Home Tools
Log in
Cart

Opioid Receptor

Opioid receptors belong to the large superfamily of seven transmembrane-spanning (7TM) G protein-coupled receptors (GPCRs). As a class, GPCRs are of fundamental physiological importance mediating the actions of the majority of known neurotransmitters and hormones.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T38193L β-Endorphin (1-27) (human) acetate 96.52%
β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity. β-Endorphin (1-27) (human) acetate is...
TP2105L UFP-101 acetate TP2105L 95.92%
UFP-101 acetate
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
TQ0267 Endomorphin 1 189388-22-5 95.92%
Endomorphin 1
Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).
TP1882L1 Orphanin FQ(1-11) acetate(178249-41-7 free base) TP1882L1 95.54%
Orphanin FQ(1-11) acetate(178249-41-7 free base)
Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, in...
T22752L (D-Ser2)-Leu-Enkephalin-Thr T22752L 94.17%
(D-Ser2)-Leu-Enkephalin-Thr
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.
T8455 Spinorphin 137201-62-8 100%
Spinorphin
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
T39529 AT-121 hydrochloride 2099681-71-5 100%
AT-121 hydrochloride
AT-121 hydrochloride is a dual agonist of nociception and mu opioid receptor with Ki values of 3.67 and 16.49 nM, respectively.AT-121 hydrochloride is a safe, no...
T31081 CP-866087 519052-04-1 100%
CP-866087
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.
T7567L Adrenorphin 3TFA(88377-68-8(free base)) T7567L 100%
Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
TP1905 BW-180C 63631-40-3 100%
BW-180C
BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.
T7639 Deltorphin 2 122752-16-3 100%
Deltorphin 2
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.
T8557 N-terminally acetylated Leu-enkephalin T8557 100%
N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous peptide consisting of five amino acids, functions as an agonist at opioid receptors. The N-terminally acetylated form of this compo...
T7748 Dermorphin TFA 78331-26-7 100%
Dermorphin TFA
Dermorphin TFA is a new class of opioids-like peptides
T7637 Deltorphin I 122752-15-2 100%
Deltorphin I
Deltorphin I is an agonist of δ-opioid receptor.
T7665 [Leu5]-Enkephalin TFA(58822-25-6(free bas)) 73563-78-7
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago
T39284 EST73502 HCl 2307458-82-6 98%
EST73502 HCl
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
T76341L [DPro10] Dynorphin A (1-11)acetate,porcine 98%
[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-...
T25354L DuP 747 HCl 115904-74-0 98%
DuP 747 HCl
DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.
T3417 Amentoflavone 1617-53-4 98%
Amentoflavone
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
TQ0082 Aticaprant 1174130-61-0 98%
Aticaprant
Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).
β-Endorphin (1-27) (human) acetate
T38193L
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity. β-Endorphin (1-27) (human) acetate is...
UFP-101 acetate
TP2105L
UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
Endomorphin 1
TQ0267
Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).
Orphanin FQ(1-11) acetate(178249-41-7 free base)
TP1882L1
Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, in...
(D-Ser2)-Leu-Enkephalin-Thr
T22752L
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.
Spinorphin
T8455
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
AT-121 hydrochloride
T39529
AT-121 hydrochloride is a dual agonist of nociception and mu opioid receptor with Ki values of 3.67 and 16.49 nM, respectively.AT-121 hydrochloride is a safe, no...
CP-866087
T31081
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.
Adrenorphin 3TFA(88377-68-8(free base))
T7567L
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
BW-180C
TP1905
BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.
Deltorphin 2
T7639
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.
N-terminally acetylated Leu-enkephalin
T8557
Leu-enkephalin, an endogenous peptide consisting of five amino acids, functions as an agonist at opioid receptors. The N-terminally acetylated form of this compo...
Dermorphin TFA
T7748
Dermorphin TFA is a new class of opioids-like peptides
Deltorphin I
T7637
Deltorphin I is an agonist of δ-opioid receptor.
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
T7665
[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago
EST73502 HCl
T39284
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
[DPro10] Dynorphin A (1-11)acetate,porcine
T76341L
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-...
DuP 747 HCl
T25354L
DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.
Amentoflavone
T3417
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
Aticaprant
TQ0082
Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).
1 2 3 4 5 6 7
TargetMol