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Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
TP1071 Nociceptin 170713-75-4 99.35%
Nociceptin
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.
T0137 Mirtazapine 85650-52-8 99.3%
Mirtazapine
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
T31081L CP 866087 519052-02-9 99.28%
CP 866087
CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
T7173L [Leu5]-Enkephalin acetate(58822-25-6 free base) T7173L 99.28%
[Leu5]-Enkephalin acetate(58822-25-6 free base)
[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4....
T6553 JTC-801 244218-51-7 99.27%
JTC-801
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.
T28453L Propiram fumarate HCl 945013-73-0 99.25%
Propiram fumarate HCl
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
T3417 Amentoflavone 1617-53-4 99.22%
Amentoflavone
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
T8991 BMS986187 684238-37-7 99.19%
BMS986187
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
T22810 GR 89696 fumarate 126766-32-3 99.19%
GR 89696 fumarate
GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.
TP1179L Porcine dynorphin A(1-13) acetate TP1179L 99.14%
Porcine dynorphin A(1-13) acetate
Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiol...
T31750 Faxeladol 433265-65-7 99.11%
Faxeladol
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
T23335 SCH 221510 322473-89-2 99.10%
SCH 221510
SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used t...
T23306 Salvinorin A 83729-01-5 99.06%
Salvinorin A
Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
T21757 BRL 52537 hydrochloride 112282-24-3 99.04%
BRL 52537 hydrochloride
BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury[1]. It is used for res...
T1407 (-)-Menthol 2216-51-5 99.01%
(-)-Menthol
(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local a...
T4691 Asimadoline hydrochloride 185951-07-9 98.94%
Asimadoline hydrochloride
Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also ...
T23076L Nociceptin (1-7) acetate T23076L 98.92%
Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor. Nociceptin (1-7) combines with nociceptin reduces hyperalgesia and has a...
T39988 6'-GNTI dihydrochloride 2410327-94-3 98.91%
6'-GNTI dihydrochloride
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
T4351 DAMGO 78123-71-4 98.83%
DAMGO
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents. Possible analgesic agent due to μ-opiod receptor intera...
T22870 IPAG 193527-91-2 98.8%
IPAG
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
Nociceptin
TP1071
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.
Mirtazapine
T0137
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
CP 866087
T31081L
CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
[Leu5]-Enkephalin acetate(58822-25-6 free base)
T7173L
[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4....
JTC-801
T6553
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.
Propiram fumarate HCl
T28453L
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
Amentoflavone
T3417
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
BMS986187
T8991
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
GR 89696 fumarate
T22810
GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.
Porcine dynorphin A(1-13) acetate
TP1179L
Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiol...
Faxeladol
T31750
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
SCH 221510
T23335
SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used t...
Salvinorin A
T23306
Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
BRL 52537 hydrochloride
T21757
BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury[1]. It is used for res...
(-)-Menthol
T1407
(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local a...
Asimadoline hydrochloride
T4691
Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also ...
Nociceptin (1-7) acetate
T23076L
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor. Nociceptin (1-7) combines with nociceptin reduces hyperalgesia and has a...
6'-GNTI dihydrochloride
T39988
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
DAMGO
T4351
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents. Possible analgesic agent due to μ-opiod receptor intera...
IPAG
T22870
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
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TargetMol