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Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling
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Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

FDA-Approved Kinase Inhibitor Library

Catalog No. L1610
  Library Compound List   Excel SDF

Kinases are a class of enzymes that facilitates phosphorylation, by transferring phosphate groups from high-energy donor molecules, such as ATP, to specific target molecules. A common group of kinases are the protein kinases, which act on specific proteins to phosphorylate them and alter their activity. Protein kinases are involved in a range of cell signaling and regulatory processes and play an important role in cell growth, metabolism, differentiation and apoptosis. Protein kinases have been associated with many diseases, including cancer, inflammatory diseases, cardiovascular diseases and neurological disorders. Therefore, targeting protein kinases has emerged as a promising therapeutic strategy for the treatment of related diseases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 280 kinase inhibitors for specific targeting of kinases, ready for high-throughput screening and high-content screening.
  • All compounds have undergone preclinical studies and clinical trials, approved for marketing by FDA, EMA, PMDA, etc., with proven biological activity and safety.
  • Detailed instructions, compound structures, target information, IC50 values, activity descriptions, etc.
  • NMR, HPLC/LCMS and other assay techniques to ensure the correct structure and high purity of the product and reduce false positives.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L1610)

Library Composition

Autophagy (72)
Apoptosis (67)
Reactive Oxygen Species (33)
Endogenous Metabolite (31)
VEGFR (27)
EGFR (24)
c-Kit (24)
PDGFR (24)
Antibacterial (18)
Antibiotic (15)
FLT (14)
FGFR (14)
Parasite (13)
ROS (13)
Potassium Channel (12)
Bcr-Abl (12)
Tyrosine Kinases (11)
Calcium Channel (11)
c-Met/HGFR (11)
Src (11)
ALK (10)
NF-κB (10)
Raf (10)
Ferroptosis (10)
PKC (10)
JAK (9)
5-HT Receptor (9)
c-RET (9)
Mitophagy (9)
Adrenergic Receptor (8)
AMPK (8)
CaMK (8)
HER (7)
PI3K (7)
CDK (7)
Sodium Channel (7)
AChR (6)
HIV Protease (6)
COX (6)
mTOR (6)
MEK (6)
STAT (6)
Influenza Virus (6)
Histamine Receptor (6)
PKA (6)
P450 (6)
Trk receptor (6)
PDE (5)
TNF (5)
BTK (5)
ROCK (5)
GSK-3 (5)
DNA/RNA Synthesis (5)
TAM Receptor (5)
IκB/IKK (4)
ERK (4)
Xanthine Oxidase (4)
Phosphatase (4)
Dopamine Receptor (4)
SARS-CoV (4)
Antifungal (4)
c-Fms (3)
Microtubule Associated (3)
IGF-1R (3)
Adenosine Receptor (3)
p38 MAPK (3)
NADPH (3)
Ras (3)
Syk (3)
Virus Protease (3)
Tyrosinase (3)
HCV Protease (3)
Mitochondrial Metabolism (3)
Topoisomerase (3)
Dehydrogenase (3)
IRE1 (2)
Caspase (2)
MAPK (2)
Lipoxygenase (2)
Estrogen/progestogen Receptor (2)
FAK (2)
Glucokinase (2)
Glutathione Peroxidase (2)
Hexokinase (2)
HSV (2)
Aryl Hydrocarbon Receptor (2)
Norepinephrine (2)
Serotonin Transporter (2)
S1P Receptor (2)
Serine/threonin kinase (2)
PAK (2)
Nucleoside Antimetabolite/Analog (2)
Serine Protease (2)
Akt (2)
TRP/TRPV Channel (2)
PLK (2)
Retinoid Receptor (1)
HIF/HIF Prolyl-Hydroxylase (1)
HIF (1)
ROR (1)
S6 Kinase (1)
HDAC (1)
HMG-CoA Reductase (1)
Hck (1)
HBV (1)
GST (1)
GRK (1)
Glutathione reductase (1)
RAAS (1)
Antiviral (1)
Proton pump (1)
Phosphorylase (1)
PAD (1)
PDK (1)
Melatonin Receptor (1)
P-gp (1)
Phospholipase (1)
LPL Receptor (1)
LDL (1)
Hydroxylase (1)
JNK (1)
PKM (1)
PPAR (1)
Interleukin (1)
Integrin (1)
Prostaglandin Receptor (1)
Proteasome (1)
IL Receptor (1)
Gap Junction Protein (1)
GluR (1)
NOD-like Receptor (NLR) (1)
NADPH-oxidase (1)
Na-K-Cl cotransporter (1)
Neurokinin receptor (1)
Chloride channel (1)
Chk (1)
CFTR (1)
AChE (1)
CSF-1R (1)
ACK (1)
ADC Cytotoxin (1)
AhR (1)
Beta Amyloid (1)
Antifolate (1)
Aurora Kinase (1)
ATPase (1)
Na+/Ca2+ Exchanger (1)
CXCR (1)
ATP Citrate Lyase (1)
Ephrin Receptor (1)
SGLT (1)
Sigma receptor (1)
Sirtuin (1)
TGF-beta/Smad (1)
Thrombin (1)
TLR (1)
TOPK (1)
Decarboxylase (1)
Transferase (1)
YAP (1)
DNA Alkylator/Crosslinker (1)
DNA Alkylation (1)
DNA (1)
DHFR (1)
Monoamine Transporter (1)
MMP (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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