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FDA-Approved & Pharmacopeia Drug Library

Catalog No. L1010
  Library Compound List   Excel SDF

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

Approved drugs all have known and well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization. Hits from this set will provide a significant head start in any drug optimization program. In addition, a growing number of compounds have been identified from this library that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules.

TargetMol’s FDA-Approved & Pharmacopeia Drug Library collects 3158 compounds from approved institutions such as FDA, EMA, PMDA, NMPA, etc. or pharmacopoeia such as USP, BP, JP, etc., which can be used for drug repositioning and cell induction.

In addtion, we put the compounds that should be provided in the form of dry powder together to form Part B in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Please contact us for prices and availability for the specification of product you are interested at.
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If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • 3158 compounds from marketed drugs for high throughput screening (HTS) and high content screening (HCS);
  • All compounds collected in this library are drugs approved by FDA, EMA, PMDA, NMPA, etc. or included in pharmacopoeia such as USP, BP, JP, etc.;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas, such as Cancer, Cardiovascular disease, Neuroscience, Immunology/Inflammation, respiratory system disease, etc.
  • More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L1010)

Library Composition

Antibacterial (459)
Antibiotic (427)
Autophagy (373)
Endogenous Metabolite (332)
Apoptosis (293)
Adrenergic Receptor (172)
5-HT Receptor (168)
AChR (146)
COX (131)
Parasite (129)
Dopamine Receptor (118)
Histamine Receptor (105)
Antifungal (104)
DNA/RNA Synthesis (92)
HIV Protease (87)
Sodium Channel (86)
Calcium Channel (79)
Potassium Channel (76)
Topoisomerase (56)
Reactive Oxygen Species (56)
Estrogen/progestogen Receptor (55)
Glucocorticoid Receptor (54)
Ferroptosis (53)
NF-κB (52)
Influenza Virus (52)
P450 (50)
PDE (49)
GABA Receptor (43)
SARS-CoV (40)
RAAS (39)
Mitophagy (37)
Dehydrogenase (36)
EGFR (33)
HCV Protease (33)
ribosome (32)
AChE (31)
PPAR (31)
VEGFR (31)
HSV (30)
c-Kit (30)
PDGFR (29)
MAO (29)
Microtubule Associated (29)
Serotonin Transporter (29)
Nucleoside Antimetabolite/Analog (29)
Estrogen Receptor/ERR (28)
Prostaglandin Receptor (28)
Reverse Transcriptase (27)
Norepinephrine (25)
Virus Protease (24)
ATPase (24)
Proteasome (24)
Opioid Receptor (23)
HBV (23)
Progesterone Receptor (23)
iGluR (23)
Antifection (22)
Proton pump (21)
Monoamine Oxidase (21)
TNF (20)
Antioxidant (20)
TRP/TRPV Channel (20)
DNA Alkylator/Crosslinker (20)
Thrombin (18)
Androgen Receptor (18)
Carbonic Anhydrase (18)
HDAC (18)
Adenosine Receptor (17)
ROS (17)
FLT (17)
FGFR (17)
MMP (17)
MRP (15)
c-Met/HGFR (15)
PKC (15)
GNRH Receptor (15)
JAK (15)
Lipoxygenase (14)
Bcr-Abl (14)
DPP-4 (14)
Phosphatase (14)
NMDAR (14)
IL Receptor (14)
Src (14)
Antifolate (14)
GluR (13)
NO Synthase (13)
Phospholipase (13)
Tyrosine Kinases (13)
AMPK (13)
Antiviral (13)
Retinoid Receptor (13)
Drug Metabolite (13)
Tyrosinase (12)
Mitochondrial Metabolism (12)
Raf (12)
Transferase (12)
Beta Amyloid (12)
HMG-CoA Reductase (12)
Amino Acids and Derivatives (12)
Thyroid hormone receptor(THR) (12)
DHFR (12)
CDK (12)
PI3K (11)
ERK (11)
P-gp (11)
PARP (11)
STAT (11)
ALK (10)
CaMK (10)
c-RET (10)
HIF/HIF Prolyl-Hydroxylase (10)
P2 Receptor (10)
Factor Xa (10)
DNA gyrase (10)
Interleukin (9)
Akt (9)
MEK (9)
DNA (9)
DNA Alkylation (9)
CAT (8)
Vasopressin Receptor (8)
NADPH (8)
mTOR (8)
SGLT (8)
Serine Protease (8)
Chloride channel (8)
p38 MAPK (8)
ABC (8)
PKA (7)
Neurokinin receptor (7)
TLR (7)
Reductase (7)
HSP (7)
IκB/IKK (7)
Aromatase (7)
Integrin (7)
Guanylate cyclase (7)
CFTR (7)
Trk receptor (7)
HER (7)
GPR (7)
Wnt/beta-catenin (7)
Monoamine Transporter (6)
Anti-infection (6)
Caspase (6)
BCL (6)
ADC Cytotoxin (6)
BTK (6)
NOS (6)
TAM Receptor (6)
Hedgehog/Smoothened (6)
Sigma receptor (6)
Oxytocin Receptor (6)
Cysteine Protease (6)
ROCK (6)
Glutathione Peroxidase (6)
Glucagon Receptor (6)
S1P Receptor (6)
Serine/threonin kinase (5)
Xanthine Oxidase (5)
TGF-beta/Smad (5)
LPL Receptor (5)
IGF-1R (5)
Lipid (5)
Annexin A (5)
Cell wall (5)
Histone Demethylase (5)
Histone Methyltransferase (5)
Hydroxylase (5)
CaSR (5)
Cannabinoid Receptor (5)
DNA Methyltransferase (5)
GSK-3 (5)
Endothelin Receptor (5)
Fatty Acid Synthase (5)
Smo (4)
Somatostatin (4)
LTR (4)
Leukotriene Receptor (4)
Decarboxylase (4)
Neprilysin (4)
FXR (4)
FAK (4)
NOD (4)
UGT (4)
NOD-like Receptor (NLR) (4)
Glucokinase (4)
Ras (4)
Melatonin Receptor (4)
PLK (3)
p53 (3)
GPCR19 (3)
Complement System (3)
CXCR (3)
Free radical scavengers (3)
PAK (3)
GST (3)
PGE Synthase (3)
Gap Junction Protein (3)
Gamma-secretase (3)
Glutathione reductase (3)
CETP (3)
cholecystokinin (3)
Indoleamine 2,3-Dioxygenase (IDO) (3)
Adenosine deaminase (3)
c-Fms (3)
Melanocortin Receptor (3)
AhR (3)
CCR (3)
Sirtuin (3)
Syk (3)
Aminopeptidase (3)
MT Receptor (3)
Arginase (3)
Aryl Hydrocarbon Receptor (3)
Acyltransferase (2)
Protease-activated Receptor (2)
Adiponectin receptor (2)
Thrombopoietin Receptor (2)
DYRK (2)
DUB (2)
TOPK (2)
RSV (2)
Telomerase (2)
Rho (2)
Epigenetic Reader Domain (2)
CRM1 (2)
ROR (2)
CGRP Receptor (2)
S6 Kinase (2)
Ephrin Receptor (2)
YAP (2)
Na-K-Cl cotransporter (2)
Hexokinase (2)
Monocarboxylate transporter (2)
Integrase (2)
P2X Receptor (2)
GlyT (2)
IRE1 (2)
HIF (2)
Isocitrate Dehydrogenase (IDH) (2)
JNK (2)
LDL (2)
GluCls (2)
Histone Acetyltransferase (2)
MAPK (2)
Platelet aggregation (2)
OAT (2)
Beta-Secretase (1)
Bradykinin Receptor (1)
Immunology/Inflammation related (1)
MTH1 (1)
Taste receptor (1)
BACE (1)
IRAK (1)
Aurora Kinase (1)
ATP Citrate Lyase (1)
IFNAR (1)
Angiotensin-converting Enzyme (ACE) (1)
advanced glycation end products (1)
VDA (1)
Mdm2 (1)
Lipase (1)
ACK (1)
cAMP (1)
Epoxide Hydrolase (1)
Na+/Ca2+ Exchanger (1)
p97 (1)
Liver X Receptor (1)
PDK (1)
Pyroptosis (1)
Dynamin (1)
GHSR (1)
RAR/RXR  (1)
PD-1/PD-L1 (1)
PAFR (1)
PAD (1)
CSF-1R (1)
CRISPR/Cas9 (1)
Casein Kinase (1)
GRK (1)
OX Receptor (1)
Hck (1)
Chk (1)
Nrf2 (1)
NPC1L1 (1)
Hydrogenase (1)
FAAH (1)
NADPH-oxidase (1)
IAP (1)
PKM (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE