T14831 |
Bryostatin 1
|
83314-01-6
|
98%
|
|
Bryostatin 1 is a natural macrolide isolated from the bryozoan Bugula neritina and is a CNS)permeable PKC modulator. Bryostatin 1 binds to the isolated C1 domain...
|
T15683 |
L-689502
|
138483-63-3
|
98%
|
|
L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).
|
TN3119 |
5-Hydroxy-7,8-dimethoxyflavanone
|
113981-49-0
|
98%
|
|
5-Hydroxy-7,8-dimethoxyflavanone is isolated from Andrographis paniculata Nees. leaves and roots with anti-inflammatory activity.
|
TN4705 |
Oleoside
|
178600-68-5
|
98%
|
|
Oleoside can be extracted from Olea europaea and Zizyphus lotus L. twigs and may be used to inhibit HIV-1 protease.
|
T35617 |
Mitoguazone
|
459-86-9
|
98%
|
|
Mitoguazone (Methyl-GAG) is a selective S-adenosyl-methionine decarboxylase inhibitor that penetrates the blood-brain barrier and disrupts polyamine biosynthesis...
|
TN4605 |
Myriceric acid B
|
55497-79-5
|
98%
|
|
Myriceric acid B is a potent HIV-1 entry inhibitor targeting gp41 and can serve as a lead compound for developing novel anti-HIV-1 drug. Myriceric acid B scaveng...
|
T8156 |
Saquinavir mesylate
|
149845-06-7
|
98%
|
|
Saquinavir mesylate (Ro 31-8959/003) is an Inhibitor of HIV Proteaseused in antiretroviral therapy
|
TN5191 |
Tsugafolin
|
66568-97-6
|
98%
|
|
Tsugafolin has weak anti-HIV activity.
|
TN1194 |
16beta,17-Dihydroxy-ent-kaurane-19-oic acid
|
74365-74-5
|
98%
|
|
16beta,17-Dihydroxy-ent-kaurane-19-oic acid as an anti-HIV principle, it showed significant activity against HIV replication in H9 lymphocyte cells with an EC50 ...
|
T10111L |
3-Deazaadenosine
|
6736-58-9
|
98%
|
|
3-Deazaadenosine is an inhibitor of S-adenosylhomocysteine hydrolase, with a Ki of 3.9 µM, and it has anti-inflammatory, anti-proliferative and anti-HIV activity...
|
T22468 |
1-Deoxymannojirimycin hydrochloride
|
73465-43-7
|
98%
|
|
α-mannosidase I inhibitor
|
TN5133 |
3',5,5',7-Tetrahydroxy-4',6-dimethoxyflavone
|
125537-92-0
|
98%
|
|
5,7,3',5'-tetrahydroxy-6,4'-dimethoxyflavone exhibits anti-HIV-1 activity in the anti-syncytium assay using (∆Tat/rev)MC99 virus and 1A2 cell line system, it sho...
|
TN1348 |
8-Prenylluteone
|
125002-91-7
|
98%
|
|
8-Prenylluteone can potently inhibit HIV-1 PR activity.
|
TN1708 |
Gomisin M2
|
82425-45-4
|
98%
|
|
Gomisin M2 is an anti-HIV agent.
|
TN3152 |
6-Acetonyldihydrochelerythrine
|
22864-92-2
|
98%
|
|
6-Acetonyldihydrochelerythrine exhibits significant antioxidant activities, it exhibits significant anti-HIV activity in H9 lymphocytes with EC50 and TI (Therape...
|
T10928 |
Cytochalasin A
|
14110-64-6
|
98%
|
|
Cytochalasin A is a cell-permeable fungal toxin and is an oxidized derivative of cytochalasin B. Cytochalasin A is an inhibitor of HIV-1 protease (IC50 = 3 μM), ...
|
TN4584 |
Morolic acid
|
559-68-2
|
98%
|
|
Morolic acid and moronic acid have shown sustained antidiabetic and antihyperglycemic action possibly mediated by an insulin sensitization with consequent change...
|
T14307 |
Aplaviroc
|
461443-59-4
|
98%
|
|
Aplaviroc (AK 602), a SDP derivative, is a CCR5 antagonist. With IC50s of 0.1-0.4 nM for HIV-1Ba-L, HIV-1JRFL and HIV-1MOKW.
|
T14559 |
BI 224436
|
1155419-89-8
|
98%
|
|
BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.
|
TN3777 |
Daurichromenic acid
|
82003-90-5
|
98%
|
|
Daurichromenic acid is a terpenophenol with a potent anti-HIV activity.
|