Estrogen/progestogen Receptor

Estrogen receptors are a group of proteins found inside cells. They are receptors that are activated by the hormone estrogen (17β-estradiol). Two classes of estrogen receptor exist: ER, which is a member of the nuclear hormone family of intracellular receptors, and GPER (GPR30), which is a member of the rhodopsin-like family of G protein-coupled receptors.The progesterone receptor (PR), also known as NR3C3 or nuclear receptor subfamily 3, group C, member 3, is a protein found inside cells. It is activated by the steroid hormone progesterone.

Cat. No.	Product name	CAS No.	Purity
T7644	DPN	1428-67-7	98.85%
T7644	DPN (Diarylpropionitrile) is an selective agonist of estrogen receptor β (ERβ) .
T7709	(E/Z)-GSK5182	T7709	98.83%
T7709	(E/Z)-GSK5182 (GSK5182(Z/E)) is a racemic mixture comprising (E)-GSK5182 and (Z)-GSK5182 isomers. It acts as a highly selective and orally active inverse agonist...
T25534	Indazole-Cl	848142-62-1	98.72%
T25534	Indazole-Cl is a selective ERß agonist and a selective estrogen receptor modifier (SERM).
T5118	Brilanestrant	1365888-06-7	98.71%
T5118	Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).
T0301	Ethisterone	434-03-7	98.51%
T0301	Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.
T3975	AZD9496	1639042-08-2	98.47%
T3975	AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.
T8984	FLTX1	1481401-71-1	98.46%
T8984	FLTX1 is a fluorescent derivative of Tamoxifen, designed to efficiently target and label intracellular Tamoxifen-binding sites (estrogen receptors) both under pe...
T1193	Clomiphene citrate	50-41-9	98.45%
T1193	Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.
T16566	Propyl pyrazole triol	263717-53-9	98.39%
T16566	Propyl pyrazole triol (PPT) is a selective agonist of estrogen receptor alpha. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 4...
T4000	(±)-Equol	94105-90-5	98.28%
T4000	(±)-Equol ((R,S)-Equol) is a non-steroidal estrogen produced from the metabolism of the isoflavonoid phytoestrogen daidzen by human intestinal microflora. The es...
T12832	Amcenestrant	2114339-57-8	98.13%
T12832	Amcenestrant (SAR439859) is an orally active, nonsteroidal and selective degrader of estrogen receptor (SERD). SAR439859 is a potent antagonist of ER (with an EC...
T2810	(20S)-Protopanaxatriol	34080-08-5	98.12%
T2810	(20S)-Protopanaxatriol (g-PPT)(g-PPT), a metabolite of ginsenoside, could regulate endothelial cell functions through the estrogen receptor and glucocorticoid re...
T77552	SLU-PP-1072	2285432-57-5	98.1%
T77552	SLU-PP-1072 is an ERRα and ERRγ inverse dual agonist that disrupts PCa cell metabolism and induces apoptosis through cell cycle dysregulation.SLU-PP-1072 is used...
T11915	LY88074	177744-96-6	98.05%
T11915	LY88074 is a raloxifene analog in which the basic side chain has been removed. LY88074 is an agonist of ERβ (EC50 = 232 nM).This compound stimulates uterine cel...
T0040	Quinestrol	152-43-2	98%
T0040	Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer and prostate...
T5835	PROTAC ERRα ligand 2	2306388-57-6	98%
T5835	PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
T2544	Bazedoxifene acetate	198481-33-3	98%
T2544	Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).
T13768	(+)-Medicarpin	33983-39-0	97.8%
T13768	(+)-Medicarpin, a pterocarpan, is an isoflavonoid compound derived from multiple medicinal plant species such as Sophora japonica, Zollernia paraensis, Platymisc...
T7904	SR 19881	2213490-89-0	97.76%
T7904	SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).
T8370	GSK5182	877387-37-6	97.63%
T8370	GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)