Dopamine Receptor

Dopamine receptors are a class of G protein-coupled receptors that are prominent in the vertebrate central nervous system (CNS). Dopamine receptors activate different effectors through not only G-protein coupling, but also signaling through different protein (dopamine receptor-interacting proteins) interactions.

Cat. No.	Product name	CAS No.	Purity
T33816	Ordopidine	871351-60-9	99.52%
T33816	Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity. Ordopi...
T2190	Methiothepin mesylate	74611-28-2	99.51%
T2190	Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.
T9081	FAUC 346	474432-65-0	99.51%
T9081	FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.
T13110	Tedatioxetine hydrobromide	960151-65-9	99.50%
T13110	Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and an antagonist of 5-HT2A, 5-HT2C, 5-HT3, and α...
T21337	Lurasidone	367514-87-2	99.5%
T21337	Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6....
T2132	Buspirone hydrochloride	33386-08-2	99.5%
T2132	Buspirone hydrochloride (Buspar) is a 5HT(1A) receptor agonist, used to treat generalized anxiety disorder (GAD).
T27677	JNJ-37822681	935776-74-2	99.48%
T27677	JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.
T10232	Acetophenazine dimaleate	5714-00-1	99.48%
T10232	Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.
T10705	CCG 203769	410074-60-1	99.46%
T10705	CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.
T32737	Liafensine	1198790-53-2	99.46%
T32737	Liafensine(BMS-820836) is a novel and selective triple monoamine reuptake inhibitor with inhibitory effects on the reuptake of serotonin, norepinephrine, and dop...
T23483	U 99194 maleate	234757-41-6	99.45%
T23483	U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.
T4576	Perospirone	150915-41-6	99.45%
T4576	Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agon...
TQ0311	GSK163090	844903-58-8	99.45%
TQ0311	GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).
T11463	GR 103691	162408-66-4	99.44%
T11463	GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM). It shows more than 100-fold selectivity for human dopamine human (h)D3 over hD4 an...
T11011	Dexpramipexole dihydrochloride	104632-27-1	99.44%
T11011	Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine agon...
T5S2059	Glaucine	475-81-0	99.42%
T5S2059	Glaucine has antitussive, antioxidative potential and antiviral activities, it may be an anti-arthritic agent, it can enhance LPS and zymosan-induced IL-10 produ...
T38754	Trazpiroben	1352993-39-5	99.41%
T38754	Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.
T8959	OS-3-106	1580000-17-4	99.4%
T8959	OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.
T1292	Tiapride hydrochloride	51012-33-0	99.4%
T1292	Tiapride is a selective blocker of D2/3 dopamine receptors in the brain. It is used in the therapy of various psychiatric and neurological disorders containing d...
T21432	Molindone	7416-34-4	99.37%
T21432	Molindone ((±)-Molindone) is a therapeutic antipsychotic used to treat schizophrenia by blocking the action of dopamine in the brain. molindone is often used in ...