Bioactive Lipid Compound Library

Catalog No. L7000

Library Compound List Excel SDF

Bioactive lipids have been shown to provide health benefits either through modification of tissue fatty acid composition or induction of cell signaling pathways, due to their pivotal role in immune regulation, inflammation, and maintenance of tissue homeostasis. While some health benefits are derived from consumption of short to medium-chain fatty acids, evidence suggests that the polyunsaturated fatty acids (PUFAs) are the most important bioactive lipids. PUFAs are found mostly in plant seed oils and are important substrates for the biosynthesis of cellular hormones (eicosanoids) and other signaling compounds that modulate human health. The beneficial health effects of PUFAs seem to be dependent on their isomer configuration as the cis-isomer is the predominant bioactive form which enhances membrane fluidity when incorporated into cells. Increased membrane fluidity enhances cell to cell communication and helps maintain normal homeostasis or prevent the development of metabolic disorders.

The TargetMol’s Bioactive Lipid Inhibitor Library, a unique collection of 385 bioactive lipids related compounds, can be used for research in bioactive lipids, and high throughput screening (HTS) and high content screening (HCS).

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)

Request for Quote

If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com

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Product Description

A unique collection of 385 bioactive lipids related compounds for high throughput screening (HTS) and high content screening (HCS), including Agonists & Antagonists, Endocannabinoids, Farnesyl/geranylgeranyl derivates, HETEs deHETEs, hepoxilins, Polyunsaturated fatty acids, Leukotrienes, lipoxins, LPA & phosphatidic acids, Octadecanoids, PAFs, Prostaglandins & thromboxanes, Retinoids, vitamin D metabolites, Sphingolipids, etc.;
Targets include GPCR, HDAC, PPAR, DNA Alkylating, EGFR, etc.;
Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
Structurally diverse, medicinally active, and cell permeable;
NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files

Publications Cited TargetMol Libraries

1. Cell Stem Cell. 2022 Apr 29(4) 545–558. 2. Science Bulletin. 2022. 3. Science Translational Medicine. 2022, 14(656): eabn3231. 4. Science Advances. 2023, 9(9): eade3760. 5. Nature. 2020, 582: 289-293. 6. Nature Biotechnology. 2021, 39(11): 1444-1452. 7. Nature Communications. 2022, 13(1): 1-15.. 8. Nature Communications. 2023, 14(1): 1020.. 9. Nature Communications. 2023, 14(1): 2756..

10. Blood. 2021, 137(11): 1478-1490. 11. Nucleic Acids Research. 2021. 12. Nature Communications. 2023, 14(1): 7574. 13. Advanced Science. 2020, 7(16): 2000925. 14. Angewandte Chemie. 2021. 15. Acta Pharmaceutica Sinica B. 2022. 16. Protein & Cell. 2021, 12(11): 877-888. 17. Bone Research. 2023, 11(1): 54. 18. Pharmacology & Therapeutics. (2021): 107930. 19. Nature Communications. 2021, 12(1): 1-12. 20. Journal of Cell Biology. 2022, 221(5): e202112024.

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Library Composition

Endogenous Metabolite (91)

Autophagy (82)

Apoptosis (53)

PDE (48)

COX (25)

PPAR (20)

Estrogen/progestogen Receptor (19)

Antibacterial (18)

Phospholipase (17)

MAO (15)

Ferroptosis (13)

TRP/TRPV Channel (11)

Antifungal (10)

HMG-CoA Reductase (10)

P450 (10)

Lipoxygenase (10)

Prostaglandin Receptor (10)

HDAC (9)

Thrombin (9)

Mitophagy (9)

HIV Protease (9)

Antibiotic (8)

Adenosine Receptor (8)

FXR (8)

Cannabinoid Receptor (8)

Estrogen Receptor/ERR (8)

NF-κB (8)

Monoamine Oxidase (8)

Glucocorticoid Receptor (8)

Potassium Channel (7)

Retinoid Receptor (7)

Lipase (7)

Reactive Oxygen Species (7)

PI3K (7)

Virus Protease (6)

Fatty Acid Synthase (6)

TNF (6)

Factor Xa (6)

AhR (6)

Lipid (6)

Parasite (5)

Aryl Hydrocarbon Receptor (5)

Casein Kinase (5)

Adrenergic Receptor (5)

Sirtuin (5)

Calcium Channel (5)

Progesterone Receptor (5)

Dehydrogenase (5)

AChR (5)

p38 MAPK (4)

GABA Receptor (4)

Influenza Virus (4)

PKC (4)

CETP (4)

Histamine Receptor (4)

GPR (4)

Nrf2 (4)

FAAH (3)

PLK (3)

Akt (3)

HIF (3)

5-HT Receptor (3)

DNA/RNA Synthesis (3)

IκB/IKK (3)

Androgen Receptor (3)

GPCR19 (3)

Sodium Channel (3)

p53 (3)

Antioxidant (3)

Phosphatase (3)

Liver X Receptor (3)

Glutathione Peroxidase (2)

MMP (2)

Acyltransferase (2)

AChE (2)

RSV (2)

ERK (2)

Histone Demethylase (2)

LPA Receptor (2)

DNA-PK (2)

CaMK (2)

DNA (2)

LTR (2)

LPL Receptor (2)

mTOR (2)

GSK-3 (2)

PAK (2)

TGF-beta/Smad (2)

Chloride channel (2)

Caspase (2)

Leukotriene Receptor (2)

LDL (2)

CDK (2)

PARP (2)

Mitochondrial Metabolism (2)

ROS (2)

Opioid Receptor (2)

BCL (2)

MRP (2)

Mdm2 (2)

HIF/HIF Prolyl-Hydroxylase (1)

PKM (1)

PAI-1 (1)

ALK (1)

S1P Receptor (1)

MLK (1)

MEK (1)

FAK (1)

Microtubule Associated (1)

ATM/ATR (1)

Acetyl-CoA Carboxylase (1)

Tyrosinase (1)

c-RET (1)

Ras (1)

NOD (1)

AMPK (1)

NADPH-oxidase (1)

Platelet aggregation (1)

Hydroxylase (1)

STAT (1)

Proteasome (1)

Histone Acetyltransferase (1)

NADPH (1)

iGluR (1)

VEGFR (1)

Cysteine Protease (1)

Nucleoside Antimetabolite/Analog (1)

Wnt/beta-catenin (1)

Tyrosine Kinases (1)

HBV (1)

PKA (1)

ABC (1)

Melatonin Receptor (1)

DYRK (1)

Topoisomerase (1)

Reductase (1)

DNA Alkylator/Crosslinker (1)

c-Met/HGFR (1)

Src (1)

ROR (1)

Dopamine Receptor (1)

Monocarboxylate transporter (1)

Transferase (1)

NOS (1)

ATPase (1)

IAP (1)

Annexin A (1)

SARS-CoV (1)

IL Receptor (1)

HSP (1)

P-gp (1)

MNK (1)

PGE Synthase (1)

EGFR (1)

Epigenetic Reader Domain (1)

GluR (1)

Epoxide Hydrolase (1)

Xanthine Oxidase (1)

PAD (1)

HSV (1)

RIP kinase (1)

Hedgehog/Smoothened (1)

PDGFR (1)

Smo (1)

Guanylate cyclase (1)

NMDAR (1)

P2X Receptor (1)

Phosphorylase (1)

Drug Metabolite (1)

Gamma-secretase (1)

UGT (1)

NO Synthase (1)

Library Information Sample

Empty	1000025-07-9	1000413-72-8	229005-80-5	1000787-75-6	946387-07-1	1000998-59-3	1175526-27-8	1001288-58-9	1001350-96-4	1001404-83-6	Empty
Empty	Vadadustat	TAK875	TAK-779	Tegobuvir	RN-1734	BMS-687453	AM211	FT011	BMS754807	AAI101	Empty
Empty	1001625-82-6	1001645-58-4	1001753-24-7	1001908-89-9	1002304-34-8	1002-84-2	100291-86-9	100299-08-9	10030-52-1	10040-45-6	Empty
Empty	RPW-24	SRT1720 hydrochloride	INH6	SRT 2183	AMG208	Pentadecanoic acid	Apiopaeonoside	Pemirolast potassium	L-Anserine nitrate salt	Sodium Picosulfate	Empty
Empty	100427-26-7	1004316-88-4	10045-45-1	100462-37-1	1004990-28-6	100-51-6	1005-24-9	1005264-47-0	1005334-57-5	1005342-46-0	Empty
Empty	Lercanidipine	Cobicistat	1-Ethyl-2-benzimidazolinone	ROSIRIDIN	PF-AKT400	Benzyl alcohol	1-Methylnicotinamide chloride	MX69	CVT-10216	LCL161	Empty
Empty	1005491-05-3	100-55-0	1005504-62-0	1005883-72-6	100643-71-8	1007207-67-1	10075-50-0	1007647-73-5	100784-20-1	10083-24-6	Empty
Empty	Tirasemtiv	Roniacol	Rg3039	Z433927330	Desloratadine	CH5132799	5-Bromoindole	Smurf1-IN-A01	Halosulfuron-methyl	Piceatannol	Empty
Empty	100872-83-1	100874-08-6	1009119-64-5	1009119-65-6	100929-71-3	1009298-09-2	1009298-59-2	100929-99-5	1009734-33-1	10097-84-4	Empty
Empty	ML346	SB 4	Daclatasvir	Daclatasvir dihydrochloride	NADPH (tetracyclohexanamine)	AZD8055	Vistusertib	PAβN dihydrochloride	HZ1157	Rotundine	Empty
Empty	1009816-48-1	1009817-63-3	1009820-21-6	100986-85-4	101001-34-7	1010411-21-8	1010-60-2	1011244-68-0	1011301-27-1	1011529-10-4	Empty
Empty	Thiamet G	B-AP15	Silmitasertib	Levofloxacin	Pamicogrel	GSK369796 Dihydrochloride	2-Chloronaphthoquinone	TFAP	Tenovin3	Azvudine	Empty
Empty	101152-94-7	101155-02-6	1011557-82-6	1011-74-1	101-20-2	1012054-59-9	101-21-3	101-26-8	101303-98-4	1013101-36-4	Empty
Empty	Milnacipran hydrochloride	BW-A78U	Tenovin-6	DL-Normetanephrine hydrochloride	Triclocarban	CUDC101	Chlorpropham	Mestinon	Zacopride hydrochloride	PF04691502	Empty
Empty	101-31-5	1013-69-0	1013750-77-0	1013753-99-5	10138-52-0	1013920-15-4	1013937-63-7	1014691-61-2	101477-54-7	101494-95-5	Empty
Empty	L-Hyoscyamine	Noreugenin	ML-030	BC-1382	Gadolinium chloride	Vorolanib	VTP-27999 TFA	GSK0660	Lomerizine hydrochloride	8-CHLOROQUINAZOLIN-4(1H)-ONE	Empty