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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively. Inhibitor library is a unique collection of 9730 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9730 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
CDK
COX
Antibiotic
AChR
PI3K
EGFR
Endogenous Metabolite
HIV Protease
DNA/RNA Synthesis
Adrenergic Receptor
Dopamine Receptor
NF-κB
PDE
Calcium Channel
VEGFR
Epigenetic Reader Domain
Histamine Receptor
Dehydrogenase
P450
Histone Methyltransferase
Potassium Channel
Sodium Channel
HDAC
JAK
Parasite
Phosphatase
Antifungal
mTOR
FLT
Src
Microtubule Associated
Topoisomerase
TRP/TRPV Channel
SARS-CoV
PDGFR
AChE
PARP
FGFR
PKC
Wnt/beta-catenin
Raf
Akt
HCV Protease
p38 MAPK
Influenza Virus
STAT
RAAS
ERK
c-Kit
GSK-3
MAO
Prostaglandin Receptor
GABA Receptor
Lipoxygenase
c-Met/HGFR
Bcr-Abl
ALK
TNF
MMP
NMDAR
Proteasome
Adenosine Receptor
BCL
Reactive Oxygen Species
GluR
Phospholipase
Ferroptosis
DUB
HSP
Aurora Kinase
BTK
Virus Protease
Kras
Histone Demethylase
Tyrosinase
TGF-beta/Smad
GPR
Tyrosine Kinases
CCR
Ras
Transferase
ROCK
iGluR
MAPK
HER
ATPase
IL Receptor
E1/E2/E3 Enzyme
MEK
Integrin
Casein Kinase
Beta Amyloid
NO Synthase
Caspase
Monoamine Oxidase
JNK
PKA
PPAR
Antiviral
Serine/threonin kinase
Serotonin Transporter
Carbonic Anhydrase
IκB/IKK
Reverse Transcriptase
DNA-PK
Antioxidant
Mitophagy
Cysteine Protease
HBV
Mitochondrial Metabolism
HSV
Androgen Receptor
Sirtuin
AMPK
CXCR
c-RET
Reductase
NOS
Norepinephrine
HIF
TAM Receptor
ADC Cytotoxin
Estrogen/progestogen Receptor
Serine Protease
RIP kinase
P2X Receptor
ROS
IGF-1R
P-gp
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
CaMK
Histone Acetyltransferase
Gamma-secretase
Glucosidase
Drug Metabolite
TLR
HIF/HIF Prolyl-Hydroxylase
Proton pump
Interleukin
Trk receptor
FAK
Hedgehog/Smoothened
FAAH
Acyltransferase
c-Fms
PLK
S6 Kinase
Cannabinoid Receptor
ATM/ATR
Neurokinin receptor
Syk
p53
Glucocorticoid Receptor
Opioid Receptor
DPP-4
NOD
HMG-CoA Reductase
Pim
Endothelin Receptor
Chk
Fatty Acid Synthase
Kinesin
Chloride channel
DYRK
Antifection
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
Thrombin
LTR
NADPH
Factor Xa
Rho
Leukotriene Receptor
LRRK2
transporter
Anti-infection
DNA Methyltransferase
IRAK
Mdm2
BACE
Lipase
Xanthine Oxidase
PDK
PD-1/PD-L1
LPL Receptor
Immunology/Inflammation related
S1P Receptor
P2Y Receptor
PERK
Glutathione Peroxidase
Smo
Nrf2
Hydroxylase
Sigma receptor
DHFR
MRP
PAK
Epoxide Hydrolase
cAMP
Retinoid Receptor
Complement System
Glucokinase
OX Receptor
LPA Receptor
PI4K
cholecystokinin
ROS Kinase
YAP
c-Myc
IRE1
Neuropeptide Y Receptor
GTPase
Aryl Hydrocarbon Receptor
CSF-1R
IAP
Myosin
Ephrin Receptor
ribosome
Aromatase
Antifolate
DNA
PGE Synthase
Aminopeptidase
Protease-activated Receptor
AhR
Telomerase
Beta-Secretase
RSV
Discoidin Domain Receptor (DDR)
Monocarboxylate transporter
CETP
ABC
IDO
DNA gyrase
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
Vasopressin Receptor
Acetyl-CoA Carboxylase
Platelet aggregation
NOD-like Receptor (NLR)
Glutaminase
GRK
Bradykinin Receptor
Lipid
PAI-1
Melanocortin Receptor
NADPH-oxidase
CFTR
MLK
GNRH Receptor
NAMPT
Phosphorylase
ATP Citrate Lyase
BCRP
MNK
STING
Neprilysin
SGK
Dynamin
Ligands for Target Protein for PROTAC
Tie-2
SIK
PAFR
LDL
Glucagon Receptor
GlyT
PAD
OAT
Porcupine
ASK
GST
Carboxypeptidase
Adenylyl cyclase
CRM1
Na+/Ca2+ Exchanger
LIM Kinase
Neurotensin Receptor
PYK2
UGT
Guanylate cyclase
APC
MAGL
DNA Alkylation
Angiotensin-converting Enzyme (ACE)
CRFR
GPX
p97
Thyroid hormone receptor(THR)
ROR
DNA Alkylator/Crosslinker
Progesterone Receptor
FLAP
MT Receptor
AAK1 (AP2 associated kinase 1)
Transketolase
Wee1
cGAS
MELK
Methionine Adenosyltransferase (MAT)
Protease
Ligand for E3 Ligase
Gap Junction Protein
Melanin-concentrating Hormone Receptor (MCHR)
PROTACs
MALT
DprE1
MyD88
Amino Acids and Derivatives
Amylase
MTH1
Bombesin Receptor
ACK
Survivin
CD73
Decarboxylase
Hippo pathway
CRISPR/Cas9
Aquaporin
GHSR
Adenosine deaminase
CGRP Receptor
DAPK
BMI-1
advanced glycation end products
NPC1L1
CD38
NEDD8
TOPK
Melatonin Receptor
Galectin
CaSR
VDAC
Hexokinase
HCN Channel
PTEN
KSP
Pyroptosis
Drug-Linker Conjugates for ADC
Imidazoline Receptor
PKM
Apelin receptor
CAT
Transaminase
Arginase
IFNAR
Arrestin
Necroptosis
Hck
Liver X Receptor
Haspin Kinase
Mucin
OXPHOS
PSMA
HuR
Oxytocin Receptor
Glyoxalase
GSNOR
NUDIX hydrolase
EBI2/GPR183
Sodium-dependent phosphate transporter
gp120/CD4
Kisspeptin
FXR
Vitamin
FOXO1
Prolyl Endopeptidase (PREP)
Na-K-Cl cotransporter
Molecular Glues
Integrase
Somatostatin
AIM2
hCE
TSH Receptor
KLF
Taste receptor
stilbene oxidase
Piezo Channel
Procollagen C Proteinase
Neuropeptide W
aconitase
RAR/RXR 
Cell wall
LHRH
VDA
OCT
N-Acetylglucosaminyltransferase
Stemness kinase
RANKL/RANK
Annexin A
Adiponectin receptor
Fas/FasL
FABP
PACAP
Anion Exchanger
Thioredoxin
PGC-1α
Glutathione reductase
MRGPR
GPCR19
CPT
GluCls
Fer/FerT kinase
lysosomal autophagy