Home > HIV Protease

HIV Protease

T0100	Atazanavir sulfate	Atazanavir sulfate is an azapeptide and HIV-PROTEASE INHIBITOR that is used in the treatment of HIV INFECTIONS and AIDS in combination with other ANTI-HIV AGENT...
T0100L	Atazanavir	Atazanavir(BMS-232632) is an highly effective HIV-1 protease inhibitor.
T0110	Zalcitabine	Zalcitabine(Dideoxycytidine;ddC; 2',3'-Dideoxycytidine) is a nucleoside analog reverse transcriptase inhibitor (NRTI); At low concentrations, It can potently in...
T1267	Abacavir	Abacavir is a nucleoside reverse transcriptase inhibitor analog of guanosine. This agent decreases HIV viral loads, retards or prevents the damage to the immune...
T1525	Ritonavir	Ritonavir is a peptidomimetic agent that inhibits both HIV-1 and HIV-2 proteases. Ritonavir is highly inhibited by serum proteins but boosts the effect of other...
T1595	Nevirapine	Nevirapine is a benzodiazepine non-nucleoside reverse transcriptase inhibitor. In combination with other antiretroviral drugs, nevirapine reduces HIV viral load...
T1623	Lopinavir	Lopinavir is a peptidomimetic HIV protease inhibitor that retains activity against HIV protease with the Val 82 mutation. Lopinavir is less affected by binding ...
T1815	Dapivirine	Dapivirine is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.
T1883	Des(benzylpyridyl) Atazanavi	Atazanavir is a highly effective HIV-1 protease inhibitor.
T2239	Raltegravir potassium	Raltegravir potassium salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.
T2324	Darunavir	Darunavir is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS. Due to the emergence of ANTIVIRAL DRUG RESISTANCE when used alo...
T2329	Dolutegravir sodium	Dolutegravir sodium salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature mutants Y143R, Q1...
T2332	Elvitegravir	Elvitegravir is a Human Immunodeficiency Virus Integrase Strand Transfer Inhibitor. The mechanism of action of elvitegravir is as an HIV Integrase Inhibitor, an...
T2393	Efavirenz	Efavirenz is a Human Immunodeficiency Virus 1 Non-Nucleoside Analog Reverse Transcriptase Inhibitor. The mechanism of action of efavirenz is as a Non-Nucleoside...
T2409L	Tenofovir Disoproxil Fumarate	Tenofovir Disoproxil Fumarate is a pro-drug, fumaric acid salt form of tenofovir, a nucleoside reverse transcriptase inhibitor analog of adenosine. Tenofovir di...
T2728	Limonin	Limonin is a triterpenoid enriched in citrus fruits, which has antivirus and antitumor ability.
T2830	Betulinic acid	Betulinic acid is a pentacyclic lupane-type triterpene derivative of betulin (isolated from the bark of Betula alba, the common white birch) which has antiretro...
T3172	Trovirdine	Trovirdine is a thiourea non-nucleoside reverse transcriptase inhibitor.
T3335	Darunavir Ethanolate	Darunavir ethanolate is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS. Due to the emergence of ANTIVIRAL DRUG RESISTANCE wh...
T3523	Fostemsavir	BMS-663068 is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.
T3632	Doravirine	Doravirine is a non-nucleoside reverse transcriptase inhibitor, used in the treatment of HIV/AIDS.
T3683	lithospermic acid	lithospermic acid is a potent anti-HIV agent and shows anti-gonadotrophic and anti-thyroidal effects.
T3732	Sebacic acid	Sebacic acid is a saturated, straight-chain naturally occurring dicarboxylic acid.
T6001	Nelfinavir Mesylate	Nelfinavir Mesylate is an effective HIV protease inhibitor (Ki: 2 nM).
T6065	Triciribine	Triciribine is a DNA synthesis inhibitor, and it also inhibits Akt and HIV-1/2.
T6098	Cabotegravir	Cabotegravir (GSK744, GSK1265744) is a long-acting HIV integrase inhibitor and inhibits the HIV-1 integrase catalyzed strand transfer reaction (IC50: 3.0 nM).
T6198	Dolutegravir	Dolutegravir (IC50=2.7 nM), a two-metal-binding HIV integrase inhibitor, exhibits medium activity against raltegravir-resistant signature mutants Y143R, Q148K, ...
T6367	Abacavir sulfate	Abacavir， a nucleoside analogue，effectively utilize its antiviral activity
T6388	Amprenavir	Amprenavir is a synthetic derivative of hydroxyethylamine sulfonamide that selectively binds to and inhibits human immunodeficiency virus (HIV) protease.
T6420	BMS-707035	BMS-707035 is a specific HIV-I integrase (IN) inhibitor with IC50 of 15 nM. Phase 2.
T6653	Salmeterol Xinafoate	Salmeterol Xinafoate is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma symptoms and chronic obstr...
T3S2007	MRE-269	Ursonic acid belongs to the family of Ursane Triterpenes whose structure is based on the pentacyclic ursane skeleton. It has potential as HIV-1 Protease Inhibit...
T4S0295	Cosmosiin	1. Cosmosiin is a anti-HIV agent. 2. Cosmosiin may be beneficial for diabetic complications through their enhanced adiponectin secretion, tyrosine phosphorylati...
T5S0983	Absinthiin	1. Absinthiin is a weak HIV-1 protease inhibitor.
T2S0223	Isosinensetin	1. Isosinensetin shows antioxidant and HIV-1 protease inhibiting activities.
T4493	Bictegravir	Bictegravir is a potent inhibitor of HIV-1 integrase (IC50: 7.5 nM).
TL0006	Chicoric Acid	Chicoric Acid is a potent inhibitor of human immunodeficiency virus type-1 (HIV-1) integrase and the replication in tissues. It also a class of cannabinomimetic...
T4S1999	Valepotriate	Valepotriate fraction can have sedative effects and affect behavioral parameters related to recognition memory. Valepotriates, a new class of cytotoxic and anti...
T4962	Ginsenoside Z-R1	Zingibroside R1 has anti-HIV-1 activity.
T4S1718	Punicalin	Punicalin exerts anti-inflammatory, antioxidative, and anti-hepatotoxic activities, it shows inhibitory activity on HIV-1 reverse transcriptase in a dose-depend...

Prev 1 Next