T11021 |
DHODH-IN-12
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1263303-93-0
|
100%
|
|
DHODH-IN-12 is a leflunomide derivative and a weak dihydrorotate dehydrogenase (DHODH) inhibitor with a pKa of 5.07.
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T10140 |
4-Diethylaminobenzaldehyde
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120-21-8
|
|
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4-Diethylaminobenzaldehyde is a reversible aldehyde dehydrogenase (ALDH) inhibitor (Ki: 4 nM for ALDH1). It displays a potent anti-androgenic effect (IC50: 1.71μ...
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T19831 |
Sodium Oxamate
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565-73-1
|
98%
|
|
Sodium Oxamate (Oxamic acid sodium salt) is an LDH inhibitor. Sodium oxamate induces G2/M cell cycle arrest via downregulation of the CDK1/cyclin B1 pathway and ...
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T4173 |
R162
|
64302-87-0
|
98%
|
|
R162 is an effective glutamate dehydrogenase 1 (GDH1) inhibitor.
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T2901 |
Daidzin
|
552-66-9
|
98%
|
|
Daidzin (Daidzoside) is an isoflavone isolated from soya bean with anti-oxidant, anti-carcinogenic, and anti-atherosclerotic activities.
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T73143 |
PHGDH-IN-3
|
2893778-31-7
|
98%
|
|
PHGDH-IN-3 is an orally active phosphoglycerate dehydrogenase (PHGDH) inhibitor with an IC50 of 2.8 μM against PHGDH. PHGDH-IN-3 can be used in studies about can...
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T73446 |
BI‑3231
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2894848-07-6
|
98%
|
|
BI‑3231 is a selective and potent inhibitor of hydroxysteroid 17ß-dehydrogenase 13 HSD17B13, inhibiting hHSD17B13 and mHSD17B13.BI-3231 can be used for the study...
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T9494 |
Imidazole-5-propionic acid
|
1074-59-5
|
98%
|
|
Imidazole-5-propionic acid (Imidazolylpropionic acid) is a product of histidine metabolism and may involve oxidation or transamination. Imidazole-5-propionic aci...
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T0494 |
Tetramisole hydrochloride
|
5086-74-8
|
98%
|
|
Tetramisole hydrochloride (Tetramisole HCl) inhibits alkaline phosphatase and is a high-purity antiparasitic agent.
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T2650 |
MK-8245
|
1030612-90-8
|
98%
|
|
MK-8245 is a liver-targeting SCD inhibitor for human SCD1 (IC50: 1 nM) and for rat/mouse SCD1 (IC50: 3 nM), with anti-diabetic and anti-dyslipidemic function.
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T77576 |
17β-HSD10-IN-1
|
2316765-78-1
|
98%
|
|
17β-HSD10-IN-1 is an orally available 17β-hydroxysteroid dehydrogenase type 10 (17β-HSD10) inhibitor with blood-brain permeability and potency for the study of A...
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T12196 |
NCT-505
|
2231079-74-4
|
98%
|
|
NCT-505 is a potent and selective inhibitor of aldehyde dehydrogenase (ALDH1A1, IC50 = 7 nM) and a weak inhibitor of hALDH1A2, hALDH1A3, hALDH2, hALDH3A1 with IC...
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T10146 |
4-Hydroxyderricin
|
55912-03-3
|
98%
|
|
4-Hydroxyderricin, a potent and selective MAO-B inhibitor (IC50: 3.43 μM), is the main active ingredient of Angelica sinensis, which mildly inhibits dopamine β-h...
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T12438 |
PfDHODH-IN-1
|
183945-55-3
|
98%
|
|
PfDHODH-IN-1 is an analogue of the active Leflunomide metabolite, has antimalarial activity.
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T0897 |
Nitrofurazone
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59-87-0
|
98%
|
|
Nitrofurazone (Furacilin) is a topical anti-infective agent effective against gram-negative and gram-positive bacteria. It is used for superficial WOUNDS AND INJ...
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T0647 |
Tryptamine
|
61-54-1
|
98%
|
|
Tryptamine is a monoamine alkaloid found in animals, plants, and fungi. It contains an indole ring structure and is structurally analogous to the tryptophan. It ...
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T1809 |
AGI-6780
|
1432660-47-3
|
98%
|
|
AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant.
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T6157 |
Devimistat
|
95809-78-2
|
98%
|
|
Devimistat (6,8-Bis(benzylthio)octanoic acid) , a lipoate analog, inhibits mitochondrial enzymes pyruvate dehydrogenase (PDH) and α-ketoglutarate dehydrogenase, ...
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T40686 |
Tiazofurin
|
60084-10-8
|
98%
|
|
Tiazofurin (NSC-286193) is a synthetic nucleoside analogue with antineoplastic activity. Tiazofurin is anabolized intracellularly to tiazole-4-carboxamide adenin...
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T37190 |
L-Allylglycine
|
16338-48-0
|
98%
|
|
L-Allylglycine is an amino acid derivative that reduces glutamate decarboxylase (GAD) activity by 60% when administered at a dose of 39.8 μmol/g per hour ex vivo...
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