T20166L |
Deltorphin acetate
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98.93%
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Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioid receptor...
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T4411 |
DAMGO TFA (78123-71-4(Free base))
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T4411
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98.67%
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Potent, selective agonist of Mu-opioid receptor. Antinociceptive. Stimulates calcium-activated adenylyl cyclases related cAMP production. Expresses chemokines an...
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TP1793 |
Nociceptin (1-13), amide
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178064-02-3
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100%
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Nociceptin (1-13), amide is a potent ORL1 (OP4) receptor agonist with a pEC50 of 7.9 for mouse vas deferens and a Ki of 0.75 nM for binding to rat forebrain memb...
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T7567 |
Adrenorphin
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88377-68-8
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Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
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T4633 |
Asimadoline
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153205-46-0
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Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany. Asimadoline was originally develo...
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T7404 |
Dermorphin
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77614-16-5
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Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
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T11479 |
GSK1521498
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1426543-84-1
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98%
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GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive consumption of food, alcohol, ...
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T11478 |
GSK1521498 free base (hydrochloride)
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1007578-24-6
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98%
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GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR). It is being used for the treatment of disorders of compulsive cons...
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T79060 |
MOR agonist-1
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2305781-14-8
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98%
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MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated disorders...
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T79430 |
μ opioid receptor agonist 3
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2378397-91-0
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98%
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Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM. It holds promise for research into pain m...
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T79431 |
Mu opioid receptor antagonist 7
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2378397-30-7
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98%
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Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (IC...
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T79547 |
MOR agonist-2
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98%
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Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM. This compound holds pote...
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T79848 |
Icalcaprant
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2227384-17-8
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98%
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Icalcaprant is a kappa-opioid receptor antagonist [1].
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T80086 |
DALDA TFA
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98%
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DALDA TFA is a potent, μ-opioid receptor agonist exhibiting high selectivity and an affinity constant (K i) of 1.69 nM. It demonstrates antinociceptive propertie...
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T80421 |
CSD-CH2(1,8)-NH2
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98%
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CSD-CH2(1,8)-NH2 is a selective and competitive kappa-opioid receptor (KOR) antagonist with a K i of 6.8 nM. It inhibits calcium mobilization in dorsal root gang...
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T80463 |
Dynorphin B (1-9)
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126050-26-8
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98%
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Dynorphin B (1-9), a neuropeptide and the N-terminal cleavage product of dynorphin B, has its formation inhibited by N-ethylmaleimide (NEM), a non-selective cyst...
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T80515 |
β-Endorphin (1-27) (human)
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76622-84-9
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98%
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β-Endorphin (1-27) (human) is an opioid antagonist that selectively binds to μ-, δ-, and κ-opioid receptors, with dissociation constants (Kis) of 5.31, 6.17, and...
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T81938 |
Leumorphin, human
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88846-98-4
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98%
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Leumorphin, human, is a potent agonist of the kappa opioid receptor (κ opioid receptor) and inhibits the contraction of the guinea pig ileum's myenteric plexus-l...
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TP1367L |
[D-Ala2]leucine-enkephalin acetate
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TP1367L
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98%
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[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study the signaling pathway of d...
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TN5017 |
Sideritoflavone
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70360-12-2
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98%
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Sideritoflavone has anti-inflammatory effect, it is a selective inhibitor of lipoxygenase activity in vitro.
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