T23306 |
Salvinorin A
|
83729-01-5
|
99.06%
|
|
Salvinorin A is a non-nitrogenous κ-opioid selective agonist.
|
T76341L |
[DPro10] Dynorphin A (1-11)acetate,porcine
|
|
99.05%
|
|
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-...
|
T21757 |
BRL 52537 hydrochloride
|
112282-24-3
|
99.04%
|
|
BRL 52537 hydrochloride is a selective and specific KOR agonist which has been implicated in neuroprotection from ischemic neuronal injury[1]. It is used for res...
|
T1407 |
(-)-Menthol
|
2216-51-5
|
99.01%
|
|
(-)-Menthol (Levomenthol) is a levo isomer of menthol, an organic compound made synthetically or obtained from peppermint or mint oils with flavoring and local a...
|
T21660L |
B-Casomorphin (1-3) Acetate
|
T21660L
|
98.99%
|
|
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.
|
T4691 |
Asimadoline hydrochloride
|
185951-07-9
|
98.94%
|
|
Asimadoline hydrochloride (EMD-61753 hydrochloride) is a κ-opioid receptor agonist potentially for the treatment of pruritus. Asimadoline hydrochloride has also ...
|
T23076L |
Nociceptin (1-7) acetate
|
T23076L
|
98.92%
|
|
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor. Nociceptin (1-7) combines with nociceptin reduces hyperalgesia and has a...
|
T39988 |
6'-GNTI dihydrochloride
|
2410327-94-3
|
98.91%
|
|
6'-GNTI dihydrochloride is a κ-opioid receptor (KOR) agonist that favors activation of G-protein-mediated signaling over recruitment of β-aspirin 2. 6'-GNTI dihy...
|
T0963 |
Naltrexone hydrochloride
|
16676-29-2
|
98.9%
|
|
Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.
|
T4351 |
DAMGO
|
78123-71-4
|
98.83%
|
|
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents. Possible analgesic agent due to μ-opiod receptor intera...
|
T22870 |
IPAG
|
193527-91-2
|
98.8%
|
|
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
|
T20435L |
Leuphasyl TFA
|
67586-27-0
|
98.79%
|
|
Leuphasyl TFA is an amid peptide, a δ-opioid receptor agonist, is a degradation resistant long-acting Leu-enkephalin analog used to study the signaling pathway o...
|
T8992 |
BMS986188
|
1776115-10-6
|
98.76%
|
|
BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.
|
T23074 |
NNC 63-0532
|
250685-44-0
|
98.75%
|
|
NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.
|
T4411 |
DAMGO TFA (78123-71-4(Free base))
|
T4411
|
98.67%
|
|
Potent, selective agonist of Mu-opioid receptor. Antinociceptive. Stimulates calcium-activated adenylyl cyclases related cAMP production. Expresses chemokines an...
|
T8414 |
SNC 80
|
156727-74-1
|
98.67%
|
|
SNC 80 (NIH 10815) is a potent, highly selective and non-peptide δ-opioid receptor agonist, Ki = 1.78 nM, IC50 = 2.73 nM. SNC80 also selectively activates μ-δ he...
|
T23002 |
ML-335
|
1069498-96-9
|
98.52%
|
|
ML-335 is a μ-δ isomer-targeted agonist, a μOR-δOR-biased ligand that can serve as a scaffold for the development of unique types of (isomer-biased) drugs.ML-335...
|
T5158 |
N-Desmethylclozapine
|
6104-71-8
|
98.45%
|
|
N-Desmethylclozapine (Desmethylclozapine) is an antagonist of serotonin (5-HT) receptor subtype 5-HT2C (IC50: 7.1 nM). It also is an antagonist at dopamine D4 re...
|
T14835 |
BTRX-335140
|
2244614-14-8
|
98.45%
|
|
BTRX-335140 (CYM-53093) is a potent and selective, orally active κ opioid receptor (KOR) antagonist, has antagonist activity for κOR, μOR and δOR with IC50 value...
|
T26869 |
BMS-986122
|
313669-88-4
|
98.42%
|
|
BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 ...
|