Home Tools
Log in
Cart

Anti-Cancer Metabolism Compound Library

Catalog No. L2130
  Library Compound List   Excel SDF

Cancer metabolism has emerged as an important area of research in recent years. Reprogramming of the cellular energy metabolism, essential for cancer cell proliferation and tumor development, constitutes an emerging hallmark of cancer and may serve as a biochemical basis for new therapeutic intervention. From the abnormal aerobic glycolysis effect in tumor cells was first discovered by German scientist Warburg in the early 1920s to now on all aspects of tumor metabolic activity (sugar, fat, amino acids, etc.) analysis and complex metabolic regulation network discovery, the study of tumor metabolism has entered into a more striking height. Distinct metabolic pathways (glycolysis and glutaminolysis), key regulators of aerobic glycolysis (AMPK, mTOR, HIF-1, c-Myc, p53, etc.), and key metabolism enzymes (PKM, HK, PFK, PK, IDH, GLS) might be the key targets for tumor therapeutics. Developing inhibitors targeting dysregulated metabolic enzymes and pathways may represent a promising strategy to overcome drug resistance in cancer therapy.

A unique collection of 1280 cancer cellular metabolism related compounds by TargetMol can be used for cancer related research and high throughput and high content screening for anti-cancer drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Please contact us for prices and availability for the specification of product you are interested at.
Get quote
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
Request Library
Get quote

Product Description

  • A unique collection of 1280 cancer cellular metabolism related compounds for cancer research and high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials;
  • Covers 16 major targets related to cancer cellular metabolism (glucose, proteins, lipids and nucleic acids) including ACL, CA, FASN, GLUT, GLS, HMG-CoA, MAGL, MCTs, PDH, PDK, PKM, etc.; Effect tool for research in cancer metabolism and anti-cancer drug screening.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2130)

Library Composition

PI3K (103)
Dehydrogenase (93)
Src (69)
PPAR (61)
mTOR (57)
Bcr-Abl (46)
Glucocorticoid Receptor (37)
Akt (36)
Raf (34)
GSK-3 (32)
AMPK (32)
Carbonic Anhydrase (30)
p53 (28)
CDK (27)
DNA-PK (26)
HIF (25)
P450 (23)
Ras (23)
Glucokinase (22)
Phospholipase (21)
Phosphatase (21)
COX (21)
c-Kit (20)
GluR (20)
ERK (20)
Sirtuin (20)
VEGFR (20)
PDGFR (19)
ATPase (19)
Lipoxygenase (19)
S6 Kinase (18)
ATM/ATR (18)
NF-κB (17)
MEK (17)
FLT (16)
IDO (16)
Reductase (16)
EGFR (15)
HMG-CoA Reductase (15)
DPP-4 (15)
Autophagy (14)
PDK (13)
Fatty Acid Synthase (13)
IGF-1R (13)
FGFR (13)
Mdm2 (12)
FXR (12)
DNA/RNA Synthesis (12)
SGLT (12)
Mitochondrial Metabolism (11)
Aurora Kinase (11)
Liver X Receptor (10)
PKC (10)
Apoptosis (10)
HIF/HIF Prolyl-Hydroxylase (10)
c-Met/HGFR (9)
c-RET (9)
Rho (9)
FAAH (9)
PKA (8)
ROR (8)
Potassium Channel (8)
c-Myc (8)
Wnt/beta-catenin (8)
c-Fms (7)
DHFR (7)
AChR (7)
Estrogen/progestogen Receptor (7)
PKM (7)
JAK (7)
STAT (7)
Lipase (7)
Chk (6)
LRRK2 (6)
MMP (6)
Amino Acids and Derivatives (6)
Sodium Channel (6)
NADPH (6)
p38 MAPK (6)
Casein Kinase (6)
Calcium Channel (6)
transporter (6)
NAMPT (5)
NADPH-oxidase (5)
NOS (5)
Epigenetic Reader Domain (5)
Endogenous Metabolite (5)
Acetyl-CoA Carboxylase (5)
Lipid (5)
PDE (5)
Nrf2 (5)
Histone Methyltransferase (4)
GABA Receptor (4)
FAK (4)
MAPK (4)
ALK (4)
BCL (4)
CETP (4)
TNF (4)
Tyrosine Kinases (4)
NMDAR (4)
SGK (4)
TAM Receptor (4)
ROS (4)
NPC1L1 (4)
BTK (3)
IL Receptor (3)
ATP Citrate Lyase (3)
Adrenergic Receptor (3)
Tyrosinase (3)
Glutaminase (3)
TRP/TRPV Channel (3)
Caspase (3)
CAT (3)
Antiviral (3)
Microtubule Associated (3)
MTH1 (3)
Hck (3)
ROCK (3)
Acyltransferase (3)
GlyT (3)
Retinoid Receptor (3)
Syk (3)
Serine Protease (3)
Histone Demethylase (3)
Histamine Receptor (3)
MAO (3)
CSF-1R (3)
Monocarboxylate transporter (3)
Hexokinase (2)
HDAC (2)
Antifection (2)
HIV Protease (2)
HSV (2)
Reactive Oxygen Species (2)
IAP (2)
Antibacterial (2)
Annexin A (2)
Indoleamine 2,3-Dioxygenase (IDO) (2)
Integrin (2)
JNK (2)
LTR (2)
AhR (2)
SIK (2)
Trk receptor (2)
UGT (2)
ACAT (2)
HCV Protease (2)
Glutathione reductase (2)
GTPase (2)
PI4K (2)
MLK (2)
Antioxidant (2)
ABC (2)
PLK (2)
DNA Alkylation (2)
MPO (2)
MRP (2)
Ephrin Receptor (2)
CaMK (2)
CFTR (2)
Chloride channel (2)
PARP (2)
Arginase (2)
GPCR19 (2)
Glutathione Peroxidase (2)
GPR (2)
Parasite (2)
ACK (1)
Vitamin (1)
S1P Receptor (1)
RAAS (1)
OXPHOS (1)
NO Synthase (1)
PYK2 (1)
Serine/threonin kinase (1)
PTEN (1)
Proteasome (1)
PAK (1)
Prostaglandin Receptor (1)
Transferase (1)
Topoisomerase (1)
p97 (1)
PAI-1 (1)
Stearoyl-CoA Desaturase (SCD) (1)
Phosphorylase (1)
Thrombin (1)
Pim (1)
Melatonin Receptor (1)
RAR/RXR (1)
iGluR (1)
Hedgehog/Smoothened (1)
GPX (1)
Antifungal (1)
Histone Acetylation (1)
Opioid Receptor (1)
Antibiotic (1)
HSP (1)
Glucagon Receptor (1)
Hydroxylase (1)
BACE (1)
BMI-1 (1)
Ferroptosis (1)
FABP (1)
Reverse Transcriptase (1)
Isocitrate Dehydrogenase (IDH) (1)
IκB/IKK (1)
Cannabinoid Receptor (1)
Keap1-Nrf (1)
LDL (1)
cell cycle arrest (1)
Decarboxylase (1)
Androgen Receptor (1)
Cysteine Protease (1)
CPT (1)
MELK (1)
cholecystokinin (1)
5-HT Receptor (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE