Cart
GPCR/G Protein Glucagon Receptor

Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Cat No. product name
T11408 GLP-1 receptor agonist 1 GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
T12878 Semaglutide TFA Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor.
T3967 Exendin-4 Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer...
T7364 NNC-0640 NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
T8748 Exendin-4 acetate
TP1469 Lixisenatide acetate Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
TP1796 Albiglutide TFA Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
TQ0124 BETP BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
TQ0239 PF-06291874 PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
GLP-1 receptor agonist 1
T11408CAS 2212020-52-3
GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
Semaglutide TFA
T12878CAS T12878
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
GRA-Ex-25
T3422CAS 307983-31-9
GRA-Ex-25 is an inhibitor of glucagon receptor.
Exendin-4
T3967CAS 141758-74-9
Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer...
NNC-0640
T7364CAS 307986-98-7
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
Exendin-4 acetate
T8748CAS 914454-01-6
Lixisenatide acetate
TP1469CAS 1997361-87-1
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
Albiglutide TFA
TP1796CAS TP1796
Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
BETP
TQ0124CAS 1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
PF-06291874
TQ0239CAS 1393124-08-7
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.