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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 2545 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2545 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
DNA/RNA Synthesis
Antibacterial
Dopamine Receptor
Antibiotic
COX
Histamine Receptor
VEGFR
Sodium Channel
Calcium Channel
EGFR
PI3K
Potassium Channel
FLT
CDK
PDGFR
P450
Glucocorticoid Receptor
JAK
c-Kit
HIV Protease
Parasite
Reactive Oxygen Species
Topoisomerase
FGFR
PPAR
mTOR
HDAC
Microtubule Associated
c-Met/HGFR
Dehydrogenase
Ferroptosis
Prostaglandin Receptor
NF-κB
AChR
Src
Mitophagy
Antifungal
GABA Receptor
Nucleoside Antimetabolite/Analog
Tyrosine Kinases
SARS-CoV
GPR
Estrogen/progestogen Receptor
Adenosine Receptor
Influenza Virus
Bcr-Abl
Raf
Androgen Receptor
HER
iGluR
PDE
Opioid Receptor
Akt
Estrogen Receptor/ERR
PARP
Aurora Kinase
Epigenetic Reader Domain
MEK
BTK
p38 MAPK
P-gp
HSP
Serotonin Transporter
HSV
Norepinephrine
RAAS
ERK
Trk receptor
ALK
c-RET
ATPase
DNA Alkylator/Crosslinker
HBV
TRP/TRPV Channel
ROS
HCV Protease
GSK-3
NMDAR
CXCR
HIF/HIF Prolyl-Hydroxylase
Proton pump
Phosphatase
Virus Protease
PKC
Endothelin Receptor
SGLT
c-Fms
TAM Receptor
DNA-PK
E1/E2/E3 Enzyme
Guanylate cyclase
BCL
Chk
Retinoid Receptor
STAT
TNF
Proteasome
Carbonic Anhydrase
LPL Receptor
Progesterone Receptor
Caspase
Reverse Transcriptase
AMPK
HIF
S1P Receptor
Histone Methyltransferase
GNRH Receptor
Antifolate
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DNA Alkylation
IL Receptor
MMP
CFTR
p53
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P2X Receptor
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Hedgehog/Smoothened
IGF-1R
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Nrf2
Syk
Transferase
DHFR
P2Y Receptor
Wnt/beta-catenin
CSF-1R
Antifection
Vasopressin Receptor
Interleukin
Cannabinoid Receptor
HMG-CoA Reductase
S6 Kinase
FAK
JNK
MRP
PKA
ROCK
IAP
OX Receptor
GluR
Lipoxygenase
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TLR
Casein Kinase
ATM/ATR
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PLK
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ROS Kinase
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Integrin
Pim
MAO
Drug Metabolite
Smo
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DNA Methyltransferase
Sigma receptor
Kinesin
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RIP kinase
Glucagon Receptor
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
DNA
IκB/IKK
Phospholipase
IRAK
NADPH
Histone Demethylase
Tie-2
Glutathione Peroxidase
Serine Protease
Leukotriene Receptor
DPP-4
CCR
AChE
Ephrin Receptor
GHSR
Hydroxylase
Thrombin
NO Synthase
Chloride channel
IFNAR
Melatonin Receptor
CaSR
Aryl Hydrocarbon Receptor
IDO
Monoamine Transporter
Molecular Glues
Fatty Acid Synthase
Xanthine Oxidase
KSP
CaMK
Wee1
PGE Synthase
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Aminopeptidase
GPCR19
CRFR
ribosome
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CGRP Receptor
cholecystokinin
AhR
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YAP
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MT Receptor
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STING
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Oxytocin Receptor
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Ligands for Target Protein for PROTAC
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PYK2
IRE1
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transporter
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LPA Receptor
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Discoidin Domain Receptor (DDR)
p97
NOD-like Receptor (NLR)
MLK
advanced glycation end products
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NPC1L1
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Hydrogenase
MALT
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DYRK
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Hck
Glucokinase
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Glutaminase
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UGT
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GRK
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ACK
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ASK
GluCls
PAI-1
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MELK
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Neprilysin
KLF
PI4K
Aquaporin
SGK
Complement System
NOD
NADPH-oxidase
BMI-1
Tyrosinase
Imidazoline Receptor

Keywords