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Drug Repurposing Compound Library

Catalog No. L9200
  Library Compound List   Excel SDF

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

The Drug Repurposing Compound Library by TargetMol, containing 4240 approved and clinical drugs, which have undergone extensive preclinical studies and have well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization, is a good tool for drug repurposing and cell induction.

In addtion, we put the compounds that should be provided in the form of dry powder together to form Part B in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Please contact us for prices and availability for the specification of product you are interested at.
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If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 4240 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS);
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • All approved drugs collected in this library are approved by Food and Drug Administration (FDA), the European Medicine Agency (EMA), or National Medical Products Administration (NMPA), or included in the US Pharmacopeia (USP) Dictionary, the British Pharmacopoeia (BP), the European Pharmacopoeia (EP), the Japanese Pharmacopoeia (JP), or Chinese Pharmacopoeia (CP) Dictionary;
  • Covers various research areas, such as cancer, cardiovascular disease, immunology, respiratory system, etc.
  • Covers various targets, such as 5-HT Receptor, Sodium Channel, p38 MAPK, PI3K, MEK, etc.
  • Detailed compound information with structure, target, activity, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L9200)

Library Composition

Autophagy (465)
Antibacterial (434)
Apoptosis (420)
Antibiotic (398)
Endogenous Metabolite (338)
5-HT Receptor (194)
Adrenergic Receptor (171)
AChR (149)
COX (132)
Dopamine Receptor (130)
DNA/RNA Synthesis (114)
Histamine Receptor (110)
Parasite (108)
HIV Protease (103)
Antifungal (96)
Sodium Channel (93)
Potassium Channel (87)
Calcium Channel (79)
VEGFR (75)
Topoisomerase (68)
Reactive Oxygen Species (64)
EGFR (63)
PI3K (62)
Influenza Virus (61)
Glucocorticoid Receptor (61)
PDE (60)
Ferroptosis (58)
Estrogen/progestogen Receptor (58)
P450 (57)
GABA Receptor (55)
Dehydrogenase (54)
FLT (52)
NF-κB (52)
PPAR (49)
PDGFR (48)
CDK (47)
SARS-CoV (47)
HCV Protease (46)
JAK (46)
c-Kit (44)
FGFR (44)
HDAC (43)
Microtubule Associated (42)
RAAS (41)
c-Met/HGFR (40)
Mitophagy (39)
Prostaglandin Receptor (39)
mTOR (37)
Nucleoside Antimetabolite/Analog (34)
Reverse Transcriptase (33)
Estrogen Receptor/ERR (32)
Src (32)
Adenosine Receptor (31)
Opioid Receptor (31)
ribosome (31)
HBV (31)
HSV (30)
Serotonin Transporter (30)
Proteasome (30)
Androgen Receptor (29)
Virus Protease (29)
iGluR (29)
Bcr-Abl (28)
AChE (28)
Norepinephrine (27)
Raf (27)
TNF (26)
Tyrosine Kinases (26)
MAO (25)
ATPase (25)
GPR (25)
NMDAR (24)
Carbonic Anhydrase (23)
Phosphatase (23)
Progesterone Receptor (23)
DNA Alkylator/Crosslinker (22)
PARP (22)
ROS (22)
Antifection (22)
Beta Amyloid (21)
Akt (21)
GluR (21)
Proton pump (21)
Epigenetic Reader Domain (20)
MEK (20)
HSP (20)
TRP/TRPV Channel (20)
Monoamine Oxidase (20)
Antioxidant (19)
IL Receptor (19)
P-gp (19)
BTK (19)
p38 MAPK (19)
Mitochondrial Metabolism (19)
PKC (19)
c-RET (18)
HER (18)
AMPK (18)
Thrombin (18)
ALK (18)
Transferase (18)
GNRH Receptor (17)
ERK (17)
MMP (17)
Interleukin (17)
DPP-4 (17)
Drug Metabolite (17)
TAM Receptor (16)
Retinoid Receptor (16)
Thyroid hormone receptor(THR) (16)
Caspase (16)
HIF/HIF Prolyl-Hydroxylase (16)
Trk receptor (16)
GSK-3 (15)
Phospholipase (15)
BCL (15)
NO Synthase (15)
Antifolate (14)
Antiviral (14)
Gamma-secretase (14)
CXCR (14)
Aurora Kinase (14)
MRP (14)
E1/E2/E3 Enzyme (14)
DNA Alkylation (13)
NADPH (13)
Endothelin Receptor (13)
c-Fms (13)
Lipoxygenase (13)
STAT (13)
Glucagon Receptor (13)
Glucokinase (13)
Chk (12)
DNA-PK (12)
CCR (12)
CFTR (12)
HMG-CoA Reductase (12)
Guanylate cyclase (12)
P2 Receptor (12)
TLR (12)
p53 (11)
Histone Methyltransferase (11)
Factor Xa (11)
Neurokinin receptor (11)
DHFR (11)
DNA gyrase (11)
FAK (11)
Amino Acids and Derivatives (11)
S1P Receptor (11)
Vasopressin Receptor (11)
PKA (11)
Integrin (10)
Chloride channel (10)
Sigma receptor (10)
CSF-1R (10)
LPL Receptor (10)
Syk (10)
IGF-1R (10)
HIF (10)
CaMK (10)
Wnt/beta-catenin (10)
SGLT (10)
ROCK (10)
Reductase (10)
Glutathione Peroxidase (10)
Hedgehog/Smoothened (10)
Cannabinoid Receptor (10)
Serine Protease (9)
IAP (9)
S6 Kinase (9)
FXR (9)
TGF-beta/Smad (9)
DNA Methyltransferase (9)
PLK (9)
OX Receptor (9)
Tyrosinase (8)
ADC Cytotoxin (8)
Hydroxylase (8)
JNK (8)
Sirtuin (8)
DNA (8)
ABC (8)
Indoleamine 2,3-Dioxygenase (IDO) (8)
Histone Demethylase (8)
CAT (8)
Aminopeptidase (7)
ATM/ATR (7)
Mdm2 (7)
NOS (7)
Ras (7)
Smo (7)
Aryl Hydrocarbon Receptor (7)
Xanthine Oxidase (7)
Aromatase (7)
LTR (7)
RSV (6)
Isocitrate Dehydrogenase (IDH) (6)
IκB/IKK (6)
AhR (6)
Kinesin (6)
Complement System (6)
Leukotriene Receptor (6)
BACE (6)
CETP (6)
Beta-Secretase (6)
Monoamine Transporter (6)
Cysteine Protease (6)
Fatty Acid Synthase (6)
Casein Kinase (6)
cholecystokinin (6)
PAK (6)
Acyltransferase (6)
Oxytocin Receptor (5)
ROR (5)
IDO (5)
UGT (5)
IFNAR (5)
RIP kinase (5)
Cell wall (5)
NOD (5)
Ephrin Receptor (5)
Anti-infection (5)
Pim (5)
GHSR (5)
Gap Junction Protein (5)
FAAH (5)
Liver X Receptor (5)
Bradykinin Receptor (4)
GPCR19 (4)
Melatonin Receptor (4)
GST (4)
Annexin A (4)
PDK (4)
Serine/threonin kinase (4)
PGE Synthase (4)
Decarboxylase (4)
CaSR (4)
CGRP Receptor (4)
Lipid (4)
Acetyl-CoA Carboxylase (4)
Somatostatin (4)
DprE1 (4)
Tie-2 (4)
NOD-like Receptor (NLR) (4)
Neprilysin (4)
Free radical scavengers (3)
Glutathione reductase (3)
Rho (3)
Arginase (3)
DYRK (3)
MAPK (3)
GlyT (3)
NAMPT (3)
Melanocortin Receptor (3)
Telomerase (3)
STING (3)
Monocarboxylate transporter (3)
MT Receptor (3)
Myosin (3)
KSP (3)
Hexokinase (3)
NADPH-oxidase (3)
Neuropeptide Y Receptor (3)
IRAK (3)
CRM1 (3)
Nrf2 (3)
OAT (3)
TOPK (3)
P2X Receptor (3)
Adenosine deaminase (3)
VDA (2)
Thrombopoietin Receptor (2)
Stearoyl-CoA Desaturase (SCD) (2)
advanced glycation end products (2)
Taste receptor (2)
YAP (2)
LPA Receptor (2)
LDL (2)
Histone Acetyltransferase (2)
Discoidin Domain Receptor (DDR) (2)
Integrase (2)
IRE1 (2)
Lipase (2)
PAI-1 (2)
PD-1/PD-L1 (2)
PYK2 (2)
Na-K-Cl cotransporter (2)
Galectin (2)
BCRP (2)
PKM (2)
DUB (2)
Porcupine (2)
ATP Citrate Lyase (2)
c-Myc (2)
Protease-activated Receptor (2)
CRFR (2)
NEDD8 (2)
LHRH (1)
KLF (1)
CRISPR/Cas9 (1)
Hydrogenase (1)
Thioredoxin (1)
Pyroptosis (1)
transporter (1)
Hck (1)
GTPase (1)
GRK (1)
Glutaminase (1)
GluCls (1)
VDAC (1)
ACK (1)
Wee1 (1)
Dynamin (1)
FLAP (1)
GSNOR (1)
Stemness kinase (1)
MELK (1)
PAD (1)
ASK (1)
RAR/RXR  (1)
Aquaporin (1)
Platelet aggregation (1)
PI4K (1)
Phosphorylase (1)
BMI-1 (1)
PERK (1)
cAMP (1)
PAFR (1)
p97 (1)
Survivin (1)
Anion Exchanger (1)
SGK (1)
OXPHOS (1)
NPC1L1 (1)
Angiotensin-converting Enzyme (ACE) (1)
N-Acetylglucosaminyltransferase (1)
Na+/Ca2+ Exchanger (1)
MTH1 (1)
MNK (1)
MLK (1)
Epoxide Hydrolase (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE