Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Anti-Cancer Approved Drug Library

Catalog No. L2110

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 1779 approved anti-cancer drugs based on published literatures and database to form this collection that can be used as positive controls in biological cancer investigation and cancer correlation study.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L2110

Anti-Cancer Approved Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 1779 approved anti-cancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • These FDA, EMA, or NMPA approved anti-cancer drugs have annotated bioactivity, safety, and bioavailability;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Adrenergic Receptor
5-HT Receptor
COX
Dopamine Receptor
Histamine Receptor
Antibacterial
Antibiotic
Sodium Channel
Calcium Channel
Potassium Channel
DNA/RNA Synthesis
AChR
Glucocorticoid Receptor
P450
Parasite
VEGFR
c-Kit
HIV Protease
PDGFR
Antifungal
EGFR
Estrogen/progestogen Receptor
PPAR
GABA Receptor
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
SARS-CoV
Prostaglandin Receptor
Endogenous Metabolite
Ferroptosis
Serotonin Transporter
Norepinephrine
Proton pump
Mitophagy
PDE
FLT
Src
Dehydrogenase
Topoisomerase
JAK
RAAS
Bcr-Abl
Androgen Receptor
NF-κB
FGFR
ATPase
DNA Alkylator/Crosslinker
ADC Cytotoxin
c-Met/HGFR
HDAC
Microtubule Associated
Reactive Oxygen Species
HSV
Influenza Virus
HBV
Tyrosine Kinases
iGluR
ALK
Progesterone Receptor
GNRH Receptor
PARP
CDK
Opioid Receptor
SGLT
Antifolate
Raf
c-RET
Carbonic Anhydrase
Virus Protease
PKC
MAO
NMDAR
P-gp
Reverse Transcriptase
Retinoid Receptor
HER
Proteasome
DHFR
HCV Protease
P2Y Receptor
Adenosine Receptor
MRP
TRP/TRPV Channel
BTK
ROS
DNA Alkylation
PI3K
Phosphatase
Drug Metabolite
Antifection
Guanylate cyclase
CaMK
Trk receptor
MEK
TAM Receptor
Thrombin
Monoamine Oxidase
Hedgehog/Smoothened
Kras
Aromatase
AMPK
Phospholipase
TNF
Neurokinin receptor
HMG-CoA Reductase
ROS Kinase
CFTR
Chloride channel
Histone Methyltransferase
ABC
ROCK
ERK
Monoamine Transporter
IL Receptor
Vasopressin Receptor
Endothelin Receptor
MMP
GluR
DNA
mTOR
Interleukin
STAT
DNA Methyltransferase
S1P Receptor
Transferase
LPL Receptor
NADPH
CaSR
Annexin A
Smo
DPP-4
Lipoxygenase
PGE Synthase
Antiviral
TLR
ribosome
GPR
HIF
Sigma receptor
HIF/HIF Prolyl-Hydroxylase
NO Synthase
Antioxidant
Glutathione Peroxidase
Melatonin Receptor
PKA
Serine Protease
Serine/threonin kinase
Cysteine Protease
Leukotriene Receptor
Caspase
P2X Receptor
Na-K-Cl cotransporter
Mitochondrial Metabolism
Molecular Glues
Isocitrate Dehydrogenase (IDH)
BCL
Fatty Acid Synthase
Xanthine Oxidase
IGF-1R
Akt
AChE
HSP
Free radical scavengers
Ligand for E3 Ligase
c-Fms
Melanocortin Receptor
Oxytocin Receptor
Hydroxylase
Adenosine deaminase
Syk
FAK
AhR
NOS
CAT
Integrin
CRM1
p38 MAPK
Ligands for Target Protein for PROTAC
YAP
IFNAR
GSK-3
Wnt/beta-catenin
Rho
FXR
IRE1
Gamma-secretase
MT Receptor
Hexokinase
Somatostatin
Beta-Secretase
MAPK
OAT
Ephrin Receptor
Nrf2
RSV
IκB/IKK
GST
Beta Amyloid
GHSR
CGRP Receptor
Gap Junction Protein
Ras
cholecystokinin
Tyrosinase
Protease-activated Receptor
Thyroid hormone receptor(THR)
NPC1L1
Monocarboxylate transporter
ROR
Amino Acids and Derivatives
LTR
Reductase
Na+/Ca2+ Exchanger
RAR/RXR 
Histone Demethylase
JNK
TOPK
VDA
Hck
Aryl Hydrocarbon Receptor
CSF-1R
Immunology/Inflammation related
Adiponectin receptor
UGT
PAFR
MTH1
LDL
GRK
Glucagon Receptor
DNA gyrase
PROTAC Linker
HCN Channel
PAK
FAAH
CCR
Bradykinin Receptor
CXCR
Chk
ACK
Aurora Kinase
cAMP
Thrombopoietin Receptor
Epigenetic Reader Domain
DUB
TGF-beta/Smad
ATP Citrate Lyase
Aminopeptidase
GPCR19
Decarboxylase
Pyroptosis
Neprilysin
PLK
Complement System
Cannabinoid Receptor
NADPH-oxidase
NOD
S6 Kinase
NOD-like Receptor (NLR)
Imidazoline Receptor
PD-1/PD-L1

Keywords