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Search Result

Search Results for " leukotriene receptor "

Targets

Leukotriene Receptor Leukotriene Receptor Lipoxygenase LTR

70

Compounds

6

Natural Products

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T1677 Montelukast Singular Leukotriene Receptor , Lipoxygenase , LTR
Montelukast (Singular) is an orally available leukotriene receptor antagonist which is widely used for the prophylaxis and chronic treatment of asthma and has been linked to rare cases of clinically apparent liver injury...
T16280 Nedocromil FPL 59002 Leukotriene Receptor , Prostaglandin Receptor , Histamine Receptor
Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
T26519 Ablukast Ro 23-3544 Leukotriene Receptor
Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.
T22946 LY255283 LY 255283 Leukotriene Receptor
LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human peripheral blood polymorphonuclear leukocytes (PMNL) and in monocytes activated by calcium ionophore A2318...
T1677L Montelukast sodium MK0476 Leukotriene Receptor , LTR
Montelukast sodium (MK0476) is an orally available leukotriene receptor antagonist which is widely used for the prophylaxis and chronic treatment of asthma and has been linked to rare cases of clinically apparent liver i...
T6893 MK-886 MK886,L 663536 Apoptosis , Leukotriene Receptor , COX , PPAR , FLAP
MK-886 (L 663536) is an inhibitor of leukotriene biosynthesis, inhibiting 5-lipoxygenase-activating protein (FLAP). It is also a moderately potent PPARα antagonist.
T0694 Pranlukast ONO-1078 Leukotriene Receptor , IL Receptor , Others , TNF , NF-κB , LTR
Pranlukast (ONO-1078) is a cysteinyl leukotriene receptor-1 antagonist. It antagonizes or reduces bronchospasm caused, principally in asthmatics, by an allergic reaction to accidentally or inadvertently encountered aller...
T6736 Zafirlukast Vanticon,ICI 204219,Accolate Leukotriene Receptor
Zafirlukast (ICI 204219) is an orally available leukotriene receptor antagonist which is widely used for the prophylaxis and chronic treatment of asthma.
T20615 Olsalazine Dipentium,Salicylic acid Others
Olsalazine (Dipentium), an anti-inflammatory drug, is used in the treatment of inflammatory bowel disease. It is also a novel DNA hypomethylating agent.
T22358 Etalocib LY293111,VML295 Apoptosis , Leukotriene Receptor , LTR
Etalocib (LY293111) is a novel diaryl ether carboxylic acid derivative, is a selective and potent inhibitor of the lipoxygenase pathway either via antagonism of the leukotriene B4 (LTB4) receptor or directly through 5'-l...
T3148 MK-571 sodium L-660711 (sodium salt),L-660711 sodium salt,Verlukast sodium,L-660711,MK571,MK-571 sodium salt,Propanoic acid Leukotriene Receptor , LTR
MK-571 sodium (L-660711 sodium salt) is a selective, orally active antagonist of the CysLT1 receptor. MK-571 sodium is a multidrug resistance protein-2 (ABCC2, Mrp2) inhibitor used to demonstrate the role of Mrp2 in the ...
T22787 FPL 55712 Others
Leukotriene receptor antagonist
T27979 Masilukast ICI-D-3523,ZD-3523,ICI D-3523,MCC-847,SA-09012,D-3523 Leukotriene Receptor
Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated with inflammation.
T15002 CP-105696 Pfizer 105696 LTR
CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.
T16395 ONO4057 ONO-LB457 Leukotriene Receptor
ONO4057 is a potent and orally active Leukotriene B4 receptor antagonist with an IC50 value of 0.7±0.3 μM. Immunosuppressive effect of ONO4057 on rat allografts.
T15647 Tipelukast MN 001,KCA 757 Leukotriene Receptor
Tipelukast (KCA 757) is a novel orally available leukotriene receptor antagonist with anti-inflammatory activity that reduces fibrosis and down-regulates TIMP-1, type 1 collagen.Tipelukast is used in the study of asthma.
T68130 Pobilukast SKF 104353 Z2,SKF 104353 Leukotriene Receptor
Pobilukast (SKF 104353) is a selective cysteinyl leukotriene receptor antagonist that blocks phosphatidylinositol metabolism and leukotriene D-induced thromboxane synthesis, and can be used to study limiting myocardial d...
T68119 Ontazolast BIRM-270 LTR
Ontazolast is a small molecule leukotriene B4 receptor (LTB4R) antagonist for the treatment of immune system disorders and respiratory diseases.Ontazolast is a candidate compound for the treatment of asthma.
T28974 Ticolubant Calcium Channel , LTR
Ticolubant is orally active leukotriene B4 antagonist with high affinity for the human neutrophil LTB4 receptor (Ki = 0.78 nM), blocks LTB4-induced Ca2+ migration with an IC50 of 6.6 ± 1.5 nM, and shows topical anti-inf...
T68108L Moxilubant HCl Moxilubant hcl(146978-48-5 Free base) LTR
Moxilubant HCl is a small molecule leukotriene B4 receptor 1 (LTB4R) antagonist for the treatment of immune system disorders, skin and musculoskeletal disorders, and may be used in studies of psoriasis and rheumatoid art...
T4657 WHI-P97 JAK
WHI-P97 is a rationally designed potent inhibitor of JAK-3. IC50 value: Target: JAK3 Treatment of mast cells with WHI-P97 inhibited the translocation of 5-lipoxygenase (5-LO) from the nucleoplasm to the nuclear membrane ...
T27916 LY 306669 LY-306669,LY306669
LY 306669 is an antagonist of leukotriene B4 receptor.
T28527 RG 14893
RG 14893 is a antagonist of high-affinity leukotriene B4 receptor.
T71043 MDL-43291
MDL-43291 is a leukotriene receptor antagonist.
T26809 BIIL 260 BIIL260,BIIL-260
BIIL 260 is a leukotriene B4 (BLT1) receptor antagonist with anti-inflammatory activity.
T22668 Cinalukast Others
CysLT1 leukotriene receptor antagonist
T30827 Cgp 33304 Cgp-33304,Cgp33304
CGP 33304 is a dual leukotriene receptor antagonist and phospholipase A2 inhibitor. It prevents hypoxia secondary to bronchial constriction induced by leukotriene in a shocking state.
T27912 LY 290324 LY-290324,LY290324
LY 290324 is an orally active, potent and selective antagonist of cysteinyl leukotriene (LTD4) receptor.
T11764 KP496 Others
KP496 is a selective, dual antagonist for Thromboxane A2 receptor and Leukotriene D4 receptor.
T24304 L 648051 4-Apsob,L48051,L-648051
L 648051 is a leukotriene D4 receptor antagonist.
T27896 LY 213024 LY-213024,LY213024
LY 213024 is an antagonist of leukotriene B4 receptor.
T27893 LY 203647 LY203647,LY-203647
LY 203647 is a antagonist of leukotriene D4 and E4 receptor.
T27913 LY 292728 LY292728,LY-292728
LY 292728 is a highly potent antagonist of leukotriene B4 receptor.
T69278 FPL-55712
FPL-55712 is a CysLT1 leukotriene receptor antagonist.
T28699 SC-41930 CGS 24115,SC41930,CGS24115
SC-41930 is a potent and selective antagonist of leukotriene B4 receptor.
T15801 LY210073 Others
LY210073 is an antagonist of the Leukotriene B4 (LTB4) receptor (IC50: 6.2 nM).
T73793 20-Carboxy-Leukotriene B4
20-Carboxy-Leukotriene B4 (20-COOH LTB4), a metabolite of Leukotriene B4 (LTB4), exhibits high affinity binding to the BLT1 receptor. It notably inhibits LTB4-mediated neutrophil responses, including migration, degranula...
T68831 Furodysinin
Furodysinin is an agonist of human leukotriene B4 receptor.
T70477 SC 53228
SC 53228 is a specific leukotriene B4 receptor antagonist.
T68418 Furodysinin lactone
Furodysinin lactone is an agonist of human leukotriene B4 receptor.
T10872 CP-96021 hydrochloride Others
CP-96021 hydrochloride is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor receptor (Kis: 34 nM and 37 nM).
T68348 Montelukast methylstyrene
Montelukast methylstyrene is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and to relieve symptoms of seasonal allergies.
T15803 LY223982 SKF107324,CGS23131 Others
LY223982 is an effective and specific inhibitor of the leukotriene B4 receptor (IC50: 13.2 nM). It also can against [3H]LTB4 binding to LTB4 receptor.
T27815 Leucettamol A Leucettamine A
Leucettamol A is a leukotriene B4 receptor antagonist isolated from the marine sponge Leucetta microraphis. It inhibits the formation of a complex composed of the ubiquitin E2 enzyme Ubc13 and Uev1A.
T10873 CP-96486 Others
CP-96486 is a potent and orally active antagonist of leukotriene D4 (LTD4)/platelet activating factor (PAF) receptor (Kis: 20 and 24 nM).
T21821 REV 5901
REV 5901 is a competitive and orally effective antagonist of leukotriene receptor, with a Ki of 0.7 μM. REV 5901 is also a 5-lipoxygenase inhibitor. REV 5901 can be used for the research of asthma in which leukotriene re...
T68496 Montelukast cyclopropaneacetamide
Montelukast cyclopropaneacetamide is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and to relieve symptoms of seasonal allergies.
T69501 Montelukast alcohol
Montelukast alcohol is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and to relieve symptoms of seasonal allergies.
T71369 Montelukast sulfoxide
Montelukast sulfoxide is a leukotriene receptor antagonist (LTRA) used for the maintenance treatment of asthma and to relieve symptoms of seasonal allergies.
T26958 CAY10583 CAY 10583,CAY-10583
CAY10583 is an agonist of leukotriene B4 receptor type 2 (BLT2). CAY10583 directly promotes keratinocyte migration and indirectly enhances fibroblast proliferation by increasing keratinocyte production of bFGF1 and TGF-β...

Compounds

Montelukast
T1677
Synonym: Singular
Target: Leukotriene Receptor, Lipoxygenase, LTR
Nedocromil
T16280
Synonym: FPL 59002
Target: Leukotriene Receptor, Prostaglandin Receptor, Histamine Receptor
Ablukast
T26519
Synonym: Ro 23-3544
Target: Leukotriene Receptor
LY255283
T22946
Synonym: LY 255283
Target: Leukotriene Receptor
Montelukast sodium
T1677L
Synonym: MK0476
Target: Leukotriene Receptor, LTR
MK-886
T6893
Synonym: MK886,L 663536
Target: Apoptosis, Leukotriene Receptor, COX, PPAR, FLAP
Pranlukast
T0694
Synonym: ONO-1078
Target: Leukotriene Receptor, IL Receptor, Others, TNF, NF-κB, LTR
Zafirlukast
T6736
Synonym: Vanticon,ICI 204219,Accolate
Target: Leukotriene Receptor
Olsalazine
T20615
Synonym: Dipentium,Salicylic acid
Target: Others
Etalocib
T22358
Synonym: LY293111,VML295
Target: Apoptosis, Leukotriene Receptor, LTR
MK-571 sodium
T3148
Synonym: L-660711 (sodium salt),L-660711 sodium salt,Verlukast sodium,L-660711,MK571,MK-571 sodium salt,Propanoic acid
Target: Leukotriene Receptor, LTR
FPL 55712
T22787
Synonym:
Target: Others
Masilukast
T27979
Synonym: ICI-D-3523,ZD-3523,ICI D-3523,MCC-847,SA-09012,D-3523
Target: Leukotriene Receptor
CP-105696
T15002
Synonym: Pfizer 105696
Target: LTR
ONO4057
T16395
Synonym: ONO-LB457
Target: Leukotriene Receptor
Tipelukast
T15647
Synonym: MN 001,KCA 757
Target: Leukotriene Receptor
Pobilukast
T68130
Synonym: SKF 104353 Z2,SKF 104353
Target: Leukotriene Receptor
Ontazolast
T68119
Synonym: BIRM-270
Target: LTR
Ticolubant
T28974
Synonym:
Target: Calcium Channel, LTR
Moxilubant HCl
T68108L
Synonym: Moxilubant hcl(146978-48-5 Free base)
Target: LTR
WHI-P97
T4657
Synonym:
Target: JAK
LY 306669
T27916
Synonym: LY-306669,LY306669
Target:
RG 14893
T28527
Synonym:
Target:
MDL-43291
T71043
Synonym:
Target:
BIIL 260
T26809
Synonym: BIIL260,BIIL-260
Target:
Cinalukast
T22668
Synonym:
Target: Others
Cgp 33304
T30827
Synonym: Cgp-33304,Cgp33304
Target:
LY 290324
T27912
Synonym: LY-290324,LY290324
Target:
KP496
T11764
Synonym:
Target: Others
L 648051
T24304
Synonym: 4-Apsob,L48051,L-648051
Target:
LY 213024
T27896
Synonym: LY-213024,LY213024
Target:
LY 203647
T27893
Synonym: LY203647,LY-203647
Target:
LY 292728
T27913
Synonym: LY292728,LY-292728
Target:
FPL-55712
T69278
Synonym:
Target:
SC-41930
T28699
Synonym: CGS 24115,SC41930,CGS24115
Target:
LY210073
T15801
Synonym:
Target: Others
20-Carboxy-Leukotriene B4
T73793
Synonym:
Target:
Furodysinin
T68831
Synonym:
Target:
SC 53228
T70477
Synonym:
Target:
Furodysinin lactone
T68418
Synonym:
Target:
CP-96021 hydrochloride
T10872
Synonym:
Target: Others
Montelukast methylstyrene
T68348
Synonym:
Target:
LY223982
T15803
Synonym: SKF107324,CGS23131
Target: Others
Leucettamol A
T27815
Synonym: Leucettamine A
Target:
CP-96486
T10873
Synonym:
Target: Others
REV 5901
T21821
Synonym:
Target:
Montelukast cyclopropaneacetamide
T68496
Synonym:
Target:
Montelukast alcohol
T69501
Synonym:
Target:
Montelukast sulfoxide
T71369
Synonym:
Target:
CAY10583
T26958
Synonym: CAY 10583,CAY-10583
Target:
1 2
Cat No. Product Name Synonyms Targets
T7786 Tryptanthrin DNA gyrase
Tryptanthrin is a natural DNA gyrase inhibitor.
T5714 5-O-Demethylnobiletin 5-DEMETHYLNOBILETIN Leukotriene Receptor , Lipoxygenase
5-O-Demethylnobiletin (5-DEMETHYLNOBILETIN) is a natual product, has anti-inflammatory activity, it may act through a direct inhibition of 5-LOX, without affecting the expression of COX-2.
TN1182 11-​Keto-​beta-​boswellic acid 11-Keto-beta-boswellic acid Leukotriene Receptor , NF-κB , Lipoxygenase
11-Keto-beta-boswellic acid, a novel Nrf2 activator, and a selective 5-lipoxygenase (5-LOX) inhibitor; it exerts dose dependent cardioprotective effect manifested by dose-dependent reduction in serum lactate dehydrogenas...
T21504 γ-Linolenic Acid methyl ester Methyl gamma-linolenate LTR
γ-Linolenic Acid methyl ester (Methyl gamma-linolenate) is a weak leukotriene B4 (LTB4) receptor antagonist.
T4973 Paraxanthine 1,7-DIMETHYLXANTHINE Endogenous Metabolite
Paraxanthine (1,7-dimethylxanthine) is a metabolite of caffeine (sc-202514) which functions as an adenosine receptor ligand and a PARP-1 inhibitor in pulmonary epithelial cells. Studies suggest that Paraxanthine is struc...
T37972 12-OxoETE
12-OxoETE is synthesized by human platelets and Aplysia nervous tissue after incubation with arachidonic acid. Microsomal fractions of various tissues will reduce 12-oxoETE to 12(S)-HETE or a mixture of 12(S)- and 12(R)-...

Natural Products

Tryptanthrin
T7786
Synonym:
Target: DNA gyrase
5-O-Demethylnobiletin
T5714
Synonym: 5-DEMETHYLNOBILETIN
Target: Leukotriene Receptor, Lipoxygenase
11-​Keto-​beta-​boswellic acid
TN1182
Synonym: 11-Keto-beta-boswellic acid
Target: Leukotriene Receptor, NF-κB, Lipoxygenase
γ-Linolenic Acid methyl ester
T21504
Synonym: Methyl gamma-linolenate
Target: LTR
Paraxanthine
T4973
Synonym: 1,7-DIMETHYLXANTHINE
Target: Endogenous Metabolite
12-OxoETE
T37972
Synonym:
Target:

Recombinant Proteins

Species：
Human (2)
Mouse (1)
Expression System：
E. coli (2)
in vitro E. coli expression system (1)
Tag：
His (2)
N-terminal 10xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPH-03749 CYSLTR1 Protein, Human, Recombinant (His) Human in vitro E. coli expression system
Receptor for cysteinyl leukotrienes mediating bronchoconstriction of individuals with and without asthma. Stimulation by LTD4 results in the contraction and proliferation of smooth muscle, edema, eosinophil migration and...
TMPY-06837 PPAR alpha/PPARA Protein, Mouse, Recombinant (His) Mouse E. coli
Peroxisome proliferators include hypolipidemic drugs, herbicides, leukotriene antagonists, and plasticizers; this term arises because they induce an increase in the size and number of peroxisomes. Peroxisomes are subcell...
TMPY-06830 PPAR alpha/PPARA Protein, Human, Recombinant (His) Human E. coli
Peroxisome proliferators include hypolipidemic drugs, herbicides, leukotriene antagonists, and plasticizers; this term arises because they induce an increase in the size and number of peroxisomes. Peroxisomes are subcell...
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