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Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T4499 Mequitazine 29216-28-2 99.95%
Mequitazine
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
T0031 Ziprasidone hydrochloride monohydrate 138982-67-9 99.95%
Ziprasidone hydrochloride monohydrate
Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic ac...
T0211L Azelastine hydrochloride 79307-93-0 99.94%
Azelastine hydrochloride
Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.
T0081 Lafutidine 118288-08-7 99.94%
Lafutidine
Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.
T0217 Levodropropizine 99291-25-5 99.93%
Levodropropizine
Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
T29096 Vapitadine dihydrochloride 279253-83-7 99.92%
Vapitadine dihydrochloride
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
T0217L (+)-Dropropizine 99291-24-4 99.92%
(+)-Dropropizine
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex and by interfering...
T6488 Epinastine hydrochloride 108929-04-0 99.92%
Epinastine hydrochloride
Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
T1822L Clemizole hydrochloride 1163-36-6 99.91%
Clemizole hydrochloride
Clemizole hydrochloride is an antagonist for H1 histamine receptor. According to the research, Clemizole hydrochloride can inhibit hepatitis C virus (HCV) replic...
T1540 Doxepin hydrochloride 1229-29-4 99.91%
Doxepin hydrochloride
Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
T1469 Levocetirizine 130018-77-8 99.9%
Levocetirizine
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.
T0381 Amodiaquine dihydrochloride dihydrate 6398-98-7 99.9%
Amodiaquine dihydrochloride dihydrate
Amodiaquine dihydrochloride dihydrate (Amodiaquine hydrochloride) is the hydrochloride salt of amodiaquine, an orally active 4-aminoquinoline derivative with ant...
T1425 Pemirolast potassium 100299-08-9 99.89%
Pemirolast potassium
Pemirolast Potassium is the potassium salt form of pemirolast, a pyrimidinone derivative with antiallergic property. Pemirolast potassium (TWT-8152) exerts its a...
T0330 Diphenhydramine hydrochloride 147-24-0 99.89%
Diphenhydramine hydrochloride
Diphenhydramine hydrochloride (DPH) is a histamine H1 antagonist used as an antitussive and antiemetic. It is also used for pruritus and dermatoses, for hypersen...
T16759 Ritanserin 87051-43-2 99.89%
Ritanserin
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine ...
T0246 Betahistine dihydrochloride 5579-84-0 99.88%
Betahistine dihydrochloride
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.
T41247 Thioperamide maleate 148440-81-7 99.88%
Thioperamide maleate
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31 ...
T21390 Fexofenadine 83799-24-0 99.87%
Fexofenadine
Fexofenadine (Carboxyterfenadine), an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. C...
T0678 Amitriptyline hydrochloride 549-18-8 99.87%
Amitriptyline hydrochloride
Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive ...
T2848 Osthole 484-12-8 99.87%
Osthole
Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.
Mequitazine
T4499
Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.
Ziprasidone hydrochloride monohydrate
T0031
Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic ac...
Azelastine hydrochloride
T0211L
Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.
Lafutidine
T0081
Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.
Levodropropizine
T0217
Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
Vapitadine dihydrochloride
T29096
Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
(+)-Dropropizine
T0217L
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved in the cough reflex and by interfering...
Epinastine hydrochloride
T6488
Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.
Clemizole hydrochloride
T1822L
Clemizole hydrochloride is an antagonist for H1 histamine receptor. According to the research, Clemizole hydrochloride can inhibit hepatitis C virus (HCV) replic...
Doxepin hydrochloride
T1540
Doxepin hydrochloride (Aponal) is a dibenzoxepin tricyclic compound. It displays a range of pharmacological actions including maintaining adrenergic innervation....
Levocetirizine
T1469
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.
Amodiaquine dihydrochloride dihydrate
T0381
Amodiaquine dihydrochloride dihydrate (Amodiaquine hydrochloride) is the hydrochloride salt of amodiaquine, an orally active 4-aminoquinoline derivative with ant...
Pemirolast potassium
T1425
Pemirolast Potassium is the potassium salt form of pemirolast, a pyrimidinone derivative with antiallergic property. Pemirolast potassium (TWT-8152) exerts its a...
Diphenhydramine hydrochloride
T0330
Diphenhydramine hydrochloride (DPH) is a histamine H1 antagonist used as an antitussive and antiemetic. It is also used for pruritus and dermatoses, for hypersen...
Ritanserin
T16759
Ritanserin (R 55667) is a highly effective, relatively selective, long-acting antagonist of 5-HT2 receptor (IC50: 0.9 nM), less active on Histamine H1, Dopamine ...
Betahistine dihydrochloride
T0246
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.
Thioperamide maleate
T41247
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31 ...
Fexofenadine
T21390
Fexofenadine (Carboxyterfenadine), an antihistamine pharmaceutical drug, is used to treat allergy symptoms, such as nasal congestion, hay fever, and urticaria. C...
Amitriptyline hydrochloride
T0678
Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive ...
Osthole
T2848
Osthole (Osthol), a potential inhibitor of histamine H1 receptor, has been shown to stimulate osteoblast proliferation and differentiation.
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TargetMol