T9035 |
Testosterone undecanoate
|
5949-44-0
|
98.47%
|
|
Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.
|
T0272 |
Nilutamide
|
63612-50-0
|
98.45%
|
|
Nilutamide (RU23908), an antineoplastic hormonal agent, is mainly used in the treatment of prostate Y. Nilutamide is a pure, nonsteroidal anti-androgen with affi...
|
T1167 |
Cyproterone acetate
|
427-51-0
|
98.43%
|
|
Cyproterone acetate (Cyproterone 17-O-acetate) binds the androgen receptor (AR), thereby preventing androgen-induced receptor activation in target tissues and in...
|
T8933 |
JNJ-63576253 free base
|
2110426-27-0
|
98.32%
|
|
JNJ-63576253 free base (TRC253) is a potent and orally active full antagonist of androgen receptor (AR), with IC50s of 37 and 54 nM for F877L mutant AR and wild-...
|
T11410L |
GLPG0492
|
1215085-92-9
|
98.27%
|
|
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic act...
|
T20761 |
RU 59063
|
155180-53-3
|
98.21%
|
|
RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands.
|
T1596 |
Chlormadinone acetate
|
302-22-7
|
98.18%
|
|
Chlormadinone acetate (Gestafortin) is an orally active synthetic progestational hormone used often in combinations as an oral contraceptive.
|
T9752 |
3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
|
2759137-87-4
|
98.15%
|
|
3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.
|
T2207 |
Adrenosterone
|
382-45-6
|
98.13%
|
|
Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.
|
T13273 |
UT-34
|
2168525-92-4
|
98.1%
|
|
UT-34 is a selective and orally active antagonist of second-generation pan-androgen receptor (AR) and degrader(IC50s of 211.7 nM, 262.4 nM and 215.7 nM for wild-...
|
TN2245 |
Sunset Yellow FCF
|
2783-94-0
|
98.03%
|
|
Sunset Yellow FCF (Sunset yellow) is an orange azo dye with pH-dependent absorbance.Sunset Yellow FCF is used in food, cosmetics and pharmaceuticals.It is used a...
|
T7440 |
P,p'-DDE
|
72-55-9
|
98%
|
|
p,p'-DDE (p,p'-dichlorodiphenyldichloroethylene) is a metabolite and degradation product of the organochlorine pesticide DDT
|
T3393 |
Triptophenolide
|
74285-86-2
|
98%
|
|
Triptophenolide (Hypolide) is a compound isolated from Tripterygium wilfordii Hook with anti-inflammatory activity.
|
T7358 |
YK11
|
1370003-76-1
|
98%
|
|
YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when use...
|
T12146 |
N-Desmethyl-Apalutamide
|
1332391-11-3
|
97.83%
|
|
N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.
|
T21740 |
RD162
|
915087-27-3
|
97.74%
|
|
RD162 is a non-steroidal antiandrogen (NSAA) specifically binding to the androgen receptor (AR).
|
T6400 |
AZD3514
|
1240299-33-5
|
96.6%
|
|
AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression.Phase 1.
|
TQ0214 |
Dimethylcurcumin
|
52328-98-0
|
95.77%
|
|
Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer. It effectively suppresses castration-resistant prostate cancer cell proliferatio...
|
T6002 |
Enzalutamide
|
915087-33-1
|
100%
|
|
Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP). Enzalutamide activates autophagy, has antitumor activity, and is commonly u...
|
T75129 |
Luxdegalutamide
|
2750830-09-0
|
100%
|
|
Luxdegalutamide (ARV-766) is an orally available and effective protein degrader of protein hydrolysis-targeted chimeras (PROTAC).Luxdegalutamide degrades the wil...
|