Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.

Cat. No.	Product name	CAS No.	Purity
TP1211L	BAM 22P acetate	TP1211L	99.87%
TP1211L	BAM 22P acetate is a potent opioid agonist.
T7173	[Leu5]-Enkephalin	58822-25-6	99.87%
T7173	[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4.0 and 3.4 nM,...
T5S2360	Corydaline	518-69-4	99.86%
T5S2360	1. Corydaline (Corydalin), an isoquinoline alkaloid, is one of the major active constituents in a new prokinetic botanical agent. 2. Corydaline promotes gastric ...
T5167	Cebranopadol	863513-91-1	99.86%
T5167	Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP) an...
T25354L	DuP 747 HCl	115904-74-0	99.81%
T25354L	DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.
TP1254	[Met5]-Enkephalin, amide TFA	TP1254	99.81%
TP1254	[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.
T2921	Sinomenine hydrochloride	6080-33-7	99.79%
T2921	Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.
T0209	Loperamide hydrochloride	34552-83-5	99.78%
T0209	Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.
T0929	Docusate sodium	577-11-7	99.77%
T0929	Docusate sodium (Aerosol OT) is an orally available, over-the-counter laxative and stool softener used to treat or prevent constipation. Docusate has not been li...
T1197	Trimebutine maleate	34140-59-5	99.76%
T1197	Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects. Trimebutine is an agonist of peripheral mu, delta, and kappa opiate r...
T4407	SR17018	2134602-45-0	99.73%
T4407	SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.
TP1826L	Dynorphin B (1-13) acetate(83335-41-5 free base)	TP1826L	99.72%
TP1826L	Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.
T6175	ADL-5859	850173-95-4	99.71%
T6175	ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the ...
TP2040L	Dynorphin A acetate(80448-90-4 free base)	TP2040L	99.69%
TP2040L	Dynorphin A acetate is an Endogenous kappa receptor agonist.
T4236	AR-M 1000390 hydrochloride	209808-47-9	99.68%
T4236	AR-M 1000390 hydrochloride (ARM-390 HCl) , also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. D...
TP1404L	Hemorphin-7 acetate(152685-85-3 free base)	TP1404L	99.66%
TP1404L	Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin. Hemorphin peptides exhibits antinociceptive and ...
T0783	Mianserin hydrochloride	21535-47-7	99.63%
T0783	Mianserin hydrochloride (Org GB 94) is a tetracyclic compound with antidepressant effects. it apparently blocks alpha-adrenergic, histamine H1, and some types of...
T7665	[Leu5]-Enkephalin TFA(58822-25-6(free bas))	73563-78-7	99.63%
T7665	[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago
TP2050L	CTAP(TFA） (103429-32-9 free base)	TP2050L	99.62%
TP2050L	CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM. It displays over 12...
T67888L	Samidorphan HCl	2328045-02-7	99.60%
T67888L	Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors. Samidorphan HC...