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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2545 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2545 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Targetmol Compound Libraries
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
5-HT Receptor
Adrenergic Receptor
Dopamine Receptor
DNA/RNA Synthesis
Histamine Receptor
VEGFR
COX
EGFR
Sodium Channel
Antibacterial
Calcium Channel
PI3K
Antibiotic
FLT
CDK
Potassium Channel
PDGFR
c-Kit
P450
Glucocorticoid Receptor
JAK
FGFR
c-Met/HGFR
mTOR
HDAC
Src
HIV Protease
PPAR
Parasite
Prostaglandin Receptor
Topoisomerase
AChR
Dehydrogenase
Tyrosine Kinases
Bcr-Abl
GABA Receptor
Nucleoside Antimetabolite/Analog
GPR
Microtubule Associated
Raf
Ferroptosis
Antifungal
Reactive Oxygen Species
Androgen Receptor
SARS-CoV
Estrogen/progestogen Receptor
Adenosine Receptor
Estrogen Receptor/ERR
PARP
Aurora Kinase
HER
BTK
Epigenetic Reader Domain
Akt
NF-κB
MEK
Mitophagy
p38 MAPK
PDE
Opioid Receptor
Norepinephrine
Endogenous Metabolite
Serotonin Transporter
iGluR
HSP
Trk receptor
ALK
c-RET
ADC Cytotoxin
RAAS
P-gp
DNA Alkylator/Crosslinker
Endothelin Receptor
ATPase
Phosphatase
GSK-3
HBV
TRP/TRPV Channel
ERK
CXCR
SGLT
c-Fms
TAM Receptor
Proton pump
DNA-PK
Guanylate cyclase
HSV
Chk
Influenza Virus
Proteasome
HCV Protease
E1/E2/E3 Enzyme
NMDAR
ROS
Retinoid Receptor
Histone Methyltransferase
LPL Receptor
Progesterone Receptor
Virus Protease
PKC
DNA Alkylation
Reverse Transcriptase
HIF/HIF Prolyl-Hydroxylase
CFTR
S1P Receptor
Carbonic Anhydrase
GNRH Receptor
Antifolate
Gamma-secretase
STAT
AMPK
TNF
FAK
P2Y Receptor
Caspase
CSF-1R
Hedgehog/Smoothened
IL Receptor
Vasopressin Receptor
Interleukin
HIF
Syk
S6 Kinase
DHFR
JNK
ROCK
P2X Receptor
IGF-1R
Indoleamine 2,3-Dioxygenase (IDO)
ATM/ATR
Kras
Cannabinoid Receptor
ROS Kinase
p53
Kinesin
Mdm2
Transferase
PKA
Wnt/beta-catenin
Mitochondrial Metabolism
Antifection
Smo
BCL
OX Receptor
GluR
DNA
TGF-beta/Smad
TLR
PLK
Neurokinin receptor
Sigma receptor
Integrin
Pim
MAO
IAP
RIP kinase
Drug Metabolite
Glucagon Receptor
Isocitrate Dehydrogenase (IDH)
MMP
Casein Kinase
Beta Amyloid
Ligand for E3 Ligase
Phospholipase
DNA Methyltransferase
IRAK
HMG-CoA Reductase
Monoamine Oxidase
Histone Demethylase
Tie-2
MRP
Serine Protease
Leukotriene Receptor
DPP-4
CCR
Bradykinin Receptor
Ephrin Receptor
Nrf2
GHSR
Hydroxylase
Thrombin
Antioxidant
IFNAR
CaSR
IDO
Molecular Glues
Fatty Acid Synthase
PAK
KSP
Lipoxygenase
Wee1
PGE Synthase
STING
Sirtuin
CRFR
Aromatase
CGRP Receptor
cholecystokinin
NO Synthase
Chloride channel
PROTACs
CRM1
YAP
NADPH
Glutathione Peroxidase
Melatonin Receptor
Rho
Serine/threonin kinase
NAMPT
Annexin A
Na-K-Cl cotransporter
Monoamine Transporter
Neuropeptide Y Receptor
Somatostatin
Xanthine Oxidase
CaMK
DUB
PSMA
AChE
OAT
Antiviral
Free radical scavengers
RSV
IκB/IKK
ribosome
Melanocortin Receptor
Adenosine deaminase
Ras
Protease-activated Receptor
AhR
PD-1/PD-L1
NOS
ROR
NEDD8
Ligands for Target Protein for PROTAC
LTR
Reductase
PERK
VDA
ABC
Cysteine Protease
Liver X Receptor
FXR
PYK2
IRE1
MT Receptor
HCN Channel
Telomerase
BCRP
Beta-Secretase
MAPK
Porcupine
GPCR19
CD73
transporter
Drug-Linker Conjugates for ADC
GST
LPA Receptor
Oxytocin Receptor
Gap Junction Protein
Discoidin Domain Receptor (DDR)
p97
NOD-like Receptor (NLR)
MLK
advanced glycation end products
CAT
NPC1L1
Monocarboxylate transporter
MALT
DYRK
RAR/RXR 
TOPK
GTPase
Factor Xa
c-Myc
Galectin
Kisspeptin
N-Acetylglucosaminyltransferase
Hck
Glucokinase
Stemness kinase
Glutaminase
Aryl Hydrocarbon Receptor
Myosin
Motilin Receptor
PAFR
MTH1
LDL
GRK
DNA gyrase
GlyT
Hexokinase
Anion Exchanger
PROTAC Linker
Thioredoxin
ACK
ATP Citrate Lyase
Acyltransferase
Survivin
MNK
Aminopeptidase
Decarboxylase
ASK
PAI-1
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Neprilysin
Hippo pathway
PI4K
KLF
PDK
Aquaporin
SGK
Complement System
NADPH-oxidase
BMI-1
NOD
Imidazoline Receptor

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