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Kinase Inhibitor Library

Catalog No. L1600
  Library Compound List   Excel SDF

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. A protein kinase modifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved in signal transduction. Various other kinases act on small molecules such as lipids, carbohydrates, amino acids, and nucleotides, either for signaling or to prime them for metabolic pathways.

TargetMol’s Tyrosine Kinase Inhibitors Library, containing 2160 kinase inhibitors, can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
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Product Description

  • A unique collection of 2160 kinase inhibitors for high throughput screening and high content screening for drug discovery in kinase related diseases;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include MAPK, PI3K, JAK, STAT, CDK, MEK, Insulin/IGF receptors, CaM Kinease II, PKA, JNK, PKC, RAF, EGFR, SAPK, GSK, MLCK, Src-family, IKK, PDGFR, VEGFR, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L1600)

Library Composition

Apoptosis (387)
Autophagy (288)
PI3K (146)
Reactive Oxygen Species (142)
EGFR (137)
CDK (136)
VEGFR (130)
Endogenous Metabolite (85)
JAK (81)
Akt (78)
mTOR (77)
FLT (76)
Src (75)
PDGFR (75)
NF-κB (73)
Antibacterial (69)
ERK (69)
FGFR (69)
p38 MAPK (69)
PKC (60)
Raf (58)
STAT (57)
AMPK (55)
c-Kit (55)
c-Met/HGFR (53)
Ras (49)
ROS (45)
GSK-3 (45)
ALK (45)
Bcr-Abl (43)
MEK (39)
Tyrosine Kinases (38)
JNK (38)
Glucokinase (37)
Aurora Kinase (37)
IκB/IKK (37)
TGF-beta/Smad (35)
MAPK (34)
BTK (34)
PKA (33)
Parasite (33)
DNA-PK (32)
c-RET (30)
HER (30)
Casein Kinase (30)
TAM Receptor (29)
Trk receptor (29)
ROCK (28)
S6 Kinase (28)
COX (27)
Influenza Virus (26)
Ferroptosis (26)
IGF-1R (26)
Antibiotic (25)
Serine/threonin kinase (24)
CaMK (24)
ATM/ATR (23)
PLK (23)
Potassium Channel (23)
Antifungal (23)
FAK (22)
HIV Protease (22)
TNF (22)
Aryl Hydrocarbon Receptor (20)
c-Fms (19)
Tyrosinase (19)
Mitophagy (19)
P450 (18)
Chk (17)
Antioxidant (17)
Syk (17)
RIP kinase (17)
Caspase (17)
DNA/RNA Synthesis (16)
PDK (16)
LRRK2 (16)
Mitochondrial Metabolism (15)
Calcium Channel (15)
Phosphatase (14)
PPAR (14)
PERK (14)
AChR (13)
AhR (13)
Dehydrogenase (13)
5-HT Receptor (13)
IL Receptor (12)
Interleukin (12)
IRAK (12)
MMP (12)
IRE1 (12)
Wnt/beta-catenin (11)
S1P Receptor (11)
Pim (11)
Rho (11)
Serine Protease (10)
PAK (10)
CSF-1R (10)
Virus Protease (10)
Adrenergic Receptor (10)
HSV (10)
Epigenetic Reader Domain (9)
Lipoxygenase (9)
Kinesin (9)
Ephrin Receptor (9)
SARS-CoV (8)
PDE (8)
DYRK (8)
Histamine Receptor (8)
PI4K (8)
Microtubule Associated (8)
PKM (8)
BCL (8)
Sodium Channel (8)
Adenosine Receptor (8)
HCV Protease (7)
Estrogen/progestogen Receptor (7)
IFNAR (7)
Topoisomerase (7)
HSP (7)
Discoidin Domain Receptor (DDR) (7)
HDAC (6)
MLK (6)
MNK (6)
Tie-2 (6)
Myosin (6)
SGK (6)
Estrogen Receptor/ERR (6)
Drug Metabolite (6)
NO Synthase (6)
GRK (6)
ACK (5)
Xanthine Oxidase (5)
LIM Kinase (5)
NADPH (5)
PYK2 (5)
E1/E2/E3 Enzyme (5)
SIK (5)
HIF/HIF Prolyl-Hydroxylase (5)
p53 (5)
TLR (5)
Beta Amyloid (5)
Antiviral (5)
ATPase (5)
Carbonic Anhydrase (4)
ASK (4)
Histone Methyltransferase (4)
P-gp (4)
Phospholipase (4)
TRP/TRPV Channel (4)
PARP (4)
Dopamine Receptor (4)
AChE (4)
HBV (4)
Integrin (4)
PTEN (4)
TOPK (4)
RAAS (4)
GABA Receptor (3)
PAI-1 (3)
c-Myc (3)
YAP (3)
Reverse Transcriptase (3)
Chloride channel (3)
Cannabinoid Receptor (3)
Prostaglandin Receptor (3)
Proteasome (3)
STING (3)
Transferase (3)
transporter (3)
Wee1 (3)
NOS (3)
OXPHOS (3)
Histone Acetyltransferase (3)
DNA Alkylation (3)
MAO (3)
LPL Receptor (3)
Hexokinase (3)
Hck (3)
Glutathione Peroxidase (3)
Fatty Acid Synthase (2)
MELK (2)
Anti-infection (2)
cAMP (2)
Aromatase (2)
LDL (2)
Sirtuin (2)
Antifection (2)
KSP (2)
DUB (2)
Beta-Secretase (2)
BCRP (2)
Retinoid Receptor (2)
HIF (2)
Serotonin Transporter (2)
BACE (2)
ROR (2)
Haspin Kinase (2)
Phosphorylase (2)
GTPase (2)
Nucleoside Antimetabolite/Analog (2)
GluR (2)
NAMPT (2)
Na+/Ca2+ Exchanger (2)
cholecystokinin (2)
CRISPR/Cas9 (2)
PD-1/PD-L1 (2)
Nrf2 (2)
NPC1L1 (2)
Norepinephrine (2)
NADPH-oxidase (2)
SGLT (1)
Gap Junction Protein (1)
Sigma receptor (1)
Gamma-secretase (1)
Glucagon Receptor (1)
Free radical scavengers (1)
Hippo pathway (1)
UGT (1)
VDA (1)
GST (1)
APC (1)
Stemness kinase (1)
Hedgehog/Smoothened (1)
Glutathione reductase (1)
GPR (1)
Antifolate (1)
Thrombin (1)
advanced glycation end products (1)
hCE (1)
Histone Demethylase (1)
GPX (1)
Fer/FerT kinase (1)
NOD (1)
RAR/RXR  (1)
ATP Citrate Lyase (1)
DHFR (1)
PGE Synthase (1)
CFTR (1)
cGAS (1)
Monoamine Oxidase (1)
Monoamine Transporter (1)
MRP (1)
PAD (1)
cell cycle arrest (1)
p97 (1)
Na-K-Cl cotransporter (1)
P2X Receptor (1)
P2 Receptor (1)
Neurokinin receptor (1)
Opioid Receptor (1)
Decarboxylase (1)
DNA (1)
CaSR (1)
FAAH (1)
Proton pump (1)
RSV (1)
HMG-CoA Reductase (1)
Hydroxylase (1)
Immunology/Inflammation related (1)
Indoleamine 2,3-Dioxygenase (IDO) (1)
Epoxide Hydrolase (1)
NOD-like Receptor (NLR) (1)
Leukotriene Receptor (1)
Melatonin Receptor (1)
Lipid (1)
Progesterone Receptor (1)
BMI-1 (1)
Bombesin Receptor (1)
Porcupine (1)
Platelet aggregation (1)
DNA Alkylator/Crosslinker (1)
FXR (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE