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Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Preclinical Compound Library

Catalog No. L3410
  Library Compound List   Excel SDF

Preclinical Compound Library is a collection of 709 compounds that are in preclinical phase with clear targets and detailed information on disease indication and reference.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
Get quote

Product Description

  • A unique collection of 709 preclinical compounds for high throughput screening (HTS) and high content screening (HCS);
  • Hot lead compounds for new drug discovery and development;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L3410)

Library Composition

Apoptosis (130)
Autophagy (113)
Endogenous Metabolite (37)
Antibacterial (36)
Antibiotic (34)
VEGFR (24)
CDK (23)
PDGFR (20)
PI3K (19)
DNA/RNA Synthesis (18)
HIV Protease (18)
FGFR (18)
Influenza Virus (17)
NF-κB (17)
EGFR (17)
Adrenergic Receptor (15)
JAK (14)
FLT (13)
Epigenetic Reader Domain (12)
Histamine Receptor (12)
Src (12)
c-Kit (12)
5-HT Receptor (12)
Microtubule Associated (12)
Parasite (12)
mTOR (12)
Dopamine Receptor (12)
Sodium Channel (11)
Calcium Channel (11)
HDAC (11)
c-RET (10)
Ferroptosis (10)
PDE (10)
BCL (10)
Phosphatase (10)
AChR (9)
Reactive Oxygen Species (9)
Adenosine Receptor (9)
Raf (9)
ATM/ATR (9)
PPAR (9)
Potassium Channel (9)
HSP (9)
E1/E2/E3 Enzyme (9)
MEK (9)
Bcr-Abl (9)
Mitophagy (9)
SARS-CoV (8)
PKC (8)
COX (8)
c-Met/HGFR (8)
GluR (8)
PLK (8)
iGluR (8)
Aurora Kinase (8)
p53 (8)
ALK (8)
DNA-PK (8)
GSK-3 (7)
ROS (7)
p38 MAPK (7)
NMDAR (7)
STAT (7)
Antifungal (7)
Akt (7)
Dehydrogenase (7)
DNA Alkylator/Crosslinker (7)
Trk receptor (7)
Mdm2 (6)
Casein Kinase (6)
Beta Amyloid (6)
IGF-1R (6)
Topoisomerase (6)
Ras (6)
Proteasome (6)
P450 (6)
Opioid Receptor (6)
Histone Methyltransferase (6)
FXR (5)
Chk (5)
TGF-beta/Smad (5)
GABA Receptor (5)
Cannabinoid Receptor (5)
PDK (5)
TAM Receptor (5)
AMPK (5)
S6 Kinase (5)
Tyrosine Kinases (5)
Sigma receptor (5)
Lipoxygenase (5)
Reverse Transcriptase (5)
PKA (4)
TNF (4)
PARP (4)
Pim (4)
TRP/TRPV Channel (4)
Hydroxylase (4)
BTK (4)
LPL Receptor (4)
Wnt/beta-catenin (4)
IL Receptor (4)
Retinoid Receptor (4)
FAK (4)
Gamma-secretase (4)
Serine Protease (4)
Sirtuin (4)
Estrogen/progestogen Receptor (4)
HBV (4)
ERK (4)
Endothelin Receptor (4)
RAAS (4)
LPA Receptor (3)
Estrogen Receptor/ERR (3)
MAPK (3)
ROCK (3)
MELK (3)
Serine/threonin kinase (3)
Aminopeptidase (3)
Mitochondrial Metabolism (3)
HER (3)
MMP (3)
Cysteine Protease (3)
DUB (3)
MRP (3)
Virus Protease (3)
NADPH (3)
Nucleoside Antimetabolite/Analog (3)
Nrf2 (3)
Norepinephrine (3)
Hedgehog/Smoothened (3)
Glucokinase (3)
HCV Protease (3)
Proton pump (3)
TLR (3)
CRM1 (3)
Glucocorticoid Receptor (3)
Smo (3)
Complement System (3)
Integrin (3)
Prostaglandin Receptor (3)
Interleukin (3)
HIF (3)
ATPase (3)
Phospholipase (3)
JNK (3)
Transferase (3)
Guanylate cyclase (3)
Syk (2)
NOS (2)
ROR (2)
Progesterone Receptor (2)
transporter (2)
Vasopressin Receptor (2)
Oxytocin Receptor (2)
STING (2)
TOPK (2)
ribosome (2)
PAI-1 (2)
Reductase (2)
S1P Receptor (2)
IκB/IKK (2)
Xanthine Oxidase (2)
HMG-CoA Reductase (2)
Acetyl-CoA Carboxylase (2)
Caspase (2)
IRE1 (2)
IFNAR (2)
IAP (2)
HSV (2)
Histone Demethylase (2)
Liver X Receptor (2)
Histone Acetyltransferase (2)
HIF/HIF Prolyl-Hydroxylase (2)
GPR (2)
c-Fms (2)
CRISPR/Cas9 (2)
FAAH (2)
Leukotriene Receptor (2)
Kinesin (2)
Androgen Receptor (2)
NADPH-oxidase (2)
Wee1 (1)
advanced glycation end products (1)
Adenylyl cyclase (1)
cell cycle arrest (1)
Adenosine deaminase (1)
Chloride channel (1)
Tie-2 (1)
UGT (1)
CSF-1R (1)
CXCR (1)
Discoidin Domain Receptor (DDR) (1)
AChE (1)
DNA (1)
DNA Alkylation (1)
SIK (1)
Amino Acids and Derivatives (1)
Thrombin (1)
CCR (1)
CaSR (1)
Antifolate (1)
Antioxidant (1)
Aryl Hydrocarbon Receptor (1)
ASK (1)
BCRP (1)
DPP-4 (1)
Carboxypeptidase(CPG2) (1)
Taste receptor (1)
BMI-1 (1)
Telomerase (1)
Bradykinin Receptor (1)
Carbonic Anhydrase (1)
DNA Methyltransferase (1)
NOD (1)
DprE1 (1)
Monocarboxylate transporter (1)
MALT (1)
PAFR (1)
Melanocortin Receptor (1)
MNK (1)
Monoamine Transporter (1)
P2 Receptor (1)
OXPHOS (1)
lysosomal autophagy (1)
OX Receptor (1)
Na+/Ca2+ Exchanger (1)
NAMPT (1)
NEDD8 (1)
NPC1L1 (1)
Neurokinin receptor (1)
NO Synthase (1)
PAK (1)
LTR (1)
Ephrin Receptor (1)
GlyT (1)
RIP kinase (1)
Epoxide Hydrolase (1)
Rho (1)
Factor Xa (1)
FLAP (1)
NOD-like Receptor (NLR) (1)
Glutathione Peroxidase (1)
GNRH Receptor (1)
Lipid (1)
PYK2 (1)
GPCR19 (1)
Platelet aggregation (1)
PKM (1)
Isocitrate Dehydrogenase (IDH) (1)
P-gp (1)
PERK (1)
Gap Junction Protein (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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