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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 9019 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 9019 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
COX
DNA/RNA Synthesis
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Reactive Oxygen Species
Histamine Receptor
Calcium Channel
VEGFR
Antibiotic
Cytochromes P450
Sodium Channel
HDAC
GABA Receptor
PPAR
Parasite
TRP/TRPV Channel
mTOR
Akt
GPR
ERK
AChR
JAK
Wnt/beta-catenin
Antifungal
Src
Prostaglandin Receptor
HIV Protease
STAT
FLT
Adenosine Receptor
Estrogen Receptor/ERR
PARP
Opioid Receptor
p38 MAPK
PDGFR
Microtubule Associated
Dehydrogenase
Nucleoside Antimetabolite/Analog
AMPK
GSK-3
FGFR
Raf
Topoisomerase
Epigenetic Reader Domain
TNF
Estrogen/progestogen Receptor
Bcl-2 Family
Influenza Virus
Caspase
Glucocorticoid Receptor
iGluR
Antioxidant
c-Met/HGFR
Histone Methyltransferase
Androgen Receptor
Ferroptosis
c-Kit
HSP
Cannabinoid Receptor
Bcr-Abl
PKC
MMP
ALK
ATPase
Sirtuin
TGF-beta/Smad
Phosphatase
Kras
IL Receptor
Ras
Aurora Kinase
PDE
HER
JNK
MAPK
Tyrosine Kinases
MEK
DUB
IκB/IKK
NO Synthase
ROCK
P-gp
ADC Cytotoxin
Mitophagy
p53
ROS
Lipoxygenase
SARS-CoV
Serine/threonin kinase
Virus Protease
NMDAR
CXCR
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
DNA-PK
Hedgehog/Smoothened
HSV
IGF-1R
Neurokinin receptor
PKA
RIP kinase
P2X Receptor
Nrf2
NOD
LPL Receptor
BTK
E1/E2/E3 Enzyme
Drug Metabolite
c-RET
TLR
S6 Kinase
FAK
Antiviral
Cholinesterase (ChE)
HIF
Interleukin
ATM/ATR
PLK
Sigma receptor
NOS
Mitochondrial Metabolism
GluR
TAM Receptor
Chloride channel
Proton pump
PERK
Serotonin Transporter
Casein Kinase
Tyrosinase
Proteasome
HBV
Chk
Norepinephrine
RAAS
Trk receptor
Phospholipase
Mdm2
HCV Protease
Rho
Gamma-secretase
Protease-activated Receptor
DNA Alkylator/Crosslinker
Histone Demethylase
Pim
Endothelin Receptor
Beta Amyloid
Carbonic Anhydrase
Neuropeptide Y Receptor
IRAK
PROTACs
Glucagon Receptor
SGLT
Retinoid Receptor
PDK
Syk
P2Y Receptor
MAO
Antifection
Guanylate cyclase
Smo
Bradykinin Receptor
DHFR
Fatty Acid Synthase
Vasopressin Receptor
cAMP
transporter
Reverse Transcriptase
c-Fms
Melanocortin Receptor
PD-1/PD-L1
Transferase
DYRK
c-Myc
DNA
Histone Acetyltransferase
LPA Receptor
DNA Methyltransferase
cholecystokinin
CFTR
DNA Alkylation
OX Receptor
CaMK
Anti-infection
ROS Kinase
Integrin
GNRH Receptor
Leukotriene Receptor
IRE1
Kinesin
NADPH
Progesterone Receptor
Antifolate
IAP
ABC Transporter
PI4K
NOD-like Receptor (NLR)
Monoamine Oxidase
YAP
GTPase
Serine Protease
Neurotensin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Somatostatin
GHSR
HMG-CoA Reductase
Monocarboxylate transporter
Reductase
MRP
CSF-1R
Immunology/Inflammation related
Aromatase
GRK
CCR
GPCR19
Ligand for E3 Ligase
AhR
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Melatonin Receptor
CaSR
Aryl Hydrocarbon Receptor
Bombesin Receptor
FXR
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Apelin receptor
LTR
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Glucosidase
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PAK
Wee1
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Acyltransferase
STING
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Tie-2
OCT
Cysteine Protease
Glutaminase
SIK
Annexin A
UGT
LDL
Molecular Glues
Isocitrate Dehydrogenase (IDH)
PTEN
GPX
Hydroxylase
MLK
Melanin-concentrating Hormone Receptor (MCHR)
CRM1
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Liver X Receptor
PYK2
Glucokinase
NAMPT
PAFR
MT Receptor
Lipid
PSMA
Survivin
OAT
CRFR
MELK
RSV
GST
ribosome
SGK
Cell Cycle Arrest
MTH1
DPP-4
FAAH
ACK1
Xanthine Oxidase
Beta-Secretase
Porcupine
ASK
Methionine Adenosyltransferase (MAT)
CRISPR/Cas9
Oxytocin Receptor
CGRP Receptor
Discoidin Domain Receptor (DDR)
Platelet aggregation
BMI-1
PKM
NPC1L1
MALT
ROR
TOPK
Kisspeptin
VDAC
Vitamin
IDO
Adiponectin Receptor
DNA gyrase
Hexokinase
PAD
KSP
ATP Citrate Lyase
LRRK2
Aminopeptidase
Decarboxylase
TSH Receptor
PAI-1
Hippo pathway
Aquaporin
Adenosine Deaminase
p97
Adenylyl Cyclase
RAR/RXR 
Galectin
AAK1
Hck
RANKL/RANK
Haspin Kinase
Na-K-Cl cotransporter
HCN Channel
Epoxide Hydrolase
Transketolase
CD73
Pyroptosis
Carboxypeptidase
KLF
Complement System
NADPH-oxidase
Imidazoline Receptor
EBI2/GPR183
NEDD8
MyD88
Arginase
Sodium-dependent phosphate transporter
Cell wall
Lipase
gp120/CD4
VDA
Factor Xa
OXPHOS
Glutathione reductase
AIM2
GluCls
HuR
Protease
RXFP receptor
Gap Junction Protein
DAPK
Lysosomal Autophagy
Thyroid hormone receptor(THR)
Advanced Glycation End Products
Transaminase
Hydrogenase
CD38
CYP19A1
NUDIX hydrolase
Piezo Channel
Dynamin
Neuropeptide W
Necroptosis
N-Acetylglucosaminyltransferase
Stemness kinase
Amylase
FLAP
Phosphorylase
GlyT
Anion Exchanger
PROTAC Linker
Thioredoxin
Stearoyl-CoA Desaturase (SCD)
Angiotensin-converting Enzyme (ACE)
Thrombopoietin Receptor
cGAS
hCE
Neprilysin

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