Histamine Receptor

The histamine receptors are a class of G protein–coupled receptors which bind histamine as their primary endogenous ligand.

Cat. No.	Product name	CAS No.	Purity
T20597	Alginic acid	9005-32-7	98%
T20597	Alginic acid is a natural polysaccharide extracted from brown seaweeds with anti-anaphylactic and anti-inflammatory activities. Alginic acid inhibits histamine r...
TN1661	Ganoderic acid C2	103773-62-2	98%
TN1661	Ganoderic acid C2 has anti-inflammatory,and anti-tumor-promoting activities. Ganoderic acid C2 can inhibit histamine release, it also has inhibitory effects on t...
T5829	H4 Receptor antagonist 1	848217-00-5	98%
T5829	H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.
T8599	Betazole dihydrochloride	138-92-1	98%
T8599	Betazole hydrochloride is an agonist of H2 receptor.
T25875	Noberastine	110588-56-2	98%
T25875	Noberastine is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.
T0053	Hydroxyzine Pamoate	10246-75-0	98%
T0053	Hydroxyzine pamoate is a histamine H1 receptor antagonist that is effective in the treatment of chronic urticaria, dermatitis, and histamine-mediated pruritus. U...
T1269	Tripelennamine hydrochloride	154-69-8	98%
T1269	Tripelennamine hydrochloride is a histamine H1 antagonist with low sedative action but frequent gastrointestinal irritation.
T1115	Doxylamine succinate	562-10-7	98%
T1115	Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties. Doxylamine succinate competitively blocks the histamine ...
T0174	Cyproheptadine hydrochloride sesquihydrate	41354-29-4	98%
T0174	Cyproheptadine hydrochloride sesquihydrate, an antihistamine, is an antagonist of serotonin and histamine2.
T0903	Cinnarizine	298-57-7	98%
T0903	Cinnarizine is a piperazine derivative having histamine H1-receptor and calcium-channel blocking activity with vasodilating and antiemetic properties but it indu...
T3723	Dioxopromethazine hydrochloride	15374-15-9	98%
T3723	Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.
T0172	Maprotiline hydrochloride	10347-81-6	98%
T0172	Maprotiline hydrochloride is a bridged-ring tetracyclic antidepressant that is both mechanistically and functionally similar to the tricyclic antidepressants, in...
T22724	Dimaprit dihydrochloride	23256-33-9	98%
T22724	Dimaprit dihydrochloride is a selective histamine H2 receptor agonist. Dimaprit dihydrochloride also inhibits nNOS with an IC50 of 49 μM. It can stimulate gastri...
T6534	Histamine dihydrochloride	56-92-8	98%
T6534	Histamine, an organic nitrogen compound, works on target cells in the mammalian brain by stimulating of Histamine 1/2.
T0298	Dimenhydrinate	523-87-5	98%
T0298	Dimenhydrinate is an ethanolamine and histamine antagonist with anti-allergic activity.
T1470L	Fexofenadine hydrochloride	138452-21-8	98%
T1470L	Fexofenadine Hydrochloride is a carboxylated metabolic derivative of terfenadine and long-lasting selective histamine H1 receptor antagonist, with antihistaminic...
T6535	Histamine Phosphate	51-74-1	98%
T6535	Histamine acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.
T16280	Nedocromil	69049-73-6	98%
T16280	Nedocromil inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
T40652	Meclizine	569-65-3	98%
T40652	Meclizine (Meclozine) shows antihistamine activity and reversibly inhibits the interaction of histamine at the H1 receptors . Meclizine is a member of the pipera...
T0445L	Promethazine hydrochloride	58-33-3	98%
T0445L	Promethazine HCl(NSC-231688), the first-generation antihistamine, is a strong antagonist of the H1 receptor and a moderate antagonist of the mACh receptor, moder...