Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 3150 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L2150

Anti-Cancer Drug Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 3150 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Antibacterial
COX
Dopamine Receptor
Histamine Receptor
Antibiotic
DNA/RNA Synthesis
Sodium Channel
Calcium Channel
VEGFR
Potassium Channel
EGFR
AChR
Parasite
PI3K
Glucocorticoid Receptor
Reactive Oxygen Species
P450
Topoisomerase
CDK
FLT
HIV Protease
NF-κB
JAK
PDGFR
PPAR
GABA Receptor
c-Kit
FGFR
HDAC
Microtubule Associated
Estrogen/progestogen Receptor
Ferroptosis
Dehydrogenase
Antifungal
c-Met/HGFR
Estrogen Receptor/ERR
mTOR
Prostaglandin Receptor
Mitophagy
Influenza Virus
Src
Nucleoside Antimetabolite/Analog
Tyrosine Kinases
Androgen Receptor
SARS-CoV
iGluR
Bcr-Abl
Adenosine Receptor
PDE
Raf
GPR
ADC Cytotoxin
HER
Serotonin Transporter
TRP/TRPV Channel
Akt
ATPase
PARP
Opioid Receptor
Norepinephrine
Aurora Kinase
HSP
p38 MAPK
Virus Protease
PKC
HSV
Epigenetic Reader Domain
P-gp
ALK
MEK
TNF
Proton pump
NMDAR
BTK
DNA Alkylator/Crosslinker
RAAS
Phosphatase
ERK
ROS
c-RET
HIF/HIF Prolyl-Hydroxylase
Histone Methyltransferase
HBV
Endothelin Receptor
Trk receptor
HCV Protease
GSK-3
Drug Metabolite
MMP
AMPK
Carbonic Anhydrase
Progesterone Receptor
Caspase
BCL
CXCR
SGLT
STAT
c-Fms
Chk
Retinoid Receptor
TAM Receptor
Proteasome
DNA-PK
GNRH Receptor
E1/E2/E3 Enzyme
Guanylate cyclase
DNA Alkylation
IL Receptor
Reverse Transcriptase
FAK
p53
S1P Receptor
LPL Receptor
MAO
P2X Receptor
TGF-beta/Smad
HIF
CFTR
Transferase
DHFR
MRP
PKA
Antifolate
Gamma-secretase
Mitochondrial Metabolism
Hedgehog/Smoothened
GluR
Lipoxygenase
IGF-1R
Interleukin
Neurokinin receptor
HMG-CoA Reductase
Monoamine Oxidase
Antioxidant
P2Y Receptor
Wnt/beta-catenin
ROCK
IAP
Vasopressin Receptor
AChE
TLR
Nrf2
PLK
Cannabinoid Receptor
Syk
ROS Kinase
Mdm2
Chloride channel
CSF-1R
Indoleamine 2,3-Dioxygenase (IDO)
ATM/ATR
Beta Amyloid
S6 Kinase
NADPH
JNK
Antifection
Smo
CCR
CaMK
Antiviral
Kras
Phospholipase
DNA Methyltransferase
Sigma receptor
Kinesin
Integrin
ABC
Glucagon Receptor
Monoamine Transporter
OX Receptor
DNA
Sirtuin
Casein Kinase
Ligand for E3 Ligase
Aromatase
cholecystokinin
Thrombin
Histone Demethylase
Glutathione Peroxidase
Pim
Leukotriene Receptor
RIP kinase
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
IRAK
NO Synthase
IFNAR
Tie-2
Serine Protease
FXR
Molecular Glues
DPP-4
Fatty Acid Synthase
PGE Synthase
GPCR19
Ephrin Receptor
GHSR
Hydroxylase
NOD
Tyrosinase
Amino Acids and Derivatives
YAP
LTR
Melatonin Receptor
CaSR
Serine/threonin kinase
Aryl Hydrocarbon Receptor
IDO
Annexin A
DNA gyrase
Neuropeptide Y Receptor
Somatostatin
Xanthine Oxidase
KSP
Wee1
STING
Aminopeptidase
CRFR
ribosome
Melanocortin Receptor
PDK
Oxytocin Receptor
CGRP Receptor
Ras
AhR
PD-1/PD-L1
PROTACs
NOS
Monocarboxylate transporter
ROR
CRM1
Reductase
Rho
Cysteine Protease
Liver X Receptor
NAMPT
PYK2
UGT
MT Receptor
Na-K-Cl cotransporter
Hexokinase
DUB
PSMA
MAPK
OAT
Free radical scavengers
transporter
RSV
GST
Adenosine deaminase
Protease-activated Receptor
NOD-like Receptor (NLR)
CAT
NEDD8
Ligands for Target Protein for PROTAC
Arginase
Cell wall
PERK
VDA
Factor Xa
Vitamin
IRE1
LDL
Glucosidase
PROTAC Linker
HCN Channel
Telomerase
ATP Citrate Lyase
BCRP
Beta-Secretase
Acyltransferase
Porcupine
CD73
Decarboxylase
Drug-Linker Conjugates for ADC
LPA Receptor
Gap Junction Protein
Discoidin Domain Receptor (DDR)
p97
MLK
Imidazoline Receptor
advanced glycation end products
NPC1L1
Hydrogenase
MALT
BACE
Na+/Ca2+ Exchanger
DYRK
RAR/RXR 
Lipase
TOPK
GTPase
c-Myc
Galectin
Kisspeptin
N-Acetylglucosaminyltransferase
Hck
Neurotensin Receptor
Glucokinase
Glutaminase
Stemness kinase
Immunology/Inflammation related
Myosin
Adiponectin receptor
PAFR
MTH1
GRK
GlyT
Anion Exchanger
Thioredoxin
FAAH
PAD
ACK
cAMP
Thrombopoietin Receptor
Lipid
Glutathione reductase
MNK
Survivin
Histone Acetyltransferase
ASK
GluCls
PAI-1
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
Neprilysin
PI4K
KLF
Aquaporin
SGK
Complement System
Platelet aggregation
NADPH-oxidase
BMI-1

Keywords