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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T2535 | Ivabradine hydrochloride | S 16257-2,Ivabradine HCl | Adrenergic Receptor |
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hyperpolarization-activated, cyclic nucleotide-gat... | |||
T7516 | ZD7288 | ICI D7288 | HCN Channel |
ZD7288 (ICI D7288), a selective hyperpolarization-activated cyclic nucleotide-gated channel blocker, inhibits hippocampal synaptic plasticity. | |||
T10813 | Cilobradine hydrochloride | DK-AH 269 | HCN Channel |
Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels. | |||
T13387L | Zatebradine hydrochloride | UL-FS-49CL,UL-FS-49 | Others , HCN Channel |
Zatebradine hydrochloride (UL-FS-49CL) is a highly effective and effective HCN Channel inhibitor (IC50:1.96 µM). HCN Channel is an effective hyperpolarization activated loop nucleotide gated channel. Zatebradine hydrochl... | |||
T70573 | Cilobradine | ||
Cilobradine is an HCN Channel blocker; an open channel blocker of neuronal Ih and related cardiac If channels. | |||
T37160 | 8-Demethyl Ivabradine | ||
8-Demethyl Ivabradine is a metabolite derived from Ivabradine, an orally bioavailable cyclic nucleotide-gated (HCN) channel blocker with hyperpolarization-activated properties[1]. | |||
T73975 | Ivabradine impurity 1 | ||
Ivabradine Impurity 1, identified as an impurity of Ivabradine, is an orally bioavailable compound that functions as a blocker of the hyperpolarization-activated, cyclic nucleotide-gated (HCN) channel [1]. | |||
T63014 | Ivabradine | ||
Ivabradine is a potent, orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits pacemaker current (If). ivabradine decreases heart rate in a dose-dependent manner and does no... |