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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 3580 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3580 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
DNA/RNA Synthesis
CDK
EGFR
PI3K
VEGFR
Microtubule Associated
NF-κB
Topoisomerase
Epigenetic Reader Domain
PDGFR
Antibiotic
mTOR
FLT
Antifungal
Histone Methyltransferase
FGFR
c-Kit
Akt
HDAC
Dehydrogenase
c-Met/HGFR
Parasite
COX
HIV Protease
Reactive Oxygen Species
PARP
STAT
Raf
Src
Nucleoside Antimetabolite/Analog
JAK
HSP
Bcl-2 Family
Wnt/beta-catenin
Estrogen/progestogen Receptor
Estrogen Receptor/ERR
Antioxidant
Bcr-Abl
ERK
ADC Cytotoxin
Ferroptosis
Kras
Phosphatase
Aurora Kinase
Influenza Virus
PKC
TNF
p38 MAPK
Androgen Receptor
Cytochromes P450
BTK
ALK
MMP
Mitophagy
Caspase
IL Receptor
MEK
p53
Calcium Channel
AMPK
HER
E1/E2/E3 Enzyme
FAK
PPAR
c-RET
Chk
DUB
DNA-PK
GSK-3
ROS
HSV
IGF-1R
Antiviral
AChR
Ras
DNA Alkylator/Crosslinker
Virus Protease
Lipoxygenase
Trk receptor
Sirtuin
TAM Receptor
Mdm2
Histone Demethylase
Tyrosine Kinases
PDE
MAPK
P-gp
TLR
Retinoid Receptor
Proteasome
Gamma-secretase
TGF-beta/Smad
Nrf2
ATM/ATR
HIF
Potassium Channel
Pim
SARS-CoV
c-Fms
HIF/HIF Prolyl-Hydroxylase
Hedgehog/Smoothened
CXCR
PLK
DNA Methyltransferase
GABA Receptor
Sodium Channel
S6 Kinase
ROS Kinase
HBV
TRP/TRPV Channel
JNK
Adrenergic Receptor
Mitochondrial Metabolism
Smo
DNA Alkylation
Casein Kinase
PDK
5-HT Receptor
Kinesin
Carbonic Anhydrase
Transferase
Histamine Receptor
PKA
Histone Acetyltransferase
Tyrosinase
Dopamine Receptor
HCV Protease
Integrin
Serine/threonin kinase
CSF-1R
IAP
IκB/IKK
Phospholipase
Syk
PROTACs
Adenosine Receptor
Rho
Drug Metabolite
Fatty Acid Synthase
Indoleamine 2,3-Dioxygenase (IDO)
Interleukin
Prostaglandin Receptor
Aromatase
NO Synthase
NOS
Antifolate
MAO
DNA
PSMA
S1P Receptor
ATPase
YAP
c-Myc
Serine Protease
Cholinesterase (ChE)
CaMK
transporter
Beta Amyloid
Anti-infection
PD-1/PD-L1
Monocarboxylate transporter
DHFR
Reductase
Progesterone Receptor
Glucokinase
ROCK
Glucocorticoid Receptor
Antifection
Isocitrate Dehydrogenase (IDH)
Telomerase
Reverse Transcriptase
Ligand for E3 Ligase
GPR
DYRK
NADPH
PERK
GNRH Receptor
Liver X Receptor
Glutaminase
Aryl Hydrocarbon Receptor
P2X Receptor
PAK
Transketolase
Wee1
STING
Ephrin Receptor
GPX
IRAK
cholecystokinin
AhR
LPL Receptor
Tie-2
Glutathione Peroxidase
Cysteine Protease
iGluR
IRE1
RIP kinase
CCR
Endothelin Receptor
Lipid
BCRP
Survivin
Discoidin Domain Receptor (DDR)
NOD
Chloride channel
Proton pump
ROR
Ligands for Target Protein for PROTAC
IFNAR
RAAS
GTPase
Cell Cycle Arrest
PYK2
NAMPT
IDO
Myosin
UGT
MTH1
NMDAR
Hexokinase
Molecular Glues
KSP
GluR
Acyltransferase
Aminopeptidase
MELK
LPA Receptor
Platelet aggregation
BMI-1
Thrombin
Monoamine Oxidase
PKM
CRM1
Factor Xa
ABC Transporter
Opioid Receptor
FAAH
PAD
cAMP
OXPHOS
MNK
CD73
PAI-1
Methionine Adenosyltransferase (MAT)
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
Complement System
Cannabinoid Receptor
HMG-CoA Reductase
MALT
NEDD8
Amino Acids and Derivatives
LTR
RAR/RXR 
Lipase
TOPK
Galectin
CaSR
MRP
Serotonin Transporter
Neurotensin Receptor
Leukotriene Receptor
FXR
Vitamin
Immunology/Inflammation related
Annexin A
Adiponectin Receptor
DNA gyrase
Glucosidase
Bombesin Receptor
ACK1
PTEN
Somatostatin
ATP Citrate Lyase
Porcupine
GPCR19
Decarboxylase
ASK
HuR
RSV
Drug-Linker Conjugates for ADC
GST
Protease
ribosome
PI4K
KLF
Neurokinin receptor
APC/C
Protease-activated Receptor
p97
Lysosomal Autophagy
NOD-like Receptor (NLR)
Advanced Glycation End Products
Adenylyl Cyclase
NPC1L1
CD38
CYP19A1
NUDIX hydrolase
MyD88
Arginase
Arrestin
Na+/Ca2+ Exchanger
VDA
Melatonin Receptor
OCT
Kisspeptin
AAK1
Hck
LIM Kinase
Stemness kinase
RANKL/RANK
Amylase
SIK
FLAP
PAFR
Haspin Kinase
GRK
DPP-4
Neuropeptide Y Receptor
Thioredoxin
Xanthine Oxidase
SGLT
PGE Synthase
Glutathione reductase
LRRK2
Free radical scavengers
GluCls
Pyroptosis
Hippo pathway
Carboxypeptidase
GHSR
SGK
DAPK
Sigma receptor
MLK

Keywords