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Anti-Cancer Approved Drug Library

Catalog No. L2110
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 1825 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 1825 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2110)

Publications Cited TargetMol Libraries

1. Oncogene. 2021: 1-13.. 2. Cell Death & Disease. 2023, 14(4): 272. 3. British Journal of Cancer. 2023: 1-12. 4. Molecular oncology. 2022, 16(5): 1091. 5. Oncology Reports. 2023, 50(6): 1-11. 6. bioRxiv. 2023: 2023.01. 16.523559. 7. Cell Stem Cell. 2022 Apr 29(4) 545–558. 8. Science Bulletin. 2022. 9. Science Translational Medicine. 2022, 14(656): eabn3231.
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Library Composition

Autophagy (337)
Apoptosis (249)
Adrenergic Receptor (159)
5-HT Receptor (158)
Endogenous Metabolite (152)
Antibacterial (137)
COX (120)
Antibiotic (114)
Dopamine Receptor (108)
Histamine Receptor (104)
DNA/RNA Synthesis (80)
Sodium Channel (78)
Calcium Channel (75)
Potassium Channel (72)
AChR (67)
Parasite (53)
Glucocorticoid Receptor (52)
P450 (44)
HIV Protease (42)
Reactive Oxygen Species (38)
Ferroptosis (37)
Antifungal (36)
NF-κB (36)
EGFR (34)
Estrogen/progestogen Receptor (33)
GABA Receptor (33)
c-Kit (32)
VEGFR (32)
Mitophagy (31)
Topoisomerase (30)
PDGFR (29)
Nucleoside Antimetabolite/Analog (29)
PPAR (29)
SARS-CoV (28)
Influenza Virus (27)
Estrogen Receptor/ERR (27)
Dehydrogenase (27)
Prostaglandin Receptor (26)
PDE (25)
Serotonin Transporter (23)
Microtubule Associated (23)
Proton pump (22)
ATPase (20)
DNA Alkylator/Crosslinker (20)
Norepinephrine (20)
iGluR (19)
Androgen Receptor (19)
FLT (18)
HDAC (18)
JAK (17)
RAAS (17)
FGFR (17)
HSV (17)
Bcr-Abl (16)
Opioid Receptor (15)
c-Met/HGFR (15)
Virus Protease (15)
Adenosine Receptor (15)
Src (15)
TRP/TRPV Channel (14)
HBV (14)
Tyrosine Kinases (14)
Antifolate (13)
TNF (13)
Progesterone Receptor (13)
PKC (12)
CDK (12)
GNRH Receptor (12)
ROS (12)
Retinoid Receptor (12)
Raf (12)
SGLT (11)
ALK (11)
MAO (11)
DHFR (11)
NMDAR (11)
MRP (11)
P-gp (11)
Carbonic Anhydrase (10)
HMG-CoA Reductase (10)
Reverse Transcriptase (10)
AChE (10)
Proteasome (10)
Drug Metabolite (10)
PARP (10)
Antifection (9)
CaMK (9)
Phosphatase (9)
c-RET (9)
AMPK (9)
HCV Protease (9)
Lipoxygenase (8)
DNA Alkylation (8)
MMP (8)
mTOR (8)
PI3K (8)
BTK (8)
P2Y Receptor (8)
Monoamine Oxidase (8)
GluR (8)
HIF/HIF Prolyl-Hydroxylase (8)
Guanylate cyclase (7)
Monoamine Transporter (7)
Phospholipase (7)
TAM Receptor (7)
Trk receptor (7)
ABC (7)
Chloride channel (7)
HER (7)
STAT (7)
CFTR (7)
Thrombin (7)
GPR (7)
NADPH (7)
MEK (7)
Neurokinin receptor (7)
BCL (6)
DNA (6)
DNA Methyltransferase (6)
Interleukin (6)
Aromatase (6)
ribosome (6)
IL Receptor (6)
Vasopressin Receptor (6)
S1P Receptor (6)
Hedgehog/Smoothened (6)
P2X Receptor (6)
Mitochondrial Metabolism (6)
Transferase (6)
ERK (6)
LPL Receptor (5)
PKA (5)
Wnt/beta-catenin (5)
Nrf2 (5)
TLR (5)
ROCK (5)
Histone Methyltransferase (5)
Endothelin Receptor (5)
Caspase (5)
Ras (5)
FXR (5)
Akt (5)
CaSR (5)
ROS Kinase (5)
Glutathione Peroxidase (5)
HIF (5)
PGE Synthase (4)
HSP (4)
Fatty Acid Synthase (4)
NO Synthase (4)
Tyrosinase (4)
DPP-4 (4)
Annexin A (4)
GPCR19 (4)
NOD (4)
Leukotriene Receptor (4)
Oxytocin Receptor (4)
p38 MAPK (4)
IκB/IKK (4)
Antiviral (4)
Antioxidant (4)
Beta Amyloid (4)
Melatonin Receptor (4)
Smo (4)
GSK-3 (4)
Amino Acids and Derivatives (4)
Sigma receptor (4)
LTR (3)
Adenosine deaminase (3)
Serine/threonin kinase (3)
Syk (3)
Serine Protease (3)
Aminopeptidase (3)
Ligand for E3 Ligase (3)
Integrin (3)
Hydroxylase (3)
Melanocortin Receptor (3)
Cysteine Protease (3)
GST (3)
c-Fms (3)
Free radical scavengers (3)
Molecular Glues (3)
cholecystokinin (3)
IGF-1R (3)
AhR (3)
Isocitrate Dehydrogenase (IDH) (3)
Gamma-secretase (3)
Na-K-Cl cotransporter (3)
TGF-beta/Smad (3)
Xanthine Oxidase (3)
UGT (3)
FAK (3)
PAK (3)
MT Receptor (3)
CXCR (3)
MAPK (2)
LDL (2)
TOPK (2)
Gap Junction Protein (2)
Arginase (2)
Ligands for Target Protein for PROTAC (2)
NOS (2)
Cell wall (2)
GHSR (2)
Reductase (2)
IFNAR (2)
DNA gyrase (2)
PLK (2)
Cannabinoid Receptor (2)
CGRP Receptor (2)
CCR (2)
NOD-like Receptor (NLR) (2)
CAT (2)
Monocarboxylate transporter (2)
Beta-Secretase (2)
OAT (2)
Lipid (2)
Aryl Hydrocarbon Receptor (2)
ROR (2)
Rho (2)
IRE1 (2)
Protease-activated Receptor (2)
YAP (2)
Ephrin Receptor (2)
Decarboxylase (2)
Aurora Kinase (2)
Somatostatin (2)
CRM1 (2)
Hexokinase (2)
RSV (2)
Glutathione reductase (2)
PD-1/PD-L1 (1)
Hydrogenase (1)
NPC1L1 (1)
NADPH-oxidase (1)
Platelet aggregation (1)
Complement System (1)
p53 (1)
Mdm2 (1)
Imidazoline Receptor (1)
S6 Kinase (1)
GluCls (1)
BACE (1)
PAFR (1)
Epigenetic Reader Domain (1)
Adiponectin receptor (1)
Thrombopoietin Receptor (1)
cAMP (1)
ACK (1)
PAD (1)
Chk (1)
Immunology/Inflammation related (1)
OX Receptor (1)
Bradykinin Receptor (1)
MTH1 (1)
FAAH (1)
GRK (1)
Glucagon Receptor (1)
PROTAC Linker (1)
CSF-1R (1)
DUB (1)
Na+/Ca2+ Exchanger (1)
Factor Xa (1)
RAR/RXR  (1)
Histone Demethylase (1)
PDK (1)
Lipase (1)
JNK (1)
VDA (1)
Neprilysin (1)
IAP (1)
Pyroptosis (1)
Histone Acetyltransferase (1)
Sirtuin (1)
Hck (1)
Liver X Receptor (1)
ATP Citrate Lyase (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Thyroid hormone receptor(THR) (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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