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TargetMol | Compound Library

Anti-Cancer Active Compound Library

Catalog No. L2160

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 3970 compounds with known anti-tumor activity as Anticancer Active Compound Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2160

Anti-Cancer Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3970 compounds with known anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
Endogenous Metabolite
CDK
DNA/RNA Synthesis
EGFR
VEGFR
PI3K
NF-κB
Microtubule Associated
Topoisomerase
Antibiotic
Epigenetic Reader Domain
PDGFR
mTOR
Histone Methyltransferase
FLT
Antifungal
Akt
FGFR
Dehydrogenase
Parasite
HDAC
c-Kit
c-Met/HGFR
PARP
HIV Protease
STAT
COX
Antioxidant
Raf
Reactive Oxygen Species
Bcl-2 Family
Src
Estrogen Receptor/ERR
Wnt/beta-catenin
Nucleoside Antimetabolite/Analog
Estrogen/progestogen Receptor
ERK
JAK
Phosphatase
HSP
Influenza Virus
ADC Cytotoxin
Ferroptosis
TNF
Bcr-Abl
PKC
Androgen Receptor
Kras
MMP
Aurora Kinase
ALK
p38 MAPK
Cytochromes P450
BTK
IL Receptor
MEK
Caspase
AMPK
FAK
p53
Mitophagy
Calcium Channel
DUB
c-RET
PPAR
E1/E2/E3 Enzyme
ROS
HER
Antiviral
TLR
AChR
Ras
DNA Alkylator/Crosslinker
Histone Demethylase
Chk
IGF-1R
P-gp
GSK-3
Virus Protease
Nrf2
TAM Receptor
DNA-PK
HSV
Lipoxygenase
Sirtuin
Mdm2
Tyrosine Kinases
PDE
TGF-beta/Smad
SARS-CoV
Trk receptor
ATM/ATR
Retinoid Receptor
Proteasome
Gamma-secretase
MAPK
HIF
Potassium Channel
JNK
Pim
Hedgehog/Smoothened
c-Fms
GABA Receptor
5-HT Receptor
DNA Methyltransferase
HIF/HIF Prolyl-Hydroxylase
TRP/TRPV Channel
CXCR
PLK
S6 Kinase
PROTACs
DNA Alkylation
Histone Acetyltransferase
Sodium Channel
ROS Kinase
Kinesin
NO Synthase
Integrin
Histamine Receptor
PKA
HBV
Adrenergic Receptor
IAP
Mitochondrial Metabolism
PDK
Tyrosinase
Transferase
Dopamine Receptor
Smo
Fatty Acid Synthase
Casein Kinase
Phospholipase
Carbonic Anhydrase
IκB/IKK
NOS
HCV Protease
YAP
Serine/threonin kinase
MAO
CSF-1R
Cholinesterase (ChE)
DNA
Indoleamine 2,3-Dioxygenase (IDO)
Interleukin
GPR
Syk
PD-1/PD-L1
S1P Receptor
Adenosine Receptor
Rho
Serine Protease
Drug Metabolite
Antifection
Prostaglandin Receptor
transporter
Aromatase
DHFR
Antifolate
CaMK
Ligand for E3 Ligase
Anti-infection
ATPase
Reductase
PERK
c-Myc
ROCK
Beta Amyloid
Monocarboxylate transporter
Progesterone Receptor
GNRH Receptor
Cholecystokinin Receptor
Glutaminase
Aryl Hydrocarbon Receptor
Glucocorticoid Receptor
Isocitrate Dehydrogenase (IDH)
Telomerase
Wee1
Ephrin Receptor
GPX
Reverse Transcriptase
AhR
DYRK
NADPH
Glutathione Peroxidase
Immunology/Inflammation related
RIP kinase
P2X Receptor
Molecular Glues
PAK
CCR
PSMA
STING
NOD
IRAK
Chloride channel
LPL Receptor
IFNAR
RAAS
Tie-2
Cysteine Protease
Liver X Receptor
Glucokinase
NAMPT
iGluR
IRE1
ABC Transporter
Endothelin Receptor
Lipid
MNK
Survivin
Acyltransferase
Methionine Adenosyltransferase (MAT)
Cannabinoid Receptor
Discoidin Domain Receptor (DDR)
Proton pump
MALT
ROR
Ligands for Target Protein for PROTAC
GTPase
Cell Cycle Arrest
PYK2
Vitamin
IDO
Myosin
UGT
MTH1
NMDAR
Glucosidase
Hexokinase
KSP
cAMP
BCRP
Aminopeptidase
MELK
LPA Receptor
BMI-1
HMG-CoA Reductase
Thrombin
Monoamine Oxidase
PKM
CRM1
Galectin
Leukotriene Receptor
Opioid Receptor
Bombesin Receptor
FAAH
PAD
Transketolase
GluR
CD73
Decarboxylase
PAI-1
ribosome
CRISPR/Cas9
Hydroxylase
Adenosine Deaminase
Complement System
Neurokinin receptor
Platelet aggregation
APC/C
Protease-activated Receptor
p97
NEDD8
MyD88
Amino Acids and Derivatives
LTR
Arrestin
RAR/RXR 
Lipase
TOPK
Factor Xa
Kisspeptin
CaSR
MRP
Serotonin Transporter
Neurotensin Receptor
FXR
Annexin A
Adiponectin Receptor
GRK
DNA gyrase
ACK1
PTEN
Somatostatin
Xanthine Oxidase
ATP Citrate Lyase
OXPHOS
Porcupine
GPCR19
ASK
HuR
RSV
GST
Protease
KLF
PI4K
SGK
Lysosomal Autophagy
NOD-like Receptor (NLR)
Advanced Glycation End Products
Adenylyl Cyclase
NPC1L1
CD38
CYP19A1
NUDIX hydrolase
Dynamin
Arginase
BACE
Na+/Ca2+ Exchanger
gp120/CD4
VDA
Melatonin Receptor
OCT
AAK1
Hck
LIM Kinase
Stemness kinase
RANKL/RANK
SIK
FLAP
PAFR
Haspin Kinase
LDL
DPP-4
Neuropeptide Y Receptor
Thioredoxin
Vasopressin Receptor
Epoxide Hydrolase
SGLT
PGE Synthase
Beta-Secretase
Glutathione reductase
LRRK2
Free radical scavengers
GluCls
Pyroptosis
Hippo pathway
Carboxypeptidase
GHSR
RXFP receptor
DAPK
NADPH-oxidase
Sigma receptor
MLK

Keywords