Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Drug Repurposing Compound Library

Catalog No. L9200

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds. The Drug Repurposing Compound Library by TargetMol, containing 4960 approved and clinical drugs, which have undergone extensive preclinical studies and have well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization, is a good tool for drug repurposing and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L9200

Drug Repurposing Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 4960 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS);
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • All approved drugs collected in this library are approved by Food and Drug Administration (FDA), the European Medicine Agency (EMA), or National Medical Products Administration (NMPA), or included in the US Pharmacopeia (USP) Dictionary, the British Pharmacopoeia (BP), the European Pharmacopoeia (EP), the Japanese Pharmacopoeia (JP), or Chinese Pharmacopoeia (CP) Dictionary;
  • Covers various research areas, such as cancer, cardiovascular disease, immunology, respiratory system, etc.
  • Covers various targets, such as 5-HT Receptor, Sodium Channel, p38 MAPK, PI3K, MEK, etc.
  • Detailed compound information with structure, target, activity, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Autophagy
Antibacterial
Apoptosis
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
AChR
Dopamine Receptor
Histamine Receptor
COX
HIV Protease
Parasite
DNA/RNA Synthesis
Antifungal
Sodium Channel
Potassium Channel
Calcium Channel
VEGFR
EGFR
Topoisomerase
PDE
Glucocorticoid Receptor
PI3K
Reactive Oxygen Species
SARS-CoV
Cytochromes P450
CDK
Estrogen/progestogen Receptor
Dehydrogenase
HCV Protease
FLT
Influenza Virus
GABA Receptor
Ferroptosis
PPAR
NF-κB
PDGFR
Microtubule Associated
JAK
c-Kit
HDAC
FGFR
RAAS
c-Met/HGFR
Estrogen Receptor/ERR
mTOR
HBV
Prostaglandin Receptor
Mitophagy
Nucleoside Antimetabolite/Analog
Src
Adenosine Receptor
Androgen Receptor
Reverse Transcriptase
Tyrosine Kinases
Serotonin Transporter
iGluR
Bcr-Abl
NMDAR
HSV
Cholinesterase (ChE)
GPR
TRP/TRPV Channel
Norepinephrine
Proteasome
BTK
GluR
Virus Protease
MAO
Raf
HER
ATPase
ADC Cytotoxin
Phosphatase
PARP
Antiviral
ribosome
TNF
Progesterone Receptor
Opioid Receptor
Epigenetic Reader Domain
Akt
HSP
p38 MAPK
Antioxidant
ROS
Carbonic Anhydrase
Transferase
Beta Amyloid
PKC
Aurora Kinase
ALK
IL Receptor
P-gp
HIF/HIF Prolyl-Hydroxylase
Proton pump
Histone Methyltransferase
Antifection
MMP
MEK
Thyroid hormone receptor(THR)
DPP-4
Monoamine Oxidase
DNA Alkylator/Crosslinker
Drug Metabolite
Mitochondrial Metabolism
Endothelin Receptor
TLR
c-RET
Thrombin
ERK
Interleukin
Trk receptor
Bcl-2 Family
AMPK
Phospholipase
GSK-3
P2X Receptor
CXCR
Retinoid Receptor
c-Fms
HMG-CoA Reductase
GNRH Receptor
MRP
Caspase
ROCK
CCR
Lipoxygenase
SGLT
STAT
TAM Receptor
S1P Receptor
Integrin
PKA
Vasopressin Receptor
Chk
Neurokinin receptor
FAK
p53
NO Synthase
DNA-PK
NADPH
E1/E2/E3 Enzyme
Gamma-secretase
Guanylate cyclase
DNA Alkylation
HIF
Cannabinoid Receptor
Syk
CFTR
LPL Receptor
Reductase
Factor Xa
Wnt/beta-catenin
Antifolate
TGF-beta/Smad
Nrf2
Kras
DHFR
Amino Acids and Derivatives
P2Y Receptor
Glutathione Peroxidase
Serine Protease
FXR
DNA gyrase
Hedgehog/Smoothened
IGF-1R
RSV
Sigma receptor
ROS Kinase
Histone Demethylase
CSF-1R
IAP
ATM/ATR
Hydroxylase
PLK
Tyrosinase
Mdm2
Chloride channel
NOS
CETP
Leukotriene Receptor
ABC Transporter
Glucosidase
OX Receptor
CaMK
Indoleamine 2,3-Dioxygenase (IDO)
DNA Methyltransferase
S6 Kinase
Kinesin
BACE
JNK
Cysteine Protease
Vitamin
Smo
Xanthine Oxidase
Ligand for E3 Ligase
NOD
cholecystokinin
Glucokinase
Aryl Hydrocarbon Receptor
RIP kinase
Glucagon Receptor
DNA
Beta-Secretase
Acyltransferase
Aminopeptidase
Sirtuin
Casein Kinase
Aromatase
ROR
Pim
Monoamine Transporter
Molecular Glues
Isocitrate Dehydrogenase (IDH)
Fatty Acid Synthase
PAK
Bradykinin Receptor
PGE Synthase
IκB/IKK
GHSR
CGRP Receptor
Gap Junction Protein
IRAK
AhR
LTR
IFNAR
Cell wall
Tie-2
Serine/threonin kinase
IDO
MT Receptor
GlyT
FAAH
MAPK
GPCR19
Ephrin Receptor
CRFR
Melanocortin Receptor
Complement System
NADPH-oxidase
Imidazoline Receptor
PROTACs
CRM1
DprE1
YAP
Melatonin Receptor
CaSR
Liver X Receptor
Annexin A
UGT
Neuropeptide Y Receptor
Somatostatin
KSP
Lipid
Wee1
OAT
STING
Decarboxylase
Neprilysin
GST
Acetyl-CoA Carboxylase
LPA Receptor
PDK
Anti-infection
Ras
Protease-activated Receptor
NOD-like Receptor (NLR)
PD-1/PD-L1
Monocarboxylate transporter
Arginase
PERK
Rho
PYK2
NAMPT
Glutaminase
Myosin
LDL
Na-K-Cl cotransporter
Hexokinase
Epoxide Hydrolase
Mucin
DUB
Telomerase
Free radical scavengers
transporter
Oxytocin Receptor
Adenosine Deaminase
Advanced Glycation End Products
Taste receptor
GSNOR
NEDD8
Ligands for Target Protein for PROTAC
Lipase
TOPK
VDA
Galectin
c-Myc
Kisspeptin
IRE1
FLAP
Phosphorylase
Integrase
HCN Channel
Thrombopoietin Receptor
ATP Citrate Lyase
BCRP
Glutathione reductase
Porcupine
CD73
GluCls
PAI-1
Aquaporin
Discoidin Domain Receptor (DDR)
p97
MLK
PKM
Apelin receptor
Adenylyl Cyclase
NPC1L1
Hydrogenase
MALT
Dynamin
Arrestin
Na+/Ca2+ Exchanger
RAR/RXR 
DYRK
gp120/CD4
GTPase
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
LIM Kinase
Neurotensin Receptor
Stemness kinase
Immunology/Inflammation related
SIK
Adiponectin Receptor
PAFR
MTH1
Fas/FasL
GRK
Anion Exchanger
PROTAC Linker
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
ACK1
Angiotensin-converting Enzyme (ACE)
PAD
cAMP
Huntingtin
Survivin
MNK
Histone Acetyltransferase
ASK
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
KLF
PI4K
CRISPR/Cas9
RXFP receptor
SGK
Platelet aggregation
BMI-1