1353749-74-2 99.47%
CSRM617 hydrochloride
CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 ( OC2, a master regulator of androgen receptor) with a K d of 7...
T8709 Nandrolone phenylpropionate 62-90-8 99.46%
Nandrolone phenylpropionate
Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis
T1261 Medroxyprogesterone Acetate 71-58-9 99.45%
Medroxyprogesterone Acetate
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective ...
T3137 Boldenone Undecylenate 13103-34-9 99.39%
Boldenone Undecylenate
Boldenone Undecylenate (Parenabol) is a synthetic steroid.
T26539 AC-262536 870888-46-3 99.38%
AC-262536
AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.
T15816 LY341495 201943-63-7 99.37%
LY341495
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
T29111 VPC-13566 218464-59-6 99.37%
VPC-13566
VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the B...
T3618 GSK-2881078 1539314-06-1 99.33%
GSK-2881078
GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting t...
T14008 2,2,5,7,8-Pentamethyl-6-Chromanol 950-99-2 99.3%
2,2,5,7,8-Pentamethyl-6-Chromanol
2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol), which has potent androgen receptor (AR) signaling modulation and ...
TCS1372 Atraric acid 4707-47-5 99.27%
Atraric acid
Atraric acid derivatives as a new chemical lead structure for novel therapeutic compounds as AR antagonists, that can be used for prophylaxis or treatment of pro...
T9246 JNJ-63576253 2110428-64-1 99.27%
JNJ-63576253
JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).
T3357 Clascoterone 19608-29-8 99.26%
Clascoterone
Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.
T16090L MK-0773 FA 99.17%
MK-0773 FA
MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is a selective androgen receptor modulator with an IC50 value of 6.6 nM for AR, which can be used for the prevent...
T8217 Enzalutamide carboxylic acid 1242137-15-0 99.17%
Enzalutamide carboxylic acid
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
T6915 Darolutamide 1297538-32-9 99.14%
Darolutamide
Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).
T22263 Bavdegalutamide 2222112-77-6 99.04%
Bavdegalutamide
Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR). Bavdegalutamide can be used in studies about prostate cancer. Bavdegalutamide shows ora...
T5100 DJ-V-159 2253744-53-3 99%
DJ-V-159
DJ-V-159 (DJ-V159) is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A).
T19213 Boldenone Cypionate 106505-90-2 98.78%
Boldenone Cypionate
Boldenone Cypionate is an androgenic anabolic steroid used by recreational bodybuilders and regular gym members.
T2895 Lupeol 545-47-1 98.64%
Lupeol
Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
Enzalutamide
T6002
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP). Enzalutamide activates autophagy, has antitumor activity, and is commonly u...
CSRM617 hydrochloride
T10896L
CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 ( OC2, a master regulator of androgen receptor) with a K d of 7...
Nandrolone phenylpropionate
T8709
Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis
Medroxyprogesterone Acetate
T1261
Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a long-acting contraceptive that is effective ...
Boldenone Undecylenate
T3137
Boldenone Undecylenate (Parenabol) is a synthetic steroid.
AC-262536
T26539
AC-262536 is a selective androgen receptor (SAR) modulator. It has partial agonist activity with respect to testosterone and suppresses luteinizing hormone.
LY341495
T15816
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
VPC-13566
T29111
VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the B...
GSK-2881078
T3618
GSK-2881078 is a selective androgen receptor modulator (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting t...
2,2,5,7,8-Pentamethyl-6-Chromanol
T14008
2,2,5,7,8-Pentamethyl-6-Chromanol (PMC) is the anti-oxidant moiety of vitamin E (α-tocopherol), which has potent androgen receptor (AR) signaling modulation and ...
Atraric acid
TCS1372
Atraric acid derivatives as a new chemical lead structure for novel therapeutic compounds as AR antagonists, that can be used for prophylaxis or treatment of pro...
JNJ-63576253
T9246
JNJ-63576253 is a Clinical Stage Androgen Receptor Antagonist for F877L Mutant and Wild-Type Castration-Resistant Prostate Cancer (mCRPC).
Clascoterone
T3357
Clascoterone (CB-03-01) is a new topical and peripherally selective androgen antagonist.
MK-0773 FA
T16090L
MK-0773 FA (MK-0773 FA (606101-58-0 Free base)) is a selective androgen receptor modulator with an IC50 value of 6.6 nM for AR, which can be used for the prevent...
Enzalutamide carboxylic acid
T8217
Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .
Darolutamide
T6915
Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).
Bavdegalutamide
T22263
Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR). Bavdegalutamide can be used in studies about prostate cancer. Bavdegalutamide shows ora...
DJ-V-159
T5100
DJ-V-159 (DJ-V159) is an agonist for G protein-coupled receptor family C group 6 member A (GPRC6A).
Boldenone Cypionate
T19213
Boldenone Cypionate is an androgenic anabolic steroid used by recreational bodybuilders and regular gym members.
Lupeol
T2895
Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.
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TargetMol