TP1071 |
Nociceptin
|
170713-75-4
|
99.35%
|
|
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.
|
T0137 |
Mirtazapine
|
85650-52-8
|
99.3%
|
|
Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy can be associated with transient asy...
|
T31081L |
CP 866087
|
519052-02-9
|
99.28%
|
|
CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.
|
T7173L |
[Leu5]-Enkephalin acetate(58822-25-6 free base)
|
T7173L
|
99.28%
|
|
[Leu5]-Enkephalin acetate(58822-25-6 free base) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and μ-opioid receptors (Kis = 4....
|
T6553 |
JTC-801
|
244218-51-7
|
99.27%
|
|
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.
|
T28453L |
Propiram fumarate HCl
|
945013-73-0
|
99.25%
|
|
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
|
T3417 |
Amentoflavone
|
1617-53-4
|
99.22%
|
|
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
|
T8991 |
BMS986187
|
684238-37-7
|
99.19%
|
|
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
|
T22810 |
GR 89696 fumarate
|
126766-32-3
|
99.19%
|
|
GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.
|
TP1179L |
Porcine dynorphin A(1-13) acetate
|
TP1179L
|
99.14%
|
|
Porcine dynorphin A(1-13) acetate (Dynorphin A Porcine Fragment 1-13 acetate) is a potent, endogenous κ opioid receptor agonist and is antinociceptive at physiol...
|
T31750 |
Faxeladol
|
433265-65-7
|
99.11%
|
|
Faxeladol, a potent adrenergic absorption inhibitor and serotonin reuptake inhibitor, is a small-molecule Opioid receptor agonist that can be used to study neuro...
|
T23335 |
SCH 221510
|
322473-89-2
|
99.10%
|
|
SCH 221510 is an orally available, selective and potent NOP agonist with an EC50 of 12 nM and a Ki of 0.3 nM.SCH 221510 has anxiolytic activity and can be used t...
|
T23306 |
Salvinorin A
|
83729-01-5
|
99.06%
|
|
Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
|
T21757 |
BRL 52537 hydrochloride
|
112282-24-3
|
99.04%
|
|
BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury[1]. It is used for res...
|
T1407 |
(-)-Menthol
|
2216-51-5
|
99.01%
|
|
(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local a...
|
T4691 |
Asimadoline hydrochloride
|
185951-07-9
|
98.94%
|
|
Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also ...
|
T23076L |
Nociceptin (1-7) acetate
|
T23076L
|
98.92%
|
|
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor. Nociceptin (1-7) combines with nociceptin reduces hyperalgesia and has a...
|
T39988 |
6'-GNTI dihydrochloride
|
2410327-94-3
|
98.91%
|
|
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
|
T4351 |
DAMGO
|
78123-71-4
|
98.83%
|
|
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents. Possible analgesic agent due to μ-opiod receptor intera...
|
T22870 |
IPAG
|
193527-91-2
|
98.8%
|
|
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
|