T38193L |
β-Endorphin (1-27) (human) acetate
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96.52%
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β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity. β-Endorphin (1-27) (human) acetate is...
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TP2105L |
UFP-101 acetate
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TP2105L
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95.92%
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UFP-101 acetate is a selective and competitive antagonist of the NOP receptor (pKi = 10.24) with >3000-fold selectivity over δ, μ, and κ opioid receptors.
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TQ0267 |
Endomorphin 1
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189388-22-5
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95.92%
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Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).
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TP1882L1 |
Orphanin FQ(1-11) acetate(178249-41-7 free base)
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TP1882L1
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95.54%
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Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, in...
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T22752L |
(D-Ser2)-Leu-Enkephalin-Thr
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T22752L
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94.17%
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(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.
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T8455 |
Spinorphin
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137201-62-8
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100%
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Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
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T39529 |
AT-121 hydrochloride
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2099681-71-5
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100%
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AT-121 hydrochloride is a dual agonist of nociception and mu opioid receptor with Ki values of 3.67 and 16.49 nM, respectively.AT-121 hydrochloride is a safe, no...
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T31081 |
CP-866087
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519052-04-1
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100%
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CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.
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T7567L |
Adrenorphin 3TFA(88377-68-8(free base))
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T7567L
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100%
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Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
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TP1905 |
BW-180C
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63631-40-3
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100%
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BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.
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T7639 |
Deltorphin 2
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122752-16-3
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100%
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Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.
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T8557 |
N-terminally acetylated Leu-enkephalin
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T8557
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100%
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Leu-enkephalin, an endogenous peptide consisting of five amino acids, functions as an agonist at opioid receptors. The N-terminally acetylated form of this compo...
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T7748 |
Dermorphin TFA
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78331-26-7
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100%
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Dermorphin TFA is a new class of opioids-like peptides
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T7637 |
Deltorphin I
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122752-15-2
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100%
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Deltorphin I is an agonist of δ-opioid receptor.
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T7665 |
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
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73563-78-7
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[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago
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T39284 |
EST73502 HCl
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2307458-82-6
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98%
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EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.
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T76341L |
[DPro10] Dynorphin A (1-11)acetate,porcine
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98%
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[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-...
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T25354L |
DuP 747 HCl
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115904-74-0
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98%
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DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two conformations.
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T3417 |
Amentoflavone
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1617-53-4
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98%
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Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications. CYP3A4 and CYP2C9 are proteins used for ...
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TQ0082 |
Aticaprant
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1174130-61-0
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98%
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Aticaprant (LY-2456302) (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).
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