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Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
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Kinase Inhibitor Library

Catalog No. L1600
  Library Compound List   Excel SDF

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. A protein kinase modifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved in signal transduction. Various other kinases act on small molecules such as lipids, carbohydrates, amino acids, and nucleotides, either for signaling or to prime them for metabolic pathways.

TargetMol’s Kinase Inhibitor Library, containing 2720 kinase inhibitors/regulators , can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 2720 kinase inhibitors for high throughput screening and high content screening for drug discovery in kinase related diseases;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include MAPK, PI3K, JAK, STAT, CDK, MEK, Insulin/IGF receptors, CaM Kinease II, PKA, JNK, PKC, RAF, EGFR, SAPK, GSK, MLCK, Src-family, IKK, PDGFR, VEGFR, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files
Request Library Compound List (L1600)

Publications Cited TargetMol Libraries

1. Cancer Cell. 2019, 35(1): 125-139. e9. 2. Journal of Experimental & Clinical Cancer Research. 2023, 42(1): 1-22.. 3. Biochimica et Biophysica Acta (BBA)-Reviews on Cancer. 2023: 189021. 4. Frontiers in Cell and Developmental Biology. 2022.1. 5. International Journal of Molecular Sciences. 2022, 23(3): 1906. 6. International Journal of Molecular Sciences. 2022, 23(2): 776. 7. International Journal of Molecular Sciences. 2019, 20(22): 5780. 8. bioRxiv. 2023: 2023.06. 22.546046.. 9. Cell Stem Cell. 2022 Apr 29(4) 545–558.
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Library Composition

Apoptosis (388)
Autophagy (292)
CDK (231)
PI3K (202)
EGFR (190)
VEGFR (164)
JAK (111)
mTOR (111)
Akt (103)
p38 MAPK (102)
FLT (101)
ERK (101)
Src (100)
PDGFR (94)
PKC (87)
AMPK (84)
FGFR (83)
GSK-3 (82)
Raf (81)
c-Kit (75)
Ras (73)
NF-κB (71)
c-Met/HGFR (69)
Bcr-Abl (67)
Aurora Kinase (57)
ALK (57)
MAPK (56)
BTK (56)
JNK (52)
MEK (49)
Tyrosine Kinases (48)
Casein Kinase (47)
ROCK (47)
PKA (46)
Antibacterial (41)
Endogenous Metabolite (41)
Serine/threonin kinase (40)
IGF-1R (40)
DNA-PK (38)
c-RET (38)
TAM Receptor (37)
TGF-beta/Smad (36)
Epigenetic Reader Domain (36)
IκB/IKK (35)
CaMK (34)
Trk receptor (34)
S6 Kinase (33)
Glucosidase (32)
FAK (32)
RIP kinase (31)
HER (30)
PLK (30)
Glucokinase (30)
STAT (29)
TNF (28)
ATM/ATR (28)
c-Fms (28)
Parasite (27)
Syk (27)
Chk (25)
Pim (25)
PERK (24)
ROR (23)
IRAK (22)
DYRK (21)
Caspase (21)
COX (20)
LRRK2 (20)
PDK (19)
Mitophagy (19)
Antibiotic (19)
Influenza Virus (18)
Wnt/beta-catenin (18)
HIV Protease (18)
PAK (18)
DNA/RNA Synthesis (16)
IRE1 (16)
Tyrosinase (16)
Rho (16)
Reactive Oxygen Species (16)
PI4K (15)
Calcium Channel (15)
IL Receptor (15)
Ferroptosis (14)
Phosphatase (14)
ROS Kinase (14)
Ephrin Receptor (13)
5-HT Receptor (12)
P450 (12)
BCL (12)
AChR (12)
Antifungal (12)
PPAR (12)
Potassium Channel (11)
S1P Receptor (11)
CSF-1R (11)
Adrenergic Receptor (11)
MMP (11)
ROS (10)
PDE (10)
MNK (10)
MLK (10)
GRK (10)
Discoidin Domain Receptor (DDR) (10)
SGK (9)
HSV (9)
Kinesin (9)
Serine Protease (9)
NO Synthase (9)
Microtubule Associated (9)
Adenosine Receptor (9)
PKM (9)
Dehydrogenase (9)
Wee1 (8)
Sodium Channel (8)
Antiviral (8)
SARS-CoV (8)
Beta Amyloid (8)
PARP (8)
Interleukin (7)
HDAC (7)
Tie-2 (7)
Lipoxygenase (7)
AAK1 (AP2 associated kinase 1) (7)
Virus Protease (7)
Mitochondrial Metabolism (7)
SIK (7)
AChE (6)
TOPK (6)
Drug Metabolite (6)
P-gp (6)
MELK (6)
Topoisomerase (6)
Nrf2 (6)
Histamine Receptor (6)
LIM Kinase (6)
ACK (5)
TLR (5)
Integrin (5)
transporter (5)
LDL (5)
Histone Methyltransferase (5)
Ligand for E3 Ligase (5)
PYK2 (5)
Antioxidant (5)
HCV Protease (5)
Dopamine Receptor (5)
ASK (5)
Hippo pathway (5)
Carbonic Anhydrase (4)
Myosin (4)
Carboxypeptidase (4)
LPL Receptor (4)
DAPK (4)
TRP/TRPV Channel (4)
GTPase (4)
Estrogen/progestogen Receptor (4)
GluR (4)
HSP (3)
NOS (3)
Prostaglandin Receptor (3)
Sirtuin (3)
Transferase (3)
p53 (3)
PAI-1 (3)
Indoleamine 2,3-Dioxygenase (IDO) (3)
Ligands for Target Protein for PROTAC (3)
YAP (3)
Haspin Kinase (3)
Antifection (3)
Hexokinase (3)
Aryl Hydrocarbon Receptor (3)
MAO (3)
DNA Alkylation (3)
Hck (3)
ATPase (3)
Estrogen Receptor/ERR (3)
HBV (3)
cholecystokinin (3)
Glutathione Peroxidase (3)
HIF/HIF Prolyl-Hydroxylase (3)
IFNAR (3)
BACE (3)
E1/E2/E3 Enzyme (3)
Phospholipase (2)
HIF (2)
NADPH-oxidase (2)
Anti-infection (2)
Reverse Transcriptase (2)
Cannabinoid Receptor (2)
CRISPR/Cas9 (2)
PTEN (2)
Gamma-secretase (2)
Beta-Secretase (2)
RAAS (2)
DUB (2)
NADPH (2)
Serotonin Transporter (2)
Nucleoside Antimetabolite/Analog (2)
BCRP (2)
PROTACs (2)
FXR (2)
Proton pump (2)
Histone Acetyltransferase (2)
Chloride channel (2)
cAMP (2)
NAMPT (1)
Gap Junction Protein (1)
gp120/CD4 (1)
Liver X Receptor (1)
cell cycle arrest (1)
BMI-1 (1)
Antifolate (1)
MRP (1)
Melatonin Receptor (1)
RSV (1)
Sigma receptor (1)
Necroptosis (1)
CETP (1)
Fer/FerT kinase (1)
Histone Demethylase (1)
p97 (1)
RAR/RXR  (1)
Arrestin (1)
AhR (1)
MyD88 (1)
DHFR (1)
PD-1/PD-L1 (1)
NPC1L1 (1)
Protease-activated Receptor (1)
Phosphorylase (1)
Stemness kinase (1)
Norepinephrine (1)
Decarboxylase (1)
STING (1)
GPX (1)
Porcupine (1)
Acyltransferase (1)
Retinoid Receptor (1)
PGE Synthase (1)
Lipid (1)
Protease (1)
Aromatase (1)
ATP Citrate Lyase (1)
Androgen Receptor (1)
GPR (1)
DNA (1)
Thrombopoietin Receptor (1)
iGluR (1)
GABA Receptor (1)
Hydroxylase (1)
PAD (1)
FAAH (1)
Hedgehog/Smoothened (1)
RXFP receptor (1)
Bombesin Receptor (1)
Fatty Acid Synthase (1)
PROTAC Linker (1)
Opioid Receptor (1)
Monoamine Transporter (1)
NMDAR (1)
P2X Receptor (1)
cGAS (1)
Proteasome (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
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