T4688 |
Pipequaline hydrochloride
|
80221-58-5
|
99.43%
|
|
Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It ...
|
T11684 |
Isoguvacine hydrochloride
|
68547-97-7
|
99.41%
|
|
Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist. Isoguvacine hydrochloride binds to rat synapti...
|
T0702 |
Gabapentin
|
60142-96-3
|
99.39%
|
|
Gabapentin (Neurontin) is an Anti-epileptic Agent. The physiologic effect of gabapentin is by means of Decreased Central Nervous System Disorganized Electrical A...
|
T34146 |
Propanidid
|
1421-14-3
|
99.39%
|
|
Propanidid (Sombrevin) is a gamma-aminobutyric acid type A receptor (GABAA) agonist and a fast-acting intravenous anesthetic that lowers arterial blood pressure....
|
T20242 |
Chlorothymol
|
89-68-9
|
99.37%
|
|
Chlorothymol (AI3-00120) is a disinfectant used in oral.
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T15775 |
Lotilaner
|
1369852-71-0
|
99.32%
|
|
Lotilaner is a parasiticide. It is used as a potent non-competitive antagonist of insects GABACl receptors (IC50 of 23.84 nM for Drosophila melanogaster GABA rec...
|
T8887 |
2'MeO6MF
|
89112-85-6
|
99.26%
|
|
2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional re...
|
T13690 |
Etifoxine hydrochloride
|
56776-32-0
|
99.25%
|
|
Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug. Unlike benzodiazepines, Etifoxine hydrochloride appears to produce i...
|
T26891 |
BPDBA
|
312281-74-6
|
99.24%
|
|
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and m...
|
T2407 |
Tiagabine
|
115103-54-3
|
99.24%
|
|
Tiagabine (NO050328) is an Anti-epileptic Agent. The physiologic effect of tiagabine is by means of Decreased Central Nervous System Disorganized Electrical Acti...
|
T2983 |
3,4,5-Trimethoxycinnamic acid
|
90-50-6
|
99.19%
|
|
3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the GA...
|
T4363 |
CGP52432
|
139667-74-6
|
99.16%
|
|
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
|
T3S2100 |
(-)-Securinine
|
5610-40-2
|
99.12%
|
|
(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.
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T77568 |
6,7-dimethylisatin
|
20205-43-0
|
99.09%
|
|
6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.
|
T23470 |
Tracazolate hydrochloride
|
1135210-68-2
|
99.07%
|
|
Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity. Tracazolate hydrochlori...
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T17144 |
TPA 023
|
252977-51-8
|
99.06%
|
|
TPA 023 is a selective agonist of GABAA α2/α3 subtype (Kis = 0.19 - 0.41 nM).
|
T0627 |
β-Alanine
|
107-95-9
|
99%
|
|
β-Alanine (3-Aminopropanoic acid) is a naturally occurring beta amino acid formed in vivo by the degradation of dihydrouracil and carnosine. It acts as a neurotr...
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T0883 |
Tramiprosate
|
3687-18-1
|
99%
|
|
Tramiprosate (Alzhemed) is an orally active, blood-brain-barrier-crossing, naturally occurring amino acid found in a variety of red seaweeds that binds soluble A...
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T1602 |
Valproic acid sodium salt
|
1069-66-5
|
99%
|
|
Valproic acid sodium salt (Sodium Valproate) is the sodium salt form of valproic acid with anti-epileptic activity. Valproic acid sodium salt is converted into i...
|
T2775 |
Baicalin
|
21967-41-9
|
98.96%
|
|
Baicalin (Baicalein 7-O-β-D-glucuronide) is a prolyl endopeptidase inhibitor isolated from scutellaria baicalensis, with antioxidant, anti-tumor, anti-HIV proper...
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