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Inhibitor Library

Catalog No. L2000
  Library Compound List   Excel SDF

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively.

Inhibitor library is a unique collection of 5700 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
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Product Description

  • A unique collection of 5700 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2000)

Library Composition

Apoptosis (652)
Autophagy (495)
Antibacterial (198)
5-HT Receptor (143)
CDK (141)
COX (135)
PI3K (134)
NF-κB (133)
Endogenous Metabolite (130)
DNA/RNA Synthesis (128)
HIV Protease (127)
AChR (123)
EGFR (122)
VEGFR (117)
Antibiotic (115)
Epigenetic Reader Domain (98)
Dopamine Receptor (94)
Calcium Channel (91)
P450 (91)
Dehydrogenase (91)
HDAC (90)
PDE (90)
Histone Methyltransferase (84)
Histamine Receptor (81)
Parasite (78)
Adrenergic Receptor (77)
Src (76)
JAK (75)
FLT (75)
PDGFR (73)
Influenza Virus (73)
mTOR (70)
Potassium Channel (69)
Phosphatase (67)
Antifungal (65)
Sodium Channel (65)
FGFR (62)
AChE (59)
STAT (59)
Raf (58)
Topoisomerase (58)
c-Kit (57)
Microtubule Associated (56)
PARP (56)
p38 MAPK (55)
Akt (55)
ERK (54)
c-Met/HGFR (53)
RAAS (53)
HCV Protease (53)
PKC (52)
TRP/TRPV Channel (52)
Ferroptosis (52)
SARS-CoV (51)
Ras (48)
Reactive Oxygen Species (48)
Proteasome (48)
ALK (47)
TNF (46)
GABA Receptor (46)
BCL (45)
Bcr-Abl (45)
Wnt/beta-catenin (44)
GSK-3 (42)
MAO (42)
Prostaglandin Receptor (41)
MMP (40)
Lipoxygenase (39)
Mitophagy (39)
HSP (38)
TGF-beta/Smad (38)
Aurora Kinase (37)
JNK (35)
DNA-PK (35)
Adenosine Receptor (35)
E1/E2/E3 Enzyme (35)
Tyrosinase (35)
Tyrosine Kinases (35)
Virus Protease (35)
DUB (34)
MEK (34)
IL Receptor (33)
Monoamine Oxidase (32)
NO Synthase (32)
Reverse Transcriptase (32)
BTK (32)
Beta Amyloid (32)
Phospholipase (32)
GluR (31)
PPAR (31)
HSV (31)
ATPase (31)
IκB/IKK (31)
iGluR (31)
ROCK (30)
P2 Receptor (30)
NMDAR (30)
TAM Receptor (30)
Mitochondrial Metabolism (29)
HER (29)
Glucokinase (29)
Histone Demethylase (29)
Caspase (29)
Casein Kinase (28)
GPR (28)
ROS (28)
MAPK (28)
Serine/threonin kinase (28)
Serotonin Transporter (28)
HBV (27)
Nucleoside Antimetabolite/Analog (26)
Sirtuin (26)
P-gp (26)
PKA (26)
HIF/HIF Prolyl-Hydroxylase (26)
Interleukin (26)
CCR (26)
c-RET (26)
Integrin (25)
Histone Acetyltransferase (25)
Transferase (25)
AMPK (25)
S6 Kinase (24)
Androgen Receptor (24)
Gamma-secretase (24)
Trk receptor (24)
Proton pump (23)
CaMK (23)
Cysteine Protease (23)
Carbonic Anhydrase (22)
p53 (22)
IGF-1R (22)
HIF (22)
FAK (22)
Serine Protease (21)
Estrogen/progestogen Receptor (21)
Opioid Receptor (21)
TLR (21)
NOS (20)
DPP-4 (20)
ATM/ATR (20)
Hedgehog/Smoothened (20)
Drug Metabolite (20)
Estrogen Receptor/ERR (20)
PLK (20)
Indoleamine 2,3-Dioxygenase (IDO) (19)
Reductase (19)
Chk (19)
Norepinephrine (19)
Glucocorticoid Receptor (18)
CXCR (18)
Syk (18)
Chloride channel (18)
HMG-CoA Reductase (18)
c-Fms (18)
FAAH (18)
RIP kinase (18)
Kinesin (18)
LRRK2 (17)
LPL Receptor (16)
Fatty Acid Synthase (16)
SGLT (16)
Cannabinoid Receptor (16)
Acyltransferase (15)
NADPH (15)
Antifection (14)
Anti-infection (14)
transporter (14)
S1P Receptor (14)
Aryl Hydrocarbon Receptor (14)
Endothelin Receptor (14)
PDK (14)
OX Receptor (14)
Lipase (13)
Rho (13)
PAK (13)
P2X Receptor (13)
NOD (13)
Thrombin (13)
DNA Methyltransferase (13)
Smo (13)
IAP (12)
Neurokinin receptor (12)
Epoxide Hydrolase (12)
Glutathione Peroxidase (12)
c-Myc (12)
IRE1 (12)
Antioxidant (12)
Mdm2 (12)
PI4K (11)
LTR (11)
CSF-1R (11)
Retinoid Receptor (11)
BACE (11)
Pim (11)
MRP (11)
ribosome (11)
NOD-like Receptor (NLR) (11)
AhR (11)
Leukotriene Receptor (11)
Hydroxylase (11)
PERK (11)
IRAK (11)
Antiviral (11)
Antifolate (10)
IDO (10)
Factor Xa (10)
Isocitrate Dehydrogenase (IDH) (10)
Xanthine Oxidase (10)
Aminopeptidase (10)
PD-1/PD-L1 (9)
LPA Receptor (9)
PGE Synthase (9)
Ephrin Receptor (9)
Beta-Secretase (9)
Nrf2 (9)
Sigma receptor (9)
Stearoyl-CoA Desaturase (SCD) (9)
NAMPT (8)
RSV (8)
PAD (8)
Acetyl-CoA Carboxylase (8)
Telomerase (8)
STING (8)
Protease-activated Receptor (8)
Phosphorylase (7)
Vasopressin Receptor (7)
DYRK (7)
SGK (7)
DNA gyrase (7)
Discoidin Domain Receptor (DDR) (7)
DHFR (7)
Monocarboxylate transporter (7)
PAI-1 (7)
ABC (7)
BCRP (7)
Complement System (7)
MLK (7)
ATP Citrate Lyase (7)
Myosin (7)
p97 (6)
MNK (6)
UGT (6)
GNRH Receptor (6)
Tie-2 (6)
cAMP (6)
GTPase (6)
Neprilysin (6)
LIM Kinase (6)
Na+/Ca2+ Exchanger (6)
Immunology/Inflammation related (6)
ASK (6)
Neuropeptide Y Receptor (6)
Porcupine (6)
SIK (5)
Platelet aggregation (5)
PTEN (5)
TOPK (5)
PYK2 (5)
Bradykinin Receptor (5)
ACK (5)
BMI-1 (5)
cGAS (5)
YAP (5)
NADPH-oxidase (5)
Glutaminase (5)
GlyT (5)
GRK (5)
Guanylate cyclase (5)
Dynamin (5)
DprE1 (5)
DNA Alkylator/Crosslinker (5)
CRM1 (5)
CRISPR/Cas9 (5)
Melanocortin Receptor (5)
cholecystokinin (5)
Monoamine Transporter (5)
DNA (5)
NPC1L1 (5)
CETP (5)
DNA Alkylation (4)
APC (4)
advanced glycation end products (4)
Arginase (4)
Aromatase (4)
GPX (4)
Decarboxylase (4)
GST (4)
Adenosine deaminase (4)
MAGL (4)
Lipid (4)
OAT (4)
Progesterone Receptor (4)
MELK (4)
VDAC (4)
FLAP (4)
IFNAR (3)
Hippo pathway (3)
KSP (3)
Hexokinase (3)
NEDD8 (3)
OXPHOS (3)
Thyroid hormone receptor(THR) (3)
PAFR (3)
Liver X Receptor (3)
Free radical scavengers (3)
Carboxypeptidase(CPG2) (3)
Hck (3)
Wee1 (3)
PKM (3)
MTH1 (3)
CFTR (3)
Gap Junction Protein (3)
Neurotensin Receptor (3)
CAT (3)
Bombesin Receptor (3)
Adenylyl cyclase (2)
FXR (2)
Galectin (2)
Survivin (2)
Amino Acids and Derivatives (2)
GHSR (2)
Glucagon Receptor (2)
Haspin Kinase (2)
EBI2/GPR183 (2)
Aquaporin (2)
MT Receptor (2)
Pyroptosis (2)
CRFR (2)
ROR (2)
KLF (2)
MALT (2)
Melatonin Receptor (2)
Integrase (2)
MyD88 (2)
VDA (1)
aconitase (1)
FOXO1 (1)
Protease (1)
CGRP Receptor (1)
Melanin-concentrating Hormone Receptor (MCHR) (1)
TSH Receptor (1)
FABP (1)
Fer/FerT kinase (1)
N-Acetylglucosaminyltransferase (1)
Somatostatin (1)
lysosomal autophagy (1)
Transaminase (1)
Taste receptor (1)
Anion Exchanger (1)
Stemness kinase (1)
stilbene oxidase (1)
HCN Channel (1)
CaSR (1)
GSNOR (1)
Oxytocin Receptor (1)
hCE (1)
Thioredoxin (1)
Thrombopoietin Receptor (1)
LDL (1)
GPCR19 (1)
gp120/CD4 (1)
Apelin receptor (1)
Na-K-Cl cotransporter (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE