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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 7234 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 7234 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
COX
Antibacterial
Adrenergic Receptor
DNA/RNA Synthesis
NF-κB
CDK
PI3K
Potassium Channel
EGFR
Reactive Oxygen Species
Calcium Channel
P450
VEGFR
Antibiotic
Sodium Channel
Dopamine Receptor
GABA Receptor
HDAC
PPAR
Parasite
Histamine Receptor
TRP/TRPV Channel
JAK
mTOR
Akt
p38 MAPK
Antifungal
AChR
Src
ERK
Wnt/beta-catenin
FLT
PDGFR
Estrogen Receptor/ERR
STAT
HIV Protease
AMPK
FGFR
PARP
Dehydrogenase
Nucleoside Antimetabolite/Analog
GSK-3
iGluR
Raf
Influenza Virus
Microtubule Associated
Glucocorticoid Receptor
Caspase
BCL
Estrogen/progestogen Receptor
c-Met/HGFR
Topoisomerase
TNF
c-Kit
Androgen Receptor
Epigenetic Reader Domain
Ras
Ferroptosis
Bcr-Abl
Sirtuin
HSP
Aurora Kinase
PKC
MMP
TGF-beta/Smad
ATPase
Histone Methyltransferase
ALK
Antioxidant
JNK
Mitophagy
PDE
MAPK
Prostaglandin Receptor
MEK
Tyrosine Kinases
IL Receptor
ROCK
HER
IκB/IKK
DUB
Serine/threonin kinase
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p53
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DNA-PK
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NO Synthase
NMDAR
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Adenosine Receptor
IGF-1R
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P2X Receptor
S6 Kinase
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DHFR
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IRE1
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transporter
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DNA Alkylation
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ABC
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ROS Kinase
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Serine Protease
CSF-1R
IAP
DNA
SGLT
GPCR19
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Sigma receptor
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YAP
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Reductase
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STING
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Bradykinin Receptor
Angiotensin-converting Enzyme (ACE)
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cGAS
hCE
CRFR
HuR
Neprilysin
CGRP Receptor

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