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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively. Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
Antibacterial
5-HT Receptor
CDK
COX
Antibiotic
AChR
EGFR
PI3K
HIV Protease
Endogenous Metabolite
DNA/RNA Synthesis
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
PDE
NF-κB
Epigenetic Reader Domain
VEGFR
Dehydrogenase
Histamine Receptor
Histone Methyltransferase
Cytochromes P450
Potassium Channel
Sodium Channel
Parasite
HDAC
Phosphatase
JAK
Antifungal
mTOR
Src
FLT
Microtubule Associated
Topoisomerase
TRP/TRPV Channel
SARS-CoV
PDGFR
Cholinesterase (ChE)
PKC
PARP
Raf
FGFR
Wnt/beta-catenin
p38 MAPK
Influenza Virus
STAT
HCV Protease
RAAS
ERK
GSK-3
Akt
MAO
Prostaglandin Receptor
c-Kit
GABA Receptor
Lipoxygenase
Bcr-Abl
c-Met/HGFR
ALK
NMDAR
MMP
TNF
Proteasome
Reactive Oxygen Species
Adenosine Receptor
GluR
Bcl-2 Family
DUB
Phospholipase
Aurora Kinase
HSP
Ferroptosis
BTK
Histone Demethylase
Virus Protease
Kras
TGF-beta/Smad
Tyrosinase
GPR
Tyrosine Kinases
ROCK
iGluR
IL Receptor
MAPK
Ras
ATPase
Transferase
HER
E1/E2/E3 Enzyme
CCR
Casein Kinase
NO Synthase
Integrin
PKA
Beta Amyloid
MEK
Monoamine Oxidase
PPAR
Serine/threonin kinase
Antiviral
JNK
Serotonin Transporter
Caspase
Carbonic Anhydrase
IκB/IKK
Reverse Transcriptase
Antioxidant
Cysteine Protease
Androgen Receptor
DNA-PK
Mitophagy
HBV
Mitochondrial Metabolism
HSV
Sirtuin
CXCR
AMPK
c-RET
Reductase
NOS
ROS
Norepinephrine
HIF
ADC Cytotoxin
Estrogen/progestogen Receptor
Serine Protease
RIP kinase
P2X Receptor
IGF-1R
P-gp
Estrogen Receptor/ERR
CaMK
Histone Acetyltransferase
TAM Receptor
Nucleoside Antimetabolite/Analog
Gamma-secretase
Drug Metabolite
Glucosidase
TLR
HIF/HIF Prolyl-Hydroxylase
Interleukin
Trk receptor
FAK
Proton pump
Hedgehog/Smoothened
FAAH
Acyltransferase
c-Fms
PLK
S6 Kinase
Cannabinoid Receptor
Opioid Receptor
ATM/ATR
Neurokinin receptor
Syk
p53
Glucocorticoid Receptor
DPP-4
Endothelin Receptor
NOD
Pim
Chk
HMG-CoA Reductase
Fatty Acid Synthase
Kinesin
Chloride channel
DYRK
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Anti-infection
IRAK
Thrombin
LTR
Factor Xa
Rho
Leukotriene Receptor
LRRK2
transporter
Mdm2
LPL Receptor
BACE
NADPH
Lipase
Xanthine Oxidase
PDK
DNA Methyltransferase
PD-1/PD-L1
Immunology/Inflammation related
Nrf2
Sigma receptor
S1P Receptor
P2Y Receptor
PERK
Glutathione Peroxidase
Smo
cAMP
Hydroxylase
MRP
PAK
Epoxide Hydrolase
Retinoid Receptor
Complement System
DHFR
Glucokinase
OX Receptor
LPA Receptor
PI4K
cholecystokinin
ROS Kinase
YAP
c-Myc
IRE1
Neuropeptide Y Receptor
ribosome
GTPase
Aryl Hydrocarbon Receptor
CSF-1R
IAP
Myosin
Ephrin Receptor
Aromatase
AhR
DNA
PGE Synthase
Aminopeptidase
Protease-activated Receptor
Antifolate
ABC Transporter
Monoamine Transporter
Telomerase
Beta-Secretase
RSV
Discoidin Domain Receptor (DDR)
Monocarboxylate transporter
CETP
Glutaminase
IDO
DNA gyrase
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
Vasopressin Receptor
Acetyl-CoA Carboxylase
Platelet aggregation
NOD-like Receptor (NLR)
GRK
Bradykinin Receptor
Lipid
PAI-1
Melanocortin Receptor
NADPH-oxidase
CFTR
MLK
GNRH Receptor
LIM Kinase
NAMPT
Phosphorylase
ATP Citrate Lyase
BCRP
MNK
STING
Neprilysin
SGK
Dynamin
Ligands for Target Protein for PROTAC
Tie-2
SIK
PAFR
Glucagon Receptor
GlyT
OAT
Porcupine
ASK
GST
Carboxypeptidase
Adenylyl Cyclase
CRM1
Na+/Ca2+ Exchanger
AAK1
Neurotensin Receptor
PYK2
UGT
LDL
MAGL
DNA Alkylation
Angiotensin-converting Enzyme (ACE)
PAD
Wee1
CRFR
GPX
APC/C
p97
Thyroid hormone receptor(THR)
ROR
Progesterone Receptor
FLAP
MT Receptor
Guanylate cyclase
Transketolase
cGAS
MELK
Methionine Adenosyltransferase (MAT)
Ligand for E3 Ligase
Protease
CGRP Receptor
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
MyD88
Amino Acids and Derivatives
DprE1
DNA Alkylator/Crosslinker
Amylase
Bombesin Receptor
ACK1
Survivin
CD73
Decarboxylase
Pyroptosis
Hippo pathway
CRISPR/Cas9
GHSR
Aquaporin
Adenosine Deaminase
Gap Junction Protein
DAPK
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
NEDD8
Melatonin Receptor
Galectin
CaSR
VDAC
MTH1
Hexokinase
HCN Channel
PTEN
KSP
Drug-Linker Conjugates for ADC
Imidazoline Receptor
PKM
Apelin receptor
Transaminase
Arginase
Arrestin
IFNAR
Necroptosis
TOPK
Hck
Liver X Receptor
Haspin Kinase
Mucin
OXPHOS
PSMA
TSH Receptor
HuR
Oxytocin Receptor
Glyoxalase
GSNOR
NUDIX hydrolase
EBI2/GPR183
Sodium-dependent phosphate transporter
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
Vitamin
FOXO1
Prolyl Endopeptidase (PREP)
Na-K-Cl cotransporter
Molecular Glues
Integrase
Somatostatin
AIM2
hCE
KLF
Taste receptor
stilbene oxidase
Piezo Channel
Procollagen C Proteinase
Aconitase
Neuropeptide W
RAR/RXR 
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
FXR
Stemness kinase
RANKL/RANK
Adiponectin Receptor
Fas/FasL
FABP
PACAP
Anion Exchanger
Thioredoxin
PGC-1α
Glutathione reductase
MRGPR
GPCR19
CPT
GluCls
Fer/FerT kinase
Lysosomal Autophagy