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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively. Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
Antibacterial
5-HT Receptor
CDK
COX
Antibiotic
AChR
PI3K
EGFR
HIV Protease
Endogenous Metabolite
DNA/RNA Synthesis
Adrenergic Receptor
Dopamine Receptor
Calcium Channel
PDE
NF-κB
VEGFR
Epigenetic Reader Domain
Dehydrogenase
Histamine Receptor
Histone Methyltransferase
Cytochromes P450
Potassium Channel
Sodium Channel
Parasite
HDAC
Phosphatase
JAK
Antifungal
mTOR
Src
FLT
Microtubule Associated
Topoisomerase
TRP/TRPV Channel
SARS-CoV
PDGFR
Cholinesterase (ChE)
PARP
FGFR
PKC
Raf
Wnt/beta-catenin
Akt
STAT
p38 MAPK
Influenza Virus
HCV Protease
RAAS
ERK
c-Kit
GSK-3
Prostaglandin Receptor
MAO
GABA Receptor
c-Met/HGFR
Lipoxygenase
Bcr-Abl
ALK
TNF
NMDAR
MMP
Proteasome
Reactive Oxygen Species
Adenosine Receptor
GluR
Bcl-2 Family
DUB
HSP
Phospholipase
Ferroptosis
Aurora Kinase
Histone Demethylase
Virus Protease
TGF-beta/Smad
Tyrosinase
GPR
ROCK
iGluR
IL Receptor
MAPK
Ras
Transferase
Tyrosine Kinases
ATPase
HER
E1/E2/E3 Enzyme
CCR
Integrin
PKA
Casein Kinase
MEK
NO Synthase
Beta Amyloid
JNK
PPAR
Caspase
Antiviral
Monoamine Oxidase
Serine/threonin kinase
Carbonic Anhydrase
Serotonin Transporter
IκB/IKK
Reverse Transcriptase
Antioxidant
Mitophagy
Cysteine Protease
Androgen Receptor
DNA-PK
HBV
Mitochondrial Metabolism
HSV
AMPK
CXCR
Sirtuin
c-RET
Reductase
NOS
ROS
Norepinephrine
HIF
TAM Receptor
Estrogen/progestogen Receptor
RIP kinase
P2X Receptor
IGF-1R
P-gp
Estrogen Receptor/ERR
Serine Protease
CaMK
Histone Acetyltransferase
Nucleoside Antimetabolite/Analog
Gamma-secretase
Drug Metabolite
Glucosidase
TLR
HIF/HIF Prolyl-Hydroxylase
Interleukin
Trk receptor
FAK
Proton pump
Hedgehog/Smoothened
FAAH
Acyltransferase
c-Fms
PLK
S6 Kinase
Cannabinoid Receptor
Opioid Receptor
ATM/ATR
Neurokinin receptor
Syk
p53
Glucocorticoid Receptor
DPP-4
Endothelin Receptor
NOD
HMG-CoA Reductase
Pim
Chk
Fatty Acid Synthase
Kinesin
Chloride channel
DYRK
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Anti-infection
IRAK
LTR
NADPH
Rho
Leukotriene Receptor
LRRK2
transporter
Thrombin
Mdm2
LPL Receptor
BACE
Lipase
Factor Xa
Xanthine Oxidase
PDK
DNA Methyltransferase
Immunology/Inflammation related
Nrf2
Sigma receptor
PD-1/PD-L1
S1P Receptor
BTK
P2Y Receptor
PERK
Glutathione Peroxidase
Smo
cAMP
Kras
Hydroxylase
DHFR
MRP
PAK
Epoxide Hydrolase
Retinoid Receptor
Cholecystokinin Receptor
Glucokinase
OX Receptor
LPA Receptor
PI4K
Complement System
ROS Kinase
YAP
c-Myc
IRE1
Neuropeptide Y Receptor
ribosome
GTPase
Aryl Hydrocarbon Receptor
IAP
CSF-1R
Myosin
Ephrin Receptor
Aromatase
AhR
Antifolate
DNA
PGE Synthase
Aminopeptidase
Protease-activated Receptor
ABC Transporter
Monoamine Transporter
Telomerase
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ADC Cytotoxin
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CETP
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IDO
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Stearoyl-CoA Desaturase (SCD)
Vasopressin Receptor
Acetyl-CoA Carboxylase
Platelet aggregation
NOD-like Receptor (NLR)
GRK
DNA gyrase
Bradykinin Receptor
Lipid
PAI-1
Melanocortin Receptor
NADPH-oxidase
CFTR
MLK
GNRH Receptor
LIM Kinase
NAMPT
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BCRP
MNK
STING
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SGK
Dynamin
Ligands for Target Protein for PROTAC
Tie-2
PAFR
LDL
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Phosphorylase
GlyT
PAD
OAT
Porcupine
ASK
Carboxypeptidase
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CRM1
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AAK1
Neurotensin Receptor
PYK2
SIK
UGT
MAGL
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Wee1
CRFR
GST
GPX
APC/C
p97
Thyroid hormone receptor(THR)
ROR
Progesterone Receptor
FLAP
MT Receptor
Guanylate cyclase
cGAS
MELK
Methionine Adenosyltransferase (MAT)
Ligand for E3 Ligase
Protease
CGRP Receptor
Gap Junction Protein
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
Amino Acids and Derivatives
MyD88
DprE1
DNA Alkylator/Crosslinker
Amylase
MTH1
Bombesin Receptor
ACK1
Survivin
CD73
Decarboxylase
Pyroptosis
Hippo pathway
CRISPR/Cas9
Aquaporin
GHSR
Adenosine Deaminase
DAPK
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
NEDD8
Melatonin Receptor
Galectin
CaSR
VDAC
Hexokinase
HCN Channel
PTEN
KSP
Imidazoline Receptor
Apelin receptor
Transaminase
Arginase
Arrestin
IFNAR
Necroptosis
TOPK
Hck
Liver X Receptor
Haspin Kinase
OXPHOS
TSH Receptor
HuR
Oxytocin Receptor
PKM
GSNOR
NUDIX hydrolase
EBI2/GPR183
Glutaminyl Cyclase
gp120/CD4
Kisspeptin
FXR
FOXO1
Prolyl Endopeptidase (PREP)
Na-K-Cl cotransporter
Molecular Glues
Integrase
Somatostatin
Transketolase
AIM2
hCE
KLF
Drug-Linker Conjugates for ADC
Taste receptor
stilbene oxidase
RAR/RXR
Piezo Channel
Procollagen C Proteinase
Aconitase
Neuropeptide W
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Stemness kinase
RANKL/RANK
Adiponectin Receptor
Fas/FasL
FABP
PACAP
Anion Exchanger
Thioredoxin
Mucin
PSMA
Glutathione reductase
MRGPR
GPCR19
CPT
GluCls
Fer/FerT kinase
Lysosomal Autophagy
Glyoxalase
Sodium-dependent phosphate transporter
Vitamin
PGC-1α