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Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
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Anti-Cancer Approved Drug Library

Catalog No. L2110
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1726 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 1726 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2110)

Library Composition

Autophagy (338)
Autophagy (322)
Apoptosis (246)
Apoptosis (230)
Antibacterial (212)
Antibiotic (202)
Adrenergic Receptor (165)
5-HT Receptor (160)
Endogenous Metabolite (152)
Endogenous Metabolite (149)
Antibacterial (136)
COX (118)
Antibiotic (113)
Adrenergic Receptor (113)
Dopamine Receptor (107)
AChR (99)
Histamine Receptor (98)
COX (97)
5-HT Receptor (96)
DNA/RNA Synthesis (82)
DNA/RNA Synthesis (80)
Sodium Channel (78)
Potassium Channel (74)
Calcium Channel (74)
Histamine Receptor (67)
Parasite (66)
AChR (62)
Potassium Channel (61)
HIV Protease (56)
Glucocorticoid Receptor (53)
Parasite (52)
Topoisomerase (48)
Dopamine Receptor (48)
Sodium Channel (46)
P450 (45)
Antifungal (44)
Estrogen/progestogen Receptor (43)
HIV Protease (42)
Ferroptosis (40)
Reactive Oxygen Species (39)
Ferroptosis (38)
GABA Receptor (37)
PDE (36)
Antifungal (36)
EGFR (35)
Calcium Channel (35)
NF-κB (34)
Influenza Virus (33)
NF-κB (33)
Glucocorticoid Receptor (33)
P450 (33)
Estrogen/progestogen Receptor (32)
Dehydrogenase (32)
EGFR (32)
c-Kit (31)
Topoisomerase (31)
Mitophagy (31)
VEGFR (31)
VEGFR (30)
c-Kit (30)
Nucleoside Antimetabolite/Analog (30)
RAAS (30)
Mitophagy (30)
Nucleoside Antimetabolite/Analog (29)
Reactive Oxygen Species (29)
PDGFR (28)
PPAR (28)
PDGFR (28)
Microtubule Associated (28)
GABA Receptor (27)
SARS-CoV (27)
Influenza Virus (27)
PPAR (27)
SARS-CoV (25)
Prostaglandin Receptor (25)
Dehydrogenase (25)
Estrogen Receptor/ERR (24)
PDE (23)
Microtubule Associated (23)
Proton pump (22)
Serotonin Transporter (22)
Estrogen Receptor/ERR (22)
AChE (21)
Antifection (21)
Norepinephrine (20)
DNA Alkylator/Crosslinker (20)
iGluR (20)
DNA Alkylator/Crosslinker (19)
Androgen Receptor (19)
HDAC (19)
ATPase (19)
Progesterone Receptor (18)
HDAC (18)
Reverse Transcriptase (17)
FLT (17)
JAK (17)
RAAS (17)
Androgen Receptor (17)
FLT (17)
Opioid Receptor (17)
HSV (16)
TNF (16)
Serotonin Transporter (16)
HSV (16)
Virus Protease (16)
FGFR (16)
MAO (16)
Virus Protease (16)
Carbonic Anhydrase (15)
Tyrosine Kinases (15)
Bcr-Abl (15)
FGFR (15)
c-Met/HGFR (15)
c-Met/HGFR (15)
Adenosine Receptor (14)
Bcr-Abl (14)
TRP/TRPV Channel (14)
HBV (14)
ATPase (14)
GNRH Receptor (14)
Proteasome (14)
Src (14)
HBV (14)
Prostaglandin Receptor (14)
Adenosine Receptor (13)
TRP/TRPV Channel (13)
Antifolate (13)
TNF (13)
Antifolate (13)
NMDAR (13)
Src (13)
HCV Protease (13)
Proton pump (13)
Retinoid Receptor (12)
Retinoid Receptor (12)
MRP (12)
JAK (12)
Raf (12)
Thrombin (12)
CDK (12)
Raf (12)
PKC (12)
Progesterone Receptor (12)
Phosphatase (12)
ROS (11)
HMG-CoA Reductase (11)
Norepinephrine (11)
CDK (11)
Tyrosine Kinases (11)
PKC (11)
ROS (11)
DHFR (11)
MAO (11)
DHFR (11)
Amino Acids and Derivatives (11)
MRP (11)
P-gp (11)
GNRH Receptor (10)
ALK (10)
ALK (10)
Proteasome (10)
c-RET (10)
IL Receptor (10)
Drug Metabolite (10)
Monoamine Oxidase (10)
SGLT (10)
Reverse Transcriptase (10)
c-RET (10)
iGluR (10)
Carbonic Anhydrase (10)
CaMK (10)
Lipoxygenase (10)
PARP (10)
HMG-CoA Reductase (9)
Lipoxygenase (9)
P-gp (9)
DNA Alkylation (9)
AMPK (9)
DNA gyrase (9)
PARP (9)
Antifection (9)
Phosphatase (9)
ribosome (9)
Opioid Receptor (9)
Mitochondrial Metabolism (9)
MMP (9)
Transferase (9)
MMP (9)
DNA Alkylation (9)
NMDAR (9)
AChE (9)
AMPK (9)
ABC (8)
PI3K (8)
CaMK (8)
Chloride channel (8)
HER (8)
Phospholipase (8)
Monoamine Oxidase (8)
DNA (8)
STAT (8)
GluR (8)
HCV Protease (8)
Thrombin (7)
HER (7)
Phospholipase (7)
MEK (7)
STAT (7)
MEK (7)
Mitochondrial Metabolism (7)
mTOR (7)
Interleukin (7)
P2Y Receptor (7)
Guanylate cyclase (7)
Monoamine Transporter (7)
NADPH (7)
BTK (7)
HIF/HIF Prolyl-Hydroxylase (7)
Neurokinin receptor (7)
CFTR (7)
PI3K (7)
ABC (7)
Serine Protease (7)
GPR (7)
DNA Methyltransferase (6)
DNA (6)
TAM Receptor (6)
Trk receptor (6)
TAM Receptor (6)
Aromatase (6)
S1P Receptor (6)
Chloride channel (6)
BCL (6)
mTOR (6)
BCL (6)
Drug Metabolite (6)
Vasopressin Receptor (6)
Hedgehog/Smoothened (6)
NADPH (6)
Aromatase (6)
Interleukin (6)
IL Receptor (6)
ERK (6)
ribosome (6)
NO Synthase (6)
HIF/HIF Prolyl-Hydroxylase (6)
Hedgehog/Smoothened (6)
CFTR (6)
S1P Receptor (6)
CAT (6)
Trk receptor (6)
BTK (6)
Tyrosinase (6)
Transferase (6)
Caspase (5)
CaSR (5)
Beta Amyloid (5)
Wnt/beta-catenin (5)
Fatty Acid Synthase (5)
Thyroid hormone receptor(THR) (5)
ROCK (5)
Factor Xa (5)
ERK (5)
GluR (5)
Glutathione Peroxidase (5)
DNA Methyltransferase (5)
Nrf2 (5)
Ras (5)
LPL Receptor (5)
LPL Receptor (5)
Neurokinin receptor (5)
Leukotriene Receptor (5)
Glutathione Peroxidase (5)
Caspase (5)
TLR (5)
FXR (5)
PKA (5)
Endothelin Receptor (5)
Beta Amyloid (5)
Sigma receptor (5)
GSK-3 (4)
Fatty Acid Synthase (4)
PKA (4)
PGE Synthase (4)
DPP-4 (4)
p38 MAPK (4)
Oxytocin Receptor (4)
NO Synthase (4)
Tyrosinase (4)
Smo (4)
NOD (4)
ROS Kinase (4)
Melatonin Receptor (4)
LTR (4)
CXCR (4)
IκB/IKK (4)
HSP (4)
Histone Methyltransferase (4)
GPCR19 (4)
Wnt/beta-catenin (4)
Decarboxylase (4)
Ras (4)
UGT (4)
TLR (4)
Smo (4)
IκB/IKK (4)
Reductase (4)
Integrin (4)
Cysteine Protease (4)
Xanthine Oxidase (4)
FXR (4)
HSP (4)
Histone Methyltransferase (4)
GPR (4)
GSK-3 (4)
Guanylate cyclase (4)
NOS (4)
Vasopressin Receptor (4)
SGLT (4)
Antiviral (4)
Akt (4)
Antiviral (4)
Annexin A (4)
Amino Acids and Derivatives (4)
TGF-beta/Smad (3)
Na-K-Cl cotransporter (3)
LTR (3)
DPP-4 (3)
IGF-1R (3)
FAK (3)
Hydroxylase (3)
MT Receptor (3)
FAK (3)
Free radical scavengers (3)
Free radical scavengers (3)
PGE Synthase (3)
Aminopeptidase (3)
Hydroxylase (3)
Gap Junction Protein (3)
Aryl Hydrocarbon Receptor (3)
AhR (3)
PAK (3)
Antioxidant (3)
PAK (3)
GPCR19 (3)
Adenosine deaminase (3)
P2X Receptor (3)
p38 MAPK (3)
Isocitrate Dehydrogenase (IDH) (3)
GST (3)
Histone Demethylase (3)
NOD (3)
HIF (3)
Xanthine Oxidase (3)
Syk (3)
UGT (3)
CXCR (3)
Somatostatin (3)
Leukotriene Receptor (3)
cholecystokinin (3)
Adenosine deaminase (3)
Melatonin Receptor (3)
Cannabinoid Receptor (3)
Aminopeptidase (3)
TGF-beta/Smad (3)
CaSR (3)
CCR (3)
Serine/threonin kinase (3)
Cysteine Protease (3)
Serine Protease (3)
Arginase (3)
Syk (3)
Akt (3)
AhR (3)
c-Fms (3)
IGF-1R (3)
ROCK (3)
Integrin (3)
NOD-like Receptor (NLR) (3)
Melanocortin Receptor (3)
Serine/threonin kinase (3)
HIF (3)
c-Fms (3)
Monoamine Transporter (3)
Monocarboxylate transporter (2)
IRE1 (2)
Lipid (2)
Histone Demethylase (2)
LDL (2)
Isocitrate Dehydrogenase (IDH) (2)
Aryl Hydrocarbon Receptor (2)
NOD-like Receptor (NLR) (2)
Complement System (2)
Acyltransferase (2)
Annexin A (2)
TOPK (2)
Somatostatin (2)
Sirtuin (2)
Cell wall (2)
RSV (2)
ROR (2)
cholecystokinin (2)
Rho (2)
Reductase (2)
NOS (2)
CRM1 (2)
Protease-activated Receptor (2)
Endothelin Receptor (2)
Ephrin Receptor (2)
PLK (2)
Gamma-secretase (2)
GHSR (2)
Glucokinase (2)
Glutathione reductase (2)
OAT (2)
Hexokinase (2)
Lipid (2)
YAP (2)
LDL (2)
DNA gyrase (2)
Hexokinase (2)
Oxytocin Receptor (2)
Decarboxylase (2)
Sirtuin (2)
P2 Receptor (2)
P2X Receptor (2)
GST (2)
Sigma receptor (2)
RSV (2)
Neprilysin (2)
ROR (2)
Glutathione reductase (2)
Rho (2)
Ephrin Receptor (2)
GHSR (2)
Gap Junction Protein (2)
Gamma-secretase (2)
PLK (2)
TOPK (2)
CRM1 (2)
Cell wall (2)
CAT (2)
Arginase (2)
MAPK (2)
Beta-Secretase (2)
IRE1 (2)
Cannabinoid Receptor (2)
IFNAR (2)
YAP (2)
Protease-activated Receptor (2)
CCR (2)
Aurora Kinase (1)
advanced glycation end products (1)
CRISPR/Cas9 (1)
VDA (1)
BACE (1)
CSF-1R (1)
CGRP Receptor (1)
ACK (1)
Aurora Kinase (1)
RAR/RXR  (1)
Epigenetic Reader Domain (1)
RAR/RXR  (1)
Pyroptosis (1)
Pyroptosis (1)
FAAH (1)
ATP Citrate Lyase (1)
DUB (1)
BACE (1)
Complement System (1)
Beta-Secretase (1)
Thrombopoietin Receptor (1)
Factor Xa (1)
CSF-1R (1)
Telomerase (1)
cAMP (1)
Antioxidant (1)
Anti-infection (1)
ACK (1)
Chk (1)
S6 Kinase (1)
Chk (1)
CETP (1)
VDA (1)
Bradykinin Receptor (1)
CGRP Receptor (1)
S6 Kinase (1)
cAMP (1)
PKM (1)
DUB (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Neprilysin (1)
NADPH-oxidase (1)
NADPH-oxidase (1)
Na+/Ca2+ Exchanger (1)
Na+/Ca2+ Exchanger (1)
IAP (1)
MTH1 (1)
MTH1 (1)
IFNAR (1)
Hydrogenase (1)
IAP (1)
Integrase (1)
Na-K-Cl cotransporter (1)
MT Receptor (1)
Monocarboxylate transporter (1)
Imidazoline Receptor (1)
Immunology/Inflammation related (1)
Mdm2 (1)
MAPK (1)
Mdm2 (1)
Lipase (1)
ATP Citrate Lyase (1)
Liver X Receptor (1)
JNK (1)
Hydrogenase (1)
Histone Acetyltransferase (1)
Epigenetic Reader Domain (1)
PAFR (1)
Platelet aggregation (1)
Platelet aggregation (1)
FAAH (1)
Lipase (1)
Phosphorylase (1)
PDK (1)
GluCls (1)
PD-1/PD-L1 (1)
PD-1/PD-L1 (1)
GlyT (1)
PAFR (1)
PAD (1)
Histone Acetyltransferase (1)
p53 (1)
PAD (1)
p53 (1)
GRK (1)
GRK (1)
OX Receptor (1)
Hck (1)
Hck (1)
NPC1L1 (1)
Nrf2 (1)
NPC1L1 (1)
Liver X Receptor (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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