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Search Result

Search Results for " neurokinin receptor "

Targets

Neurokinin receptor Neurokinin receptor

90

Compounds

1

Natural Products

1

Recombinant Proteins

Cat No. Product Name Synonyms Targets
TP1008 Neurokinin A α-Neurokinin,Substance K,Neuromedin L Neurokinin receptor
Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.
TP1087 Substance P Neurokinin P Endogenous Metabolite , Neurokinin receptor
Substance P (Neurokinin P) (SP) is an undecapeptide (a peptide composed of a chain of 11 amino acid residues) member of the tachykinin neuropeptide family.
T7633 Senktide Neurokinin receptor
Senktide is an agonist of tachykinin NK3 receptor.
T23316 SB 218795 Neurokinin receptor
SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.
T16849 SB-222200 Neurokinin receptor
SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).
TP1086 Men 10376 TFA(135306-85-3,free) Men 10376 TFA,Neurokinin-2 receptor antagonist TFA Neurokinin receptor
Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4 M for the nk-2 receptor in the small intestine of rats.
T7209 Maropitant Neurokinin receptor
Maropitant is a selective neurokinin (NK1) receptor antagonist.
TP1572 GR-73632 Neurokinin receptor
Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).
T38144 Elinzanetant Neurokinin receptor
Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.
T15278 Fezolinetant ESN-364 Neurokinin receptor
Fezolinetant (ESN-364) is an antagonist of the neurokinin 3 receptor (NK3R). It is used for the treatment of menopausal hot flushes.
T7549 Talnetant SB 223412 Neurokinin receptor
Talnetant (SB 223412) is a selective, competitive, brain-penetrant NK3 receptor antagonist with the ability to modulate mesolimbic and mesocortical dopaminergic neurotransmission
T76429 Neurokinin Receptor (393-407), rat
Neurokinin Receptor (393-407), rat (SPR393–407), a fragment of the rat neurokinin 1 receptor (NK1R), undergoes rapid endocytosis and subsequent recycling to the plasma membrane upon substance P (SP) binding. This compoun...
T8235 L-732138 Neurokinin receptor
L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)
TP1883 [Lys5,MeLeu9,Nle10]-NKA(4-10) Neurokinin receptor
Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
T17156 Tradipitant VLY-686,LY686017 Neurokinin receptor
Tradipitant (VLY-686) is an antagonist of neurokinin-1.
T7554 Substance P (7-11) Substance P 7-11(TFA) Others , Neurokinin receptor
Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .
T16038 Men 10376 Neurokinin-2 receptor antagonist CDK
Men 10376 is a selective antagonist of tachykinin NK-2 receptor. It has a Ki of 4.4 μM for rat small intestine NK-2 receptor.
T6905 Netupitant Ro 67-31898/000,CID 6451149 Neurokinin receptor
Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).
T3716 Rolapitant SCH619734 Neurokinin receptor
Rolapitant (SCH619734) Hydrochloride is the hydrochloride salt form of rolapitant, an orally bioavailable, centrally-acting, selective, neurokinin 1 receptor (NK1-receptor) antagonist with potential antiemetic activity. ...
T7559 Neurokinin A(4-10) Neurokinin A(4-10)(TFA) Neurokinin receptor
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
T1743 Aprepitant MK-869,MK-0869,L-754030,Aprepitant` HIV Protease , Antibacterial , Antibiotic , Neurokinin receptor
Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist. The mechanism of action of aprepitant is as a Neurokinin 1 Antagonist, and Cytochrome P450 3A4 Inhibitor, and Cytochrome P450 2C9 Inducer, and C...
T13306L Vapreotide acetate RC-160 acetate,BMY-41606 acetate Neurokinin receptor
Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).
T1790 Fosaprepitant dimeglumine L785298,MK-0517,Fosaprepitant dimeglumine salt Neurokinin receptor
Fosaprepitant dimeglumine (MK-0517) is the dimeglumine salt form of fosaprepitant, the water-soluble, N-phosphorylated prodrug of aprepitant, with antiemetic activity. Upon intravenous administration and rapid conversion...
T3034 Eprazinone dihydrochloride Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl Others , Neurokinin receptor
Eprazinone dihydrochloride (NSC 317935) is a mucolytic with antitussive and mucolytic effect.
T7828 [Sar9,Met(O2)11]-Substance P Bhsar-sp,NA Neurokinin receptor
[Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
T7396 Substance P(1-7) Substance P 1-7 Others , Neurokinin receptor
Substance P(1-7) (Substance P 1-7) is the major bioactive metabolite formed after proteolytic degradation of the tachykinin substance P (SP),with anti-inflammatory, anti-nociceptive and anti-hyperalgesic effects
T7631 Eledoisin Related Peptide Eledoisin RP,Eledoisin-Related Peptide,Eledoisin Related Peptide(2TFA) Neurokinin receptor
Eledoisin Related Peptide (Eledoisin RP) is a tachykinin receptor ligand.
T29157 WIN 51,708 WIN51,708,WIN-51,708
WIN 51,708 is an antagonist of neurokinin-1 receptor.
TP1363L Neurokinin B acetate(86933-75-7 free base) Neurokinin K Neurokinin receptor
Neurokinin B acetate(86933-75-7 free base) is the acetate form of Neurokinin B, which belongs to the tachykinin family. Neurokinin binds to neurokinin receptor 1 (NK1R), nk2r and NK3R, and mediates its biological effects...
TP1385 Neurokinin A(4-10) TFA(97559-35-8 free base) Neurokinin A(4-10) TFA Neurokinin receptor
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].
T68068 Ezlopitant CJ 11974,CJ-11974,CJ11974 Neurokinin receptor
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.
T69140 Burapitant SSR 240600 Neurokinin receptor
Burapitant (SSR 240600) is a novel non-peptide tachykinin neurokinin 1 (NK) receptor antagonist with anti-coke oven and antidepressant activity.
T68068L (R)-CJ 11974 Neurokinin receptor
(R)-CJ 11974 is a novel non-peptide neurokinin NK1 substance P receptor antagonist with potential analgesic activity that can be used to study chemotherapy-induced vomiting.
TP1851L Scyliorhinin II acetate Neurokinin receptor
Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.
T19518L Physalaemin acetate Neurokinin receptor
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.
T25616 Lanepitant 2HCl LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride Neurokinin receptor
Lanepitant 2HCl is a non-peptide neurokinin-1 receptor antagonist with analgesic and anti-inflammatory activity.Lanepitant 2HCl inhibits the binding of Substance P to the neurokinin-1 receptor, inhibits neurogenic inflam...
T16114 Pavinetant AZD4901,MLE-4901,AZD2624 MEK
Pavinetant is a small molecule orally active and selective neurokinin-3 (NK3) receptor antagonist for the treatment of hot flashes and polycystic ovarian syndrome (PCOS), which is a potential compound for the treatment o...
T3724 Rolapitant hydrochloride Rolapitant HCl Neurokinin receptor
Rolapitant (SCH619734) hydrochloride is a potent, selective, long-acting and orally active neurokinin 1 (NK1) receptor antagonist with a K i of 0.66 nM. Rolapitant hydrochloride (Rolapitant HCl) does not interact with CY...
T9417L Gamma-preprotachykinin amide (72-92) acetate gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base) Others
gamma-preprotachykinin amide (72-92) acetate is a 21 amino acid peptide belonging to the tachykinin (TK) family and including neurokinin A (NKA) in its C-terminal sequence. gamma-preprotachykinin amide (72-92) acetate po...
T68556 GW679769
GW679769 is a neurokinin-1 receptor antagonist.
T20148 L 659,877 L 659877,L-659,877,L-659877,L659,877,L659877
L 659,877 is an antagonist of the Tachykinin and neurokinin-2 receptor.
T70587 CJ-12255
CJ-12255 is a Neurokinin-1 Receptor Antagonist.
T76427 (D-Pro2,D-Trp6,8,Nle10)-Neurokinin B
(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B functions as a competitive antagonist to the Neurokinin B receptor, exhibiting a pA2 value of 5.5. Notably, it does not affect Substance P or Neurokinin A [1].
T29210 ZD6021 ZD-6021,ZD 6021
ZD6021 is an antagonist of neurokinin 1 receptor.
T69295 DNK 333
DNK 333 is a dual neurokinin NK1/NK2 receptor antagonist.
T26169 S 16474 S16474,S-16474
S 16474 is an antagonist of Neurokinin-1 Receptor.
T34799 Telmapitant
Telmapitant is an antagonist of the neurokinin NK1 receptor.
T16406 Orvepitant maleate GW823296 maleate Neurokinin receptor
Orvepitant maleate is an effective, selective, and well-tolerated neurokinin-1 receptor (NK-1) antagonist (pKi: 10.2 for human neurokinin-1 receptor). Orvepitant maleate has the potential for depressive disorder and chro...
T27175 Dilopetine Citrate E-6006 Citrate,E-6039,E6039,E 6039
Dilopetine Citrate, a tachykinin receptor modulator and a neurokinin receptor modulator, is used potentially for the treatment of depression.
T24357 L 741671 L741671,L 741,671,L741,671,L-741,671,L-741671
L 741671 is an antagonist of the neurokinin-1 receptor.

Compounds

Neurokinin A
TP1008
Synonym: α-Neurokinin,Substance K,Neuromedin L
Target: Neurokinin receptor
Substance P
TP1087
Synonym: Neurokinin P
Target: Endogenous Metabolite, Neurokinin receptor
Senktide
T7633
Synonym:
Target: Neurokinin receptor
SB 218795
T23316
Synonym:
Target: Neurokinin receptor
SB-222200
T16849
Synonym:
Target: Neurokinin receptor
Men 10376 TFA(135306-85-3,free)
TP1086
Synonym: Men 10376 TFA,Neurokinin-2 receptor antagonist TFA
Target: Neurokinin receptor
Maropitant
T7209
Synonym:
Target: Neurokinin receptor
GR-73632
TP1572
Synonym:
Target: Neurokinin receptor
Elinzanetant
T38144
Synonym:
Target: Neurokinin receptor
Fezolinetant
T15278
Synonym: ESN-364
Target: Neurokinin receptor
Talnetant
T7549
Synonym: SB 223412
Target: Neurokinin receptor
Neurokinin Receptor (393-407), rat
T76429
Synonym:
Target:
L-732138
T8235
Synonym:
Target: Neurokinin receptor
[Lys5,MeLeu9,Nle10]-NKA(4-10)
TP1883
Synonym:
Target: Neurokinin receptor
Tradipitant
T17156
Synonym: VLY-686,LY686017
Target: Neurokinin receptor
Substance P (7-11)
T7554
Synonym: Substance P 7-11(TFA)
Target: Others, Neurokinin receptor
Men 10376
T16038
Synonym: Neurokinin-2 receptor antagonist
Target: CDK
Netupitant
T6905
Synonym: Ro 67-31898/000,CID 6451149
Target: Neurokinin receptor
Rolapitant
T3716
Synonym: SCH619734
Target: Neurokinin receptor
Neurokinin A(4-10)
T7559
Synonym: Neurokinin A(4-10)(TFA)
Target: Neurokinin receptor
Aprepitant
T1743
Synonym: MK-869,MK-0869,L-754030,Aprepitant`
Target: HIV Protease, Antibacterial, Antibiotic, Neurokinin receptor
Vapreotide acetate
T13306L
Synonym: RC-160 acetate,BMY-41606 acetate
Target: Neurokinin receptor
Fosaprepitant dimeglumine
T1790
Synonym: L785298,MK-0517,Fosaprepitant dimeglumine salt
Target: Neurokinin receptor
Eprazinone dihydrochloride
T3034
Synonym: Resplen,Mucitux,Eftapan,NSC 317935,Eprazinone 2HCl
Target: Others, Neurokinin receptor
[Sar9,Met(O2)11]-Substance P
T7828
Synonym: Bhsar-sp,NA
Target: Neurokinin receptor
Substance P(1-7)
T7396
Synonym: Substance P 1-7
Target: Others, Neurokinin receptor
Eledoisin Related Peptide
T7631
Synonym: Eledoisin RP,Eledoisin-Related Peptide,Eledoisin Related Peptide(2TFA)
Target: Neurokinin receptor
WIN 51,708
T29157
Synonym: WIN51,708,WIN-51,708
Target:
Neurokinin B acetate(86933-75-7 free base)
TP1363L
Synonym: Neurokinin K
Target: Neurokinin receptor
Neurokinin A(4-10) TFA(97559-35-8 free base)
TP1385
Synonym: Neurokinin A(4-10) TFA
Target: Neurokinin receptor
Ezlopitant
T68068
Synonym: CJ 11974,CJ-11974,CJ11974
Target: Neurokinin receptor
Burapitant
T69140
Synonym: SSR 240600
Target: Neurokinin receptor
(R)-CJ 11974
T68068L
Synonym:
Target: Neurokinin receptor
Scyliorhinin II acetate
TP1851L
Synonym:
Target: Neurokinin receptor
Physalaemin acetate
T19518L
Synonym:
Target: Neurokinin receptor
Lanepitant 2HCl
T25616
Synonym: LY303870 dihydrochloride,LY 303870 dihydrochloride,LY-303870 dihydrochloride,Lanepitant dihydrochloride
Target: Neurokinin receptor
Pavinetant
T16114
Synonym: AZD4901,MLE-4901,AZD2624
Target: MEK
Rolapitant hydrochloride
T3724
Synonym: Rolapitant HCl
Target: Neurokinin receptor
gamma-preprotachykinin amide (72-92) acetate
T9417L
Synonym: gamma-preprotachykinin amide (72-92) acetate (114882-65-4 Free base)
Target: Others
GW679769
T68556
Synonym:
Target:
L 659,877
T20148
Synonym: L 659877,L-659,877,L-659877,L659,877,L659877
Target:
CJ-12255
T70587
Synonym:
Target:
(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B
T76427
Synonym:
Target:
ZD6021
T29210
Synonym: ZD-6021,ZD 6021
Target:
DNK 333
T69295
Synonym:
Target:
S 16474
T26169
Synonym: S16474,S-16474
Target:
Telmapitant
T34799
Synonym:
Target:
Orvepitant maleate
T16406
Synonym: GW823296 maleate
Target: Neurokinin receptor
Dilopetine Citrate
T27175
Synonym: E-6006 Citrate,E-6039,E6039,E 6039
Target:
L 741671
T24357
Synonym: L741671,L 741,671,L741,671,L-741,671,L-741671
Target:
1 2
Cat No. Product Name Synonyms Targets
T8789 N-Acetyl-L-tryptophan N-acetyltryptophan Endogenous Metabolite , Neurokinin receptor
N-Acetyl-L-tryptophan (N-acetyltryptophan) is an inhibitor of neurokinin 1 receptor (NK1-receptor, NK1R).

Natural Products

N-Acetyl-L-tryptophan
T8789
Synonym: N-acetyltryptophan
Target: Endogenous Metabolite, Neurokinin receptor

Recombinant Proteins

Species：
Human (1)
Expression System：
E. coli (1)
Tag：
N-6His (1)
Cat No. Product Name Species Expression System
TMPJ-01379 TAC3 Protein, Human, Recombinant (His) Human E. coli
Tachykinin 3 (TAC3) is a secreted protein that belongs to the Tachykinin family. Tachykinins are active peptides that excite neurons and evoke behavioral responses; they are potent vasodilators and secretagogues, and con...
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