T0171 |
Norethynodrel
|
68-23-5
|
|
|
Norethynodrel (Lynestrol) is a synthetic progestational hormone with actions and uses similar to those of PROGESTERONE. It has been used in the treatment of func...
|
T77724 |
OBHSA
|
1404508-27-5
|
98%
|
|
OBHSA(Oxabicycloheptane sulfonamide) is a novel selective estrogen receptor depressant (SERD) that can be used to study breast cancer.
|
TN2045 |
Pelargonidin-3-O-glucoside chloride
|
18466-51-8
|
98%
|
|
Pelargonidin-3-O-glucopyranoside is the glucoside of Pelargonidin, an potential antidiabetic agent. Pelargonidin-3-O-glucopyranoside has antioxidant, anti-inflam...
|
TQ0149 |
Prinaberel
|
524684-52-4
|
98%
|
|
Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
|
TN2288 |
Uralenol
|
139163-15-8
|
98%
|
|
Uralenol significantly shows the inhibitory activities against the PTP1B enzyme; it also shows inhibitory activities on mushroom tyrosinase using l-tyrosine as s...
|
T6404 |
Bazedoxifene hydrochloride
|
198480-56-7
|
98%
|
|
Bazedoxifene hydrochloride (TSE-424) is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM an...
|
T12278 |
NXT629
|
1454925-59-7
|
98%
|
|
NXT629 is a selective and competitive antagonist of PPAR-α(human PPARα with an IC50 of 77 nM).
|
TN2200 |
Segetalin A
|
161875-97-4
|
98%
|
|
Segetalin A has estrogen-like activity.
|
TN3802 |
Dehydrodiconiferyl alcohol
|
4263-87-0
|
98%
|
|
Dehydrodiconiferyl alcohol (DHCA) is a lignan isolated from calabash that inhibits osteoclast differentiation and oophorectomy induced bone loss by acting as an ...
|
T6827 |
Endoxifen Z-isomer hydrochloride
|
1032008-74-4
|
98%
|
|
Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
|
T21897 |
Methylpiperidino pyrazole
|
289726-02-9
|
98%
|
|
Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.
|
TN1690 |
Glabrene
|
60008-03-9
|
98%
|
|
Glabrene, Liquiritin apioside, neolicuroside, and 18α²-glycyrrhetic acid are the predominant phenolic derivatives partitioning at the interface and most likely t...
|
TQ0163 |
Sagittatoside A
|
118525-35-2
|
98%
|
|
Sagittatoside A selectively activates estrogen response element (ERE)-luciferase activity via ERα.
|
T16351 |
NSC16168
|
6837-93-0
|
98%
|
|
NSC16168 inhibits DNA repair and potentiates CDDP efficacy in cancer. NSC16168 is a specific ERCC1-XPF inhibitor (IC50: 0.42 μM).
|
T12329 |
Ospemifene D4
|
T12329
|
98%
|
|
Ospemifene D4 is a deuterium labeled Ospemifene. Ospemifene is a selective and orally active modulator of estrogen receptor.
|
T12312 |
OP-1074
|
1443752-76-8
|
98%
|
|
OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.
|
TN1679 |
Genistein 7,4'-di-O-β-D-glucoside
|
36190-98-4
|
98%
|
|
Genistein 7,4'-di-O-beta-D-glucopyranoside shows significant estrogenic proliferative effect in MCF-7 cell in sub-cytotoxic concentration range.
|
T11222 |
ERB-196
|
550997-55-2
|
98%
|
|
Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.
|
T11231 |
ERRγ Inverse Agonist 1
|
2316832-86-5
|
98%
|
|
ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].
|
T6819 |
Desogestrel
|
54024-22-5
|
99.96%
|
|
Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.
|