TP2036 |
DPDPE
|
88373-73-3
|
98%
|
|
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
|
T76285 |
β-Endorphin (6-31), human
|
77761-27-4
|
98%
|
|
β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors. Produced by specific neurons within...
|
TN3368 |
Akuammigine
|
642-17-1
|
98%
|
|
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
|
T7306 |
Valorphin
|
144313-54-2
|
98%
|
|
Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
|
T12169 |
Naltrindole hydrochloride
|
111469-81-9
|
98%
|
|
Naltrindole hydrochloride is a selective and non-peptide δ opioid receptor antagonist(Ki = 0.02 nM).
|
TN3367 |
Akuammidine
|
639-36-1
|
98%
|
|
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
|
T13438 |
(R,S)-Ivosidenib
|
2070009-31-1
|
98%
|
|
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
|
T12314 |
Opioid receptor modulator 1
|
77514-44-4
|
98%
|
|
Opioid receptor modulator 1 is a modulator of opioid receptor.
|
T15165 |
DPI-3290
|
182417-73-8
|
98%
|
|
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
|
T27934 |
LY255582
|
119193-09-8
|
98%
|
|
LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM, respecti...
|
T11478L |
GSK1521498 free base
|
1007573-18-3
|
98%
|
|
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
|
T11198 |
Endomorphin 2 TFA
|
1276124-00-5
|
98%
|
|
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
|
T1242 |
Alvimopan
|
156053-89-3
|
99.97%
|
|
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvim...
|
TP1813L |
Dynorphin A 1-10 acetate(79994-24-4 free base)
|
TP1813L
|
99.93%
|
|
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-acti...
|
TP2322L |
Beta-Neoendorphin acetate(77739-21-0 free base)
|
78658-39-6
|
99.91%
|
|
beta-Neoendorphin acetate is an agonist of κ-opioid receptor
|
TP1082L |
Neuropeptide AF (human) acetate
|
|
99.89%
|
|
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative, w...
|
T2726 |
Sinomenine
|
115-53-7
|
99.89%
|
|
Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
|
T21422 |
Methylnaltrexone bromide
|
73232-52-7
|
99.88%
|
|
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the s...
|
T2071 |
MCOPPB triHydrochloride
|
1108147-88-1
|
99.88%
|
|
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
|
T5S2360 |
Corydaline
|
518-69-4
|
99.86%
|
|
1. Corydaline (Corydalin), an isoquinoline alkaloid, is one of the major active constituents in a new prokinetic botanical agent. 2. Corydaline promotes gastric ...
|