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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 8700 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 8700 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
COX
NF-κB
Adrenergic Receptor
DNA/RNA Synthesis
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Reactive Oxygen Species
Histamine Receptor
Calcium Channel
P450
VEGFR
Antibiotic
Sodium Channel
JAK
GABA Receptor
HDAC
Parasite
PPAR
TRP/TRPV Channel
mTOR
GPR
AChR
ERK
Akt
Antifungal
Src
Prostaglandin Receptor
HIV Protease
Wnt/beta-catenin
FLT
p38 MAPK
Adenosine Receptor
Estrogen Receptor/ERR
Opioid Receptor
PDGFR
STAT
PARP
Microtubule Associated
GSK-3
Nucleoside Antimetabolite/Analog
AMPK
Dehydrogenase
Raf
FGFR
Caspase
TNF
Topoisomerase
Estrogen/progestogen Receptor
iGluR
Influenza Virus
Glucocorticoid Receptor
BCL
Epigenetic Reader Domain
c-Kit
c-Met/HGFR
Androgen Receptor
Antioxidant
Cannabinoid Receptor
Ferroptosis
Bcr-Abl
Histone Methyltransferase
HSP
PKC
ATPase
Sirtuin
MMP
TGF-beta/Smad
IL Receptor
Aurora Kinase
Ras
PDE
ALK
JNK
MAPK
Kras
Phosphatase
HER
NO Synthase
Tyrosine Kinases
MEK
Mitophagy
P-gp
ROCK
DUB
IκB/IKK
ADC Cytotoxin
p53
Serine/threonin kinase
SARS-CoV
Lipoxygenase
NMDAR
CXCR
Virus Protease
ROS
HIF/HIF Prolyl-Hydroxylase
DNA-PK
S1P Receptor
Neurokinin receptor
P2X Receptor
HSV
IGF-1R
LPL Receptor
Hedgehog/Smoothened
PKA
E1/E2/E3 Enzyme
Drug Metabolite
Nrf2
NOD
S6 Kinase
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BTK
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HIF
FAK
NOS
GluR
ATM/ATR
PLK
Sigma receptor
Serotonin Transporter
Interleukin
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Chloride channel
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Casein Kinase
TAM Receptor
Proteasome
HBV
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Norepinephrine
Tyrosinase
Chk
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Trk receptor
HCV Protease
PERK
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Pim
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IRAK
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SGLT
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PDK
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P2Y Receptor
Antifection
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Bradykinin Receptor
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DHFR
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cAMP
DNA Methyltransferase
cholecystokinin
CFTR
Transferase
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CCR
OX Receptor
transporter
LPA Receptor
PROTACs
Histone Demethylase
GNRH Receptor
Vasopressin Receptor
CaMK
DNA
PI4K
ROS Kinase
PD-1/PD-L1
Integrin
NADPH
GTPase
Progesterone Receptor
Antifolate
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IRE1
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Kinesin
ABC
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IAP
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PTEN
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Acyltransferase
MLK
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CRM1
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Liver X Receptor
PYK2
Glutaminase
MT Receptor
APC
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PSMA
OAT
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CRFR
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Hydroxylase
cell cycle arrest
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ribosome
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Oxytocin Receptor
CGRP Receptor
SGK
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IDO
Adiponectin receptor
DNA gyrase
Hexokinase
PAD
Xanthine Oxidase
KSP
ATP Citrate Lyase
Aminopeptidase
TSH Receptor
PAI-1
Methionine Adenosyltransferase (MAT)
Hippo pathway
Aquaporin
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Discoidin Domain Receptor (DDR)
p97
Adenylyl cyclase
RAR/RXR 
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Hck
RANKL/RANK
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AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
HCN Channel
CD73
Decarboxylase
Pyroptosis
Carboxypeptidase
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Imidazoline Receptor
CAT
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gp120/CD4
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OXPHOS
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DAPK
Gap Junction Protein
lysosomal autophagy
advanced glycation end products
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CD38
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NUDIX hydrolase
Piezo Channel
Dynamin
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N-Acetylglucosaminyltransferase
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FLAP
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GlyT
Anion Exchanger
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
Thrombopoietin Receptor
cGAS
hCE
Neprilysin
RXFP receptor

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