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Search Result

Search Results for " melatonin-receptor "

24

Compounds

2

Natural Products

1

Libraries

Cat No. Product Name Synonyms Targets
T60490 Melatonin receptor agonist 1
Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].
T14042 4-P-PDOT 4-phenyl-2- propionamidotetralin Melatonin Receptor , MT Receptor
4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.
T9193 ACH-000143 Melatonin Receptor , MT Receptor
ACH-000143 have been identified as a novel agonist of the melatonin receptors MT1 and MT2.
T8600 N-ACETYLTRYPTAMINE Melatonin Receptor
N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.
T1445 Agomelatine Thymanax,S-20098,Valdoxan Melatonin Receptor , 5-HT Receptor
Agomelatine (Valdoxan) is structurally closely related to melatonin. Agomelatine is a potent agonist at melatonin receptors and an antagonist at serotonin-2C (5-HT2C) receptors, tested in an animal model of depression.
T1463 Ramelteon TAK-375 Melatonin Receptor , MT Receptor
Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.
T15795 Luzindole N-0774 Melatonin Receptor , MT Receptor
Luzindole (N-0774) is a selective melatonin receptor antagonist. Luzindole inhibits experimental autoimmune encephalomyelitis and exerts antidepressant-like activity. Luzindole preferentially targets MT2 (Mel1b) over MT1...
T3495 Tasimelteon VEC-162,BMS-214778 Melatonin Receptor , MT Receptor
Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.
T16834 S26131 N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide MT Receptor
S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of 0.5 and 112 nM respectively.
T22530 6-Chloromelatonin Melatonin Receptor , Dopamine Receptor
6-Chloromelatonin is a potent melatonin receptor agonist, a 5-methoxyindole compound that competes for the same presynaptic melatonin receptor sites in the rabbit retina and inhibits the calcium-dependent release of [3H]...
T10929L D-3263 hydrochloride EC D-3263 HCl,D3263 HCl salt TRP/TRPV Channel
D-3263 hydrochloride (D3263 HCl salt) is enteric-coated, orally bioavailable transient receptor potential melatonin member 8 (TRPM8) agonist.
T10073 2-Iodomelatonin Melatonin Receptor
2-Iodomelatonin is a potent agonist of melatonin receptor 1 (MT1) with a Ki value of 28 pM, it is more 5-fold selective for MT1 over MT2. 2-iodomelatonin can be used to identify, characterize and localize melatonin bind...
T10198 8-M-PDOT 8-Methoxy-2-propionamidotetralin,AH-002 MT Receptor
8-M-PDOT (AH-002) is a selective and potent melatonin MT2 receptor agonist that also inhibits MT1 receptors.8-M-PDOT has anxiolytic activity and may be used to study MT2-induced neuropathic pain.
T28644 S20928 S 20928,S-20928
S20928 is an antagonist of melatonin receptor.
T28645 S-22153
S22153 is an antagonist of melatonin receptor.
T29044 UCM 765 UCM-765,UCM765
UCM 765 is a partial agonist of melatonin MT(2) receptor.
T69409 DH-97
DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).
T22721 DH97 DH 97 Others
MT2 melatonin receptor antagonist
T27430 GR 196429 GR-196429,GR 196,429,GR-196,429,GR196429,GR196,429
GR 196429, a melatonin receptor agonist, exhibits selectivity for the MT1 subtype. This compound not only promotes sleep and alters circadian rhythms but also stimulates melatonin release in mice.
T27429 GR 128107 GR128107,GR-128107
GR 128107 is an antagonist of melatonin receptor.
T10929 D-3263 Others
D-3263 is an agonist of transient receptor potential melatonin member 8 (TRPM8) with potential antitumor activity.
T17095 TIK-301 PD-6735,LY-156735 5-HT Receptor
TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM, respectively). TIK-301 is also a 5-HT2B/5-HT2C receptor an...
T71963 (−)-WIN 55,212-3 mesylate
(−)-WIN 55,212-3 mesylate is an aminoalkylindole derivative which acts as a competitive neutral antagonist of the human cannabinoid CB2 receptor, blocking both the stimulating action of CP 55,940 and the inverse agonism ...
T70035 Tasimelteon-d5
Tasimelteon-d5 is intended for use as an internal standard for the quantification of tasimelteon by GC- or LC-MS. Tasimelteon is a melatonin (MT) receptor agonist. It selectively binds MT1 and MT2 receptors over a panel ...

Compounds

Melatonin receptor agonist 1
T60490
Synonym:
Target:
4-P-PDOT
T14042
Synonym: 4-phenyl-2- propionamidotetralin
Target: Melatonin Receptor, MT Receptor
ACH-000143
T9193
Synonym:
Target: Melatonin Receptor, MT Receptor
N-ACETYLTRYPTAMINE
T8600
Synonym:
Target: Melatonin Receptor
Agomelatine
T1445
Synonym: Thymanax,S-20098,Valdoxan
Target: Melatonin Receptor, 5-HT Receptor
Ramelteon
T1463
Synonym: TAK-375
Target: Melatonin Receptor, MT Receptor
Luzindole
T15795
Synonym: N-0774
Target: Melatonin Receptor, MT Receptor
Tasimelteon
T3495
Synonym: VEC-162,BMS-214778
Target: Melatonin Receptor, MT Receptor
S26131
T16834
Synonym: N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide
Target: MT Receptor
6-Chloromelatonin
T22530
Synonym:
Target: Melatonin Receptor, Dopamine Receptor
D-3263 hydrochloride
T10929L
Synonym: EC D-3263 HCl,D3263 HCl salt
Target: TRP/TRPV Channel
2-Iodomelatonin
T10073
Synonym:
Target: Melatonin Receptor
8-M-PDOT
T10198
Synonym: 8-Methoxy-2-propionamidotetralin,AH-002
Target: MT Receptor
S20928
T28644
Synonym: S 20928,S-20928
Target:
S-22153
T28645
Synonym:
Target:
UCM 765
T29044
Synonym: UCM-765,UCM765
Target:
DH-97
T69409
Synonym:
Target:
DH97
T22721
Synonym: DH 97
Target: Others
GR 196429
T27430
Synonym: GR-196429,GR 196,429,GR-196,429,GR196429,GR196,429
Target:
GR 128107
T27429
Synonym: GR128107,GR-128107
Target:
D-3263
T10929
Synonym:
Target: Others
TIK-301
T17095
Synonym: PD-6735,LY-156735
Target: 5-HT Receptor
(−)-WIN 55,212-3 mesylate
T71963
Synonym:
Target:
Tasimelteon-d5
T70035
Synonym:
Target:
Cat No. Product Name Synonyms Targets
T1659 Melatonin Melatonine,N-Acetyl-5-methoxytryptamine CaMK , Apoptosis , Mitophagy , Estrogen/progestogen Receptor , Melatonin Receptor , Glutathione Peroxidase , Endogenous Metabolite , ROR , Autophagy
Melatonin (Melatonine) is a biogenic amine that is found in animals and plants. In mammals, melatonin is produced by the PINEAL GLAND. Its secretion increases in darkness and decreases during exposure to light. Melatonin...
T1354 N-Acetyl-5-hydroxytryptamine Normelatonin,O-Demethylmelatonin,N-Acetylserotonin Trk receptor , Endogenous Metabolite
N-Acetyl-5-hydroxytryptamine (O-Demethylmelatonin) , also known as Normelatonin, is the immediate precursor of melatonin. It is produced from serotonin by the enzyme aralkylamine N-acetyltransferase and is converted to m...

Natural Products

Melatonin
T1659
Synonym: Melatonine,N-Acetyl-5-methoxytryptamine
Target: CaMK, Apoptosis, Mitophagy, Estrogen/progestogen Receptor, Melatonin Receptor, Glutathione Peroxidase, Endogenous Metabolite, ROR, Autophagy
N-Acetyl-5-hydroxytryptamine
T1354
Synonym: Normelatonin,O-Demethylmelatonin,N-Acetylserotonin
Target: Trk receptor, Endogenous Metabolite
Cat No. Product Name
L3300 Histamine & Melatonin Receptor-Targeted Compound Library

155 compounds
A unique collection of 155 compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCS) for new drugs;

Libraries

Histamine & Melatonin Receptor-Targeted Compound Library
L3300
Compounds: 155
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