T3913 |
Saikosaponin D
|
20874-52-6
|
99.09%
|
|
Saikosaponin D is a novel SERCA inhibitor by inhibiting NF-κB and STAT3 signaling to protect against acetaminophen-induced hepatotoxicity.
|
T11399 |
Giredestrant
|
1953133-47-5
|
98.96%
|
|
Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has an...
|
T7839 |
Lasofoxifene Tartrate
|
190791-29-8
|
98.96%
|
|
Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.
|
T0345 |
Estropipate
|
7280-37-7
|
98.95%
|
|
Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine.
|
T3855 |
Tracheloside
|
33464-71-0
|
98.95%
|
|
Tracheloside significantly decreases the activity of alkaline phosphatase (IC50: 0.31 μg/ml), a level of inhibition comparable to that of tamoxifen (IC50: 0.43 μ...
|
T13674 |
Elacestrant
|
722533-56-4
|
98.92%
|
|
Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant is an orally available selective estrogen receptor degrader .
|
T12482 |
Pipendoxifene hydrochloride
|
245124-69-0
|
98.9%
|
|
Pipendoxifene hydrochloride is a selective modulator of estrogen receptor.
|
T11237L |
Camizestrant TFA
|
T11237L
|
98.9%
|
|
Camizestrant TFA (AZD-9833 TFA) is a potent and orally active antagonist of estrogen receptor (ER).
|
T2231 |
Estradiol dipropionate
|
113-38-2
|
98.89%
|
|
Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.
|
T2569 |
Chlorotrianisene
|
569-57-3
|
98.88%
|
|
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen r...
|
T7644 |
DPN
|
1428-67-7
|
98.85%
|
|
DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
|
T9604 |
Beta-Estradiol 17-hemisuccinate
|
7698-93-3
|
98.72%
|
|
beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.
|
T5118 |
Brilanestrant
|
1365888-06-7
|
98.71%
|
|
Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).
|
T0301 |
Ethisterone
|
434-03-7
|
98.51%
|
|
Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.
|
T3975 |
AZD9496
|
1639042-08-2
|
98.47%
|
|
AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.
|
T8984 |
FLTX1
|
1481401-71-1
|
98.46%
|
|
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under pe...
|
T1193 |
Clomiphene citrate
|
50-41-9
|
98.45%
|
|
Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.
|
T68042 |
CHF-4227
|
444643-64-5
|
98.44%
|
|
CHF-4227 is a novel, potent and selective estrogen receptor modulator that reduces cholesterol and LDL cholesterol concentrations.
|
T16566 |
Propyl pyrazole triol
|
263717-53-9
|
98.39%
|
|
Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 4...
|
T11200 |
Endoxifen (E-isomer)
|
114828-90-9
|
98.31%
|
|
Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.
|