GABA Receptor

The GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels (also known as ionotropic receptors); whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors.

Cat. No.	Product name	CAS No.	Purity
T11307	Fluxametamide	928783-29-3	99.83%
T11307	Fluxametamide is a novel isoxazoline insecticide that acts via distinctive antagonism of insect ligand-gated chloride channels, acts as an antagonist of GABA- an...
T0349	Riluzole	1744-22-5	99.81%
T0349	Riluzole (RP-54274) is a glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMY...
T4728	4-Acetamidobutanoic acid	3025-96-5	99.79%
T4728	4-Acetamidobutanoic acid (4-ACETAMIDOBUTYRIC ACID) can be found in blood, feces, and urine, as well as in human prostate tissue. 4-Acetamidobutanoic acid exists ...
T2067	NS11394	951650-22-9	99.76%
T2067	NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(1...
T28294	Panadiplon	124423-84-3	99.75%
T28294	Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of ...
T2979	DL-Menthol	89-78-1	99.74%
T2979	DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis. (–)-Menthol is more com...
T2940	6-Hydroxyflavone	6665-83-4	99.73%
T2940	6-Hydroxyflavone (6-HF) is a noncompetitive inhibitors of cytochrome P450 2C9. It is a flavone, a type of chemical compound. It is reported in leaves of Barleria...
T7000	Tiagabine hydrochloride	145821-59-6	99.72%
T7000	Tiagabine hydrochloride (NO050328 hydrochloride) is the hydrochloride salt form of tiagabine, a nipecotic acid derivative with anticonvulsant property. A selecti...
T16581	Progabide	62666-20-0	99.7%
T16581	Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.
T3741	(-)-borneol	464-45-9	99.69%
T3741	(-)-borneol (L-Borneol) has a highly efficacious positive modulating action at GABA receptor with an EC50 of 237 μM.
T1128	Oxiracetam	62613-82-5	99.69%
T1128	Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.
T2720	Ginsenoside Rc	11021-14-0	99.66%
T2720	Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
T0024	Primidone	125-33-7	99.66%
T0024	Primidone (NCI-C56360) is a potent anticonvulsant agent. It is a neuronal voltage-gated sodium channel blocker and has value in the study of epilepsy, essential ...
T7794	Zuranolone	1632051-40-1	99.66%
T7794	Zuranolone is an agonist of GABAA receptor.
T8040	Cholesterol myristate	1989-52-2	99.65%
T8040	Cholesterol Myristate (Cholesteryl Myristate) is a natural steroid found in traditional Chinese medicine that interacts with various ion channels, including the ...
T40659L	γ-Acetylenic GABA hydrochloride	103451-26-9	99.64%
T40659L	γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.
T9113	Myristicin	607-91-0	99.63%
T9113	Myristicin (Myristicine) is a natural product found in spices and umbelliferous plants. Myristicin has anti-cholinergic, Antibacterial, and hepatoprotective effe...
T0051	Urethane	51-79-6	99.63%
T0051	Urethane (Ethylurethane) was an antineoplastic agent .Now is used for other medicinal purposes.
TNU0685	Dipropofol	2416-95-7	99.6%
TNU0685	Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.
T5734	(+)-BORNEOL	464-43-7	99.6%
T5734	(+)-BORNEOL (d-Borneol) is a natural bicyclic monoterpene used for analgesia and anesthesia in traditional Chinese medicine; enhances GABA receptor activity with...