T1893 |
ML 161 |
ML 161 is the inhibitor of protease-activated receptor 1 (PAR1)-mediated platelet activation (IC50: 0.26 μM for the inhibition of platelet P-selectin expressio...
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T1986L |
Atopaxar Hydrobromide |
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arte...
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T3098 |
Vorapaxar sulfate |
Vorapaxar sulfate is a potent and orally active thrombin receptor (PAR-1) antagonist. |
T4186 |
AC264613 |
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pr...
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T7013 |
Vorapaxar |
Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM). |
T7137 |
I-191 |
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells. |
T7496 |
Thrombin Receptor Activator for Peptide |
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of co...
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T7380 |
Protease-Activated Receptor-4 |
Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy |
T7674 |
Thrombin Receptor Activator for Peptide |
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of co...
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TQ0012 |
AZ3451 |
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM). |
T7573 |
TFLLR-NH2(2TFA) |
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM). |
T7623 |
PAR-4 Agonist Peptide, amide |
PAR-4 Agonist Peptide, amide is an agonist of proteinase-activated receptor-4 (PAR-4). |
T7625 |
TRAP-6(2TFA) |
TRAP-6(2TFA) is an agonist of protease-activated receptor 1 (PAR1). |
T7740 |
Protease-Activated Receptor-4 diTFA(245443-52-1(free base)) |
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonist |
T7573L |
TFLLR-NH2 2TFA(197794-83-5(free base)) |
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM). |
T7513 |
Protease-Activated Receptor-2, amide |
Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M) |
TP1925L |
tcY-NH2 TFA(327177-34-4 free base) |
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin. |
TP1904L |
FSLLRY-NH2 TFA(245329-02-6 free base) |
FSLLRY-NH2 TFA is a is a protease-activated receptor 2 (PAR2) inhibitor. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in I...
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TP1378 |
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) |
2-Furoyl-LIGRLO-amide is a potent and selective protease-activated receptor 2 (PAR2) agonist. |
TP1046L |
PAR-2 Activating Peptide acetate(171436-38-7 free base) |
PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2). |
TP1046L |
PAR-2 Activating Peptide acetate(171436-38-7 free base) |
PAR-2 Activating Peptide acetate is an agonist of Protease-Activated Receptor-2 (PAR-2). |
TP1065 |
PAR-4 Agonist Peptide, amide TFA |
PAR-4 Agonist Peptide, amide TFA is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocke...
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