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TargetMol | Compound Library

Anti-Cancer Drug Library

Catalog No. L2150

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 3080 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2150

Anti-Cancer Drug Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3080 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Antibacterial
COX
Dopamine Receptor
Histamine Receptor
Antibiotic
DNA/RNA Synthesis
Sodium Channel
Calcium Channel
Potassium Channel
VEGFR
EGFR
AChR
Parasite
PI3K
Glucocorticoid Receptor
Reactive Oxygen Species
P450
FLT
HIV Protease
Topoisomerase
CDK
NF-κB
PDGFR
PPAR
GABA Receptor
JAK
c-Kit
FGFR
HDAC
Ferroptosis
Prostaglandin Receptor
Estrogen/progestogen Receptor
Antifungal
mTOR
Microtubule Associated
c-Met/HGFR
Dehydrogenase
Mitophagy
Influenza Virus
Estrogen Receptor/ERR
Src
Nucleoside Antimetabolite/Analog
iGluR
SARS-CoV
Adenosine Receptor
Tyrosine Kinases
Androgen Receptor
PDE
GPR
Opioid Receptor
Bcr-Abl
Raf
Serotonin Transporter
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ATPase
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p38 MAPK
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MEK
TNF
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HSP
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ALK
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GSK-3
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AMPK
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GNRH Receptor
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Progesterone Receptor
Retinoid Receptor
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cholecystokinin
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DNA
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Serine Protease
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ribosome
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transporter
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Aquaporin
SGK
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NADPH-oxidase
BMI-1

Keywords