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GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T3927 Phellopterin 2543-94-4 99.99%
Phellopterin
Phellopterin is a partial agonist of the central benzodiazepine receptors in vitro. Phellopterin shows a cytotoxic effect on RAW264.7 cell at the concentration f...
T2850 Bicuculline 485-49-4 99.99%
Bicuculline
Bicuculline ((+)-Bicuculline) is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and...
T1396 Bemegride 64-65-3 99.97%
Bemegride
Bemegride (3-Ethyl-3-methylglutarimide) is a central nervous system stimulant and antidote for barbiturate poisoning.
T8572 CL 218872 66548-69-4 99.97%
CL 218872
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 n...
T2339 Apalutamide 956104-40-8 99.97%
Apalutamide
Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
T0715 Chlormezanone 80-77-3 99.97%
Chlormezanone
Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
T2S1464 Thiocolchicoside 602-41-5 99.94%
Thiocolchicoside
Thiocolchicoside (Thiocolchicine 2-glucoside analog) (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a ...
T5375 Loreclezole 117857-45-1 99.94%
Loreclezole
Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.
T8639 Phenibut (hydrochloride) 3060-41-1 99.93%
Phenibut (hydrochloride)
Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing v...
T13536 Afoxolaner 1093861-60-9 99.93%
Afoxolaner
Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA...
T0710 L-Cycloserine 339-72-0 99.92%
L-Cycloserine
L-Cycloserine ((-)-Cycloserine) irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminotransferase in E. coli, as well in the brains of various animals...
T7699 AZD7325 942437-37-8 99.88%
AZD7325
AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
T8036 6-Methylflavone 29976-75-8 99.86%
6-Methylflavone
6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
T1065 Baclofen 1134-47-0 99.85%
Baclofen
Baclofen (Lioresal) is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing B...
T8630 Baclofen hydrochloride 28311-31-1 99.83%
Baclofen hydrochloride
Baclofen hydrochloride (4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride) is a GAMMA-AMINOBUTYRIC ACID derivative that is a specific GABA-B RECEPTORS agon...
T11349 GABAA receptor agent 1 1571-87-5 99.83%
GABAA receptor agent 1
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
T9424 Temgicoluril 10095-06-4 99.83%
Temgicoluril
Temgicoluril (mebikar) acts on GABA Receptor.
T11307 Fluxametamide 928783-29-3 99.83%
Fluxametamide
Fluxametamide is a novel isoxazoline insecticide that acts via distinctive antagonism of insect ligand-gated chloride channels, acts as an antagonist of GABA- an...
TN2268 Tetrahydromagnolol 20601-85-8 99.82%
Tetrahydromagnolol
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
T0349 Riluzole 1744-22-5 99.81%
Riluzole
Riluzole (RP-54274) is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMY...
Phellopterin
T3927
Phellopterin is a partial agonist of the central benzodiazepine receptors in vitro. Phellopterin shows a cytotoxic effect on RAW264.7 cell at the concentration f...
Bicuculline
T2850
Bicuculline ((+)-Bicuculline) is a light-sensitive competitive antagonist of GABAA receptors. It was originally identified in 1932 in plant alkaloid extracts and...
Bemegride
T1396
Bemegride (3-Ethyl-3-methylglutarimide) is a central nervous system stimulant and antidote for barbiturate poisoning.
CL 218872
T8572
CL 218872 is a benzodiazepine agonist displaying selectivity for α1 subunit-containing GABAA receptors (Ki values are 130, 1820, 1530, > 10000, 490 and > 10000 n...
Apalutamide
T2339
Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.
Chlormezanone
T0715
Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.
Thiocolchicoside
T2S1464
Thiocolchicoside (Thiocolchicine 2-glucoside analog) (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a ...
Loreclezole
T5375
Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.
Phenibut (hydrochloride)
T8639
Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing v...
Afoxolaner
T13536
Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs. Afoxolaner acts on the insect GABA and glutamate receptors, inhibiting GABA...
L-Cycloserine
T0710
L-Cycloserine ((-)-Cycloserine) irreversibly inhibits GABA pyridoxal 5′-phosphate-dependent aminotransferase in E. coli, as well in the brains of various animals...
AZD7325
T7699
AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.
6-Methylflavone
T8036
6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.
Baclofen
T1065
Baclofen (Lioresal) is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing B...
Baclofen hydrochloride
T8630
Baclofen hydrochloride (4-amino-3-(4-chlorophenyl)butanoic acid hydron chloride) is a GAMMA-AMINOBUTYRIC ACID derivative that is a specific GABA-B RECEPTORS agon...
GABAA receptor agent 1
T11349
GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.
Temgicoluril
T9424
Temgicoluril (mebikar) acts on GABA Receptor.
Fluxametamide
T11307
Fluxametamide is a novel isoxazoline insecticide that acts via distinctive antagonism of insect ligand-gated chloride channels, acts as an antagonist of GABA- an...
Tetrahydromagnolol
TN2268
Tetrahydromagnolol can activate cannabinoid (CB) receptors.
Riluzole
T0349
Riluzole (RP-54274) is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMY...
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TargetMol