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TargetMol | Compound Library

Drug Repurposing Compound Library

Catalog No. L9200

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds. The Drug Repurposing Compound Library by TargetMol, containing 4630 approved and clinical drugs, which have undergone extensive preclinical studies and have well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization, is a good tool for drug repurposing and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9200

Drug Repurposing Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 4630 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS);
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • All approved drugs collected in this library are approved by Food and Drug Administration (FDA), the European Medicine Agency (EMA), or National Medical Products Administration (NMPA), or included in the US Pharmacopeia (USP) Dictionary, the British Pharmacopoeia (BP), the European Pharmacopoeia (EP), the Japanese Pharmacopoeia (JP), or Chinese Pharmacopoeia (CP) Dictionary;
  • Covers various research areas, such as cancer, cardiovascular disease, immunology, respiratory system, etc.
  • Covers various targets, such as 5-HT Receptor, Sodium Channel, p38 MAPK, PI3K, MEK, etc.
  • Detailed compound information with structure, target, activity, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Autophagy
Antibacterial
Apoptosis
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
AChR
COX
Dopamine Receptor
Histamine Receptor
HIV Protease
DNA/RNA Synthesis
Parasite
Antifungal
Sodium Channel
Potassium Channel
Calcium Channel
VEGFR
EGFR
Topoisomerase
PDE
PI3K
Reactive Oxygen Species
Glucocorticoid Receptor
P450
CDK
Influenza Virus
FLT
HCV Protease
Estrogen/progestogen Receptor
PPAR
Dehydrogenase
Ferroptosis
NF-κB
PDGFR
SARS-CoV
Microtubule Associated
c-Kit
JAK
FGFR
GABA Receptor
HDAC
RAAS
Prostaglandin Receptor
mTOR
c-Met/HGFR
Mitophagy
Estrogen Receptor/ERR
HBV
Src
Nucleoside Antimetabolite/Analog
Reverse Transcriptase
Tyrosine Kinases
Adenosine Receptor
Serotonin Transporter
iGluR
Androgen Receptor
ribosome
GPR
Proteasome
Virus Protease
Bcr-Abl
HSV
Raf
BTK
Norepinephrine
MAO
NMDAR
AChE
TNF
ATPase
Progesterone Receptor
TRP/TRPV Channel
GluR
PARP
Opioid Receptor
HER
Phosphatase
Epigenetic Reader Domain
Akt
Carbonic Anhydrase
Transferase
Antioxidant
Aurora Kinase
HSP
p38 MAPK
Antifection
ROS
Beta Amyloid
Proton pump
PKC
P-gp
MEK
HIF/HIF Prolyl-Hydroxylase
IL Receptor
Antiviral
Monoamine Oxidase
DPP-4
ALK
Thrombin
DNA Alkylator/Crosslinker
ERK
Drug Metabolite
MMP
c-RET
Thyroid hormone receptor(THR)
Mitochondrial Metabolism
Interleukin
Trk receptor
AMPK
Phospholipase
Histone Methyltransferase
GSK-3
BCL
CXCR
Endothelin Receptor
Retinoid Receptor
c-Fms
Caspase
SGLT
TLR
TAM Receptor
MRP
PKA
Gamma-secretase
P2X Receptor
CCR
NO Synthase
DNA-PK
ROCK
E1/E2/E3 Enzyme
Chk
Lipoxygenase
STAT
Cannabinoid Receptor
Syk
CFTR
S1P Receptor
Integrin
LPL Receptor
NADPH
GNRH Receptor
DNA Alkylation
HIF
HMG-CoA Reductase
p53
DHFR
Amino Acids and Derivatives
Factor Xa
Wnt/beta-catenin
Antifolate
DNA gyrase
Guanylate cyclase
Hedgehog/Smoothened
IGF-1R
TGF-beta/Smad
Nrf2
FAK
P2Y Receptor
Reductase
Glutathione Peroxidase
Serine Protease
FXR
CSF-1R
IAP
Vasopressin Receptor
Neurokinin receptor
Chloride channel
NOS
Histone Demethylase
CETP
ABC
Glucosidase
Indoleamine 2,3-Dioxygenase (IDO)
ATM/ATR
Hydroxylase
PLK
DNA Methyltransferase
S6 Kinase
Ras
Tyrosinase
Kinesin
Mdm2
CAT
JNK
Smo
OX Receptor
CaMK
Sirtuin
Casein Kinase
RSV
Sigma receptor
ROS Kinase
BACE
Pim
Cysteine Protease
Leukotriene Receptor
Glucokinase
Aryl Hydrocarbon Receptor
Glucagon Receptor
Monoamine Transporter
Xanthine Oxidase
Beta-Secretase
Acyltransferase
Aminopeptidase
ROR
RIP kinase
Isocitrate Dehydrogenase (IDH)
Fatty Acid Synthase
PAK
DNA
IκB/IKK
Ligand for E3 Ligase
Aromatase
IRAK
cholecystokinin
AhR
LTR
IFNAR
Tie-2
CaSR
Serine/threonin kinase
Liver X Receptor
IDO
MT Receptor
GlyT
FAAH
Bradykinin Receptor
Lipid
PGE Synthase
GPCR19
Ephrin Receptor
CRFR
GHSR
Complement System
Gap Junction Protein
NOD
NADPH-oxidase
Imidazoline Receptor
DprE1
YAP
Cell wall
Melatonin Receptor
Annexin A
UGT
Molecular Glues
Neuropeptide Y Receptor
KSP
Wee1
MAPK
Decarboxylase
Neprilysin
Acetyl-CoA Carboxylase
LPA Receptor
Melanocortin Receptor
Oxytocin Receptor
CGRP Receptor
Anti-infection
NOD-like Receptor (NLR)
PD-1/PD-L1
Monocarboxylate transporter
CRM1
Arginase
Rho
NAMPT
Glutaminase
Myosin
LDL
Na-K-Cl cotransporter
Hexokinase
Somatostatin
Epoxide Hydrolase
DUB
Telomerase
OAT
STING
Free radical scavengers
GST
PDK
Adenosine deaminase
Protease-activated Receptor
advanced glycation end products
PROTACs
Taste receptor
GSNOR
NEDD8
Ligands for Target Protein for PROTAC
Lipase
PERK
TOPK
VDA
Galectin
PYK2
IRE1
FLAP
Phosphorylase
Integrase
PROTAC Linker
Stearoyl-CoA Desaturase (SCD)
Thrombopoietin Receptor
ATP Citrate Lyase
BCRP
Glutathione reductase
Porcupine
CD73
transporter
GluCls
PAI-1
Aquaporin
Discoidin Domain Receptor (DDR)
p97
MLK
PKM
Adenylyl cyclase
NPC1L1
Hydrogenase
MALT
Dynamin
Arrestin
Na+/Ca2+ Exchanger
RAR/RXR 
DYRK
GTPase
c-Myc
Kisspeptin
N-Acetylglucosaminyltransferase
VDAC
Hck
LIM Kinase
Stemness kinase
Immunology/Inflammation related
Motilin Receptor
Adiponectin receptor
PAFR
MTH1
Fas/FasL
GRK
AAK1 (AP2 associated kinase 1)
Anion Exchanger
HCN Channel
Thioredoxin
Angiotensin-converting Enzyme (ACE)
PAD
ACK
cAMP
Survivin
MNK
Histone Acetyltransferase
ASK
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
PI4K
KLF
CRISPR/Cas9
RXFP receptor
SGK
Platelet aggregation
BMI-1

Keywords