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Compound Libraries FDA-approved Drug Library

FDA-approved Drug Library

Catalog No. L4200
  Library Compound List   Excel SDF

All compounds in FDA approved drug library have well-characterized biological activity, clear targets, safety, and bioavailability – properties which could dramatically accelerate drug development and optimization. It is an effective and ideal tool for drug repurposing and cell differentiation induction. Detailed information on each compound in this library can help scientists quickly finish drug screening or make quick judgement on cell differentiation mechanism, and create conditions for further investigation on the mechanism of action.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 7015.00
250 μL * 10 mM (in DMSO) 13790.00
1 mg 13790.00
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Product Description

  • A unique collection of 1403 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research evidence and clinical trials;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas: oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry, analgesia etc
  • Structurally diverse, medicinally active, and cell permeable;
  • Rich documentation with structure, target, IC50 value and biological activity description;
  • NMR and HPLC/LCMS validated to ensure high purity.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging and Storage

  • Powder or pre-dissolved DMSO solutions in 96 well plate with optional 2D barcode
  • Shipped with blue ice.
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Library Composition

Adrenergic Receptor (81)
AChR (77)
5-HT Receptor (74)
Dopamine Receptor (50)
Histamine Receptor (46)
COX (45)
DNA/RNA Synthesis (43)
Potassium Channel (38)
Estrogen/progestogen Receptor (35)
Sodium Channel (35)
Antibacterial (33)
GR (32)
Topoisomerase (24)
ribosome (20)
PDE (20)
Calcium Channel (20)
Dehydrogenase (19)
Norepinephrine (19)
RAAS (19)
Vitamin (19)
VEGFR (18)
GABA Receptor (18)
Antifection (18)
HIV Protease (17)
Autophagy (16)
Antibiotic (15)
Carbonic Anhydrase (15)
Microtubule Associated (14)
HCV Protease (13)
MRP (13)
PPAR (12)
EGFR (12)
DNA Alkylation (12)
Reverse Transcriptase (12)
c-Kit (11)
PDGFR (11)
P450 (11)
MAO (9)
DHFR (9)
ATPase (9)
Androgen Receptor (8)
Proton pump (8)
Tyrosine Kinases (8)
Src (8)
Retinoid Receptor (7)
Raf (7)
Opioid Receptor (7)
ROS (7)
TNF (7)
Antifungal (7)
ABC (7)
Bcr-Abl (7)
DNA gyrase (7)
FGFR (7)
GluR (7)
HDAC (7)
NADPH (7)
NMDAR (7)
NF-κB (6)
Prostaglandin Receptor (6)
HMG-CoA Reductase (6)
Amino Acids and Derivatives (6)
Thrombin (6)
Transferase (5)
Proteasome (5)
Annexin A (5)
CaMK (5)
FLT (5)
Factor Xa (5)
P2 Receptor (5)
PI3K (4)
Neurokinin 1 (4)
NOS (4)
HBV (4)
MMP (4)
IL Receptor (4)
JAK (4)
Lipoxygenase (4)
DNA Methyltransferase (4)
DPP-4 (4)
CAT (4)
CDK (4)
ALK (4)
Thyroid hormone receptor(THR) (4)
STAT (3)
SGLT (3)
Phosphatase (3)
Phospholipase (3)
Reductase (3)
Tyrosinase (3)
AhR (3)
Arginase (3)
Aromatase (3)
CFTR (3)
Fatty Acid Synthase (3)
Endothelin Receptor (3)
Glutathione reductase (3)
Glucocorticoid Receptor (3)
Influenza Virus (3)
Integrin (3)
MPO (3)
MEK (3)
GST (3)
Hedgehog/Smoothened (3)
mTOR (3)
Na-K-Cl cotransporter (3)
PKC (3)
PARP (3)
Nucleoside Antimetabolite/Analog (2)
HER (2)
HIF (2)
HSV (2)
MAPK (2)
IGF-1R (2)
LDL (2)
Lipid (2)
Glucokinase (2)
GluCls (2)
Free radical scavengers (2)
FXR (2)
Decarboxylase (2)
c-Met/HGFR (2)
c-RET (2)
Chk (2)
Chloride channel (2)
Cell wall (2)
BTK (2)
Adenosine Receptor (2)
Rho (2)
TAM Receptor (2)
TLR (2)
TRP/TRPV Channel (2)
UGT (2)
Vasopressin Receptor (2)
VDA (1)
Telomerase (1)
TGF-beta/Smad (1)
Sigma receptor (1)
Sirtuin (1)
Syk (1)
ROCK (1)
S1P Receptor (1)
S6 Kinase (1)
Serine Protease (1)
Phosphorylase (1)
Wnt/beta-catenin (1)
ACK (1)
ATM/ATR (1)
ATP Citrate Lyase (1)
AMPK (1)
BCL (1)
CETP (1)
CCR (1)
Caspase (1)
CaSR (1)
CXCR (1)
Ferroptosis (1)
DUB (1)
Epigenetic Reader Domain (1)
Gap Junction Protein (1)
GlyT (1)
GPR (1)
LTR (1)
lysosomal autophagy (1)
IκB/IKK (1)
Integrase (1)
Monoamine Transporter (1)
Melatonin Receptor (1)
Hydrogenase (1)
Hydroxylase (1)
IAP (1)
HSP (1)
Histone Demethylase (1)
Histone Methyltransferase (1)
GRK (1)
GSK-3 (1)
OAT (1)
NPC1L1 (1)
Nrf2 (1)
NKCC (1)
NADPH-oxidase (1)
MTH1 (1)
PDK (1)
PED (1)
PKM (1)
Platelet aggregation (1)
PLK (1)
Protease-activated Receptor (1)