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GPCR/G Protein Vasopressin Receptor

Vasopressin Receptor

The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into the V1 (V1A), V2, and V3 (V1B) receptor subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.
Cat No. product name
T2326 Tolvaptan Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
T2568 Felypressin Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activi...
T6288 Mozavaptan Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T6453 Conivaptan hydrochloride Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
T4355 OPC 21268 OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
T4141 RO 5028442 RO5028442 has been used in trials studying Autistic Disorder.
T5019 Desmopressin Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin ...
T5144 Desmopressin acetate Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led...
T7303 Lixivaptan Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
Tolvaptan
T2326CAS 150683-30-0
Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
Felypressin
T2568CAS 56-59-7
Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activi...
Mozavaptan
T6288CAS 137975-06-5
Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
Conivaptan hydrochloride
T6453CAS 168626-94-6
Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
OPC 21268
T4355CAS 131631-89-5
OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
RO 5028442
T4141CAS 920022-47-5
RO5028442 has been used in trials studying Autistic Disorder.
Desmopressin
T5019CAS 16679-58-6
Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin ...
Desmopressin acetate
T5144CAS 62288-83-9
Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led...
Lixivaptan
T7303CAS 168079-32-1
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)