Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.

Cat. No.	Product name	CAS No.	Purity
T12489	Pimethixene	314-03-4	99.1%
T12489	Pimethixene (Calmixen) is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist...
T2226	Pergolide mesylate	66104-23-2	99.09%
T2226	Pergolide mesylate salt(LY127809) is a long-acting dopamine agonist which has been used to treat PARKINSON DISEASE and HYPERPROLACTINEMIA but withdrawn from some...
T1871	GBR 12935 dihydrochloride	67469-81-2	99.09%
T1871	GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.
T27060	CP-226269	220941-93-5	99.08%
T27060	CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM. CP 226269 can be used to study neurological diso...
T2564	Cis-(Z)-Flupentixol dihydrochloride	51529-01-2	99.07%
T2564	cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.
T4369	SCH-23390 hydrochloride	125941-87-9	99.07%
T4369	SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).
T0255	Clomipramine hydrochloride	17321-77-6	99.07%
T0255	Clomipramine hydrochloride (Anafranil) is a tricyclic antidepressant similar to IMIPRAMINE that selectively inhibits the uptake of serotonin in the brain. It is ...
T17072	Thiethylperazine dimaleate	1179-69-7	99.07%
T17072	Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor. Thiethylperazine dimaleate is an activator of ABCC1 an...
T21855	AMI-193	510-74-7	99.04%
T21855	AMI-193 (Spiramide) is an effective and selective antagonist of 5-HT2 and D2 receptor with Kis of 2, 3, 50, 2530, and 4300 nM for 5-HT2, D2 Receptor, 5-HT1A, D1 ...
T22508	3-CPMT	14008-79-8	99.03%
T22508	3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.
T8389	Trifluoperazine	117-89-5	99.03%
T8389	Trifluoperazine (trifluoroperazine) is a Dopamine D2 receptor inhibitor(IC50 : 1.2 nM), and Treatment of schizophrenia.
T0716	Molindone hydrochloride	15622-65-8	99%
T0716	Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.
T9409	Mesdopetam hemitartrate	2562346-14-7	98.96%
T9409	Mesdopetam hemitartrate (IRL790 hemitartrate) is an antagonist of dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM for human recombinant D3 receptor). It has psychomo...
T12405	Pentiapine	81382-51-6	98.93%
T12405	Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.
T3526	Dasotraline hydrochloride	675126-08-6	98.92%
T3526	Dasotraline hydrochloride (SEP-225289 hydrochloride) (SEP-225289 hydrochloride) is a triple reuptake inhibitor that inhibits dopamine, norepinephrine, and seroto...
T28809	SLV-310	264869-71-8	98.91%
T28809	SLV-310 is a potent dopamine D2 receptor antagonist and 5-HT reuptake receptor inhibitor used in the study of neurological disorders such as bipolar disorder and...
T15686	L-741626	81226-60-0	98.9%
T15686	L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3 an...
T7728	ACEPROMAZINE MALEATE	3598-37-6	98.87%
T7728	ACEPROMAZINE MALEATE is a dopamine receptor antagonist
T9237	Rotigotine	92206-54-7	98.84%
T9237	Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.
T5047	PD-168077 maleate	630117-19-0	98.82%
T5047	PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)