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TargetMol | Compound Library

Inhibitor Library

Catalog No. L2000

Cell signalingis part of any communication process that governs basic activities of cells and coordinates all cell actions. The ability of cells to perceive and correctly respond to their microenvironment is the basis of development,tissue repair, andimmunity, as well as normal tissuehomeostasis. Errors in signaling interactions and cellularinformation processingare responsible for diseases such as cancer,auto-immunity, and diabetes.By understanding cell signaling, diseases may be treated more effectively. Inhibitor library is a unique collection of 8328 compounds, each of which has clear inhibitory targets. It is an effective tool for research in cell signaling pathways and related diseases, and high throughput screening and high content screening for new drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2000

Inhibitor Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 8328 inhibitors for research in cell signaling, high throughput screening (HTS) and high content screening (HCS) for new drugs;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Covers various major targets including MAPK, PI3K, JAK, HDAC, VEGFR, CDK, etc.;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
5-HT Receptor
CDK
COX
PI3K
Endogenous Metabolite
Antibiotic
EGFR
HIV Protease
AChR
DNA/RNA Synthesis
VEGFR
PDE
NF-κB
Epigenetic Reader Domain
Dopamine Receptor
Dehydrogenase
Adrenergic Receptor
P450
Histone Methyltransferase
Histamine Receptor
HDAC
Parasite
Potassium Channel
Calcium Channel
JAK
mTOR
Antifungal
FLT
Phosphatase
Sodium Channel
Src
PDGFR
Microtubule Associated
Topoisomerase
TRP/TRPV Channel
PARP
FGFR
Raf
AChE
Wnt/beta-catenin
c-Kit
ERK
SARS-CoV
PKC
Influenza Virus
Akt
p38 MAPK
GSK-3
HCV Protease
STAT
MAO
Ras
c-Met/HGFR
RAAS
Bcr-Abl
Prostaglandin Receptor
Proteasome
TNF
Lipoxygenase
Reactive Oxygen Species
Aurora Kinase
Ferroptosis
ALK
GABA Receptor
MMP
Phospholipase
BCL
HSP
BTK
DUB
TGF-beta/Smad
Virus Protease
Transferase
Adenosine Receptor
ROCK
Casein Kinase
Tyrosine Kinases
MAPK
Tyrosinase
NMDAR
MEK
E1/E2/E3 Enzyme
Monoamine Oxidase
ATPase
GluR
Histone Demethylase
Serine/threonin kinase
Caspase
Beta Amyloid
NO Synthase
HER
iGluR
HSV
IL Receptor
DNA-PK
JNK
PKA
CCR
Reverse Transcriptase
Carbonic Anhydrase
PPAR
Sirtuin
GPR
c-RET
Mitophagy
Serotonin Transporter
Cysteine Protease
Mitochondrial Metabolism
AMPK
IκB/IKK
TAM Receptor
Antioxidant
HBV
Integrin
Nucleoside Antimetabolite/Analog
IGF-1R
NOS
Gamma-secretase
P-gp
HIF
RIP kinase
ROS
Serine Protease
Drug Metabolite
CXCR
Norepinephrine
Glucosidase
TLR
Histone Acetyltransferase
c-Fms
S6 Kinase
HIF/HIF Prolyl-Hydroxylase
Estrogen/progestogen Receptor
Reductase
CaMK
Androgen Receptor
PLK
Proton pump
Estrogen Receptor/ERR
Interleukin
Trk receptor
P2X Receptor
FAAH
Pim
Hedgehog/Smoothened
Antiviral
Syk
DPP-4
Acyltransferase
ATM/ATR
FAK
p53
Glucocorticoid Receptor
Chk
Kinesin
Fatty Acid Synthase
Indoleamine 2,3-Dioxygenase (IDO)
Opioid Receptor
SGLT
Cannabinoid Receptor
NOD
HMG-CoA Reductase
Thrombin
DYRK
NADPH
Anti-infection
IRAK
Mdm2
Chloride channel
Xanthine Oxidase
LRRK2
transporter
PDK
DNA Methyltransferase
LPL Receptor
Lipase
Rho
Antifection
Neurokinin receptor
S1P Receptor
Factor Xa
MRP
Smo
PAK
Endothelin Receptor
Nrf2
Epoxide Hydrolase
Hydroxylase
PD-1/PD-L1
P2Y Receptor
LTR
BACE
PERK
Glutathione Peroxidase
PI4K
YAP
Glucokinase
CSF-1R
Immunology/Inflammation related
IRE1
OX Receptor
Retinoid Receptor
ribosome
Aromatase
Complement System
DHFR
GTPase
c-Myc
Leukotriene Receptor
Myosin
cAMP
Sigma receptor
ROS Kinase
Aryl Hydrocarbon Receptor
Neuropeptide Y Receptor
PGE Synthase
Aminopeptidase
Ephrin Receptor
LPA Receptor
Protease-activated Receptor
DNA gyrase
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
Lipid
Beta-Secretase
Discoidin Domain Receptor (DDR)
AhR
NOD-like Receptor (NLR)
Monocarboxylate transporter
CETP
Antifolate
IDO
DNA
PAI-1
Acetyl-CoA Carboxylase
cholecystokinin
Glutaminase
IAP
GRK
Vasopressin Receptor
Telomerase
ATP Citrate Lyase
MNK
STING
SGK
MLK
NAMPT
Phosphorylase
BCRP
Porcupine
ASK
RSV
Neprilysin
Platelet aggregation
NADPH-oxidase
CFTR
Adenylyl cyclase
Dynamin
Na+/Ca2+ Exchanger
Tie-2
ABC
SIK
UGT
GlyT
MAGL
Angiotensin-converting Enzyme (ACE)
PAD
Wee1
Carboxypeptidase
GPX
p97
Thyroid hormone receptor(THR)
DNA Alkylator/Crosslinker
Progesterone Receptor
FLAP
LDL
AAK1 (AP2 associated kinase 1)
Guanylate cyclase
DNA Alkylation
OAT
MELK
GST
NPC1L1
CRM1
DprE1
LIM Kinase
Neurotensin Receptor
PYK2
PAFR
MTH1
APC
Bombesin Receptor
ACK
Survivin
Decarboxylase
cGAS
CRFR
Methionine Adenosyltransferase (MAT)
Hippo pathway
Melanocortin Receptor
CRISPR/Cas9
Aquaporin
Adenosine deaminase
BMI-1
advanced glycation end products
MALT
ROR
NEDD8
MyD88
Amino Acids and Derivatives
TOPK
Galectin
GNRH Receptor
VDAC
Amylase
MT Receptor
Glucagon Receptor
Bradykinin Receptor
PTEN
KSP
CD73
Protease
CGRP Receptor
DAPK
Imidazoline Receptor
PKM
CAT
Transaminase
Arginase
IFNAR
Necroptosis
Melatonin Receptor
CaSR
Hck
Liver X Receptor
Haspin Kinase
Hexokinase
HCN Channel
OXPHOS
Pyroptosis
Ligand for E3 Ligase
Gap Junction Protein
Melanin-concentrating Hormone Receptor (MCHR)
GSNOR
CD38
NUDIX hydrolase
EBI2/GPR183
Arrestin
gp120/CD4
FXR
FOXO1
Prolyl Endopeptidase (PREP)
Na-K-Cl cotransporter
Integrase
AIM2
hCE
KLF
Oxytocin Receptor
GHSR
Apelin receptor
Taste receptor
stilbene oxidase
Ligands for Target Protein for PROTAC
Procollagen C Proteinase
aconitase
Neuropeptide W
RAR/RXR 
Cell wall
VDA
OCT
N-Acetylglucosaminyltransferase
Stemness kinase
RANKL/RANK
Annexin A
Adiponectin receptor
Fas/FasL
FABP
Anion Exchanger
Thioredoxin
PGC-1α
Somatostatin
Glutathione reductase
GPCR19
CPT
GluCls
TSH Receptor
HuR
Fer/FerT kinase
lysosomal autophagy

Keywords