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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 3188 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3188 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
DNA/RNA Synthesis
Endogenous Metabolite
Antibacterial
CDK
EGFR
PI3K
VEGFR
Microtubule Associated
NF-κB
PDGFR
Topoisomerase
FLT
Antibiotic
Epigenetic Reader Domain
mTOR
Antifungal
FGFR
c-Kit
c-Met/HGFR
Akt
Parasite
COX
HDAC
Dehydrogenase
Reactive Oxygen Species
HIV Protease
Raf
JAK
Histone Methyltransferase
Src
BCL
STAT
HSP
PARP
Nucleoside Antimetabolite/Analog
Estrogen Receptor/ERR
ERK
Estrogen/progestogen Receptor
Ferroptosis
Wnt/beta-catenin
Aurora Kinase
Influenza Virus
Bcr-Abl
p38 MAPK
PKC
TNF
Androgen Receptor
Antioxidant
Mitophagy
P450
MEK
Phosphatase
Caspase
IL Receptor
Ras
HER
Calcium Channel
MMP
ALK
PPAR
E1/E2/E3 Enzyme
AMPK
p53
BTK
c-RET
DNA-PK
DNA Alkylator/Crosslinker
HSV
Chk
Sirtuin
TAM Receptor
FAK
GSK-3
ROS
IGF-1R
Virus Protease
Lipoxygenase
Trk receptor
Retinoid Receptor
AChR
Proteasome
PDE
DUB
P-gp
Potassium Channel
Gamma-secretase
TGF-beta/Smad
MAPK
Tyrosine Kinases
Pim
Antiviral
TLR
SARS-CoV
c-Fms
HIF/HIF Prolyl-Hydroxylase
Mdm2
CXCR
ATM/ATR
PLK
S6 Kinase
HBV
Nrf2
HIF
DNA Methyltransferase
Sodium Channel
JNK
Mitochondrial Metabolism
Hedgehog/Smoothened
PDK
5-HT Receptor
Carbonic Anhydrase
Histamine Receptor
PKA
DNA Alkylation
Casein Kinase
GABA Receptor
Kinesin
HCV Protease
Integrin
Adrenergic Receptor
CSF-1R
IAP
Smo
Fatty Acid Synthase
Indoleamine 2,3-Dioxygenase (IDO)
Histone Acetyltransferase
ROS Kinase
Transferase
Dopamine Receptor
Histone Demethylase
Rho
Serine/threonin kinase
TRP/TRPV Channel
Aromatase
Syk
Tyrosinase
Adenosine Receptor
Antifolate
MAO
Interleukin
Prostaglandin Receptor
IκB/IKK
Ligand for E3 Ligase
ATPase
YAP
c-Myc
Serine Protease
Drug Metabolite
CaMK
AChE
Beta Amyloid
Phospholipase
Anti-infection
NO Synthase
S1P Receptor
NOS
Reductase
ROCK
Glucocorticoid Receptor
Antifection
Isocitrate Dehydrogenase (IDH)
Telomerase
transporter
Reverse Transcriptase
PERK
Progesterone Receptor
GNRH Receptor
Glucokinase
Aryl Hydrocarbon Receptor
PAK
Wee1
Ephrin Receptor
GPR
cholecystokinin
PD-1/PD-L1
PROTACs
Monocarboxylate transporter
DHFR
LPL Receptor
DYRK
NADPH
Tie-2
Glutathione Peroxidase
Cysteine Protease
iGluR
RIP kinase
P2X Receptor
Opioid Receptor
CCR
DNA
Lipid
BCRP
IRAK
Chloride channel
Proton pump
ROR
Ligands for Target Protein for PROTAC
IFNAR
GTPase
cell cycle arrest
Liver X Receptor
NAMPT
IDO
IRE1
UGT
MTH1
NMDAR
Molecular Glues
KSP
GluR
STING
Aminopeptidase
MELK
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
NOD
BMI-1
Thrombin
AhR
Monoamine Oxidase
ABC
PYK2
Glutaminase
Myosin
Hexokinase
FAAH
Endothelin Receptor
PAD
cAMP
OXPHOS
Acyltransferase
Survivin
CD73
PAI-1
Methionine Adenosyltransferase (MAT)
GPX
LPA Receptor
CRISPR/Cas9
Hydroxylase
Adenosine deaminase
Complement System
Platelet aggregation
HMG-CoA Reductase
PKM
MALT
NEDD8
CRM1
Amino Acids and Derivatives
LTR
RAR/RXR 
RAAS
Lipase
TOPK
Factor Xa
Galectin
MRP
Serotonin Transporter
Leukotriene Receptor
Immunology/Inflammation related
Annexin A
Adiponectin receptor
APC
Bombesin Receptor
PTEN
Somatostatin
ACK
ATP Citrate Lyase
MNK
Porcupine
GPCR19
Decarboxylase
ASK
RSV
GST
ribosome
PI4K
KLF
Neurokinin receptor
Protease-activated Receptor
p97
lysosomal autophagy
NOD-like Receptor (NLR)
advanced glycation end products
Adenylyl cyclase
NPC1L1
CD38
CYP19A1
NUDIX hydrolase
MyD88
Arginase
Arrestin
Na+/Ca2+ Exchanger
CETP
VDA
Melatonin Receptor
OCT
CaSR
Hck
FXR
Neurotensin Receptor
Stemness kinase
RANKL/RANK
Amylase
SIK
FLAP
PAFR
Haspin Kinase
DNA gyrase
Glucosidase
DPP-4
Thioredoxin
Xanthine Oxidase
SGLT
PGE Synthase
Glutathione reductase
LRRK2
Free radical scavengers
GluCls
HuR
Pyroptosis
Hippo pathway
Carboxypeptidase
GHSR
SGK
DAPK
Sigma receptor
MLK

Keywords