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Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
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Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
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Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 2114 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
Get quote

Product Description

  • A unique collection of 2114 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2160)

Library Composition

Apoptosis (537)
Autophagy (332)
Antibacterial (102)
Endogenous Metabolite (100)
DNA/RNA Synthesis (93)
VEGFR (87)
EGFR (86)
PI3K (85)
CDK (82)
PDGFR (60)
Microtubule Associated (57)
NF-κB (57)
FLT (56)
Topoisomerase (53)
Antibiotic (53)
c-Kit (53)
FGFR (52)
Antifungal (50)
mTOR (47)
c-Met/HGFR (46)
HDAC (44)
Parasite (42)
COX (42)
Reactive Oxygen Species (42)
Src (40)
Akt (39)
Epigenetic Reader Domain (37)
STAT (36)
Raf (36)
HIV Protease (36)
Dehydrogenase (35)
ERK (35)
Bcr-Abl (34)
Influenza Virus (33)
PARP (33)
Ferroptosis (33)
BCL (32)
HSP (32)
JAK (30)
Histone Methyltransferase (30)
PKC (28)
p38 MAPK (28)
Aurora Kinase (28)
Nucleoside Antimetabolite/Analog (27)
Estrogen/progestogen Receptor (25)
MEK (25)
Phosphatase (25)
Estrogen Receptor/ERR (25)
ALK (24)
HER (23)
DNA Alkylator/Crosslinker (23)
Caspase (23)
TNF (23)
Mitophagy (23)
P450 (22)
Antioxidant (22)
E1/E2/E3 Enzyme (20)
c-RET (20)
DNA-PK (20)
IL Receptor (20)
AMPK (20)
IGF-1R (19)
Androgen Receptor (19)
PPAR (19)
FAK (19)
Wnt/beta-catenin (19)
Virus Protease (19)
Trk receptor (18)
P-gp (18)
HSV (17)
TAM Receptor (17)
p53 (17)
Ras (17)
Calcium Channel (17)
MMP (17)
ROS (17)
Proteasome (16)
PLK (16)
Retinoid Receptor (15)
Chk (15)
GSK-3 (15)
TLR (15)
SARS-CoV (14)
AChR (14)
c-Fms (14)
Adrenergic Receptor (14)
BTK (14)
TGF-beta/Smad (14)
DNA Alkylation (14)
Histamine Receptor (13)
Potassium Channel (13)
Gamma-secretase (13)
S6 Kinase (13)
Sodium Channel (13)
HBV (13)
ATM/ATR (13)
MAPK (12)
Lipoxygenase (12)
PDE (12)
Mdm2 (12)
Mitochondrial Metabolism (12)
Indoleamine 2,3-Dioxygenase (IDO) (12)
PDK (12)
GABA Receptor (12)
5-HT Receptor (12)
CXCR (12)
Antiviral (12)
DNA Methyltransferase (12)
Tyrosine Kinases (11)
Antifolate (11)
HIF/HIF Prolyl-Hydroxylase (11)
HIF (11)
Sirtuin (10)
PKA (10)
Smo (10)
HCV Protease (10)
CSF-1R (10)
MAO (10)
JNK (10)
Casein Kinase (10)
Nrf2 (10)
Integrin (10)
Kinesin (10)
ROS Kinase (9)
Fatty Acid Synthase (9)
Serine/threonin kinase (9)
Histone Demethylase (9)
Tyrosinase (9)
CaMK (9)
DUB (9)
Hedgehog/Smoothened (9)
IAP (9)
Dopamine Receptor (9)
Pim (9)
Interleukin (8)
Anti-infection (8)
Transferase (8)
AChE (8)
GNRH Receptor (8)
IκB/IKK (7)
Serine Protease (7)
TRP/TRPV Channel (7)
Aromatase (7)
transporter (7)
S1P Receptor (7)
ATPase (7)
Carbonic Anhydrase (7)
Glucocorticoid Receptor (7)
Adenosine Receptor (7)
ROCK (7)
Histone Acetyltransferase (6)
Ephrin Receptor (6)
Beta Amyloid (6)
NO Synthase (6)
Isocitrate Dehydrogenase (IDH) (6)
Antifection (6)
Progesterone Receptor (6)
GPR (6)
Reverse Transcriptase (6)
c-Myc (6)
NOS (5)
LPL Receptor (5)
Reductase (5)
Syk (5)
PAK (5)
Phospholipase (5)
Prostaglandin Receptor (5)
Glutathione Peroxidase (5)
Tie-2 (5)
Cysteine Protease (5)
DHFR (5)
cholecystokinin (5)
Telomerase (5)
PD-1/PD-L1 (5)
STING (4)
Thrombin (4)
NOD (4)
ROR (4)
UGT (4)
Opioid Receptor (4)
Wee1 (4)
NMDAR (4)
Rho (4)
NAMPT (4)
IRE1 (4)
Aryl Hydrocarbon Receptor (4)
KSP (4)
Glucokinase (4)
AhR (4)
Liver X Receptor (4)
Monocarboxylate transporter (4)
CCR (4)
Drug Metabolite (4)
IDO (4)
Aminopeptidase (4)
LPA Receptor (4)
IFNAR (4)
iGluR (4)
Immunology/Inflammation related (3)
DNA (3)
YAP (3)
PERK (3)
DYRK (3)
CRISPR/Cas9 (3)
Hydroxylase (3)
HMG-CoA Reductase (3)
Hexokinase (3)
GPX (3)
PYK2 (3)
Discoidin Domain Receptor (DDR) (3)
Chloride channel (3)
GluR (3)
BMI-1 (3)
Adenosine deaminase (3)
Neurokinin receptor (3)
Monoamine Oxidase (3)
cell cycle arrest (3)
MELK (3)
Survivin (3)
p97 (3)
ribosome (2)
PTEN (2)
ACK (2)
CRM1 (2)
RAAS (2)
Adiponectin receptor (2)
Galectin (2)
RSV (2)
RIP kinase (2)
Cannabinoid Receptor (2)
CD73 (2)
Amino Acids and Derivatives (2)
TOPK (2)
ASK (2)
ATP Citrate Lyase (2)
BCRP (2)
Proton pump (2)
MTH1 (2)
Protease-activated Receptor (2)
NEDD8 (2)
P2X Receptor (2)
Leukotriene Receptor (2)
OXPHOS (2)
LTR (2)
lysosomal autophagy (2)
KLF (2)
ABC (2)
IRAK (2)
MNK (2)
Platelet aggregation (2)
Lipid (2)
MRP (2)
GPCR19 (2)
Porcupine (2)
NADPH (2)
advanced glycation end products (1)
CaSR (1)
Xanthine Oxidase (1)
Myosin (1)
cAMP (1)
Thioredoxin (1)
OCT (1)
MALT (1)
Acyltransferase (1)
NPC1L1 (1)
Adenylyl cyclase (1)
VDAC (1)
Melatonin Receptor (1)
Arginase (1)
LHRH (1)
NOD-like Receptor (NLR) (1)
VDA (1)
Annexin A (1)
PAI-1 (1)
Stemness kinase (1)
Endothelin Receptor (1)
Pyroptosis (1)
GST (1)
MyD88 (1)
RAR/RXR  (1)
GHSR (1)
GTPase (1)
FXR (1)
Free radical scavengers (1)
FLAP (1)
Factor Xa (1)
Hck (1)
FAAH (1)
PGE Synthase (1)
PAD (1)
Dynamin (1)
DPP-4 (1)
LDL (1)
CYP19A1 (1)
Serotonin Transporter (1)
SGK (1)
SGLT (1)
Sigma receptor (1)
SIK (1)
Glutaminase (1)
Complement System (1)
PAFR (1)
RANKL/RANK (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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