T12654 |
(Rac)-Acolbifene
|
151533-34-5
|
98.18%
|
|
(Rac)-Acolbifene (EM-343) is the racemic form of Acolbifene. Acolbifene is a estrogen receptor antagonist. (Rac)-Acolbifene exhibits anti-estrogenic and estrogen...
|
T10239 |
Acolbifene
|
182167-02-8
|
98.17%
|
|
Acolbifene (SCH 57068) is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ER...
|
T20744 |
Nylestriol
|
39791-20-3
|
98.16%
|
|
Nylestriol (LY 49825) is an agonist of estrogen receptor.
|
T15364 |
G-1
|
881639-98-1
|
98.14%
|
|
G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).
|
T15249 |
Estrogen receptor modulator 1
|
63676-22-2
|
98.14%
|
|
Estrogen receptor modulator 1 causes regression of Tamoxifen-resistant, hormone-independent xenograft tumors. Estrogen receptor modulator 1 is an orally active a...
|
T12832 |
Amcenestrant
|
2114339-57-8
|
98.13%
|
|
Amcenestrant (SAR439859) is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD). SAR439859 is a potent antagonist of ER (with an EC...
|
T2810 |
(20S)-Protopanaxatriol
|
34080-08-5
|
98.12%
|
|
(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid re...
|
T11236 |
Giredestrant tartrate
|
2407529-33-1
|
98.01%
|
|
Giredestrant tartrate (Estrogen receptor antagonist 1) is a novel, orally active, selective and effective non-steroidal estrogen receptor antagonist. Giredestran...
|
T7313 |
Enclomiphene citrate
|
7599-79-3
|
98%
|
|
Enclomiphene citrate (trans-Clomiphene citrate) is a non-steroidal estrogen receptor antagonist,with antioestrogenic property
|
T7299 |
β-Estradiol 17-acetate
|
1743-60-8
|
98%
|
|
β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) is a metabolite of estradiol.
|
T5624 |
Bisphenol B
|
77-40-7
|
98%
|
|
Bisphenol B has a binding affinity for estrogen receptors.
|
T5531 |
GSK-4716
|
101574-65-6
|
98%
|
|
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
|
T3665 |
Tectoridin
|
611-40-5
|
98%
|
|
Tectoridin (Shekanin) possesses an estrogenic and thyroid hormone-like agent by activating estrogen and thyroid hormone receptors. Tectoridin has anti-oxidant, a...
|
T0040 |
Quinestrol
|
152-43-2
|
98%
|
|
Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer and prostate...
|
T5835 |
PROTAC ERRα ligand 2
|
2306388-57-6
|
98%
|
|
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
|
T2544 |
Bazedoxifene acetate
|
198481-33-3
|
98%
|
|
Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).
|
T5S0543 |
Isocurcumenol
|
24063-71-6
|
98%
|
|
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
|
T15788 |
LSZ-102
|
2135600-76-7
|
97.84%
|
|
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
|
T2882 |
Genistin
|
529-59-9
|
97.65%
|
|
Genistin (Genistoside) is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflamm...
|
T8370 |
GSK5182
|
877387-37-6
|
97.63%
|
|
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)
|