Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.

Cat. No.	Product name	CAS No.	Purity
T1105	Penfluridol	26864-56-2	99.94%
T1105	Penfluridol (TLP-607) is a highly potent antipsychotic.
T3497	Ocaperidone	129029-23-8	99.94%
T3497	Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.
T16392	ONC206	1638178-87-6	99.93%
T16392	ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and poss...
T0455	Clozapine	5786-21-0	99.93%
T0455	Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent. It binds several types of central nervous system receptors, an...
T1567	Olanzapine	132539-06-1	99.92%
T1567	Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.
T1412	Loxapine succinate	27833-64-3	99.92%
T1412	Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.
T5397	A-381393	726174-00-1	99.92%
T5397	A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).
T14853	Cabergoline	81409-90-7	99.92%
T14853	Cabergoline (FCE-21336) is an ergot derived-dopamine D2-like receptor agonist. It has high affinity for D2, D3, and 5-HT2B receptors (Ki=0.7, 1.5, and 1.2, respe...
T1540	Doxepin hydrochloride	1229-29-4	99.91%
T1540	Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
T3278	Piribedil	3605-01-4	99.91%
T3278	Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.
T2793	Tetrahydropalmatine	2934-97-6	99.91%
T2793	Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epileptic a...
T3085	Piperacetazine	3819-00-9	99.9%
T3085	Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.
T7352	Pridopidine	346688-38-8	99.89%
T7352	Pridopidine (FR310826), a dopamine (DA) stabilizer, acts as a low affinity dopamine D2 receptor (D2R) antagonist, improves motor performance and shows neuroprote...
T2874	Tetrahydroberberine	522-97-4	99.89%
T2874	Tetrahydroberberine (Canadine) is an isoquinoline alkaloid isolated from corydalis tuber, has a micromolar affinity for dopamine D(2) receptors.
T0280	Spiperone	749-02-0	99.89%
T0280	Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds. It has been recommended in the treatment of SCHIZOPHRE...
T4S0779	D-tetrahydropalmatine	3520-14-7	99.89%
T4S0779	D-Tetrahydropalmatine is a organic cation transporter 1 (OCT1) inhibitor, it can obviously inhibit the uptake of monocrotaline (MCT) in MDCK-hOCT1 cells and isol...
T16759	Ritanserin	87051-43-2	99.89%
T16759	Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine ...
T12352L	Oxidopamine hydrobromide	636-00-0	99.88%
T12352L	Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.
T5842	Bromocriptine mesylate	22260-51-1	99.87%
T5842	Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)
T9100	BP 897	192384-87-5	99.87%
T9100	BP 897 (2-Naphthalenecarboxamide, N-[4-[4-(2-methoxyphenyl)-1-piperazinyl]butyl]-) is a potent and selective dopamine D3 receptor agonist, and a weak dopamine D2...