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Nuclear Receptor Inhibitors Library

Catalog No. L1510
  Library Compound List   Excel SDF

Nuclear receptors are a class of proteins, different from membrane receptors located in the cell membrane, found within cells that are responsible for sensing steroid and thyroid hormones and certain other molecules. Nuclear receptors have the ability to directly bind to DNA and regulate the expression of adjacent genes, hence these receptors are classified as transcription factors, thereby controlling the development, homeostasis, and metabolism of the organism. Over the last 15 years a growing number of nuclear receptors have been identified that coordinate genetic networks regulating lipid metabolism and energy utilization and underlie the pathogenesis of metabolic diseases, such as obesity, type II diabetes, hypertension, and cardiovascular disease.

TargetMol collects 420 reported compounds targeting nuclear receptors as Nuclear Receptor Compound Library, which can be used for research in nuclear receptor signaling and related diseases, and high throughput and high content screening for drug discovery.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
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Product Description

  • A unique collection of 420 nuclear receptor signaling targeted compounds for high throughput and high content screening;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

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Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
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Library Composition

Estrogen/progestogen Receptor (91)
PPAR (83)
Glucocorticoid Receptor (62)
Androgen Receptor (48)
Retinoid Receptor (20)
FXR (18)
Thyroid hormone receptor(THR) (15)
COX (10)
Liver X Receptor (10)
ROR (9)
NF-κB (8)
Vitamin (8)
P450 (8)
Estrogen Receptor/ERR (7)
Wnt/beta-catenin (6)
Autophagy (5)
Annexin A (4)
ROS (3)
Potassium Channel (3)
AMPK (3)
GPR (3)
GPCR19 (3)
Akt (3)
Adrenergic Receptor (3)
IL Receptor (3)
BCL (2)
VEGFR (2)
DNA/RNA Synthesis (2)
transporter (2)
GABA Receptor (2)
Endogenous Metabolite (2)
GR (2)
Reductase (2)
MMP (2)
RAR/RXR (2)
MPO (2)
MRP (2)
Lipoxygenase (2)
PDE (2)
Melatonin Receptor (1)
MAO (1)
LDL (1)
Antibiotic (1)
Antioxidant (1)
Apoptosis (1)
Aromatase (1)
JNK (1)
Hydroxylase (1)
Calcium Channel (1)
CaMK (1)
Cannabinoid Receptor (1)
Caspase (1)
c-Kit (1)
c-Met/HGFR (1)
HER (1)
Cysteine Protease (1)
HCV Protease (1)
AhR (1)
ABC (1)
AChR (1)
Tyrosinase (1)
RAAS (1)
Sirtuin (1)
STAT (1)
TAM Receptor (1)
Thrombin (1)
GSK-3 (1)
TNF (1)
Progesterone Receptor (1)
PKC (1)
GNRH Receptor (1)
Phosphorylase (1)
Phospholipase (1)
Phosphatase (1)
p53 (1)
Opioid Receptor (1)
Nrf2 (1)
NOS (1)
GluR (1)
EGFR (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE