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Home > Chromatin/Epigenetic > JAK > AZD1480
AZD1480  
Catalog No. T3069    CAS 935666-88-9
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5mg
9 days
43.00
10mg
9 days
68.00
50mg
9 days
170.00
100mg
9 days
306.00
200mg
9 days
553.00
1g
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0.00
5g
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0.00
10mM * 1mL (in DMSO)
9 days
47.00
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Documents and Quality Management
Purity:97.50% COA Datasheet HPLC MSDS
Biological Activity:

Product Description:

AZD1480 is a novel ATP-competitive JAK2 inhibitor with IC50 of 0.26 nM in a cell-free assay, selectivity against JAK3 and Tyk2, and to a smaller extent against JAK1. Phase 1.

Target:
JAK2;
Research Area:
Cancer
Chemical Information:
Molecular Weight 348.77
Formula C14H14ClFN8
CAS Number 935666-88-9
Solubility DMSO: 69mg/ml(197.84 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
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Reference

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