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Search Result

Search Results for " cgrp-receptor "

Targets

CGRP Receptor

29

Compounds

2

Natural Products

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T8682 Vazegepant hydrochloride Vazegepant HCl CGRP Receptor
Vazegepant hydrochloride (Vazegepant HCl) is the first intranasal gepant for the acute treatment of migraine and has announced a positive phase II/III study.
T17194 Ubrogepant MK-1602 CGRP Receptor
Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.
T12293L Olcegepant BIBN-4096,BIBN 4096BS CGRP Receptor
Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP).
TP1040 Calcitonin (salmon) Calcitonin salmon,Salmon calcitonin CGRP Receptor
Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.
T4610 Rimegepant BMS 927711,BMS-927711,BMS927711,BHV-3000 CGRP Receptor
Rimegepant (BMS 927711) is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM.
T6590 MK-3207 Hydrochloride MK-3207 HCl CGRP Receptor
MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.
T13453 CGRP antagonist 1 CGRP Receptor
CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the study of cardiovascular and neurovascular diseases.
TP1323 CGRP 8-37 (rat) CGRP Receptor
CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.
TP1200 CGRP (83-119), rat TFA Calcitonin Gene Related Peptide(83-119), rat TFA Others
CGRP (83-119), rat TFA (Calcitonin Gene Related Peptide(83-119), rat TFA) is a 37 amino acid calcitonin family of neuropeptide, acts through calcitonin receptor-like receptor.
TP1134L HCGRP-(8-37) acetate HCGRP-(8-37) acetate (119911-68-1 free base) CGRP Receptor
HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.
TP1257L Adrenomedullin (AM) (22-52), human acetate Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base） CGRP Receptor
Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an adrenomedullin receptor.
T70820 MK-8825
MK-8825 is a CGRP receptor antagonist.
TP1134 HCGRP-(8-37) Human α-CGRP (8-37)
Rat CGRP-(8-37) (VTHRLAGLLSRSGGVVKDNFVPTNVGSEAF) is a highly selective CGRP receptor antagonist
T16093 Telcagepant MK-0974 Others
Telcagepant is an orally active antagonist of calcitonin gene-related peptide (CGRP) receptor (Kis: 0.77 nM and 1.2 nM for human and rhesus CGRP receptors, respectively).
T38734 Vazegepant Zavegepant,BHV-3500
Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.
T30537 BMS-694153 BMS694153,BMS 694153
BMS-694153 is a potent and selective CGRP receptor antagonist.
TP2044 α-CGRP(human) α-CGRP (human)
Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.
T75978 β-CGRP, human TFA
Human β-CGRP TFA (β-CGRP, human TFA) is a calcitonin peptide that functions through interaction with the calcitonin-receptor-like receptor (CRLR) and receptor-activity-modifying protein (RAMP) complex, demonstrating IC50...
T76363 [Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
[Tyr22] Calcitonin Gene Related Peptide (22-37), rat, refers to a fragment (amino acids 22-37) of the rat calcitonin gene-related peptide (CGRP) that targets the CGRP receptor and adenylate cyclase. While calcitonin is p...
T39522 HTL22562
HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.
TP1203 CGRP(83-119), rat Calcitonin Gene Related Peptide (CGRP) (83-119), rat
Calcitonin Gene Related Peptide (CGRP) (83-119), rat is a 37 amino acid calcitonin family of neuropeptide, acts through calcitonin receptor-like receptor.
T26796 BI-44370
BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.
T12293 Olcegepant hydrochloride BIBN-4096 hydrochloride,BIBN4096BS hydrochloride Others
Olcegepant hydrochloride is a potent and selective non-peptidethe calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (with IC50 of 0.03 nM for human CGRP).
T73703 (3R,5R,6S)-Atogepant
Atogepant ((3R,5R,6S)-MK-8031) is the enantiomer of itself and serves as a calcitonin gene-related peptide (CGRP) receptor antagonist, primarily utilized in migraine research.
TP1131 β-CGRP, human TFA (101462-82-2 free base) CGRP-II (Human) (TFA),Human β-CGRP (TFA),β-CGRP, human TFA
β-CGRP,human tissue is one of the calcitonin peptide, through complex behavior of calcitonin receptor like receptor (CRLR) - and receptor activity - modifying proteins (increased), and 1 and 300 - nM CRLR IC50s/RAMP1 and...
T21558 MK-3207
MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC 50 = 0.12 nM; K i = 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3. IC50 Value: 0.024 nM (Ki, Human CGRP) [1] As other CGRP recep...
T76678 Eptinezumab
Eptinezumab, a human monoclonal antibody, specifically binds to and blocks the calcitonin gene-related peptide (CGRP) from binding to its receptor, thus acting as a preventive treatment for migraine in adults [1].
T75934 AC 187 TFA
AC 187 TFA, a potent and orally active amylin receptor antagonist, exhibits an IC50 of 0.48 nM and a Ki of 0.275 nM. It demonstrates greater selectivity for the amylin receptor over calcitonin and CGRP receptors and has ...
TP2049 CRSP-1
Endogenous central calcitonin (CT) receptor agonist that stimulates cAMP formation at a potency 350-fold greater than CT (ED50 values are 0.2 and 71 nM respectively). Displays no activity at calcitonin-gene related pepti...

Compounds

Vazegepant hydrochloride
T8682
Synonym: Vazegepant HCl
Target: CGRP Receptor
Ubrogepant
T17194
Synonym: MK-1602
Target: CGRP Receptor
Olcegepant
T12293L
Synonym: BIBN-4096,BIBN 4096BS
Target: CGRP Receptor
Calcitonin (salmon)
TP1040
Synonym: Calcitonin salmon,Salmon calcitonin
Target: CGRP Receptor
Rimegepant
T4610
Synonym: BMS 927711,BMS-927711,BMS927711,BHV-3000
Target: CGRP Receptor
MK-3207 Hydrochloride
T6590
Synonym: MK-3207 HCl
Target: CGRP Receptor
CGRP antagonist 1
T13453
Synonym:
Target: CGRP Receptor
CGRP 8-37 (rat)
TP1323
Synonym:
Target: CGRP Receptor
CGRP (83-119), rat TFA
TP1200
Synonym: Calcitonin Gene Related Peptide(83-119), rat TFA
Target: Others
HCGRP-(8-37) acetate
TP1134L
Synonym: HCGRP-(8-37) acetate (119911-68-1 free base)
Target: CGRP Receptor
Adrenomedullin (AM) (22-52), human acetate
TP1257L
Synonym: Adrenomedullin (AM) (22-52), human acetate（159899-65-7 Free base）
Target: CGRP Receptor
MK-8825
T70820
Synonym:
Target:
HCGRP-(8-37)
TP1134
Synonym: Human α-CGRP (8-37)
Target:
Telcagepant
T16093
Synonym: MK-0974
Target: Others
Vazegepant
T38734
Synonym: Zavegepant,BHV-3500
Target:
BMS-694153
T30537
Synonym: BMS694153,BMS 694153
Target:
α-CGRP(human)
TP2044
Synonym: α-CGRP (human)
Target:
β-CGRP, human TFA
T75978
Synonym:
Target:
[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
T76363
Synonym:
Target:
HTL22562
T39522
Synonym:
Target:
CGRP(83-119), rat
TP1203
Synonym: Calcitonin Gene Related Peptide (CGRP) (83-119), rat
Target:
BI-44370
T26796
Synonym:
Target:
Olcegepant hydrochloride
T12293
Synonym: BIBN-4096 hydrochloride,BIBN4096BS hydrochloride
Target: Others
(3R,5R,6S)-Atogepant
T73703
Synonym:
Target:
β-CGRP, human TFA (101462-82-2 free base)
TP1131
Synonym: CGRP-II (Human) (TFA),Human β-CGRP (TFA),β-CGRP, human TFA
Target:
MK-3207
T21558
Synonym:
Target:
Eptinezumab
T76678
Synonym:
Target:
AC 187 TFA
T75934
Synonym:
Target:
CRSP-1
TP2049
Synonym:
Target:
Cat No. Product Name Synonyms Targets
T21581L AC 187 Acetate AC 187 Acetate (151804-77-2 Free base) Amylin Receptor
AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.
TP2167 β-CGRP, human acetate β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate CGRP Receptor
β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor (CRLR) (IC50s: 1 nM and 300 nM for CRLR/RAMP1 and CRLR/RAMP...

Natural Products

AC 187 Acetate
T21581L
Synonym: AC 187 Acetate (151804-77-2 Free base)
Target: Amylin Receptor
β-CGRP, human acetate
TP2167
Synonym: β-CGRP, human acetate (101462-82-2 free),CGRP-II (Human) (acetate),Human β-CGRP acetate
Target: CGRP Receptor

Recombinant Proteins

Species：
Human (3)
Expression System：
HEK293 (3)
Tag：
hFc (2)
His (1)
Cat No. Product Name Species Expression System
TMPY-03280 RAMP3 Protein, Human, Recombinant (hFc) Human HEK293
RAMP3 belongs to the RAMP family. Members of this family are single-transmembrane-domain proteins, called receptor (calcitonin) activity modifying proteins (RAMPs). RAMPs have a wide biological distribution; high concent...
TMPY-00371 STC1 Protein, Human, Recombinant (His) Human HEK293
Stanniocalcin-1 (STC1) is a paracrine factor associated with inflammation and carcinogenesis. STC1 is a secreted glycoprotein hormone and involved in various types of human malignancies. Stanniocalcin-1 (STC1), which has...
TMPY-02839 Adrenomedullin Protein, Human, Recombinant (hFc) Human HEK293
Adrenomedullin consists of 52 amino acids and is a member of the adrenomedullin family. It s a a hypotensive peptide and has 1 intramolecular disulfide bond. It seems that adrenomedullin has a slight homology with the ca...
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