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GPCR/G Protein Glucagon Receptor

Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Cat No. product name
T3422 GRA-Ex-25 GRA-Ex-25 is an inhibitor of glucagon receptor.
T3967 Exendin-4 Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer...
T7364 NNC-0640 NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
TQ0124 BETP BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
TQ0239 PF-06291874 PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
T8355 Exendin-4 Exendin-4 is a glucagon-like protein-1 (GLP-1) receptor agonist
T12878 Semaglutide TFA Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T11408 GLP-1 receptor agonist 1 GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
GRA-Ex-25
T3422CAS 307983-31-9
GRA-Ex-25 is an inhibitor of glucagon receptor.
Exendin-4
T3967CAS 141758-74-9
Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer...
NNC-0640
T7364CAS 307986-98-7
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
BETP
TQ0124CAS 1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
PF-06291874
TQ0239CAS 1393124-08-7
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
Exendin-4
T8355CAS 141732-76-5
Exendin-4 is a glucagon-like protein-1 (GLP-1) receptor agonist
Semaglutide TFA
T12878CAS
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
GLP-1 receptor agonist 1
T11408CAS 2212020-52-3
GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .