FDA-Approved & Pharmacopeia Drug Library

Catalog No. L1010

Library Compound List Excel SDF

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

Approved drugs all have known and well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization. Hits from this set will provide a significant head start in any drug optimization program. In addition, a growing number of compounds have been identified from this library that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules.

TargetMol’s FDA-Approved & Pharmacopeia Drug Library collects 3158 compounds from approved institutions such as FDA, EMA, PMDA, NMPA, etc. or pharmacopoeia such as USP, BP, JP, etc., which can be used for drug repositioning and cell induction.

In addtion, we put the compounds that should be provided in the form of dry powder together to form Part B in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)

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please contact our compound library specialist for a customized compound library at inquiry@targetmol.com

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Product Description

3158 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
All compounds collected in this library are drugs approved by FDA, EMA, PMDA, NMPA, etc. or included in pharmacopoeia such as USP, BP, JP, etc.;
An effective tool for discovering new with old drugs and new drug target identification;
Covers various research areas, such as Cancer, Cardiovascular disease, Neuroscience, Immunology/Inflammation, respiratory system disease, etc.
More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
Structurally diverse, medicinally active, and cell permeable;
NMR and HPLC validated to ensure high purity and quality.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
Shipped with blue ice

Supporting Files

Library Handling Instructions (635 KB) Targetmol Library Catalog (13.2 MB) Request for Library Compostion in Excel and SDF files

Library Composition

Antibacterial (463)

Antibiotic (426)

Autophagy (373)

Endogenous Metabolite (327)

Apoptosis (291)

Adrenergic Receptor (172)

5-HT Receptor (170)

AChR (149)

COX (134)

Parasite (128)

Dopamine Receptor (118)

Histamine Receptor (106)

Antifungal (103)

DNA/RNA Synthesis (88)

Sodium Channel (88)

HIV Protease (85)

Calcium Channel (81)

Potassium Channel (78)

Topoisomerase (57)

Influenza Virus (54)

NF-κB (54)

Glucocorticoid Receptor (53)

Estrogen/progestogen Receptor (53)

Reactive Oxygen Species (52)

Ferroptosis (52)

P450 (49)

PDE (47)

GABA Receptor (44)

SARS-CoV (41)

RAAS (39)

Mitophagy (36)

Dehydrogenase (36)

HCV Protease (33)

EGFR (33)

VEGFR (32)

ribosome (31)

HSV (31)

AChE (30)

c-Kit (30)

PPAR (30)

PDGFR (29)

Nucleoside Antimetabolite/Analog (29)

Prostaglandin Receptor (29)

Serotonin Transporter (29)

Microtubule Associated (28)

Reverse Transcriptase (27)

Estrogen Receptor/ERR (27)

MAO (26)

Norepinephrine (25)

Opioid Receptor (25)

Proteasome (24)

ATPase (24)

Progesterone Receptor (24)

Virus Protease (24)

HBV (23)

iGluR (23)

TNF (22)

Antifection (22)

TRP/TRPV Channel (21)

Proton pump (21)

DNA Alkylator/Crosslinker (20)

Antioxidant (20)

Androgen Receptor (19)

Carbonic Anhydrase (19)

Monoamine Oxidase (19)

HDAC (18)

Thrombin (18)

FGFR (17)

FLT (17)

MMP (17)

ROS (16)

Adenosine Receptor (16)

Antiviral (15)

MRP (15)

JAK (15)

c-Met/HGFR (15)

IL Receptor (15)

Lipoxygenase (14)

GNRH Receptor (14)

Bcr-Abl (14)

Tyrosine Kinases (14)

NMDAR (14)

Drug Metabolite (14)

Phosphatase (14)

Antifolate (14)

DPP-4 (14)

Src (13)

PKC (13)

Retinoid Receptor (13)

GluR (13)

NO Synthase (13)

Transferase (13)

DHFR (12)

Raf (12)

Phospholipase (12)

Tyrosinase (12)

CDK (12)

Thyroid hormone receptor(THR) (12)

HMG-CoA Reductase (12)

Amino Acids and Derivatives (12)

AMPK (12)

Beta Amyloid (11)

PI3K (11)

P-gp (11)

Mitochondrial Metabolism (11)

PARP (11)

STAT (11)

ERK (11)

c-RET (10)

CaMK (10)

DNA gyrase (10)

ALK (10)

Factor Xa (10)

HIF/HIF Prolyl-Hydroxylase (9)

Nrf2 (9)

Interleukin (9)

Serine Protease (9)

MEK (9)

DNA Alkylation (9)

mTOR (8)

Vasopressin Receptor (8)

SGLT (8)

P2Y Receptor (8)

ABC (8)

Chloride channel (8)

TLR (8)

Akt (8)

CAT (8)

Neurokinin receptor (7)

Reductase (7)

HSP (7)

Aromatase (7)

p38 MAPK (7)

CFTR (7)

DNA (7)

HER (7)

Wnt/beta-catenin (7)

GPR (7)

Guanylate cyclase (7)

BCL (6)

Cysteine Protease (6)

Glutathione Peroxidase (6)

Anti-infection (6)

ROCK (6)

S1P Receptor (6)

Glucagon Receptor (6)

IκB/IKK (6)

Monoamine Transporter (6)

Integrin (6)

Sigma receptor (6)

CaSR (6)

Caspase (6)

Trk receptor (6)

NADPH (6)

TAM Receptor (6)

PKA (6)

Oxytocin Receptor (6)

Hedgehog/Smoothened (6)

BTK (6)

NOS (5)

Fatty Acid Synthase (5)

FAK (5)

DNA Methyltransferase (5)

Cell wall (5)

Histone Demethylase (5)

Cannabinoid Receptor (5)

Hydroxylase (5)

Endothelin Receptor (5)

LPL Receptor (5)

Serine/threonin kinase (5)

Lipid (5)

Histone Methyltransferase (5)

Xanthine Oxidase (5)

Annexin A (5)

TGF-beta/Smad (5)

Leukotriene Receptor (5)

PGE Synthase (5)

Neprilysin (4)

UGT (4)

Somatostatin (4)

IGF-1R (4)

NOD (4)

NOD-like Receptor (NLR) (4)

Ras (4)

Smo (4)

LTR (4)

FXR (4)

ROS Kinase (4)

GSK-3 (4)

Decarboxylase (4)

Melatonin Receptor (4)

cholecystokinin (3)

P2X Receptor (3)

Complement System (3)

CCR (3)

CETP (3)

p53 (3)

Arginase (3)

Aminopeptidase (3)

PAK (3)

CXCR (3)

c-Fms (3)

Syk (3)

Aryl Hydrocarbon Receptor (3)

Melanocortin Receptor (3)

Hexokinase (3)

Imidazoline Receptor (3)

Sirtuin (3)

GST (3)

GPCR19 (3)

Adenosine deaminase (3)

Glucosidase (3)

Glutathione reductase (3)

CGRP Receptor (3)

Gap Junction Protein (3)

Gamma-secretase (3)

MT Receptor (3)

Free radical scavengers (3)

AhR (3)

Thrombopoietin Receptor (2)

ROR (2)

Protease-activated Receptor (2)

RSV (2)

Acyltransferase (2)

S6 Kinase (2)

Adiponectin receptor (2)

Rho (2)

Telomerase (2)

TOPK (2)

YAP (2)

PLK (2)

Histone Acetyltransferase (2)

JNK (2)

Isocitrate Dehydrogenase (IDH) (2)

IRE1 (2)

Integrase (2)

Platelet aggregation (2)

Beta-Secretase (2)

HIF (2)

MAPK (2)

GlyT (2)

GluCls (2)

Epigenetic Reader Domain (2)

Ephrin Receptor (2)

DYRK (2)

DUB (2)

CRM1 (2)

LDL (2)

Indoleamine 2,3-Dioxygenase (IDO) (2)

Monocarboxylate transporter (2)

OAT (2)

PKM (2)

Na-K-Cl cotransporter (2)

PAFR (1)

Glucokinase (1)

cAMP (1)

PAD (1)

GHSR (1)

FAAH (1)

Casein Kinase (1)

Epoxide Hydrolase (1)

Phosphorylase (1)

PD-1/PD-L1 (1)

GRK (1)

Dynamin (1)

CSF-1R (1)

VDA (1)

Angiotensin-converting Enzyme (ACE) (1)

ACK (1)

CRISPR/Cas9 (1)

Chk (1)

Pyroptosis (1)

Taste receptor (1)

Hck (1)

IRAK (1)

Mdm2 (1)

MTH1 (1)

Liver X Receptor (1)

Lipase (1)

Na+/Ca2+ Exchanger (1)

NADPH-oxidase (1)

advanced glycation end products (1)

ATP Citrate Lyase (1)

NPC1L1 (1)

Aurora Kinase (1)

RAR/RXR (1)

Immunology/Inflammation related (1)

IFNAR (1)

IAP (1)

Hydrogenase (1)

RANKL/RANK (1)

Bradykinin Receptor (1)

OX Receptor (1)

BACE (1)

Library Information Sample

Empty	1000025-07-9	1000413-72-8	229005-80-5	1000787-75-6	946387-07-1	1000998-59-3	1175526-27-8	1001288-58-9	1001350-96-4	1001404-83-6	Empty
Empty	Vadadustat	TAK875	TAK-779	Tegobuvir	RN-1734	BMS-687453	AM211	FT011	BMS754807	AAI101	Empty
Empty	1001625-82-6	1001645-58-4	1001753-24-7	1001908-89-9	1002304-34-8	1002-84-2	100291-86-9	100299-08-9	10030-52-1	10040-45-6	Empty
Empty	RPW-24	SRT1720 hydrochloride	INH6	SRT 2183	AMG208	Pentadecanoic acid	Apiopaeonoside	Pemirolast potassium	L-Anserine nitrate salt	Sodium Picosulfate	Empty
Empty	100427-26-7	1004316-88-4	10045-45-1	100462-37-1	1004990-28-6	100-51-6	1005-24-9	1005264-47-0	1005334-57-5	1005342-46-0	Empty
Empty	Lercanidipine	Cobicistat	1-Ethyl-2-benzimidazolinone	ROSIRIDIN	PF-AKT400	Benzyl alcohol	1-Methylnicotinamide chloride	MX69	CVT-10216	LCL161	Empty
Empty	1005491-05-3	100-55-0	1005504-62-0	1005883-72-6	100643-71-8	1007207-67-1	10075-50-0	1007647-73-5	100784-20-1	10083-24-6	Empty
Empty	Tirasemtiv	Roniacol	Rg3039	Z433927330	Desloratadine	CH5132799	5-Bromoindole	Smurf1-IN-A01	Halosulfuron-methyl	Piceatannol	Empty
Empty	100872-83-1	100874-08-6	1009119-64-5	1009119-65-6	100929-71-3	1009298-09-2	1009298-59-2	100929-99-5	1009734-33-1	10097-84-4	Empty
Empty	ML346	SB 4	Daclatasvir	Daclatasvir dihydrochloride	NADPH (tetracyclohexanamine)	AZD8055	Vistusertib	PAβN dihydrochloride	HZ1157	Rotundine	Empty
Empty	1009816-48-1	1009817-63-3	1009820-21-6	100986-85-4	101001-34-7	1010411-21-8	1010-60-2	1011244-68-0	1011301-27-1	1011529-10-4	Empty
Empty	Thiamet G	B-AP15	Silmitasertib	Levofloxacin	Pamicogrel	GSK369796 Dihydrochloride	2-Chloronaphthoquinone	TFAP	Tenovin3	Azvudine	Empty
Empty	101152-94-7	101155-02-6	1011557-82-6	1011-74-1	101-20-2	1012054-59-9	101-21-3	101-26-8	101303-98-4	1013101-36-4	Empty
Empty	Milnacipran hydrochloride	BW-A78U	Tenovin-6	DL-Normetanephrine hydrochloride	Triclocarban	CUDC101	Chlorpropham	Mestinon	Zacopride hydrochloride	PF04691502	Empty
Empty	101-31-5	1013-69-0	1013750-77-0	1013753-99-5	10138-52-0	1013920-15-4	1013937-63-7	1014691-61-2	101477-54-7	101494-95-5	Empty
Empty	L-Hyoscyamine	Noreugenin	ML-030	BC-1382	Gadolinium chloride	Vorolanib	VTP-27999 TFA	GSK0660	Lomerizine hydrochloride	8-CHLOROQUINAZOLIN-4(1H)-ONE	Empty