Home Tools
Log in
Products Inhibitors Libraries Recombinant Proteins Kits Services Contact Us
Cart
Peptides Monoclonal Antibodies Dye Reagents PROTAC Virtual Screening TargetMol Kits Cell Counting Kit-8 (CCK-8) Inhibitor Cocktails Natural Products Phenols Alkaloids Flavonoids
Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK
Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library
TargetMol
Cytokines and Growth Factors •   Cytokines •   Growth Factors Receptor Proteins •   Fc Receptors •   Cytokines and Growth Factor Receptors
CD Proteins •   T Cell CD Proteins •   B Cell CD Proteins Immune Checkpoint Proteins •   Co-inhibitory Immune Checkpoint Proteins •   Co-stimulatory Immune Checkpoint Proteins
CAR-T Therapy Target Proteins •   Hematologic Malignancies Target Proteins •   Solid Tumors Target Proteins Enzymes •   Oxidoreductases,EC 1 •   Transferases,EC 2
Viral Proteins •   Coronavirus (CoV) Proteins •   Influenza Proteins Fluorescent Proteins Others

Anti-Cancer Drug Library

Catalog No. L2150
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 3159 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
Get quote

Product Description

  • A unique collection of 3159 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L2150)

Publications Cited TargetMol Libraries

1. Cell Stem Cell. 2022 Apr 29(4) 545–558. 2. Science Bulletin. 2022. 3. Science Translational Medicine. 2022, 14(656): eabn3231. 4. Science Advances. 2023, 9(9): eade3760. 5. Nature. 2020, 582: 289-293. 6. Nature Biotechnology. 2021, 39(11): 1444-1452. 7. Nature Communications. 2022, 13(1): 1-15.. 8. Nature Communications. 2023, 14(1): 1020.. 9. Nature Communications. 2023, 14(1): 2756..
Hide

Library Composition

Autophagy (442)
Apoptosis (419)
5-HT Receptor (203)
Endogenous Metabolite (187)
Adrenergic Receptor (171)
Antibacterial (150)
COX (137)
Dopamine Receptor (130)
Histamine Receptor (126)
Antibiotic (123)
DNA/RNA Synthesis (121)
Sodium Channel (97)
Calcium Channel (90)
Potassium Channel (86)
VEGFR (82)
EGFR (77)
AChR (72)
Parasite (68)
Reactive Oxygen Species (66)
PI3K (66)
Glucocorticoid Receptor (62)
P450 (60)
FLT (56)
CDK (54)
HIV Protease (54)
NF-κB (54)
Topoisomerase (54)
PDGFR (53)
PPAR (53)
GABA Receptor (52)
JAK (48)
c-Kit (48)
Ferroptosis (47)
FGFR (46)
HDAC (46)
Prostaglandin Receptor (42)
Microtubule Associated (42)
mTOR (42)
Estrogen/progestogen Receptor (41)
Antifungal (41)
c-Met/HGFR (40)
Dehydrogenase (39)
Mitophagy (38)
Estrogen Receptor/ERR (38)
Influenza Virus (38)
Src (35)
Nucleoside Antimetabolite/Analog (34)
iGluR (33)
SARS-CoV (32)
Adenosine Receptor (31)
Androgen Receptor (31)
Tyrosine Kinases (31)
GPR (30)
PDE (30)
Opioid Receptor (29)
Bcr-Abl (29)
Raf (28)
Serotonin Transporter (25)
HER (25)
ATPase (25)
Akt (24)
Norepinephrine (24)
DNA Alkylator/Crosslinker (24)
Aurora Kinase (23)
Proton pump (23)
PARP (23)
TNF (22)
P-gp (22)
TRP/TRPV Channel (22)
MEK (21)
Virus Protease (21)
p38 MAPK (21)
NMDAR (21)
Epigenetic Reader Domain (21)
HSV (21)
PKC (20)
BTK (20)
HSP (20)
HIF/HIF Prolyl-Hydroxylase (18)
ALK (18)
RAAS (18)
ROS (18)
ERK (18)
HBV (17)
Trk receptor (17)
c-RET (17)
CXCR (17)
BCL (16)
GSK-3 (16)
AMPK (16)
HCV Protease (16)
Phosphatase (16)
Drug Metabolite (15)
Endothelin Receptor (15)
Carbonic Anhydrase (15)
MMP (15)
E1/E2/E3 Enzyme (15)
GNRH Receptor (15)
Retinoid Receptor (15)
Caspase (15)
DNA Alkylation (15)
SGLT (15)
Proteasome (14)
c-Fms (14)
TAM Receptor (14)
Antifolate (14)
Histone Methyltransferase (14)
Progesterone Receptor (14)
STAT (14)
Guanylate cyclase (13)
IL Receptor (13)
Chk (13)
DNA-PK (13)
Reverse Transcriptase (13)
TGF-beta/Smad (12)
S1P Receptor (12)
Lipoxygenase (12)
Mitochondrial Metabolism (12)
Neurokinin receptor (12)
MRP (12)
MAO (12)
LPL Receptor (12)
CFTR (12)
p53 (12)
HIF (12)
DHFR (12)
P2X Receptor (11)
Hedgehog/Smoothened (11)
Vasopressin Receptor (11)
IGF-1R (11)
Interleukin (11)
Gamma-secretase (11)
GluR (11)
Cannabinoid Receptor (11)
Transferase (11)
HMG-CoA Reductase (11)
Wnt/beta-catenin (11)
PKA (11)
Nrf2 (11)
Monoamine Oxidase (11)
Chloride channel (10)
FAK (10)
Antioxidant (10)
AChE (10)
ROCK (10)
Syk (10)
P2Y Receptor (10)
Sigma receptor (9)
Mdm2 (9)
CaMK (9)
S6 Kinase (9)
Indoleamine 2,3-Dioxygenase (IDO) (9)
PLK (9)
TLR (9)
CSF-1R (9)
Beta Amyloid (9)
IAP (9)
Antifection (9)
Ras (8)
Casein Kinase (8)
ATM/ATR (8)
OX Receptor (8)
ROS Kinase (8)
Leukotriene Receptor (8)
Phospholipase (8)
DNA Methyltransferase (8)
NADPH (8)
Smo (8)
JNK (8)
Kinesin (7)
Integrin (7)
ABC (7)
Antiviral (7)
Sirtuin (7)
Glucagon Receptor (7)
Thrombin (7)
Aromatase (7)
cholecystokinin (7)
DNA (7)
Monoamine Transporter (7)
Pim (7)
Ligand for E3 Ligase (7)
ribosome (6)
NO Synthase (6)
IκB/IKK (6)
IRAK (6)
PAK (6)
Glutathione Peroxidase (6)
CCR (6)
Histone Demethylase (6)
Fatty Acid Synthase (6)
RIP kinase (6)
LTR (6)
Isocitrate Dehydrogenase (IDH) (6)
Bradykinin Receptor (6)
CaSR (5)
GHSR (5)
PGE Synthase (5)
Tie-2 (5)
Serine Protease (5)
FXR (5)
GPCR19 (5)
NOD (5)
IFNAR (5)
Hydroxylase (5)
Ephrin Receptor (5)
DPP-4 (5)
Molecular Glues (4)
Xanthine Oxidase (4)
CRFR (4)
PD-1/PD-L1 (4)
Annexin A (4)
Aminopeptidase (4)
IDO (4)
Aryl Hydrocarbon Receptor (4)
Serine/threonin kinase (4)
Melanocortin Receptor (4)
PDK (4)
Oxytocin Receptor (4)
KSP (4)
Somatostatin (4)
Tyrosinase (4)
Melatonin Receptor (4)
Wee1 (4)
Amino Acids and Derivatives (4)
CGRP Receptor (4)
AhR (4)
GST (3)
Reductase (3)
RSV (3)
Protease-activated Receptor (3)
Monocarboxylate transporter (3)
CRM1 (3)
Cysteine Protease (3)
Liver X Receptor (3)
ROR (3)
NOD-like Receptor (NLR) (3)
YAP (3)
Adenosine deaminase (3)
Rho (3)
NAMPT (3)
Na-K-Cl cotransporter (3)
Neuropeptide Y Receptor (3)
OAT (3)
MAPK (3)
MT Receptor (3)
STING (3)
DNA gyrase (3)
Hexokinase (3)
DUB (3)
UGT (3)
Free radical scavengers (3)
p97 (2)
PROTACs (2)
Glutathione reductase (2)
NOS (2)
CAT (2)
Beta-Secretase (2)
Factor Xa (2)
transporter (2)
TOPK (2)
BCRP (2)
PERK (2)
Gap Junction Protein (2)
Discoidin Domain Receptor (DDR) (2)
Glucosidase (2)
Cell wall (2)
Imidazoline Receptor (2)
ATP Citrate Lyase (2)
MLK (2)
Lipid (2)
NEDD8 (2)
Telomerase (2)
Arginase (2)
Ligands for Target Protein for PROTAC (2)
PROTAC Linker (2)
Histone Acetyltransferase (2)
VDA (2)
Porcupine (2)
LDL (2)
Decarboxylase (2)
CD73 (2)
Acyltransferase (2)
PYK2 (2)
IRE1 (2)
LPA Receptor (2)
Myosin (1)
Adiponectin receptor (1)
Methionine Adenosyltransferase (MAT) (1)
HCN Channel (1)
MELK (1)
PAI-1 (1)
Immunology/Inflammation related (1)
Anion Exchanger (1)
Na+/Ca2+ Exchanger (1)
Pyroptosis (1)
MNK (1)
Thioredoxin (1)
MALT (1)
FAAH (1)
Neprilysin (1)
Thrombopoietin Receptor (1)
Hydrogenase (1)
cAMP (1)
Motilin Receptor (1)
NPC1L1 (1)
GluCls (1)
PAD (1)
ASK (1)
Apelin receptor (1)
BACE (1)
NADPH-oxidase (1)
BMI-1 (1)
OXPHOS (1)
VDAC (1)
Survivin (1)
N-Acetylglucosaminyltransferase (1)
Aquaporin (1)
KLF (1)
Galectin (1)
c-Myc (1)
PI4K (1)
GRK (1)
GTPase (1)
MTH1 (1)
SGK (1)
LHRH (1)
Hippo pathway (1)
GlyT (1)
Complement System (1)
Lipase (1)
Glucokinase (1)
ACK (1)
Platelet aggregation (1)
Glutaminase (1)
Stemness kinase (1)
RAR/RXR  (1)
DYRK (1)
Hck (1)
PAFR (1)
advanced glycation end products (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
CORPORATE
About Us Careers Privacy Notice Events & News Terms & Conditions
SUPPORT
Contact Us Worldwide Distributors Quality Control Technical Support
RESOURCE
Product Catalog Product Citations Signaling Pathways Solution Calculators
FOLLOW OUR
Social Network
Newsletter Subscription
Subscribe to receive our lastest product updates and special offers!
Corporate
Support
Resource
Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
TargetMol
Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved.