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Search Result

Search Results for " retinoid-receptor "

Targets

Retinoid Receptor

26

Compounds

1

Natural Products

5

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T3955 AR7 Retinoid Receptor
AR7 is a retinoic acid receptor α (RARα) antagonist.
T7894 Tazarotenic acid AGN-190299 Others
Tazarotenic acid (AGN-190299) is a retinoid prodrug which is converted to its active form
T14912 CD3254 Retinoid Receptor
CD3254 is a selective and potent retinoid X receptor-like (RXR) agonist that inhibits neuronal cell death with OGD/reoxygenation.
T9635 Cedirogant ABBV-157 ROR
Cedirogant (ABBV-157) is an orally active retinoid-related orphan receptor-γt(RORγt) inverse agonist that is used for psoriasis study.
T23383 SR11237 SR 11237 Others , RAR/RXR 
SR11237 is a Pan retinoid X receptor (RXR) agonist. SR11237 causes RXR/RXR homodimers to form and transactivate a reporter gene containing a RXR-response element.
T7388 GSK805 ROR
GSK805 is a potent, orally bioavailable retinoid-related orphan receptor gamma t (RORγt) inverse agonist that interacts with the receptor's putative ligand binding domain without exerting significant effects on DNA bindi...
T11844 LG-100064 Retinoid Receptor , Autophagy
LG-100064 is an agonist of retinoid-X-receptor (RXR)(EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ and RXRγ)
T17209 UVI 3003 Retinoid Receptor , Autophagy
UVI 3003 is a highly selective antagonist of the retinoid X receptor. UVI 3003 inhibits Xenopus and human RXRα in Cos7 cells (IC50s: 0.22 and 0.24 μM, respectively).
T22843 HX 531 Retinoid Receptor
RXR antagonist
T11303 Fluorobexarotene Retinoid Receptor
Fluorobexarotene possesses an apparent RXR binding affinity that is 75% greater than Bexarotene. Fluorobexarotene  is a potent retinoid-X-receptor (RXR) agonist, with a Ki value of 12 nM and an EC50 value of 43 nM for RX...
TP1313L Cecropin B acetate Cecropin B acetate(80451-05-4 Free base) P450 , Retinoid Receptor , Parasite
Cecropin B acetate induces NF-κB activation and suppresses CYP3A29 by disrupting the association of the PXR/retinoid X receptor alpha (RXR-α) complex with DNA sequences. Cecropin B acetate exhibits strong antimicrobial a...
T77499 MSU-42011 NOS , Retinoid Receptor , NO Synthase , PERK , Lipid
MSU-42011 is an orally active retinoid X receptor-like (RXR) agonist.MSU-42011 potently inhibits the expression of iNOS, low SREBP-induced and activated RXR, and p-ERK at the protein level.MSU-42011 has demonstrated anti...
T25472 GW0791 GW 0791,GW-0791
GW0791 is a retinoid X receptor α (RXRα) agonist.
T23665 AGN 191701 AGN-191701,AGN191701
AGN 191701 is an agonist of the Retinoid X receptor.
T29720 Agn 190727 Agn-190727,Agn190727
Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.
T70440 AGN-191659
AGN-191659 is a Retinoid X Receptor (RXR) pan-agonist. RXR pan-agonists have been shown to modulate endothelial cell proliferation.
T69695 Izumerogant
Izumerogant is an inverse agonist of the retinoid-related orphan receptor-gamma (RORγ).
T10246 Adapalene sodium salt CD 271 sodium salt Others
Adapalene (CD 271; Differin) sodium salt is a synthetic retinoid and a Retinoic acid receptor agonist.
T24857 TBTC
TBTC is a selective agonist of retinoid X receptor α that acts by improving behavioral deficit in Alzheimer's disease model mice.
T24727 ROR Modulator I ROR-Modulator-I,RORModulatorI
ROR Modulator I is the first potent inverse agonist of the retinoid-related orphan receptor. It also has dual selectivity for RORβ and RORγt.
T70976 AGN-190121
AGN-190121 is a retinoic acid receptor (RAR) agonist. RAR and Retinoid X Receptor (RXR) ligands can act synergistically to induce hypertriglyceridemia through distinct mechanisms of action.
T19703 LG100268 LG 100268,LG-100268
LG100268 is an effective and selective rexinoid and retinoid-X receptor agonist. LG100268 binds to the α, β, and γ RXR receptors (IC50 = 3-4 nM).
T63415 RXR antagonist 1
RXR antagonist 1 is a Retinoid X Receptor (RXR) modulator that exhibits high RXR antagonism (pA2: 8.06). RXR antagonist 1 can be used to study type 2 diabetes.
T69921 BRF110
BRF110 is a brain penetrant, potent and selective agonist of nuclear receptor-related 1 (Nurr1):Retinoid X receptor α (RXRα) heterodimer. BRF110 is a neuroprotective agent that prevents dopaminergic neuron demise and str...
T37414 CAY10771
CAY10771 is a dual agonist of farnesoid X receptor (FXR) and peroxisome proliferator-activated receptor δ (PPARδ).1It activates FXR and PPARδ in reporter assays using HEK293T cells (EC50s = 0.94 and 1.5 μM, respectively)...
T35800 MD001
MD001 is a dual agonist of peroxisome proliferator-activated receptor α (PPARα) and PPARγ.1 It binds to PPARα and PPARγ (Kds = 9.55 and 0.14 μM, respectively) but does not bind to PPARβ/δ at concentrations up to 500 μM. ...
Cat No. Product Name Synonyms Targets
TN6735 Bigelovin Apoptosis , Reactive Oxygen Species , Retinoid Receptor , Autophagy , RAR/RXR 
Bigelovin is a selective retinoid X receptor α agonist. Bigelovin suppresses tumor growth through inducing apoptosis and autophagy via the inhibition of mTOR pathway regulated by ROS generation.It is also known as a pote...

Natural Products

Bigelovin
TN6735
Synonym:
Target: Apoptosis, Reactive Oxygen Species, Retinoid Receptor, Autophagy, RAR/RXR 

Recombinant Proteins

Species：
Human (3)
Cynomolgus (1)
Mouse (1)
Expression System：
Baculovirus-Insect Cells (2)
HEK293 (2)
E. coli (1)
Tag：
His (4)
N-terminal 10xHis-tagged and C-terminal Myc-tagged (1)
Cat No. Product Name Species Expression System
TMPY-00835 IGFBP-3 Protein, Human, Recombinant (His) Human HEK293
The Insulin-like Growth Factor (IGF) signaling system plays a central role in cellular growth, differentiation, and proliferation. IGFBP3 is the most abundant IGF binding protein in human serum and is a growth inhibitory...
TMPY-03251 IGFBP-3 Protein, Cynomolgus, Recombinant (His) Cynomolgus HEK293
The Insulin-like Growth Factor (IGF) signaling system plays a central role in cellular growth, differentiation, and proliferation. IGFBP3 is the most abundant IGF binding protein in human serum and is a growth inhibitory...
TMPY-02987 Vitamin D Receptor/VDR Protein, Mouse, Recombinant (His) Mouse Baculovirus-Insect Cells
VDR (vitamin D (1,25- dihydroxyvitamin D3) receptor), also known as NR1I1, belongs to the NR1I family, NR1 subfamily. It is composed of three domains: a modulating N-terminal domain, a DNA-binding domain and a C-terminal...
TMPY-02706 Vitamin D Receptor/VDR Protein, Human, Recombinant (His) Human Baculovirus-Insect Cells
VDR (vitamin D (1,25- dihydroxyvitamin D3) receptor), also known as NR1I1, belongs to the NR1I family, NR1 subfamily. It is composed of three domains: a modulating N-terminal domain, a DNA-binding domain and a C-terminal...
TMPH-01819 LXR-alpha Protein, Human, Recombinant (His & Myc) Human E. coli
Nuclear receptor that exhibits a ligand-dependent transcriptional activation activity. Interaction with retinoic acid receptor (RXR) shifts RXR from its role as a silent DNA-binding partner to an active ligand-binding su...
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