Home Tools
Log in
Cart

Estrogen Receptor/ERR

The ERRs are orphan nuclear receptors, meaning the identity of their endogenous ligand has yet to be unambiguously determined. They are named because of sequence homology with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones.There are three human estrogen related receptors:ERRα,ERRβand ERRγ .
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T3913 Saikosaponin D 20874-52-6 99.09%
Saikosaponin D
Saikosaponin D is a novel SERCA inhibitor by inhibiting NF-κB and STAT3 signaling to protect against acetaminophen-induced hepatotoxicity.
T11399 Giredestrant 1953133-47-5 98.96%
Giredestrant
Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has an...
T7839 Lasofoxifene Tartrate 190791-29-8 98.96%
Lasofoxifene Tartrate
Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.
T0345 Estropipate 7280-37-7 98.95%
Estropipate
Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine.
T3855 Tracheloside 33464-71-0 98.95%
Tracheloside
Tracheloside significantly decreases the activity of alkaline phosphatase (IC50: 0.31 μg/ml), a level of inhibition comparable to that of tamoxifen (IC50: 0.43 μ...
T13674 Elacestrant 722533-56-4 98.92%
Elacestrant
Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
T12482 Pipendoxifene hydrochloride 245124-69-0 98.9%
Pipendoxifene hydrochloride
Pipendoxifene hydrochloride is a selective modulator of estrogen receptor.
T11237L Camizestrant TFA T11237L 98.9%
Camizestrant TFA
Camizestrant TFA (AZD-9833 TFA) is a potent and orally active antagonist of estrogen receptor (ER).
T2231 Estradiol dipropionate 113-38-2 98.89%
Estradiol dipropionate
Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.
T2569 Chlorotrianisene 569-57-3 98.88%
Chlorotrianisene
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen r...
T7644 DPN 1428-67-7 98.85%
DPN
DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
T9604 Beta-Estradiol 17-hemisuccinate 7698-93-3 98.72%
beta-Estradiol 17-hemisuccinate
beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.
T5118 Brilanestrant 1365888-06-7 98.71%
Brilanestrant
Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).
T0301 Ethisterone 434-03-7 98.51%
Ethisterone
Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.
T3975 AZD9496 1639042-08-2 98.47%
AZD9496
AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.
T8984 FLTX1 1481401-71-1 98.46%
FLTX1
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under pe...
T1193 Clomiphene citrate 50-41-9 98.45%
Clomiphene citrate
Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.
T68042 CHF-4227 444643-64-5 98.44%
CHF-4227
CHF-4227 is a novel, potent and selective estrogen receptor modulator that reduces cholesterol and LDL cholesterol concentrations.
T16566 Propyl pyrazole triol 263717-53-9 98.39%
Propyl pyrazole triol
Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 4...
T11200 Endoxifen (E-isomer) 114828-90-9 98.31%
Endoxifen (E-isomer)
Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.
Saikosaponin D
T3913
Saikosaponin D is a novel SERCA inhibitor by inhibiting NF-κB and STAT3 signaling to protect against acetaminophen-induced hepatotoxicity.
Giredestrant
T11399
Giredestrant (GDC-9545) potently competes with estradiol for binding and induces a conformational change within the ER ligand binding domain. Giredestrant has an...
Lasofoxifene Tartrate
T7839
Lasofoxifene Tartrate (CP-336156) is a third-generation, non-steroidal selective estrogen receptor modulator.
Estropipate
T0345
Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine.
Tracheloside
T3855
Tracheloside significantly decreases the activity of alkaline phosphatase (IC50: 0.31 μg/ml), a level of inhibition comparable to that of tamoxifen (IC50: 0.43 μ...
Elacestrant
T13674
Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant  is an orally available selective estrogen receptor degrader .
Pipendoxifene hydrochloride
T12482
Pipendoxifene hydrochloride is a selective modulator of estrogen receptor.
Camizestrant TFA
T11237L
Camizestrant TFA (AZD-9833 TFA) is a potent and orally active antagonist of estrogen receptor (ER).
Estradiol dipropionate
T2231
Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.
Chlorotrianisene
T2569
Chlorotrianisene (tri-p-anisylchloroethylene) is an orally bioavailable, highly lipophilic, synthetic triphenylethylene (TPE) derivative and selective estrogen r...
DPN
T7644
DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
beta-Estradiol 17-hemisuccinate
T9604
beta-Estradiol 17-hemisuccinate selectively stains estrogen receptor (ER)-rich cells.
Brilanestrant
T5118
Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).
Ethisterone
T0301
Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.
AZD9496
T3975
AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.
FLTX1
T8984
FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under pe...
Clomiphene citrate
T1193
Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.
CHF-4227
T68042
CHF-4227 is a novel, potent and selective estrogen receptor modulator that reduces cholesterol and LDL cholesterol concentrations.
Propyl pyrazole triol
T16566
Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 4...
Endoxifen (E-isomer)
T11200
Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.
1 2 3 4 5 6
TargetMol