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Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TP2036 DPDPE 88373-73-3 98%
DPDPE
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
T76285 β-Endorphin (6-31), human 77761-27-4 98%
β-Endorphin (6-31), human
β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors. Produced by specific neurons within...
TN3368 Akuammigine 642-17-1 98%
Akuammigine
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
T7306 Valorphin 144313-54-2 98%
Valorphin
Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
T12169 Naltrindole hydrochloride 111469-81-9 98%
Naltrindole hydrochloride
Naltrindole hydrochloride is a selective and non-peptide δ opioid receptor antagonist(Ki = 0.02 nM).
TN3367 Akuammidine 639-36-1 98%
Akuammidine
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
T13438 (R,S)-Ivosidenib 2070009-31-1 98%
(R,S)-Ivosidenib
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
T12314 Opioid receptor modulator 1 77514-44-4 98%
Opioid receptor modulator 1
Opioid receptor modulator 1 is a modulator of opioid receptor.
T15165 DPI-3290 182417-73-8 98%
DPI-3290
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
T27934 LY255582 119193-09-8 98%
LY255582
LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM, respecti...
T11478L GSK1521498 free base 1007573-18-3 98%
GSK1521498 free base
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
T11198 Endomorphin 2 TFA 1276124-00-5 98%
Endomorphin 2 TFA
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
T1242 Alvimopan 156053-89-3 99.97%
Alvimopan
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvim...
TP1813L Dynorphin A 1-10 acetate(79994-24-4 free base) TP1813L 99.93%
Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-acti...
TP2322L Beta-Neoendorphin acetate(77739-21-0 free base) 78658-39-6 99.91%
beta-Neoendorphin acetate(77739-21-0 free base)
beta-Neoendorphin acetate is an agonist of κ-opioid receptor
TP1082L Neuropeptide AF (human) acetate 99.89%
Neuropeptide AF (human) acetate
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative, w...
T2726 Sinomenine 115-53-7 99.89%
Sinomenine
Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
T21422 Methylnaltrexone bromide 73232-52-7 99.88%
Methylnaltrexone bromide
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the s...
T2071 MCOPPB triHydrochloride 1108147-88-1 99.88%
MCOPPB triHydrochloride
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
T5S2360 Corydaline 518-69-4 99.86%
Corydaline
1. Corydaline (Corydalin), an isoquinoline alkaloid, is one of the major active constituents in a new prokinetic botanical agent. 2. Corydaline promotes gastric ...
DPDPE
TP2036
DPDPE is selective δ-opioid receptor agonist peptide. Inhibits electrically stimulated contraction of mouse vas deferens in vitro (EC50 = 5.2 nM), and is antinoc...
β-Endorphin (6-31), human
T76285
β-Endorphin is an endogenous opioid neuropeptide and opioid receptor agonist that preferentially binds to μ-opioid receptors. Produced by specific neurons within...
Akuammigine
TN3368
Akuammigine has in vitro antimalarial activity. Akuammigine competitively antagonizes the effect of noradrenaline on postsynaptic alpha-adrenoceptors, yielding p...
Valorphin
T7306
Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
Naltrindole hydrochloride
T12169
Naltrindole hydrochloride is a selective and non-peptide δ opioid receptor antagonist(Ki = 0.02 nM).
Akuammidine
TN3367
Akuammidine shows anti-inflammatory and anti-asthmatic properties, it has opioid analgesic activity, it shows a preference for mu-opioid binding sites with Ki va...
(R,S)-Ivosidenib
T13438
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
Opioid receptor modulator 1
T12314
Opioid receptor modulator 1 is a modulator of opioid receptor.
DPI-3290
T15165
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent antinocicepti...
LY255582
T27934
LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM, respecti...
GSK1521498 free base
T11478L
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor. GSK1521498 free base also has the potential for disorders of compulsive consu...
Endomorphin 2 TFA
T11198
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the...
Alvimopan
T1242
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvim...
Dynorphin A 1-10 acetate(79994-24-4 free base)
TP1813L
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor. Dynorphin A (1-10) also blocks NMDA-acti...
beta-Neoendorphin acetate(77739-21-0 free base)
TP2322L
beta-Neoendorphin acetate is an agonist of κ-opioid receptor
Neuropeptide AF (human) acetate
TP1082L
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative, w...
Sinomenine
T2726
Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
Methylnaltrexone bromide
T21422
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists. Methylnaltrexone bromide acts to reverse some of the s...
MCOPPB triHydrochloride
T2071
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
Corydaline
T5S2360
1. Corydaline (Corydalin), an isoquinoline alkaloid, is one of the major active constituents in a new prokinetic botanical agent. 2. Corydaline promotes gastric ...
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TargetMol