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Anti-Cancer Drug Library

Catalog No. L2150
  Library Compound List   Excel SDF

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 2478 anticancer drugs including FDA approved and compounds in clinical trial phases as Anticancer Drug Library that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Please contact us for prices and availability for the specification of product you are interested at.
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If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 2478 anticancer drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials), an effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug repositioning drug discovery;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc; involved in 15 different cancer research areas, such as lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2150)

Library Composition

AChR (97)
COX (91)
DNA/RNA Synthesis (73)
Adrenergic Receptor (70)
VEGFR (65)
EGFR (59)
Estrogen/progestogen Receptor (55)
PI3K (54)
Topoisomerase (53)
Potassium Channel (46)
Histamine Receptor (46)
Autophagy (45)
Dehydrogenase (45)
CDK (43)
PDE (42)
Antibacterial (42)
HDAC (41)
JAK (41)
PDGFR (40)
c-Kit (39)
FLT (38)
PPAR (36)
Microtubule Associated (35)
FGFR (35)
c-Met/HGFR (35)
Antibiotic (32)
Glucocorticoid Receptor (32)
mTOR (31)
Src (31)
GABA Receptor (30)
RAAS (30)
Sodium Channel (29)
Androgen Receptor (29)
NF-κB (26)
P450 (26)
Bcr-Abl (26)
Carbonic Anhydrase (23)
5-HT Receptor (23)
Raf (23)
Calcium Channel (22)
TNF (22)
Tyrosine Kinases (22)
Endogenous Metabolite (22)
Vitamin (20)
Dopamine Receptor (20)
Antifection (19)
MEK (18)
Epigenetic Reader Domain (18)
Akt (18)
HIV Protease (18)
DNA Alkylation (18)
MAO (18)
BTK (17)
ATPase (17)
Apoptosis (17)
HSP (16)
PKC (16)
ALK (16)
HER (16)
PARP (16)
IL Receptor (15)
p38 MAPK (15)
TAM Receptor (15)
Retinoid Receptor (14)
Reverse Transcriptase (14)
Aurora Kinase (13)
MRP (13)
c-RET (13)
HIF (12)
Chk (12)
GSK-3 (12)
CXCR (12)
DNA-PK (12)
Adenosine Receptor (12)
GPR (11)
Amino Acids and Derivatives (11)
NMDAR (11)
STAT (11)
TRP/TRPV Channel (10)
NADPH (10)
Integrin (10)
GNRH Receptor (10)
BCL (10)
Thrombin (10)
Trk receptor (10)
PKA (10)
Parasite (10)
Gamma-secretase (10)
AMPK (10)
HCV Protease (10)
Lipoxygenase (10)
Transferase (9)
Serine Protease (9)
Proteasome (9)
Caspase (9)
DNA gyrase (9)
PLK (9)
DHFR (9)
Hedgehog/Smoothened (9)
Antiviral (9)
ROS (9)
Syk (9)
Phosphatase (9)
TLR (9)
Glucokinase (8)
CSF-1R (8)
CCR (8)
IAP (8)
ribosome (8)
S1P Receptor (8)
Proton pump (8)
IGF-1R (8)
P-gp (8)
Mdm2 (8)
ERK (8)
p53 (8)
FAK (8)
MMP (8)
Phospholipase (8)
Wnt/beta-catenin (8)
HMG-CoA Reductase (7)
Prostaglandin Receptor (7)
IDO (7)
Histone Methyltransferase (7)
Hydroxylase (7)
ATM/ATR (7)
Aromatase (7)
CFTR (7)
Antioxidant (7)
Beta Amyloid (7)
JNK (7)
Tyrosinase (6)
Casein Kinase (6)
Histone Demethylase (6)
Antifungal (6)
HSV (6)
HBV (6)
S6 Kinase (6)
ABC (6)
Opioid Receptor (6)
IκB/IKK (6)
c-Fms (6)
Pim (6)
UGT (5)
NOS (5)
Kinesin (5)
E1/E2/E3 Enzyme (5)
cholecystokinin (5)
DNA Methyltransferase (5)
LTR (5)
Nucleoside Antimetabolite/Analog (5)
Sirtuin (5)
TGF-beta/Smad (5)
MPO (5)
Cysteine Protease (5)
AhR (5)
BACE (5)
SGLT (4)
NOD (4)
FXR (4)
Tie-2 (4)
Neurokinin receptor (4)
ROCK (4)
Factor Xa (4)
PAK (4)
Ephrin Receptor (4)
CaMK (4)
Chloride channel (4)
DPP-4 (4)
Fatty Acid Synthase (4)
Liver X Receptor (4)
Ras (4)
CAT (4)
Vasopressin Receptor (3)
LDL (3)
Acyltransferase (3)
Aminopeptidase (3)
Nrf2 (3)
PDK (3)
Free radical scavengers (3)
Norepinephrine (3)
HIF/HIF Prolyl-Hydroxylase (3)
CRM1 (3)
CETP (3)
Reductase (3)
Decarboxylase (3)
CaSR (3)
Na-K-Cl cotransporter (3)
DprE1 (3)
Cannabinoid Receptor (3)
GPCR19 (3)
Ferroptosis (3)
ROR (3)
Mitochondrial Metabolism (3)
Telomerase (3)
Thyroid hormone receptor(THR) (3)
Arginase (3)
Monocarboxylate transporter (2)
Monoamine Transporter (2)
Hexokinase (2)
NAMPT (2)
KSP (2)
Lipid (2)
GST (2)
Influenza Virus (2)
OX Receptor (2)
GlyT (2)
VDA (2)
Serine/threonin kinase (2)
c-Myc (2)
DNA (2)
Somatostatin (2)
PYK2 (2)
Protease-activated Receptor (2)
DUB (2)
ATP Citrate Lyase (2)
Endothelin Receptor (2)
PKM (2)
TOPK (2)
Rho (2)
Antifolate (2)
GHSR (2)
P2 Receptor (2)
GluR (2)
AChE (2)
advanced glycation end products (2)
Glutathione reductase (2)
Gap Junction Protein (2)
SARS-CoV (1)
Smo (1)
Sigma receptor (1)
SGK (1)
MNK (1)
Serotonin Transporter (1)
MELK (1)
Mitophagy (1)
MLK (1)
RAR/RXR (1)
RIP kinase (1)
PED (1)
P2X Receptor (1)
OAT (1)
p97 (1)
PAFR (1)
NPC1L1 (1)
PAI-1 (1)
NOD-like Receptor (NLR) (1)
MT Receptor (1)
Phosphorylase (1)
NO Synthase (1)
Porcupine (1)
NADPH-oxidase (1)
Reactive Oxygen Species (1)
Myosin (1)
Melatonin Receptor (1)
Lipase (1)
Stemness kinase (1)
Wee1 (1)
Oxytocin Receptor (1)
Electron transport (1)
Survivin (1)
Thioredoxin (1)
transporter (1)
Virus Protease (1)
Xanthine Oxidase (1)
Hydrogenase (1)
Hck (1)
Guanylate cyclase (1)
GTPase (1)
GluCls (1)
GRK (1)
Glutathione Peroxidase (1)
DNA Alkylator/Crosslinker (1)
Discoidin Domain Receptor (DDR) (1)
MAPK (1)
ASK (1)
STING (1)
ACAT (1)
ACK (1)
LHRH (1)
Annexin A (1)
Apoptosis inducer (1)
BCRP (1)
CPT (1)
Isocitrate Dehydrogenase (IDH) (1)
IRAK (1)
Beta-Secretase (1)
Integrase (1)
cAMP (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Cell wall (1)
OXPHOS (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE