T3552 |
CPI-455
|
1628208-23-0
|
99.02%
|
|
CPI-455 is a specific KDM5 inhibitor.
|
T39252 |
TAK-418
|
1818252-53-7
|
98.87%
|
|
TAK-418 is a selective and orally active inhibitor of LSD1/KDM1A enzyme with an IC50 of 2.9 nM. TAK-418 unlocks abnormal epigenetic mechanisms and improves autis...
|
T63140 |
LSD1-IN-20
|
1239589-91-3
|
98.72%
|
|
Lsd1-in-20 is a potent dual inhibitor of LSD1/G9a with Ki values of 0.44 and 0.68 μM, respectively. LSD1-IN-20 showed antiproliferative activity against THP-1 le...
|
T27723L |
KDM5-C49 HCl
|
|
98.59%
|
|
KDM5-C49 HCl (KDOAM-20 hydrochloride) is a potent and selective inhibitor of KDM5 demethylase. KDM5-C49 HCL(1596348-16-1 Free base) is a candidate compound for t...
|
T4383 |
GSK-J4 Hydrochloride
|
1797983-09-5
|
98.36%
|
|
GSK-J4 Hydrochloride (GSK J4 HCl) is a cell permeable, potent and selective histone demethylase(JMJD3 )inhibitor. is an ethyl ester derivative of the GSK-J1 with...
|
T10864 |
Corin
|
1808113-09-8
|
98.22%
|
|
Corin is an irreversible inhibitor of HDAC1(IC50 = 147 nM) and LSD1(Ki = 110 nM).
|
T4527 |
Seclidemstat
|
1423715-37-0
|
98.03%
|
|
Seclidemstat (SP-2577) is an effective LSD1 inhibitor, with a mean IC50 of 127 nM.
|
T1868 |
JIB-04
|
199596-05-9
|
98.02%
|
|
JIB-04 (NSC 693627) is a pan-selective Jumonji histone demethylase inhibitor.
|
T4418 |
GSK2879552 2HCl (1401966-69-5(free base))
|
T4418
|
98%
|
|
GSK2879552 is an orally available, irreversible inhibitor of lysine specific demethylase 1 (LSD1), with potential antineoplastic activity.
|
T0802 |
Procaine hydrochloride
|
51-05-8
|
98%
|
|
Procaine hydrochloride (Novocaine HCl) is the hydrochloride salt form of procaine, a benzoic acid derivative with local anesthetic and antiarrhythmic properties....
|
T5825 |
Iadademstat dihydrochloride
|
1431303-72-8
|
98%
|
|
Iadademstat dihydrochloride (ORY-1001(trans)) , a Potent and Selective Covalent KDM1A/LSD1 Inhibitor, for the Treatment of Acute Leukemia.
|
T11882 |
Pulrodemstat benzenesulfonate
|
2097523-60-7
|
97.73%
|
|
Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) is a potent and orally active inhibitor of lysine specific demethylase-1 (LSD1) with anticancer activit...
|
T39389 |
KDM2B-IN-2
|
1965248-01-4
|
97.57%
|
|
KDM2B-IN-2 is a potent histone demethylase (kdm2b) inhibitor.
|
T6593 |
ML324
|
1222800-79-4
|
97.49%
|
|
ML324(IC50=920 nM) is a specific inhibitor of jumonji histone demethylase (JMJD2).
|
T1025 |
Tranylcypromine (2-PCPA) hydrochloride
|
1986-47-6
|
97.19%
|
|
Tranylcypromine (2-PCPA) hydrochloride (SKF-385 HCl), a Monoamine Oxidase inhibitor, is effective in the treatment of major depression, dysthymic disorder, and a...
|
T3100 |
GSK-J4
|
1373423-53-0
|
97.07%
|
|
GSK-J4 (GSK J4 HCl) is a potent H3K27me3 demethylase inhibitor, with IC50s of 8.6 μM and 6.6 μM towards KDM6B and KDM6A respectively. It is the first selective i...
|
T5368 |
Eicosapentaenoic Acid
|
10417-94-4
|
96.20%
|
|
Eicosapentaenoic Acid (EPA) is a ω-3 fatty acid abundantly available in marine organisms.
|
T5484 |
GSK467
|
1628332-52-4
|
100%
|
|
GSK467 is a potent and selective inhibitor of KDM5 (JARID1)(Ki : 10 nM).
|
T22821 |
GSK J5
|
1394854-51-3
|
100%
|
|
GSK J5 is an inhibitor of schistosomes and helminths and is often used as a trematode insecticide.GSK J5 promotes schistosome mortality in a dose- and time-depen...
|
T13748 |
L-2-Hydroxyglutaric acid disodium
|
63512-50-5
|
|
|
L-2-Hydroxyglutaric acid disodium ((S)-2-Hydroxyglutaric acid disodium) is an epigenetic modifier and putative oncometabolite in renal cancer. L-2-Hydroxyglutari...
|